Page last updated: 2024-09-04

win 64338 and bradykinin

win 64338 has been researched along with bradykinin in 13 studies

Compound Research Comparison

Studies
(win 64338)
Trials
(win 64338)
Recent Studies (post-2010)
(win 64338)
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
190214,1953551,520

Protein Interaction Comparison

ProteinTaxonomywin 64338 (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (69.23)18.2507
2000's2 (15.38)29.6817
2010's2 (15.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Schölkens, BA; Wiemer, G; Wirth, KJ1
Drapeau, G; Levesque, L; Marceau, F; Rioux, F; Salvino, JM; Sawutz, DG; Seoane, PR; Wolfe, HR1
DeSiato, MA; Farmer, SG1
Bélichard, P; Defrêne, E; Luccarini, JM; Paquet, JL; Pruneau, D1
Butt, SK; Figini, M; Geppetti, P; Hall, JM1
Filteau, C; Gobeil, F; Jukic, D; Nguyen-Le, XK; Pheng, LH; Regoli, D1
Filteau, C; Gobeil, F; Nguyen-Le, XK; Pheng, LH; Regoli, D1
Dedio, J; Schölkens, BA; Wiemer, G; Wirth, K; Wohlfart, P1
Da Silva, A; Gies, JP; Lach, E; Landry, Y; Scherrer, D; Schmidlin, F1
Cheuk, BL; Ko, WH; Wong, PY1
Ouyang, A; Yu, S1
Earnest, D; Ellis, D; Hamilton, G; Jacobson, N; Katoli, P; Kelly, CR; Klekar, L; Li, L; Sharif, NA; Shepard, AR; Wang, Y; Xu, S; Yacoub, S1
Hovatta, I; Hyytiä, P; Kulesskaya, N; McEntegart, W; Mennesson, M; Misiewicz, Z; Rouhiainen, A; Saarnio, S; Sipilä, T; Sokolowska, E; Trontti, K; Urpa, L1

Other Studies

13 other study(ies) available for win 64338 and bradykinin

ArticleYear
The bradykinin B2 receptor antagonist WIN 64338 inhibits the effect of des-Arg9-bradykinin in endothelial cells.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: Animals; Aorta; Binding, Competitive; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Cells, Cultured; Cyclic GMP; Endothelium, Vascular; Naphthalenes; Nitric Oxide; Organophosphorus Compounds; Rabbits

1994
Effects of peptide and nonpeptide antagonists of bradykinin B2 receptors on the venoconstrictor action of bradykinin.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:3

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Female; Humans; In Vitro Techniques; Jugular Veins; Male; Naphthalenes; Organophosphorus Compounds; Rabbits; Umbilical Veins; Vasoconstriction

1994
Effects of a novel nonpeptide bradykinin B2 receptor antagonist on intestinal and airway smooth muscle: further evidence for the tracheal B3 receptor.
    British journal of pharmacology, 1994, Volume: 112, Issue:2

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Naphthalenes; Organophosphorus Compounds; Trachea

1994
Pharmacological evidence for a single bradykinin B2 receptor in the guinea-pig.
    British journal of pharmacology, 1995, Volume: 116, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bradykinin; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Isometric Contraction; Jugular Veins; Lung; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Naphthalenes; Organophosphorus Compounds; Receptor, Bradykinin B2; Receptors, Bradykinin; Trachea

1995
Inhibition of bradykinin-evoked trigeminal nerve stimulation by the non-peptide bradykinin B2 receptor antagonist WIN 64338 in vivo and in vitro.
    British journal of pharmacology, 1995, Volume: 116, Issue:8

    Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Eye; Guinea Pigs; Naphthalenes; Nasal Mucosa; Organophosphorus Compounds; Rabbits; Trigeminal Nerve

1995
In vitro and in vivo characterization of bradykinin B2 receptors in the rabbit and the guinea pig.
    Canadian journal of physiology and pharmacology, 1996, Volume: 74, Issue:2

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Intestines; Jugular Veins; Male; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Organophosphorus Compounds; Peptidyl-Dipeptidase A; Pulmonary Artery; Rabbits; Receptors, Bradykinin

