Page last updated: 2024-09-04

wy 26703 and clonidine

wy 26703 has been researched along with clonidine in 5 studies

Compound Research Comparison

Studies
(wy 26703)
Trials
(wy 26703)
Recent Studies (post-2010)
(wy 26703)
Studies
(clonidine)
Trials
(clonidine)
Recent Studies (post-2010) (clonidine)
110013,6922,0441,394

Protein Interaction Comparison

ProteinTaxonomywy 26703 (IC50)clonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.101
Alpha-2B adrenergic receptorHomo sapiens (human)0.0353
Alpha-2C adrenergic receptorHomo sapiens (human)0.0115
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)5.365
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-1D adrenergic receptorHomo sapiens (human)1.21
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)5.365
Alpha-2A adrenergic receptorBos taurus (cattle)0.002
NischarinRattus norvegicus (Norway rat)0.3662

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19905 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baldwin, JJ; deSolms, SJ; Guare, JP; Huff, JR; Hunt, CA; Randall, WC; Sanders, WS; Smith, SJ; Vacca, JP; Zrada, MM1
Lattimer, N; Rhodes, KF; Waterfall, JF1
Kassarich, J; Lien, EL; Morrison, A; Sullivan, D1
De Jonge, A; Doods, HN; Korstanje, C; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Wilffert, B1
Paciorek, PM; Pierce, V; Shepperson, NB; Waterfall, JF1

Other Studies

5 other study(ies) available for wy 26703 and clonidine

ArticleYear
Structure-affinity relationships of arylquinolizines at alpha-adrenoceptors.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: Algorithms; Animals; Binding, Competitive; Cattle; Clonidine; Hydrogen-Ion Concentration; Prazosin; Quinolizines; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Yohimbine

1988
Studies of alpha 2-adrenoceptor antagonist potency in vitro: comparisons in tissues from rats, rabbits, dogs and humans.
    Clinical science (London, England : 1979), 1985, Volume: 68 Suppl 10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; Dioxanes; Dogs; Humans; Idazoxan; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Platelet Aggregation; Quinolizines; Rabbits; Rats; Rats, Inbred Strains; Saphenous Vein; Species Specificity; Vas Deferens; Yohimbine

1985
Alpha-2-adrenergic control of prolactin release.
    Neuroendocrinology, 1986, Volume: 44, Issue:2

    Topics: Animals; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Female; Male; Piperoxan; Pregnancy; Prolactin; Quinolizines; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1986
Affinity of WY 26703 for central and peripheral alpha 1- and alpha 2-adrenoreceptors in the rat; comparison with yohimbine.
    Journal of autonomic pharmacology, 1984, Volume: 4, Issue:4

    Topics: Animals; Azepines; Binding, Competitive; Blood Pressure; Clonidine; In Vitro Techniques; Male; Methoxamine; Muscle, Smooth, Vascular; Myocardium; Prazosin; Quinolizines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1984
An investigation into the selectivity of a novel series of benzoquinolizines for alpha 2-adrenoceptors in vivo.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Action Potentials; Animals; Azepines; Chlorisondamine; Clonidine; Female; Indoramin; Methoxamine; Quinolizines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1984