Page last updated: 2024-09-03

wr 99210 and atovaquone

wr 99210 has been researched along with atovaquone in 2 studies

Compound Research Comparison

Studies
(wr 99210)
Trials
(wr 99210)
Recent Studies (post-2010)
(wr 99210)
Studies
(atovaquone)
Trials
(atovaquone)
Recent Studies (post-2010) (atovaquone)
59012997100420

Protein Interaction Comparison

ProteinTaxonomywr 99210 (IC50)atovaquone (IC50)
Dihydroorotate dehydrogenase Schistosoma mansoni0.431
Cytochrome bHomo sapiens (human)2.835
Dihydroorotate dehydrogenase (quinone), mitochondrialHomo sapiens (human)2.65
Dihydroorotate dehydrogenase (quinone), mitochondrialRattus norvegicus (Norway rat)0.7
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)0.23

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carlier, PR; Dalal, S; Dapper, CH; Ghavami, M; Holzschneider, K; Klemba, M1
Ager, AL; Canfield, CJ; Jacobus, DP; Lewis, NJ; Milhous, WK; Rossan, RN; Sweeney, TR1

Other Studies

2 other study(ies) available for wr 99210 and atovaquone

ArticleYear
Parallel inhibition of amino acid efflux and growth of erythrocytic Plasmodium falciparum by mefloquine and non-piperidine analogs: Implication for the mechanism of antimalarial action.
    Bioorganic & medicinal chemistry letters, 2016, 10-01, Volume: 26, Issue:19

    Topics: Animals; Antimalarials; Inhibitory Concentration 50; Mefloquine; Plasmodium falciparum

2016
PS-15: a potent, orally active antimalarial from a new class of folic acid antagonists.
    The American journal of tropical medicine and hygiene, 1993, Volume: 49, Issue:1

    Topics: Administration, Oral; Animals; Antimalarials; Aotus trivirgatus; Atovaquone; Drug Synergism; Folic Acid Antagonists; Imides; Injections, Subcutaneous; Malaria, Falciparum; Mice; Naphthoquinones; Phenyl Ethers; Plasmodium falciparum; Proguanil; Sulfamethoxazole; Triazines

1993