way 123398 has been researched along with e 4031 in 5 studies
Studies (way 123398) | Trials (way 123398) | Recent Studies (post-2010) (way 123398) | Studies (e 4031) | Trials (e 4031) | Recent Studies (post-2010) (e 4031) |
---|---|---|---|---|---|
15 | 0 | 1 | 356 | 1 | 86 |
Protein | Taxonomy | way 123398 (IC50) | e 4031 (IC50) |
---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 0.0381 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (80.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (20.00) | 2.80 |
Authors | Studies |
---|---|
Colatsky, TJ; Parsons, RW; Spinelli, W | 1 |
Colatsky, TJ; Moubarak, IF; Parsons, RW; Spinelli, W | 1 |
Arcangeli, A; Faravelli, L; Olivotto, M; Wanke, E | 1 |
Meves, H; Schwarz, JR; Wulfsen, I | 1 |
Aly, KA; Babu, M; Cayabyab, FS; Fonge, H; He, S; Islam, S; Moutaoufik, MT; Persad, A; Wu, A | 1 |
1 review(s) available for way 123398 and e 4031
Article | Year |
---|---|
HERG channel and cancer: A mechanistic review of carcinogenic processes and therapeutic potential.
Topics: Antineoplastic Agents; Apoptosis; Benzimidazoles; Carcinogenesis; Cell Movement; Cell Proliferation; Epigenesis, Genetic; ERG1 Potassium Channel; Fluoxetine; Gene Expression Regulation, Neoplastic; Humans; Integrin beta1; Long QT Syndrome; Membrane Potentials; Molecular Docking Simulation; Mutation; Myocytes, Cardiac; Neoplasms; Piperidines; Protein Conformation, alpha-Helical; Protein Interaction Mapping; Protein Structure, Quaternary; Pyridines; Signal Transduction; STAT1 Transcription Factor; Sulfanilamides | 2020 |
4 other study(ies) available for way 123398 and e 4031
Article | Year |
---|---|
Effects of WAY-123,398, a new class III antiarrhythmic agent, on cardiac refractoriness and ventricular fibrillation threshold in anesthetized dogs: a comparison with UK-68798, E-4031, and dl-sotalol.
Topics: Anesthesia; Animals; Anti-Arrhythmia Agents; Atrioventricular Node; Benzimidazoles; Dogs; Electrocardiography; Electrophysiology; Female; Heart; Heart Conduction System; Hemodynamics; In Vitro Techniques; Male; Phenethylamines; Piperidines; Purkinje Fibers; Pyridines; Refractory Period, Electrophysiological; Sotalol; Sulfanilamides; Sulfonamides; Ventricular Fibrillation | 1992 |
Cellular electrophysiology of WAY-123,398, a new class III antiarrhythmic agent: specificity of IK block and lack of reverse use dependence in cat ventricular myocytes.
Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Benzimidazoles; Cats; Cells, Cultured; Culture Techniques; Dogs; Dose-Response Relationship, Drug; Myocardium; Phenethylamines; Piperidines; Potassium Channels; Purkinje Fibers; Pyridines; Sotalol; Sulfanilamides; Sulfonamides | 1993 |
A HERG-like K+ channel in rat F-11 DRG cell line: pharmacological identification and biophysical characterization.
Topics: Animals; Anti-Arrhythmia Agents; Benzimidazoles; Brain Neoplasms; Cation Transport Proteins; Cations, Divalent; DNA-Binding Proteins; Electrophysiology; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Ganglia, Spinal; Hybrid Cells; Ion Channel Gating; Kinetics; Membrane Potentials; Mice; Models, Biological; Neuroblastoma; Patch-Clamp Techniques; Piperidines; Potassium Channels; Potassium Channels, Voltage-Gated; Pyridines; Rats; Sulfanilamides; Trans-Activators | 1996 |
Separation of M-like current and ERG current in NG108-15 cells.
Topics: Animals; Benzimidazoles; Bradykinin; Cation Transport Proteins; Ether-A-Go-Go Potassium Channels; Indoles; KCNQ2 Potassium Channel; KCNQ3 Potassium Channel; Membrane Transport Proteins; Mice; Neuroblastoma; Piperidines; Potassium Channels; Potassium Channels, Voltage-Gated; Pyridines; Rats; Sulfanilamides; Sympathetic Nervous System; Tumor Cells, Cultured | 1999 |