Page last updated: 2024-08-17

vincristine and verapamil

vincristine has been researched along with verapamil in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (3.13)18.2507
2000's14 (43.75)29.6817
2010's15 (46.88)24.3611
2020's2 (6.25)2.80

Authors

AuthorsStudies
Hosoyama, H; Kobayashi, J; Shigemori, H; Sudo, Y; Tsuruo, T; Wang, XX1
Belinsky, MG; Chen, ZS; Kruh, GD; Rea, PA; Zeng, H1
Huang, L; Humphreys, JE; Morgan, JB; Polli, JW; Serabjit-Singh, CS; Webster, LO; Wring, SA1
Borchardt, RT; Horie, K; Tang, F2
Belinsky, MG; Chen, ZS; Hopper-Borge, E; Kotova, E; Kruh, GD; Shchaveleva, I1
Bacsó, Z; Cianfriglia, M; Fenyvesi, F; Goda, K; Kappelmayer, J; Lustyik, G; Nagy, H; Szabó, G; Szilasi, M1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Burkett, BA; Chan, KF; Chan, TH; Chow, LM; Wong, IL; Zhao, Y1
Abe, M; Ando, M; Bai, J; Hasegawa, T; Hirose, K; Kawakami, J; Kikuchi, M; Matsubara, J; Sakai, J; Tomida, A; Tsuruo, T; Wang, J; Zhang, S1
Abe, M; Ando, M; Bai, J; Bai, L; Bai, Y; Dai, J; Hasegawa, T; Hirose, K; Kikuchi, M; Nishizawa, S; Sakai, J; Tomida, A; Tsuruo, T; Yamori, T1
Baubichon-Cortay, H; Chang, XB; Di Pietro, A; Perrotton, T; Trompier, D1
Ahn, CM; Cho, S; Ham, J; Kim, H; Kim, SN; Kim, YK; Lee, S; Um, Y; Woo, HB1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Jiang, HH; Kong, F; Lou, HX; Sun, B; Xi, GM; Yuan, HQ1
Chen, X; Lin, X; Skolnik, S; Wang, J1
Bastow, KF; Lee, KH; Ohkoshi, E; Shi, Q; Zhou, T1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Song, WB; Wang, WQ; Xuan, LJ; Zhang, SW1
Gan, CY; Kam, TS; Lim, SH; Low, YY; Sim, KS; Yap, WS1
Kam, TS; Lim, SH; Low, YY; Sim, DS; Sim, KS; Teoh, WY; Thomas, NF1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Abdelazeem, AH; Amjad, MW; Bukhari, SNA; Qin, HL; Raja, MAG; Youssif, BGM; Zha, GF1
Gurusamy, S; Kam, TS; Lim, SH; Low, YY; Navanesan, S; Sim, KS; Yeap, JS; Yong, KT1
Chen, X; Chen, Y; Guo, Y; Lee, KH; Li, H; Morris-Natschke, S; Wan, Q; Wang, K1
Gurusamy, S; Kam, TS; Lim, SH; Low, YY; Navanesan, S; Sim, DS; Sim, KS1
Chein, RJ; Chen, JJW; Cheng, TR; Chou, TH; Chung, WC; Hong, TM; Lee, TC; Lin, MS; Tsai, ML; Weng, CW; Wong, CH; Yang, PC; Yang, SC1
Kam, TS; Lim, SH; Low, YY; Saad, HM; Sim, KS; Tan, CH; Yeap, JS1
Bi, Y; Chen, X; Huang, W; Li, X; Liang, K; Liu, S; Ma, M; Wang, B; Wang, H; Zeng, W1
Bao, XZ; Cai, Y; Cui, ZN; Huang, Z; Li, YS; Liu, GJ; Wang, H; Wang, J; Wang, SJ; Wei, B; Wu, R; Yang, X; Ye, XY; Zhao, DS1

