Page last updated: 2024-09-03

way 100135 and ipsapirone

way 100135 has been researched along with ipsapirone in 5 studies

Compound Research Comparison

Studies
(way 100135)
Trials
(way 100135)
Recent Studies (post-2010)
(way 100135)
Studies
(ipsapirone)
Trials
(ipsapirone)
Recent Studies (post-2010) (ipsapirone)
1430343735814

Protein Interaction Comparison

ProteinTaxonomyway 100135 (IC50)ipsapirone (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)10
Alpha-2A adrenergic receptorHomo sapiens (human)1
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)10
Alpha-2B adrenergic receptorHomo sapiens (human)1
Alpha-2C adrenergic receptorHomo sapiens (human)1
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0082
D(4) dopamine receptorHomo sapiens (human)1.8
Alpha-1D adrenergic receptorHomo sapiens (human)0.5
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)10
Alpha-1A adrenergic receptorHomo sapiens (human)0.5
Alpha-1B adrenergic receptorHomo sapiens (human)0.5
D(3) dopamine receptorHomo sapiens (human)1.2
D(2) dopamine receptorRattus norvegicus (Norway rat)2.9

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chaput, C; Millan, MJ; Newman-Tancredi, A; Verrièle, L1
Emerit, MB; Hamon, M; Riad, M1
Cervo, L; Samanin, R1
Fijał, K; Gołembiowska, K; Maćkowiak, M; Wedzony, K1
Fujiwara, Y; Hamamura, T; Kuroda, S; Lee, Y1

Other Studies

5 other study(ies) available for way 100135 and ipsapirone

ArticleYear
Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Affinity Labels; Animals; Binding, Competitive; CHO Cells; Cricetinae; Guanine Nucleotides; Hippocampus; Humans; Male; Membranes; Piperazines; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

1998
Neurotrophic effects of ipsapirone and other 5-HT1A receptor agonists on septal cholinergic neurons in culture.
    Brain research. Developmental brain research, 1994, Oct-14, Volume: 82, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Autoradiography; Brain; Cell Division; Cells, Cultured; Choline O-Acetyltransferase; Dose-Response Relationship, Drug; Female; Fetus; Immunohistochemistry; Nerve Growth Factors; Neurons; Piperazines; Pregnancy; Propanolamines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes; Tritium

1994
Presynaptic 5-HT1A receptors mediate the effect of ipsapirone on punished responding in rats.
    European journal of pharmacology, 1995, Sep-25, Volume: 284, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Animals; Anti-Anxiety Agents; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Male; Piperazines; Punishment; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists

1995
Ipsapirone enhances the dopamine outflow via 5-HT1A receptors in the rat prefrontal cortex.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Buspirone; Dopamine; Homovanillic Acid; Male; Microdialysis; Piperazines; Prefrontal Cortex; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Serotonin1A receptor agonists induce Fos protein expression in the locus coeruleus of the conscious rat.
    Brain research, 1997, Jun-06, Volume: 759, Issue:1

    Topics: Animals; Isoindoles; Locus Coeruleus; Male; Neurons; Norepinephrine; Piperazines; Proto-Oncogene Proteins c-fos; Pyrimidines; Rats; Rats, Wistar; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism

1997