Page last updated: 2024-08-24

xanomeline and pilocarpine

xanomeline has been researched along with pilocarpine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (27.27)18.2507
2000's5 (45.45)29.6817
2010's2 (18.18)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Abuh, YF; Dunbar, PG; Edgar, MA; El-Assadi, AA; Fang, Z; Huzl, JJ; Liu, Y; Messer, WS; Nagy, PI; Ngur, DO; Ojo, B; Periyasamy, S; Rho, T; Roknich, S; Sbeih, S; Zhang, H1
Bymaster, FP; Calligaro, DO; DeLapp, NW; Fink-Jensen, A; Jeppesen, L; Olesen, PH; Rasmussen, T; Rimvall, K; Sauerberg, P; Shannon, HE; Sheardown, MJ; Thomsen, C; Ward, JS; Whitesitt, CA1
El-Fakahany, EE; Grant, MK1
Dei, S; Marconi, C; Pedretti, A; Romanelli, MN; Scapecchi, S; Vistoli, G1
Enomoto, T; Kitamura, A; Kiyoshi, A; Konishi, Y; Matsuda, H; Nakako, T; Sakai, M; Sumiyoshi, T; Suwa, A; Takahashi, Y; Takai, K; Tojo, K; Uematsu, Y; Uruno, Y1
Bymaster, FP; Calligaro, DO; Carter, PA; DeLapp, N; Fink-Jensen, A; Jeppesen, L; Mitch, CH; Peters, SC; Rimvall, K; Sauerberg, P; Shannon, HE; Sheardown, MJ; Ward, JS; Whitesitt, CA; Zhang, W1
Goodhead, LH; Mitchell, SN; Moss, S; Sharott, A1
Carnicella, S; Oberling, P; Pain, L1
El-Fakahany, EE; Grant, MK; Noetzel, MJ1
Gmeiner, P; Hu, Y; Hübner, H; Jin, C; Kaindl, J; Kobilka, BK; Li, H; Maeda, S; Niu, X; Risel, P; Xu, J1
Chen, H; Hou, Y; Wang, D; Wang, H; Wang, S; Xu, J; Yao, Y; Zhao, L1

Other Studies

11 other study(ies) available for xanomeline and pilocarpine

ArticleYear
Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
    Journal of medicinal chemistry, 1997, Apr-11, Volume: 40, Issue:8

    Topics: Animals; Arecoline; Brain; Carbachol; Cell Line; Models, Molecular; Muscarinic Agonists; Phosphatidylinositols; Pyrimidines; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship

1997
Identification of side chains on 1,2,5-thiadiazole-azacycles optimal for muscarinic m1 receptor activation.
    Bioorganic & medicinal chemistry letters, 1998, Oct-20, Volume: 8, Issue:20

    Topics: Animals; Cells, Cultured; CHO Cells; Cricetinae; Humans; Inhibitory Concentration 50; Muscarinic Agonists; Pyridines; Rats; Receptor, Muscarinic M1; Receptors, Muscarinic; Structure-Activity Relationship; Thiadiazoles; Transfection

1998
Persistent binding and functional antagonism by xanomeline at the muscarinic M5 receptor.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 315, Issue:1

    Topics: Animals; Carbachol; CHO Cells; Cricetinae; Inositol Phosphates; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Pilocarpine; Pyridines; Receptor, Muscarinic M5; Thiadiazoles

2005
Docking analyses on human muscarinic receptors: unveiling the subtypes peculiarities in agonists binding.
    Bioorganic & medicinal chemistry, 2008, Mar-15, Volume: 16, Issue:6

    Topics: Binding Sites; Computer Simulation; Humans; Ligands; Muscarinic Agonists; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M5; Receptors, Muscarinic

2008
Discovery of novel N-substituted oxindoles as selective m1 and m4 muscarinic acetylcholine receptors partial agonists.
    ACS medicinal chemistry letters, 2013, Feb-14, Volume: 4, Issue:2