Reviews

1 review(s) available for vincristine and verapamil

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

31 other study(ies) available for vincristine and verapamil

ArticleYear
Modulation of multidrug resistance by taxuspine C and other taxoids from Japanese yew.
    Bioorganic & medicinal chemistry letters, 1998, Jun-16, Volume: 8, Issue:12

    Topics: Animals; Bridged-Ring Compounds; Carcinoma, Squamous Cell; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Humans; Leukemia L1210; Leukemia P388; Mice; Phenylpropionates; Taxoids; Trees; Tumor Cells, Cultured; Vincristine

1998
Transport of methotrexate (MTX) and folates by multidrug resistance protein (MRP) 3 and MRP1: effect of polyglutamylation on MTX transport.
    Cancer research, 2001, Oct-01, Volume: 61, Issue:19

    Topics: 3T3 Cells; Animals; ATP-Binding Cassette Transporters; Biological Transport; Drug Resistance, Multiple; Folic Acid; Humans; Leucovorin; Methotrexate; Mice; Multidrug Resistance-Associated Proteins; Osmolar Concentration; Polyglutamic Acid; Tritium

2001
Rational use of in vitro P-glycoprotein assays in drug discovery.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:2

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Chromatography, Liquid; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; Mass Spectrometry; Pharmacology; Spodoptera

2001
Are MDCK cells transfected with the human MDR1 gene a good model of the human intestinal mucosa?
    Pharmaceutical research, 2002, Volume: 19, Issue:6

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cell Line; Digoxin; Dogs; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Genes, MDR; Humans; Intestinal Mucosa; Transfection

2002
Are MDCK cells transfected with the human MRP2 gene a good model of the human intestinal mucosa?
    Pharmaceutical research, 2002, Volume: 19, Issue:6

    Topics: Animals; Caco-2 Cells; Cell Line; Dogs; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Intestinal Mucosa; Mitochondrial Proteins; Multidrug Resistance-Associated Protein 2; Ribosomal Proteins; Saccharomyces cerevisiae Proteins; Transfection; Vinblastine

2002
Characterization of the transport properties of human multidrug resistance protein 7 (MRP7, ABCC10).
    Molecular pharmacology, 2003, Volume: 63, Issue:2

    Topics: Biological Transport; Cells, Cultured; Cyclosporine; Estradiol; Glycocholic Acid; Humans; Kinetics; Leukotriene Antagonists; Leukotriene C4; Multidrug Resistance-Associated Proteins; Osmotic Pressure; Propionates; Quinolines; Recombinant Proteins; Transfection

2003
Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.
    Biochemical and biophysical research communications, 2004, Mar-19, Volume: 315, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Anti-Bacterial Agents; Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Calcium Channel Blockers; Cyclosporine; Detergents; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Humans; Ivermectin; Mice; NIH 3T3 Cells; Substrate Specificity

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Flavonoid dimers as bivalent modulators for P-glycoprotein-based multidrug resistance: synthetic apigenin homodimers linked with defined-length poly(ethylene glycol) spacers increase drug retention and enhance chemosensitivity in resistant cancer cells.
    Journal of medicinal chemistry, 2006, Nov-16, Volume: 49, Issue:23

    Topics: Adenosine Triphosphatases; Animals; Antineoplastic Agents; Apigenin; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Dimerization; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Mice; Paclitaxel; Polyethylene Glycols; Structure-Activity Relationship; Vinblastine

2006
Structure-activity relationships of some taxoids as multidrug resistance modulator.
    Bioorganic & medicinal chemistry letters, 2007, Feb-15, Volume: 17, Issue:4

    Topics: Alkaloids; Antineoplastic Agents; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Structure-Activity Relationship; Taxoids; Taxus

2007
Synthesis and structure-activity relationships of taxuyunnanine C derivatives as multidrug resistance modulator in MDR cancer cells.
    Bioorganic & medicinal chemistry letters, 2007, Jul-01, Volume: 17, Issue:13

