Page last updated: 2024-09-04

xamoterol and colforsin

xamoterol has been researched along with colforsin in 4 studies

Compound Research Comparison

Studies
(xamoterol)
Trials
(xamoterol)
Recent Studies (post-2010)
(xamoterol)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
269801713,460461,298

Protein Interaction Comparison

ProteinTaxonomyxamoterol (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19901 (25.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Komajda, M1
Karle, CA; Kathöfer, S; Kiehn, J; Schoels, W; Zhang, W; Zitron, E1
Aiyar, N; Andreka, P; Bishopric, NH; Ohlstein, EH; Olson, LC; Turner, MS; Webster, KA; Wei, JQ1
Gutierrez, O; Pazos, A; Valdizán, EM1

Other Studies

4 other study(ies) available for xamoterol and colforsin

ArticleYear
[New cardiotonic agents].
    Annales de cardiologie et d'angeiologie, 1985, Volume: 34, Issue:10

    Topics: Aminopyridines; Amrinone; Cardiotonic Agents; Colforsin; Deoxyepinephrine; Humans; Imidazoles; Levodopa; Milrinone; Practolol; Prenalterol; Propanolamines; Pyridones; Quinazolines; Xamoterol

1985
Rapid component I(Kr) of the guinea-pig cardiac delayed rectifier K(+) current is inhibited by beta(1)-adrenoreceptor activation, via cAMP/protein kinase A-dependent pathways.
    Cardiovascular research, 2002, Feb-01, Volume: 53, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbazoles; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Enzyme Inhibitors; Guinea Pigs; Imidazoles; Indoles; Isoproterenol; Myocardium; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Pyrroles; Xamoterol

2002
Bucindolol displays intrinsic sympathomimetic activity in human myocardium.
    Circulation, 2002, May-21, Volume: 105, Issue:20

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Animals; Cell Survival; Colforsin; Culture Techniques; Cyclic AMP; Dose-Response Relationship, Drug; Female; Heart; Humans; Intracellular Fluid; Male; Middle Aged; Myocardium; Propanolamines; Rats; Sympathomimetics; Xamoterol

2002
Adenylate cyclase activity in postmortem brain of suicide subjects: reduced response to beta-adrenergic stimulation.
    Biological psychiatry, 2003, Dec-15, Volume: 54, Issue:12

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adult; Aged; Aged, 80 and over; Analysis of Variance; Case-Control Studies; Cell Membrane; Colforsin; Depressive Disorder, Major; Dose-Response Relationship, Drug; Female; Frontal Lobe; Guanine Nucleotides; Humans; In Vitro Techniques; Male; Middle Aged; Postmortem Changes; Radioligand Assay; Suicide; Xamoterol

2003