Page last updated: 2024-09-03

way 100135 and 1-(3-trifluoromethylphenyl)piperazine

way 100135 has been researched along with 1-(3-trifluoromethylphenyl)piperazine in 3 studies

Compound Research Comparison

Studies
(way 100135)
Trials
(way 100135)
Recent Studies (post-2010)
(way 100135)
Studies
(1-(3-trifluoromethylphenyl)piperazine)
Trials
(1-(3-trifluoromethylphenyl)piperazine)
Recent Studies (post-2010) (1-(3-trifluoromethylphenyl)piperazine)
143034281723

Protein Interaction Comparison

ProteinTaxonomyway 100135 (IC50)1-(3-trifluoromethylphenyl)piperazine (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.57
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.57
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.29
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.61
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.15
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.039
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.57

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kołodziejczyk, K; Maj, J; Rogóz, Z; Skuza, G1
Aguerre, S; Chaouloff, F; Mormede, P1
Heidenreich, BA; Napier, TC1

Other Studies

3 other study(ies) available for way 100135 and 1-(3-trifluoromethylphenyl)piperazine

ArticleYear
Roxindole, a dopamine autoreceptor agonist with a potential antidepressant activity. II. Effects on the 5-hydroxytryptamine system.
    Pharmacopsychiatry, 1997, Volume: 30, Issue:2

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Behavior, Animal; Body Temperature; Dopamine Agonists; Fenfluramine; Indoles; Male; Mice; Motor Activity; Oxindoles; Piperazines; Pyridines; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1997
GR 127935 and (+)-WAY 100135 do not affect TFMPP-induced inhibition of 5-HT synthesis in the midbrain and hippocampus of Wistar-Kyoto rats.
    Neuropharmacology, 1998, Volume: 37, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Hippocampus; Idazoxan; Ketanserin; Male; Mesencephalon; Mianserin; Nerve Endings; Oxadiazoles; Piperazines; Rats; Rats, Inbred WKY; Rats, Wistar; Reserpine; Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity; Tryptophan Hydroxylase

1998
Effects of serotonergic 5-HT1A and 5-HT1B ligands on ventral pallidal neuronal activity.
    Neuroreport, 2000, Sep-11, Volume: 11, Issue:13

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Dose-Response Relationship, Drug; Globus Pallidus; Male; Neurons; Piperazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists

2000