Page last updated: 2024-08-23

vx and tacrine

vx has been researched along with tacrine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Agnusdei, M; Belinskaya, T; Borriello, M; Brindisi, M; Butini, S; Campiani, G; Catalanotti, B; Fattorusso, C; Fiorini, I; Gemma, S; Nacci, V; Novellino, E; Panico, A; Persico, M; Ros, S; Saxena, A1
Bajgar, J1
Costa França, TC; da Silva, JAV; Kuca, K; Nepovimova, E; Ramalho, TC1

Other Studies

3 other study(ies) available for vx and tacrine

ArticleYear
Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Cholinesterase Inhibitors; Computational Biology; Crystallography, X-Ray; Drug Design; Humans; Models, Molecular; Protein Conformation; Structure-Activity Relationship; Tacrine

2008
Protective effect of reversible cholinesterase inhibitors (tacrine, pyridostigmine) and eqbuche against VX poisoning and brain acetylcholinesterase inhibition in rats.
    Acta medica (Hradec Kralove), 2008, Volume: 51, Issue:4

    Topics: Animals; Brain; Chemical Warfare Agents; Cholinesterase Inhibitors; Female; Neurotoxicity Syndromes; Organothiophosphorus Compounds; Pyridostigmine Bromide; Rats; Rats, Wistar; Tacrine

2008
Molecular modelling studies on the interactions of 7-methoxytacrine-4-pyridinealdoxime with VX-inhibited human acetylcholinesterase. A near attack approach to assess different spacer-lengths.
    Chemico-biological interactions, 2019, Jul-01, Volume: 307

    Topics: Acetylcholinesterase; Binding Sites; Cholinesterase Inhibitors; Humans; Ligands; Molecular Docking Simulation; Organothiophosphorus Compounds; Oximes; Protein Structure, Tertiary; Tacrine; Thermodynamics

2019