Page last updated: 2024-08-24

xanomeline and oxotremorine

xanomeline has been researched along with oxotremorine in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (8.33)18.2507
2000's3 (25.00)29.6817
2010's7 (58.33)24.3611
2020's1 (8.33)2.80

Authors

AuthorsStudies
Abuh, YF; Dunbar, PG; Edgar, MA; El-Assadi, AA; Fang, Z; Huzl, JJ; Liu, Y; Messer, WS; Nagy, PI; Ngur, DO; Ojo, B; Periyasamy, S; Rho, T; Roknich, S; Sbeih, S; Zhang, H1
Dei, S; Marconi, C; Pedretti, A; Romanelli, MN; Scapecchi, S; Vistoli, G1
Bernhardt, G; Gmeiner, P; Hübner, H; Keller, M; Pegoli, A; She, X; Wifling, D1
Butler, CR; Grimwood, S; Kablaoui, NM; Kozak, R; Lachapelle, EA; Lazzaro, JT; O'Connor, RE; Popiolek, M; Webb, D; Yang, Q; Zhang, L1
Bernhardt, G; Carpenter, J; Chen, M; Gmeiner, P; Gruber, CG; Holliday, ND; Hübner, H; Keller, M; Pegoli, A; She, X; Wan, J; Wifling, D1
Goodhead, LH; Mitchell, SN; Moss, S; Sharott, A1
Carnicella, S; Oberling, P; Pain, L1
Caine, SB; Fink-Jensen, A; Fulton, BS; Thomsen, M; Wess, J1
Christopoulos, A; Felder, C; Leach, K; Loiacono, R; Sexton, P; Suratman, S1
Hikichi, H; Maehara, S; Ohta, H1
Dolejší, E; Doležal, V; El-Fakahany, EE; Jakubík, J; Randáková, A; Rudajev, V; Zimčík, P1
Clarke, S; Reed, H; Sher, E; Zwart, R1

Other Studies

12 other study(ies) available for xanomeline and oxotremorine

ArticleYear
Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
    Journal of medicinal chemistry, 1997, Apr-11, Volume: 40, Issue:8

    Topics: Animals; Arecoline; Brain; Carbachol; Cell Line; Models, Molecular; Muscarinic Agonists; Phosphatidylinositols; Pyrimidines; Quinuclidinyl Benzilate; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Structure-Activity Relationship

1997
Docking analyses on human muscarinic receptors: unveiling the subtypes peculiarities in agonists binding.
    Bioorganic & medicinal chemistry, 2008, Mar-15, Volume: 16, Issue:6

    Topics: Binding Sites; Computer Simulation; Humans; Ligands; Muscarinic Agonists; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M5; Receptors, Muscarinic

2008
Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M
    Journal of medicinal chemistry, 2017, 04-27, Volume: 60, Issue:8

    Topics: Benzodiazepinones; Binding Sites; Molecular Dynamics Simulation; Muscarinic Antagonists; Radioisotopes; Receptor, Muscarinic M2

2017
Discovery of Selective M4 Muscarinic Acetylcholine Receptor Agonists with Novel Carbamate Isosteres.
    ACS medicinal chemistry letters, 2019, Jun-13, Volume: 10, Issue:6

    Topics:

2019
Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M
    Journal of medicinal chemistry, 2020, 04-23, Volume: 63, Issue:8

    Topics: Animals; CHO Cells; Cholinergic Agents; Cricetulus; Fluorescent Dyes; Muscarinic Antagonists; Phthalimides; Protein Structure, Secondary; Quaternary Ammonium Compounds; Receptor, Muscarinic M2

2020
Role of muscarinic receptors in the activation of the ventral subiculum and the consequences for dopamine release in the nucleus accumbens.
    European journal of pharmacology, 2003, Jan-24, Volume: 460, Issue:2-3

    Topics: Animals; Atropine; Bicuculline; Bridged-Ring Compounds; Carbachol; Cholinergic Agonists; Diamines; Dopamine; Hippocampus; Male; Microdialysis; Muscarinic Agonists; Muscarinic Antagonists; Nicotine; Nucleus Accumbens; Oxotremorine; Pilocarpine; Pyridines; Rats; Receptors, Muscarinic; Spiro Compounds; Thiadiazoles; Tropanes

2003
Cholinergic effects on fear conditioning II: nicotinic and muscarinic modulations of atropine-induced disruption of the degraded contingency effect.
    Psychopharmacology, 2005, Volume: 178, Issue:4

    Topics: Animals; Atropine; Conditioning, Classical; Fear; Male; Memory; Muscarinic Antagonists; Nicotine; Nicotinic Antagonists; Oxotremorine; Parasympathetic Fibers, Postganglionic; Pilocarpine; Psychopharmacology; Pyridines; Rats; Rats, Sprague-Dawley; Thiadiazoles

2005
Modulation of prepulse inhibition through both M(1) and M (4) muscarinic receptors in mice.
    Psychopharmacology, 2010, Volume: 208, Issue:3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Clozapine; Female; Haloperidol; Male; Mice; Mice, Knockout; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Pyridines; Receptor, Muscarinic M1; Receptor, Muscarinic M4; Reflex, Startle; Scopolamine; Thiadiazoles

2010
Impact of species variability and 'probe-dependence' on the detection and in vivo validation of allosteric modulation at the M4 muscarinic acetylcholine receptor.
    British journal of pharmacology, 2011, Volume: 162, Issue:7

    Topics: Acetylcholine; Allosteric Regulation; Allosteric Site; Animals; Cell Line; CHO Cells; Cricetinae; Cricetulus; Glycogen Synthase Kinase 3; Humans; Ligands; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Molecular Probe Techniques; Nicotinic Acids; Oxotremorine; Protein Binding; Pyridines; Receptor, Muscarinic M4; Species Specificity; Thiadiazoles; Thiophenes

2011
Behavioral effects of N-desmethylclozapine on locomotor activity and sensorimotor gating function in mice-Possible involvement of muscarinic receptors.
    Brain research, 2011, Oct-18, Volume: 1418

    Topics: Acoustic Stimulation; Animals; Antipsychotic Agents; Clozapine; Dose-Response Relationship, Drug; Drug Interactions; Mice; Motor Activity; Muscarinic Agonists; Neural Inhibition; Oxotremorine; Psychophysics; Pyridines; Receptors, Muscarinic; Scopolamine; Sensory Gating; Thiadiazoles

2011
Classical and atypical agonists activate M1 muscarinic acetylcholine receptors through common mechanisms.
    Pharmacological research, 2015, Volume: 97

    Topics: Animals; Binding Sites; Calcium; Carbachol; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Inositol Phosphates; Models, Molecular; Muscarinic Agonists; Mutation; Oxotremorine; Pyridines; Receptor, Muscarinic M1; Receptors, G-Protein-Coupled; Thiadiazoles

2015
A novel muscarinic receptor-independent mechanism of KCNQ2/3 potassium channel blockade by Oxotremorine-M.
    European journal of pharmacology, 2016, Nov-15, Volume: 791

    Topics: Animals; Humans; KCNQ2 Potassium Channel; KCNQ3 Potassium Channel; Oxotremorine; Potassium Channel Blockers; Pyridines; Receptor, Muscarinic M1; Thiadiazoles; Xenopus

2016