Page last updated: 2024-08-17

veratridine and piperidines

veratridine has been researched along with piperidines in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-19904 (14.29)18.7374
1990's17 (60.71)18.2507
2000's7 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Leidig, A; Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wirth, A1
Adam-Vizi, V; Deri, Z1
Gleitz, J; Peters, T; Tegtmeier, F; Urenjak, J; Wermelskirchen, D; Wilffert, B1
Borgers, M; Ver Donck, L1
Bielen, FV; Ver Donck, L; Verdonck, F1
Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wirth, A1
Himmel, H; Peters, T; Ravens, U; Wilhelm, D1
Adam-Vizi, V; Deri, Z; Lajtha, A; Sershen, H; Vizi, ES1
Johnson, RG; Unsworth, CD1
Cohen-Armon, M; Sokolovsky, M1
Cohen-Armon, M; Henis, YI; Kloog, Y; Sokolovsky, M1
Carroll, PT; Ivy, MT1
Carroll, PT1
Marshall, IG; Nguyen, ML; Parsons, SM; Pemberton, KE; Prior, C1
Bindels, RJ; Couwenberg, P; Jansen, JW; Rose, UM; Van Os, CH1
Campbell, GW; Dooley, DJ; Hays, SJ; Probert, AW; Roufos, I; Schwarz, RD1
Hays, S; Roufos, I; Schwarz, RD1
De la Fuente, MT; Esquerro, E; García, AG; Maroto, R; Sánchez-García, P1
Ashton, D; Clincke, G; Marrannes, R; Van Reempts, J; Willems, R; Wynants, J1
Almond, HR; Carmosin, RJ; Carson, JR; Pitis, PM; Stables, JP; Swinyard, EA; Vaught, JL; White, HS; Wolf, HH1
Cano-Abad, MF; Gandía, L; García, AG; Hernández-Guijo, JM; López, MG; Sánchez-García, P; Zapater, P1
Auld, DS; Day, JC; Mennicken, F; Quirion, R1
Gudelsky, GA; Vorhees, CV; Wallace, TL1
David, LS; Liao, C; Nicholson, RA; Zheng, J1
Abdel-Aziz, H; Ploch, M; Verspohl, EJ; Windeck, T1
Akada, Y; Amano, K; Fukudome, Y; Itoh, M; Ogawa, S; Yamamoto, I; Yamasaki, F1
Akaike, A; Akasofu, S; Hihara, H; Kosasa, T; Ogura, H; Sawada, K1
Duan, Y; Jain, S; Liao, C; Nicholson, RA1

Other Studies

28 other study(ies) available for veratridine and piperidines

ArticleYear
Veratridine activates a silent sodium channel in rat isolated aorta.
    European journal of pharmacology, 1992, Aug-25, Volume: 219, Issue:2

    Topics: Amiloride; Animals; Aorta; Benzothiazoles; Calcium; Guanidine; Guanidines; In Vitro Techniques; Piperidines; Pyrroles; Rats; Sodium Channels; Tetrodotoxin; Thiazoles; Vasodilator Agents; Veratridine

1992
Parameters not influenced by vesamicol: membrane potential, calcium uptake, and internal calcium concentration of synaptosomes.
    Neurochemical research, 1992, Volume: 17, Issue:6

    Topics: Acetylcholine; Animals; Calcium; Fura-2; Guinea Pigs; Membrane Potentials; Neuromuscular Depolarizing Agents; Piperidines; Potassium; Sodium; Synaptosomes; Veratridine

1992
Flunarizine and R 56865 suppress veratridine-induced increase in oxygen consumption and uptake of 45Ca2+ in rat cortical synaptosomes.
    Neuropharmacology, 1992, Volume: 31, Issue:3

    Topics: Animals; Benzothiazoles; Calcium; Calcium Radioisotopes; Cerebral Cortex; Flunarizine; In Vitro Techniques; Oxygen Consumption; Piperidines; Polarography; Rats; Synaptosomes; Tetrodotoxin; Thiazoles; Veratridine

1992
Myocardial protection by R 56865: a new principle based on prevention of ion channel pathology.
    The American journal of physiology, 1991, Volume: 261, Issue:6 Pt 2

