Page last updated: 2024-09-04

xamoterol and digoxin

xamoterol has been researched along with digoxin in 13 studies

Compound Research Comparison

Studies
(xamoterol)
Trials
(xamoterol)
Recent Studies (post-2010)
(xamoterol)
Studies
(digoxin)
Trials
(digoxin)
Recent Studies (post-2010) (digoxin)
269801711,4839581,289

Protein Interaction Comparison

ProteinTaxonomyxamoterol (IC50)digoxin (IC50)
STAT3, partialHomo sapiens (human)1.862
Sodium/potassium-transporting ATPase subunit alpha-1 Homo sapiens (human)0.32
Sodium/potassium-transporting ATPase subunit beta-1Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-2Rattus norvegicus (Norway rat)0.22
Sodium/potassium-transporting ATPase subunit alpha-3 Rattus norvegicus (Norway rat)0.22
Sodium/potassium-transporting ATPase subunit beta-1 Rattus norvegicus (Norway rat)0.0055
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 20.19
Sodium/potassium-transporting ATPase subunit alpha-3Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit beta-2Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-2Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-1Canis lupus familiaris (dog)0.5
Nuclear receptor ROR-gammaHomo sapiens (human)3.4798
Sodium/potassium-transporting ATPase subunit beta-3Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit gammaHomo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-4Homo sapiens (human)0.335
Sodium/potassium-transporting ATPase subunit alpha-4Rattus norvegicus (Norway rat)0.0055
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.2359

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19905 (38.46)18.7374
1990's5 (38.46)18.2507
2000's2 (15.38)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Eber, B; Klein, W; Rotman, B1
Alexander, ND; Ang, EL; Chan, WL; Cleland, JG; Krikler, SJ; Moore, D; Oakley, CM1
Armstrong, C; Blackwood, R; Bryant, B; Garnham, JC; Mayou, RA1
Timmis, AD1
Andersen, MF; Faergeman, O; Sorensen, EV; Sterndorff, B1
Bennett, DH; Coupe, MO; Molajo, AO1
Austin, CA; Channer, KS; Dent, M; Lawson-Matthew, PJ; McLean, KA1

Reviews

1 review(s) available for xamoterol and digoxin

ArticleYear
A new look at digoxin in congestive heart failure and sinus rhythm.
    Postgraduate medical journal, 1989, Volume: 65, Issue:768

    Topics: Arrhythmia, Sinus; Blood Circulation; Cardiac Glycosides; Digoxin; Heart Failure; Humans; Myocardial Contraction; Propanolamines; Xamoterol

1989

Trials

8 trial(s) available for xamoterol and digoxin

ArticleYear
Comparative effects of digoxin and xamoterol on arrhythmias in patients with mild to moderate heart failure.
    Angiology, 1992, Volume: 43, Issue:4

    Topics: Adrenergic beta-Agonists; Analysis of Variance; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Digoxin; Double-Blind Method; Electrocardiography, Ambulatory; Female; Heart Failure; Humans; Male; Middle Aged; Propanolamines; Time Factors; Xamoterol

1992
Comparative effects of xamoterol and digoxin in patients with mild to moderate heart failure. The Italian Xamoterol Multicenter Research Group.
    European heart journal, 1990, Volume: 11 Suppl A

    Topics: Adrenergic beta-Agonists; Cardiac Output, Low; Digoxin; Double-Blind Method; Drug Evaluation; Humans; Middle Aged; Multicenter Studies as Topic; Physical Exertion; Propanolamines; Xamoterol

1990
Placebo controlled trial of xamoterol versus digoxin in chronic atrial fibrillation.
    British heart journal, 1990, Volume: 64, Issue:4

    Topics: Adrenergic beta-Agonists; Aged; Aged, 80 and over; Atrial Fibrillation; Chronic Disease; Digoxin; Double-Blind Method; Electrocardiography, Ambulatory; Exercise Test; Female; Heart Rate; Humans; Male; Middle Aged; Propanolamines; Time Factors; Xamoterol

1990
Exercise capacity and quality of life in the treatment of heart failure.
    Clinical pharmacology and therapeutics, 1990, Volume: 48, Issue:3

    Topics: Adult; Aged; Digoxin; Exercise; Exercise Test; Female; Heart Failure; Humans; Male; Middle Aged; Multicenter Studies as Topic; Propanolamines; Quality of Life; Randomized Controlled Trials as Topic; Xamoterol

1990
Digoxin and xamoterol in patients with moderate chronic heart failure. A double-blind, randomized, controlled study.
    Cardiovascular drugs and therapy, 1989, Volume: 3, Issue:2

    Topics: Adrenergic beta-Agonists; Adult; Aged; Digoxin; Double-Blind Method; Echocardiography; Electrocardiography; Exercise Test; Heart Failure; Hemodynamics; Humans; Male; Middle Aged; Propanolamines; Xamoterol

1989
Double-blind placebo-controlled comparison of digoxin and xamoterol in chronic heart failure. The German and Austrian Xamoterol Study Group.
    Lancet (London, England), 1988, Mar-05, Volume: 1, Issue:8584

    Topics: Adrenergic beta-Agonists; Adult; Aged; Aged, 80 and over; Clinical Trials as Topic; Digoxin; Double-Blind Method; Exercise Test; Female; Heart Failure; Humans; Male; Middle Aged; Propanolamines; Random Allocation; Xamoterol

1988
Effect of Corwin (ICI 118587) on resting and exercise heart rate and exercise tolerance in digitalised patients with chronic atrial fibrillation.
    British heart journal, 1984, Volume: 52, Issue:4

    Topics: Adrenergic beta-Agonists; Adult; Aged; Atrial Fibrillation; Chronic Disease; Clinical Trials as Topic; Digoxin; Double-Blind Method; Drug Therapy, Combination; Electrocardiography; Female; Heart Rate; Humans; Male; Middle Aged; Physical Exertion; Propanolamines; Xamoterol

1984
Xamoterol improves the control of chronic atrial fibrillation in elderly patients.
    Age and ageing, 1995, Volume: 24, Issue:4

    Topics: Adrenergic beta-Agonists; Aged; Aged, 80 and over; Atrial Fibrillation; Chronic Disease; Cross-Over Studies; Digoxin; Double-Blind Method; Drug Administration Schedule; Drug Therapy, Combination; Electrocardiography; Exercise Test; Furosemide; Geriatric Assessment; Heart Rate; Humans; Xamoterol

1995

Other Studies

4 other study(ies) available for xamoterol and digoxin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Xamoterol versus digoxin in heart failure.
    Lancet (London, England), 1988, Apr-16, Volume: 1, Issue:8590

    Topics: Adrenergic beta-Agonists; Adult; Aged; Digoxin; Heart Failure; Humans; Middle Aged; Propanolamines; Xamoterol

1988