Page last updated: 2024-08-24

xanomeline and scopolamine hydrobromide

xanomeline has been researched along with scopolamine hydrobromide in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (28.57)29.6817
2010's5 (71.43)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bonifazi, A; Del Bello, F; Farande, A; Ferré, S; Matucci, R; Nesi, M; Petrelli, R; Piergentili, A; Quaglia, W; Vistoli, G; Yano, H1
Abou-Gharbia, M; Bartolomeo, AC; Boast, CA; Buccafusco, JJ; Husbands, MG; Kille, N; Morris, H; Moyer, JA; Rosenzweig-Lipson, S; Sabb, AL1
Nathaniel, TI; Olajuyigbe, F; Umesiri, FE1
Caine, SB; Fink-Jensen, A; Fulton, BS; Thomsen, M; Wess, J1
Barak, S; Weiner, I1
Hikichi, H; Maehara, S; Ohta, H1
Kimura, H; Kurimoto, E; Nakashima, M; Suzuki, M1

Other Studies

7 other study(ies) available for xanomeline and scopolamine hydrobromide

ArticleYear
Synthesis and biological evaluation of a novel series of heterobivalent muscarinic ligands based on xanomeline and 1-[3-(4-butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1).
    Journal of medicinal chemistry, 2014, Nov-13, Volume: 57, Issue:21

    Topics: Animals; CHO Cells; Cricetulus; Molecular Docking Simulation; Muscarinic Agonists; Piperidines; Pyridines; Quinolones; Receptor, Muscarinic M1; Structure-Activity Relationship; Thiadiazoles

2014
The preclinical pharmacological profile of WAY-132983, a potent M1 preferring agonist.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:2

    Topics: Animals; Aziridines; Behavior, Animal; Brain; Bridged-Ring Compounds; Choline; Choline O-Acetyltransferase; Cognition; Dose-Response Relationship, Drug; Drug Interactions; Female; Frontal Lobe; Hippocampus; Hypothermia; Macaca mulatta; Male; Mice; Muscarinic Agonists; Neuromuscular Blocking Agents; Pyrazines; Pyridines; Rats; Rats, Sprague-Dawley; Salivation; Scopolamine; Thiadiazoles; Time Factors; Visual Cortex

2000
Role of M1 receptor in the locomotion behavior of the African mole-rat (Cryptomys sp).
    Journal of integrative neuroscience, 2008, Volume: 7, Issue:1

    Topics: Analysis of Variance; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Locomotion; Mole Rats; Muscarinic Agonists; Muscarinic Antagonists; Pyridines; Receptor, Muscarinic M1; Scopolamine; Thiadiazoles; Time Factors

2008
Modulation of prepulse inhibition through both M(1) and M (4) muscarinic receptors in mice.
    Psychopharmacology, 2010, Volume: 208, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Clozapine; Female; Haloperidol; Male; Mice; Mice, Knockout; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Pyridines; Receptor, Muscarinic M1; Receptor, Muscarinic M4; Reflex, Startle; Scopolamine; Thiadiazoles

2010
The M₁/M₄ preferring agonist xanomeline reverses amphetamine-, MK801- and scopolamine-induced abnormalities of latent inhibition: putative efficacy against positive, negative and cognitive symptoms in schizophrenia.
    The international journal of neuropsychopharmacology, 2011, Volume: 14, Issue:9

    Topics: Amphetamine; Animals; Antimanic Agents; Behavior, Animal; Cognition Disorders; Dizocilpine Maleate; Dose-Response Relationship, Drug; Kinetics; Male; Molecular Targeted Therapy; Muscarinic Agonists; Neural Inhibition; Neurotransmitter Agents; Pyridines; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M4; Receptors, N-Methyl-D-Aspartate; Schizophrenia; Scopolamine; Tachyphylaxis; Thiadiazoles

2011
Behavioral effects of N-desmethylclozapine on locomotor activity and sensorimotor gating function in mice-Possible involvement of muscarinic receptors.
    Brain research, 2011, Oct-18, Volume: 1418

    Topics: Acoustic Stimulation; Animals; Antipsychotic Agents; Clozapine; Dose-Response Relationship, Drug; Drug Interactions; Mice; Motor Activity; Muscarinic Agonists; Neural Inhibition; Oxotremorine; Psychophysics; Pyridines; Receptors, Muscarinic; Scopolamine; Sensory Gating; Thiadiazoles

2011
TAK-071, a muscarinic M1 receptor positive allosteric modulator, attenuates scopolamine-induced quantitative electroencephalogram power spectral changes in cynomolgus monkeys.
    PloS one, 2019, Volume: 14, Issue:3

    Topics: Allosteric Regulation; Alpha Rhythm; Animals; Delta Rhythm; Donepezil; Dose-Response Relationship, Drug; Electroencephalography; Macaca fascicularis; Muscarinic Agonists; Pyridines; Receptor, Muscarinic M1; Scopolamine; Theta Rhythm; Thiadiazoles

2019