    Topics: Antineoplastic Agents; Biological Assay; Cell Line; Cell Line, Tumor; Chemistry, Pharmaceutical; Drug Design; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Fluoresceins; Humans; Inhibitory Concentration 50; Models, Chemical; Structure-Activity Relationship; Taxoids

2007
(R)- and (S)-verapamil differentially modulate the multidrug-resistant protein MRP1.
    The Journal of biological chemistry, 2007, Oct-26, Volume: 282, Issue:43

    Topics: Adenosine Triphosphatases; Animals; Cell Line; Cell Proliferation; Cell Survival; Cricetinae; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Fluoresceins; Fluorescent Dyes; Formazans; Glutathione; Inhibitory Concentration 50; Kidney; Leukotriene C4; Multidrug Resistance-Associated Proteins; Protein Conformation; Sodium Iodide; Spectrometry, Fluorescence; Stereoisomerism; Tetrazolium Salts; Transfection; Tryptophan; Verapamil

2007
Synthesis of curcumin mimics with multidrug resistance reversal activities.
    Bioorganic & medicinal chemistry, 2008, Apr-01, Volume: 16, Issue:7

    Topics: Cell Line, Tumor; Cell Survival; Cross-Linking Reagents; Curcumin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Molecular Structure; Stereoisomerism

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Bisbibenzyl derivatives sensitize vincristine-resistant KB/VCR cells to chemotherapeutic agents by retarding P-gp activity.
    Bioorganic & medicinal chemistry, 2010, Sep-15, Volume: 18, Issue:18

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bibenzyls; Catechols; Cell Line, Tumor; Doxorubicin; Drug Resistance, Neoplasm; Ethers, Cyclic; Humans; Phenyl Ethers; Rhodamine 123; Stilbenes; Vincristine

2010
Attenuation of intestinal absorption by major efflux transporters: quantitative tools and strategies using a Caco-2 model.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:2

    Topics: Adenosine; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Sub-Family B Member 4; ATP-Binding Cassette Transporters; Biological Transport; Caco-2 Cells; Chromatography, Liquid; Dibenzocycloheptenes; Diketopiperazines; Drug Discovery; Heterocyclic Compounds, 4 or More Rings; Humans; Intestinal Absorption; Mass Spectrometry; Models, Biological; Neoplasm Proteins; Pharmaceutical Preparations; Predictive Value of Tests; Propionates; Quinolines; Substrate Specificity

2011
Anti-AIDS agents 89. Identification of DCX derivatives as anti-HIV and chemosensitizing dual function agents to overcome P-gp-mediated drug resistance for AIDS therapy.
    Bioorganic & medicinal chemistry letters, 2012, May-01, Volume: 22, Issue:9

    Topics: Anti-HIV Agents; ATP Binding Cassette Transporter, Subfamily B; Cell Line, Tumor; Chromones; Drug Resistance, Multiple; Drug Resistance, Viral; Humans; Verapamil; Vincristine; Xanthones

2012
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Multidrug resistance-reversal effects of resin glycosides from Dichondra repens.
    Bioorganic & medicinal chemistry letters, 2015, Feb-15, Volume: 25, Issue:4

    Topics: Carbohydrate Sequence; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Glycosides; Humans; KB Cells; Molecular Sequence Data; Plant Leaves; Poaceae; Resins, Plant; Vincristine

2015
Aspidofractinine and Eburnane Alkaloids from a North Borneo Kopsia. Ring-Contracted, Additional Ring-Fused, and Paucidactine-Type Aspidofractinine Alkaloids from K. pauciflora.
    Journal of natural products, 2016, Jan-22, Volume: 79, Issue:1

    Topics: Antineoplastic Agents, Phytogenic; Apocynaceae; Borneo; Crystallography, X-Ray; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Indole Alkaloids; KB Cells; Malaysia; Molecular Conformation; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Plant Bark; Vincristine

2016
Vobatensines A-F, Cytotoxic Iboga-Vobasine Bisindoles from Tabernaemontana corymbosa.
    Journal of natural products, 2016, Apr-22, Volume: 79, Issue:4

