Page last updated: 2024-09-03

way 100135 and 5-carboxamidotryptamine

way 100135 has been researched along with 5-carboxamidotryptamine in 6 studies

Compound Research Comparison

Studies
(way 100135)
Trials
(way 100135)
Recent Studies (post-2010)
(way 100135)
Studies
(5-carboxamidotryptamine)
Trials
(5-carboxamidotryptamine)
Recent Studies (post-2010) (5-carboxamidotryptamine)
143034392136

Protein Interaction Comparison

ProteinTaxonomyway 100135 (IC50)5-carboxamidotryptamine (IC50)
5-hydroxytryptamine receptor 1DSus scrofa (pig)0.004

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (33.33)18.2507
2000's3 (50.00)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chaput, C; Millan, MJ; Newman-Tancredi, A; Verrièle, L1
Bill, DJ; Bill, SJ; Cliffe, IA; Dover, GM; Fletcher, A; Forster, EA; Haskins, JT; Jones, D; Mansell, HL; Reilly, Y1
Ajubita, M; Hedo, G; Lopez-Garcia, JA1
Abu-Amara, M; Aldairy, C; Hagan, JJ; Siddiqui, A; Wilson, C1
Shaharyar, S; Siddiqui, A1
Beaudet, G; Bouet, V; Boulouard, M; Dauphin, F; Freret, T; Gusmao-Montaigne, A; Nee, G; Paizanis, E1

Other Studies

6 other study(ies) available for way 100135 and 5-carboxamidotryptamine

ArticleYear
Labelling of recombinant human and native rat serotonin 5-HT1A receptors by a novel, selective radioligand, [3H]-S 15535: definition of its binding profile using agonists, antagonists and inverse agonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Affinity Labels; Animals; Binding, Competitive; CHO Cells; Cricetinae; Guanine Nucleotides; Hippocampus; Humans; Male; Membranes; Piperazines; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

1998
WAY100135: a novel, selective antagonist at presynaptic and postsynaptic 5-HT1A receptors.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Electrophysiology; Female; Guinea Pigs; Hippocampus; Hypothermia; Ileum; Male; Mice; Piperazines; Radioligand Assay; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stereoisomerism

1993
Role of serotonin1A receptors on the modulation of rat spinal mono-synaptic reflexes in vitro.
    Neuroscience letters, 2002, Dec-06, Volume: 334, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Electric Stimulation; Organ Culture Techniques; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reflex, Monosynaptic; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Spinal Nerve Roots

2002
5-HT7 receptor subtype as a mediator of the serotonergic regulation of luteinizing hormone release in the zona incerta.
    European journal of pharmacology, 2004, Apr-26, Volume: 491, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Female; Luteinizing Hormone; Male; Ovariectomy; Phenols; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Subthalamus; Sulfonamides

2004
Attenuating effects of prior oestradiol benzoate priming on 5-HT-mediated lordosis behavior in rats are dose-dependent.
    Acta physiologica Hungarica, 2007, Volume: 94, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Dopamine Antagonists; Dose-Response Relationship, Drug; Estradiol; Female; Male; Ovariectomy; Phenols; Piperazines; Posture; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin; Reflex; Serotonin; Serotonin Receptor Agonists; Sexual Behavior, Animal; Sulfonamides

2007
Modulation of 5-HT7 receptor: effect on object recognition performances in mice.
    Psychopharmacology, 2014, Volume: 231, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Male; Memory, Episodic; Mice; Oxadiazoles; Phenols; Piperazines; Receptors, Serotonin; Recognition, Psychology; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides

2014