willardiine has been researched along with 5-bromowillardiine in 4 studies
| Studies (willardiine) | Trials (willardiine) | Recent Studies (post-2010) (willardiine) | Studies (5-bromowillardiine) | Trials (5-bromowillardiine) | Recent Studies (post-2010) (5-bromowillardiine) |
|---|---|---|---|---|---|
| 43 | 0 | 10 | 11 | 0 | 0 |
| Protein | Taxonomy | willardiine (IC50) | 5-bromowillardiine (IC50) |
|---|---|---|---|
| Chain A, glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.3 | |
| Chain A, glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.3 | |
| Chain A, glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.3 | |
| Chain A, glutamate receptor 2 | Rattus norvegicus (Norway rat) | 0.3 | |
| Chain A, Glutamate Receptor 2 | Rattus norvegicus (Norway rat) | 4 | |
| Chain A, Glutamate Receptor 2 | Rattus norvegicus (Norway rat) | 4 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (50.00) | 18.2507 |
| 2000's | 2 (50.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Bleakman, D; Deverill, M; Hoo, K; Jane, DE; Kamboj, R; Mandelzys, A | 1 |
| Banke, TG; Gouaux, E; Jin, R; Mayer, ML; Traynelis, SF | 1 |
| Butini, S; Campiani, G; Christensen, JK; Coccone, SS; De Angelis, M; Fiorini, I; Gemma, S; Guarino, E; Morelli, E; Novellino, E; Pickering, DS; Schousboe, A; Trotta, F | 1 |
| Clifford, DB; Thio, LL; Zorumski, CF | 1 |
4 other study(ies) available for willardiine and 5-bromowillardiine
| Article | Year |
|---|---|
Synthesis of willardiine and 6-azawillardiine analogs: pharmacological characterization on cloned homomeric human AMPA and kainate receptor subtypes.
Topics: Alanine; Cell Line; Excitatory Amino Acid Agonists; Humans; Magnetic Resonance Spectroscopy; Molecular Structure; Pyrimidinones; Radioligand Assay; Receptors, AMPA; Receptors, Kainic Acid; Recombinant Proteins; Triazines; Uracil | 1997 |
Structural basis for partial agonist action at ionotropic glutamate receptors.
Topics: Alanine; Animals; Cell Line; Crystallography, X-Ray; Electric Conductivity; Electrophysiology; Humans; Ion Channels; Ligands; Models, Biological; Molecular Conformation; Oocytes; Pyrimidinones; Receptors, AMPA; Uracil; Xenopus laevis | 2003 |
1H-cyclopentapyrimidine-2,4(1H,3H)-dione-related ionotropic glutamate receptors ligands. structure-activity relationships and identification of potent and Selective iGluR5 modulators.
Topics: Animals; Cell Line; Electrophysiology; Excitatory Amino Acid Antagonists; Female; Humans; Ligands; Molecular Structure; Oocytes; Pyrimidinones; Rats; Receptors, Glutamate; Spodoptera; Structure-Activity Relationship; Thiophenes; Xenopus laevis | 2008 |
Effects of bromowillardiine and willardiine on non-N-methyl-D-aspartate receptors in postnatal rat hippocampal neurons.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Alanine; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Hippocampus; Membrane Potentials; Neurons; Pyrimidinones; Quinoxalines; Rats; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Uracil | 1991 |