    Topics: Antineoplastic Agents, Phytogenic; Drug Screening Assays, Antitumor; HCT116 Cells; HT29 Cells; Humans; Indole Alkaloids; KB Cells; Malaysia; Molecular Structure; Plant Leaves; Tabernaemontana

2016
Discovery of potential anticancer multi-targeted ligustrazine based cyclohexanone and oxime analogs overcoming the cancer multidrug resistance.
    European journal of medicinal chemistry, 2017, Jul-28, Volume: 135

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cyclohexanones; Dose-Response Relationship, Drug; Drug Discovery; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Molecular Docking Simulation; Molecular Structure; Oximes; Pyrazines; Structure-Activity Relationship

2017
Ajmaline, Oxindole, and Cytotoxic Macroline-Akuammiline Bisindole Alkaloids from Alstonia penangiana.
    Journal of natural products, 2018, 05-25, Volume: 81, Issue:5

    Topics: A549 Cells; Ajmaline; Alkaloids; Alstonia; Antineoplastic Agents, Phytogenic; Cell Line, Tumor; Crystallography, X-Ray; Cytotoxins; Drug Screening Assays, Antitumor; HCT116 Cells; HT29 Cells; Humans; KB Cells; MCF-7 Cells; Oxindoles; PC-3 Cells; Vincristine

2018
Seco-4-methyl-DCK derivatives as potent chemosensitizers.
    Bioorganic & medicinal chemistry letters, 2019, 01-01, Volume: 29, Issue:1

    Topics: Antineoplastic Agents; Cell Line; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Screening Assays, Antitumor; Humans; Molecular Structure; Structure-Activity Relationship

2019
Conolodinines A-D, Aspidosperma- Aspidosperma Bisindole Alkaloids with Antiproliferative Activity from Tabernaemontana corymbosa.
    Journal of natural products, 2019, 04-26, Volume: 82, Issue:4

    Topics: Aspidosperma; Cell Line, Tumor; Cell Proliferation; Drug Screening Assays, Antitumor; Humans; Indole Alkaloids; Molecular Structure; Spectrum Analysis; Tabernaemontana

2019
4(1H)-quinolone derivatives overcome acquired resistance to anti-microtubule agents by targeting the colchicine site of β-tubulin.
    European journal of medicinal chemistry, 2019, Nov-01, Volume: 181

    Topics: Antineoplastic Agents; Apoptosis; Binding Sites; Cell Proliferation; Colchicine; Drug Resistance, Neoplasm; Humans; Molecular Docking Simulation; Neoplasms; Quinolones; Tubulin; Tubulin Modulators

2019
Macroline-Sarpagine Bisindole Alkaloids with Antiproliferative Activity from
    Journal of natural products, 2019, 11-22, Volume: 82, Issue:11

    Topics: A549 Cells; Alkaloids; Alstonia; Antineoplastic Agents, Phytogenic; Cell Line, Tumor; Cell Proliferation; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; HT29 Cells; Humans; Indole Alkaloids; Molecular Structure; Oxindoles

2019
Design, synthesis, and biological evaluation of hederagenin derivatives with improved aqueous solubility and tumor resistance reversal activity.
    European journal of medicinal chemistry, 2021, Feb-05, Volume: 211

    Topics: Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Molecular Structure; Oleanolic Acid; Structure-Activity Relationship

2021
Design, synthesis and bioactivity study on 5-phenylfuran derivatives as potent reversal agents against P-glycoprotein-mediated multidrug resistance in MCF-7/ADR cell.
    European journal of medicinal chemistry, 2021, Apr-15, Volume: 216

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Line, Tumor; Cell Proliferation; Doxorubicin; Drug Design; Drug Resistance, Neoplasm; Furans; Humans; Molecular Docking Simulation; Paclitaxel; Structure-Activity Relationship; Tetrahydroisoquinolines

2021