    Topics: Animals; Benzothiazoles; Calcium; Cardiomyopathies; Heart; Lysophosphatidylcholines; Myocardial Contraction; Ouabain; Oxygen; Piperidines; Rabbits; Rats; Singlet Oxygen; Sodium; Sodium Channels; Tetrodotoxin; Thiazoles; Veratridine

1991
Preferential block of the veratridine-induced, non-inactivating Na+ current by R56865 in single cardiac Purkinje cells.
    European journal of pharmacology, 1991, Oct-22, Volume: 203, Issue:3

    Topics: Animals; Benzothiazoles; Heart; In Vitro Techniques; Membrane Potentials; Myocardium; Piperidines; Purkinje Cells; Rabbits; Sodium Channels; Tetrodotoxin; Thiazoles; Veratridine

1991
Veratridine-induced intoxication in the isolated left atrium of the rat: effects of some anti-ischemic compounds.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:1

    Topics: Animals; Atrial Function, Left; Benzothiazoles; Calcium; Coronary Disease; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Male; Piperidines; Pyrroles; Rats; Sodium; Sodium Channels; Thiazoles; Veratridine

1991
Characterization of the interaction of R 56865 with cardiac Na- and L-type Ca channels.
    British journal of pharmacology, 1991, Volume: 104, Issue:2

    Topics: Action Potentials; Animals; Benzothiazoles; Biomechanical Phenomena; Calcium Channels; Guinea Pigs; Heart; In Vitro Techniques; Myocardium; Papillary Muscles; Piperidines; Sodium; Sodium Channels; Thiazoles; Veratridine

1991
Ca2+o-independent veratridine-evoked acetylcholine release from striatal slices is not inhibited by vesamicol (AH5183): mobilization of distinct transmitter pools.
    Journal of neurochemistry, 1991, Volume: 56, Issue:1

    Topics: Acetylcholine; Animals; Calcium; Carbon Radioisotopes; Corpus Striatum; Electric Stimulation; In Vitro Techniques; Male; Perfusion; Piperidines; Rats; Rats, Inbred Strains; Veratridine

1991
Acetylcholine and ATP are coreleased from the electromotor nerve terminals of Narcine brasiliensis by an exocytotic mechanism.
    Proceedings of the National Academy of Sciences of the United States of America, 1990, Volume: 87, Issue:2

    Topics: Acetylcholine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcimycin; Electric Organ; Exocytosis; Ionomycin; Kinetics; Motor Neurons; Nerve Endings; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Potassium; Subcellular Fractions; Synaptosomes; Torpedo; Veratridine

1990
Interactions between the muscarinic receptors, sodium channels, and guanine nucleotide-binding protein(s) in rat atria.
    The Journal of biological chemistry, 1986, Sep-25, Volume: 261, Issue:27

    Topics: Acetylcholine; Animals; Batrachotoxins; Benzilates; Carbachol; Dibucaine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Ion Channels; Kinetics; Male; Mathematics; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1986
Batrachotoxin changes the properties of the muscarinic receptor in rat brain and heart: possible interaction(s) between muscarinic receptors and sodium channels.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:10

    Topics: Aconitine; Animals; Batrachotoxins; Benzilates; Binding, Competitive; Brain; Carbachol; Guanylyl Imidodiphosphate; Ion Channels; Kinetics; Macromolecular Substances; Male; Myocardium; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine

1985
Effect of 2-(4-phenylpiperidino)cyclohexanol (AH 5183) on the veratridine-induced increase in acetylcholine synthesis by rat hippocampal tissue.
    Journal of neurochemistry, 1988, Volume: 51, Issue:3

    Topics: Acetylcholine; Animals; Choline; Choline O-Acetyltransferase; Hippocampus; Isotonic Solutions; L-Lactate Dehydrogenase; Male; Naphthylvinylpyridine; Octoxynol; Phencyclidine; Piperidines; Polyethylene Glycols; Rats; Rats, Inbred Strains; Solubility; Subcellular Fractions; Veratridine; Veratrine

