Page last updated: 2024-09-04

vx 497 and etravirine

vx 497 has been researched along with etravirine in 1 studies

Compound Research Comparison

Studies
(vx 497)
Trials
(vx 497)
Recent Studies (post-2010)
(vx 497)
Studies
(etravirine)
Trials
(etravirine)
Recent Studies (post-2010) (etravirine)
253757290321

Protein Interaction Comparison

ProteinTaxonomyvx 497 (IC50)etravirine (IC50)
Chain A, Reverse transcriptase/ribonuclease HHIV-1 M:B_HXB2R0.0021
Chain B, p51 RTHIV-1 M:B_HXB2R0.0021
Chain A, Reverse transcriptase/ribonuclease HHIV-1 M:B_HXB2R0.0021
Chain B, p51 RTHIV-1 M:B_HXB2R0.0021
ATP-binding cassette sub-family C member 3Homo sapiens (human)5.1
Cytochrome P450 1A2Homo sapiens (human)0.025
ATP-dependent translocase ABCB1Homo sapiens (human)7.6
Cytochrome P450 3A4Homo sapiens (human)0.019
Cytochrome P450 2D6Homo sapiens (human)0.032
Cytochrome P450 2C9 Homo sapiens (human)0.017
Gag-Pol polyproteinHuman immunodeficiency virus type 1 (NEW YORK-5 ISOLATE)0.37
CruzipainTrypanosoma cruzi4
Multidrug resistance-associated protein 1 Homo sapiens (human)8.5
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.01
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.097
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.01
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.01
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.01
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.01
Reverse transcriptase/RNaseH Human immunodeficiency virus 10.2711
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.01
Canalicular multispecific organic anion transporter 1Homo sapiens (human)7.8
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.01
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)6
Reverse transcriptase Human immunodeficiency virus 10.0186

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Other Studies

1 other study(ies) available for vx 497 and etravirine

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023