Page last updated: 2024-09-03

xaliproden and buspirone

xaliproden has been researched along with buspirone in 2 studies

Compound Research Comparison

Studies
(xaliproden)
Trials
(xaliproden)
Recent Studies (post-2010)
(xaliproden)
Studies
(buspirone)
Trials
(buspirone)
Recent Studies (post-2010) (buspirone)
41292,096351382

Protein Interaction Comparison

ProteinTaxonomyxaliproden (IC50)buspirone (IC50)
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.025
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)1.75
Angiotensin-converting enzyme Homo sapiens (human)0.024
D(2) dopamine receptorHomo sapiens (human)0.323
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)2.125
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)4.16
DRattus norvegicus (Norway rat)0.12
D(3) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0266
D(2) dopamine receptorBos taurus (cattle)4
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)4.16
Alpha-1D adrenergic receptorHomo sapiens (human)1.077
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2AHomo sapiens (human)2.286
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.016
D(4) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)2.125
D(3) dopamine receptorHomo sapiens (human)0.044
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.75
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)4.16
D(2) dopamine receptorRattus norvegicus (Norway rat)0.2055
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.9811
Alpha-2A adrenergic receptorBos taurus (cattle)0.025
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.7
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.2666
Lysosomal alpha-glucosidaseBos taurus (cattle)0.03

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Bianchetti, A; Croci, T; Landi, M; Manara, L1

Other Studies

2 other study(ies) available for xaliproden and buspirone

ArticleYear
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Drug-induced defaecation in rats: role of central 5-HT1A receptors.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding Sites; Buspirone; Colon; Defecation; Feces; Fenclonine; Male; Naphthalenes; Pindolol; Pyridines; Rats; Receptors, Serotonin; Serotonin Receptor Agonists; Time Factors

1995