1988
The effect of the acetylcholine transport blocker 2-(4-phenylpiperidino) cyclohexanol (AH5183) on the subcellular storage and release of acetylcholine in mouse brain.
    Brain research, 1985, Dec-09, Volume: 358, Issue:1-2

    Topics: Acetylcholine; Animals; Biological Transport; Brain; Electric Organ; Mice; Mice, Inbred ICR; Phencyclidine; Piperidines; Potassium; Synaptic Vesicles; Torpedo; Veratridine

1985
Effect of veratridine on miniature endplate current amplitudes at the rat neuromuscular junction and acetylcholine uptake by Torpedo synaptic vesicles.
    Brain research, 1995, Feb-13, Volume: 671, Issue:2

    Topics: Acetylcholine; Animals; Electric Organ; Electrophysiology; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Membrane Potentials; Motor Endplate; Muscle Fibers, Skeletal; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Piperidines; Rats; Rats, Sprague-Dawley; Synaptic Vesicles; Tetrodotoxin; Torpedo; Veratridine

1995
Effects of substrate-free anoxia and veratridine on intracellular calcium concentration in isolated rat ventricular cardiomyocytes.
    Pflugers Archiv : European journal of physiology, 1994, Volume: 428, Issue:2

    Topics: Animals; Benzothiazoles; Calcium; Calcium Channel Blockers; Cell Hypoxia; Cell Separation; Cell Size; Male; Microscopy, Fluorescence; Myocardial Contraction; Myocardium; Piperidines; Rats; Rats, Wistar; Sodium; Thiazoles; Veratridine

1994
Synthesis and pharmacological evaluation of phenylacetamides as sodium-channel blockers.
    Journal of medicinal chemistry, 1994, Jan-21, Volume: 37, Issue:2

    Topics: Acetamides; Animals; Batrachotoxins; Benzeneacetamides; Cell Hypoxia; Cells, Cultured; Cerebral Cortex; CHO Cells; Cricetinae; L-Lactate Dehydrogenase; Male; Piperidines; Rats; Rats, Sprague-Dawley; Sodium; Sodium Channel Blockers; Structure-Activity Relationship; Veratridine

1994
A structure-activity relationship study of novel phenylacetamides which are sodium channel blockers.
    Journal of medicinal chemistry, 1996, Mar-29, Volume: 39, Issue:7

    Topics: Acetamides; Animals; Benzeneacetamides; CHO Cells; Cricetinae; Magnetic Resonance Spectroscopy; Molecular Structure; Piperidines; Sodium; Sodium Channel Blockers; Sodium Channels; Structure-Activity Relationship; Veratridine

1996
The actions of ouabain and lithium chloride on cytosolic Ca2+ in single chromaffin cells.
    European journal of pharmacology, 1996, Jun-13, Volume: 306, Issue:1-3

    Topics: Adrenal Glands; Animals; Antimanic Agents; Benzothiazoles; Calcium; Calcium Channel Blockers; Calcium Channels; Cattle; Cell Membrane; Cells, Cultured; Chromaffin System; Enzyme Inhibitors; Lithium Chloride; omega-Conotoxins; Ouabain; Peptides; Piperidines; Sodium; Sodium-Potassium-Exchanging ATPase; Thiazoles; Veratridine

1996
Altered Na(+)-channel function as an in vitro model of the ischemic penumbra: action of lubeluzole and other neuroprotective drugs.
    Brain research, 1997, Jan-16, Volume: 745, Issue:1-2

    Topics: Animals; Brain Ischemia; Calcium Channel Blockers; Cerebral Infarction; Cerebrovascular Circulation; Extracellular Space; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Microelectrodes; Neuroprotective Agents; Piperidines; Pyramidal Cells; Sodium Channels; Thiazoles; Veratridine

1997
Aroyl(aminoacyl)pyrroles, a new class of anticonvulsant agents.
    Journal of medicinal chemistry, 1997, May-23, Volume: 40, Issue:11

    Topics: Anesthesia; Animals; Anticonvulsants; Bicuculline; Calcium; Cerebellum; Electroshock; Mice; Models, Molecular; Molecular Structure; Pentylenetetrazole; Piperidines; Potassium; Pyrroles; Rats; Seizures; Structure-Activity Relationship; Veratridine