1996
In vivo characterization of B2 receptors mediating hypotension in anesthetized rabbits and guinea pigs.
    Immunopharmacology, 1996, Volume: 33, Issue:1-3

    Topics: Anesthesia; Animals; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Guinea Pigs; Hypotension; Naphthalenes; Organophosphorus Compounds; Rabbits; Receptor, Bradykinin B2; Receptors, Bradykinin

1996
Different B1 kinin receptor expression and pharmacology in endothelial cells of different origins and species.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Aorta; Bradykinin; Bradykinin Receptor Antagonists; Cattle; Cells, Cultured; Coronary Vessels; Cyclic GMP; DNA Primers; Endothelium, Vascular; Humans; Microcirculation; Naphthalenes; Organophosphorus Compounds; Polymerase Chain Reaction; Rats; Receptor, Bradykinin B1; Receptors, Bradykinin; Species Specificity; Transcription, Genetic; Umbilical Veins

1997
Effect of WIN 64338, a B2 bradykinin receptor antagonist on guinea-pig tracheal smooth muscle cells in culture.
    Fundamental & clinical pharmacology, 1998, Volume: 12, Issue:2

    Topics: Adrenergic beta-Antagonists; Analgesics; Animals; Binding, Competitive; Bradykinin; Bradykinin Receptor Antagonists; Cells, Cultured; Fluorescent Antibody Technique; Guinea Pigs; Inositol Phosphates; Male; Muscle, Smooth; Naphthalenes; Oligopeptides; Organophosphorus Compounds; Receptor, Bradykinin B2; Receptors, Bradykinin; Trachea

1998
COX-dependent and -independent pathways in bradykinin-induced anion secretion in rat epididymis.
    Journal of cellular physiology, 2002, Volume: 191, Issue:2

    Topics: Animals; Anions; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Calcium Signaling; Cells, Cultured; Cyclic AMP; Cyclooxygenase 1; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epididymis; Epithelial Cells; Ion Channels; Isoenzymes; Kallidin; Male; Membrane Proteins; Naphthalenes; Organophosphorus Compounds; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Signal Transduction; Vasodilator Agents

2002
TRPA1 in bradykinin-induced mechanical hypersensitivity of vagal C fibers in guinea pig esophagus.
    American journal of physiology. Gastrointestinal and liver physiology, 2009, Volume: 296, Issue:2

    Topics: Action Potentials; Animals; Bradykinin; Bradykinin B2 Receptor Antagonists; Esophagus; Guinea Pigs; Hyperalgesia; In Vitro Techniques; Isothiocyanates; Kinetics; Male; Mechanotransduction, Cellular; Naphthalenes; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neural Pathways; Nodose Ganglion; Organophosphorus Compounds; Pressure; Receptor, Bradykinin B2; Stimulation, Chemical; Transient Receptor Potential Channels; Vagus Nerve

2009
Trabecular meshwork bradykinin receptors: mRNA levels, immunohistochemical visualization, signaling processes pharmacology, and linkage to IOP reduction.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2014, Volume: 30, Issue:1

    Topics: Aged; Animals; Benzophenones; Bradykinin; Bradykinin B2 Receptor Antagonists; Bromobenzenes; Female; Humans; Immunohistochemistry; Intraocular Pressure; Kininogens; Macaca fascicularis; Male; Naphthalenes; Organophosphorus Compounds; Prostaglandins; Rabbits; Receptor, Bradykinin B2; Receptors, Bradykinin; RNA, Messenger; Signal Transduction; Trabecular Meshwork

2014
The bradykinin system in stress and anxiety in humans and mice.
    Scientific reports, 2019, 12-19, Volume: 9, Issue:1

    Topics: Adult; Animals; Anxiety Disorders; Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Brain; Disease Models, Animal; Female; Humans; Kallikrein-Kinin System; Kininogens; Male; Mice; Naphthalenes; Organophosphorus Compounds; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Polymorphism, Single Nucleotide; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Species Specificity; Stress, Psychological; Up-Regulation

2019