Page last updated: 2024-09-04

xamoterol and trimetrexate

xamoterol has been researched along with trimetrexate in 2 studies

Compound Research Comparison

Studies
(xamoterol)
Trials
(xamoterol)
Recent Studies (post-2010)
(xamoterol)
Studies
(trimetrexate)
Trials
(trimetrexate)
Recent Studies (post-2010) (trimetrexate)
26980174225021

Protein Interaction Comparison

ProteinTaxonomyxamoterol (IC50)trimetrexate (IC50)
Dihydrofolate reductase Mycobacterium avium0.3012
Dihydrofolate reductaseHomo sapiens (human)0.0207
Dihydrofolate reductaseLacticaseibacillus casei0.1435
Dihydrofolate reductaseSaccharomyces cerevisiae S288C0.042
Dihydrofolate reductaseEscherichia coli K-120.1798
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.026
Dihydrofolate reductasePneumocystis carinii0.0378
Dihydrofolate reductaseCandida albicans0.04
Dipeptidyl peptidase 4Homo sapiens (human)0.01
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.008
Bifunctional dihydrofolate reductase-thymidylate synthaseToxoplasma gondii0.5788
Bifunctional dihydrofolate reductase-thymidylate synthaseTrypanosoma cruzi0.0202
Dihydrofolate reductaseRattus norvegicus (Norway rat)0.0794

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1

Other Studies

2 other study(ies) available for xamoterol and trimetrexate

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009