1997
Effects of the neuroprotectant lubeluzole on the cytotoxic actions of veratridine, barium, ouabain and 6-hydroxydopamine in chromaffin cells.
    British journal of pharmacology, 1998, Volume: 124, Issue:6

    Topics: Adrenal Glands; Animals; Barium; Calcium; Cattle; Chromaffin Cells; Cytosol; Neuroprotective Agents; Ouabain; Oxidopamine; Penfluridol; Piperidines; Sodium; Thiazoles; Veratridine

1998
Pharmacological characterization of endogenous acetylcholine release from primary septal cultures.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:2

    Topics: Acetylcholine; Animals; Cells, Cultured; Choline; Choline O-Acetyltransferase; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Muscarinic Agonists; Neuromuscular Depolarizing Agents; Oxotremorine; Parasympatholytics; Piperidines; Pirenzepine; Potassium; Rats; Septum of Brain; Time Factors; Veratridine

2000
Effects of lubeluzole on the methamphetamine-induced increase in extracellular glutamate and the long-term depletion of striatal dopamine.
    Synapse (New York, N.Y.), 2001, Volume: 40, Issue:2

    Topics: Animals; Body Temperature; Dopamine; Drug Interactions; Extracellular Space; Glutamic Acid; Male; Methamphetamine; Neostriatum; Neurons; Neuroprotective Agents; Piperidines; Rats; Rats, Sprague-Dawley; Sodium Channels; Thiazoles; Veratridine

2001
Inhibition of voltage-sensitive sodium channels by the cannabinoid 1 receptor antagonist AM 251 in mammalian brain.
    Basic & clinical pharmacology & toxicology, 2004, Volume: 94, Issue:2

    Topics: Animals; Batrachotoxins; Brain; Cannabinoid Receptor Antagonists; Drug Interactions; Male; Membrane Potentials; Mice; Piperidines; Pyrazoles; Sodium Channels; Synaptosomes; Veratridine

2004
Mode of action of gingerols and shogaols on 5-HT3 receptors: binding studies, cation uptake by the receptor channel and contraction of isolated guinea-pig ileum.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: Animals; Binding, Competitive; Carbon Radioisotopes; Catechols; Cations; Cell Line, Tumor; Dose-Response Relationship, Drug; Fatty Alcohols; Guanidine; Guinea Pigs; Humans; Ileum; Imidazoles; In Vitro Techniques; Indoles; Ion Channels; Isotonic Contraction; Male; Mice; Organic Cation Transport Proteins; Piperidines; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Sodium Channels; Substance P; Tritium; Tropisetron; Veratridine; Zingiber officinale

2006
Potent analgesic effects of a putative sodium channel blocker M58373 on formalin-induced and neuropathic pain in rats.
    European journal of pharmacology, 2006, May-01, Volume: 536, Issue:3

    Topics: Analgesics; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Formaldehyde; Ganglia, Spinal; Hot Temperature; Hyperalgesia; Male; Mexiletine; Motor Activity; Neuralgia; Nitriles; Pain; Pain Measurement; Piperidines; Rats; Rats, Wistar; Sodium Channel Blockers; Stress, Mechanical; Substance P; Veratridine

2006
Donepezil attenuates excitotoxic damage induced by membrane depolarization of cortical neurons exposed to veratridine.
    European journal of pharmacology, 2008, Jul-07, Volume: 588, Issue:2-3

    Topics: Animals; Calcium; Caspase Inhibitors; Cells, Cultured; Cerebral Cortex; Cholinesterase Inhibitors; Donepezil; Glutamic Acid; Glycine; Indans; Membrane Potentials; Neuroprotective Agents; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Sodium; Tetrodotoxin; Veratridine

2008
The cannabinoid receptor agonist CP-55,940 and ethyl arachidonate interfere with [(3)H]batrachotoxinin A 20 alpha-benzoate binding to sodium channels and inhibit sodium channel function.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2008, Volume: 148, Issue:3

    Topics: Animals; Arachidonic Acids; Batrachotoxins; Brain; Cannabinoid Receptor Agonists; Cyclohexanols; Mice; Piperidines; Pyrazoles; Sodium Channels; Veratridine

2008