    Topics:

2013
Xanomeline compared to other muscarinic agents on stimulation of phosphoinositide hydrolysis in vivo and other cholinomimetic effects.
    Brain research, 1998, Jun-08, Volume: 795, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain Chemistry; Bridged Bicyclo Compounds, Heterocyclic; Cholinergic Agents; Cholinesterase Inhibitors; Dihydropyridines; Dose-Response Relationship, Drug; Hydrolysis; Hypothermia; Imines; Lithium; Male; Mice; Mice, Inbred Strains; Muscarinic Agonists; Oximes; Parasympathomimetics; Phosphatidylinositols; Physostigmine; Pilocarpine; Pyridines; Quinuclidines; Radioligand Assay; Salivation; Tacrine; Tetrazoles; Thiadiazoles; Tremor

1998
Role of muscarinic receptors in the activation of the ventral subiculum and the consequences for dopamine release in the nucleus accumbens.
    European journal of pharmacology, 2003, Jan-24, Volume: 460, Issue:2-3

    Topics: Animals; Atropine; Bicuculline; Bridged-Ring Compounds; Carbachol; Cholinergic Agonists; Diamines; Dopamine; Hippocampus; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nucleus Accumbens; Oxotremorine; Pilocarpine; Pyridines; Rats; Receptors, Muscarinic; Spiro Compounds; Thiadiazoles; Tropanes

2003
Cholinergic effects on fear conditioning II: nicotinic and muscarinic modulations of atropine-induced disruption of the degraded contingency effect.
    Psychopharmacology, 2005, Volume: 178, Issue:4

    Topics: Animals; Atropine; Conditioning, Classical; Fear; Male; Memory; Muscarinic Antagonists; Nicotine; Nicotinic Antagonists; Oxotremorine; Parasympathetic Fibers, Postganglionic; Pilocarpine; Psychopharmacology; Pyridines; Rats; Rats, Sprague-Dawley; Thiadiazoles

2005
Mechanisms of M3 muscarinic receptor regulation by wash-resistant xanomeline binding.
    Pharmacology, 2009, Volume: 83, Issue:5

    Topics: Animals; Atropine; Binding Sites; Carbachol; Cell Line, Transformed; Cricetinae; Drug Interactions; Female; GTP-Binding Protein alpha Subunits, Gq-G11; Humans; Muscarinic Agonists; N-Methylscopolamine; Phosphatidylinositols; Pilocarpine; Pyridines; Quinuclidinyl Benzilate; Receptor, Muscarinic M3; Thiadiazoles; Time Factors; Transfection

2009
Conformational Complexity and Dynamics in a Muscarinic Receptor Revealed by NMR Spectroscopy.
    Molecular cell, 2019, 07-11, Volume: 75, Issue:1

    Topics: Acetylcholine; Animals; Baculoviridae; Binding Sites; Carbachol; Cloning, Molecular; Gene Expression; Genetic Vectors; Humans; Isoxazoles; Kinetics; Ligands; Magnetic Resonance Spectroscopy; Molecular Dynamics Simulation; Pilocarpine; Protein Binding; Protein Conformation, alpha-Helical; Protein Conformation, beta-Strand; Protein Interaction Domains and Motifs; Pyridines; Quaternary Ammonium Compounds; Receptor, Muscarinic M2; Recombinant Proteins; Sf9 Cells; Spodoptera; Thermodynamics; Thiadiazoles

2019
Structural Insights into M1 Muscarinic Acetylcholine Receptor Signaling Bias between Gαq and β-Arrestin through BRET Assays and Molecular Docking.
    International journal of molecular sciences, 2023, Apr-16, Volume: 24, Issue:8

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; beta-Arrestin 1; beta-Arrestin 2; beta-Arrestins; Energy Transfer; GTP-Binding Proteins; HEK293 Cells; Humans; Molecular Docking Simulation; Pilocarpine; Receptor, Muscarinic M1

2023