verapamil has been researched along with verlukast in 45 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 24 (53.33) | 29.6817 |
2010's | 21 (46.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Lombardo, F; Obach, RS; Waters, NJ | 1 |
Berardi, F; Carotti, A; Cellamare, S; Colabufo, NA; Leonetti, F; Nicolotti, O; Niso, M; Pellicani, RZ; Perrone, R; Stefanachi, A | 1 |
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR | 1 |
Cory, AH; Cory, JG | 1 |
Bates, SE; Dietel, M; Hohenberger, P; Jordan, A; Lage, H; Litman, T; Stein, U; Walther, W | 1 |
Taylor, EM; Yan, R | 1 |
Buesen, R; Jacob, J; Lampen, A; Mock, M; Nau, H; Seidel, A | 1 |
Bacchelli, B; Boraldi, F; Croce, MA; Garcia Fernandez, MI; Gheduzzi, D; Pasquali Ronchetti, I; Quaglino, D; Tiozzo, R | 1 |
Candussio, L; Crivellato, E; Damiani, D; Decorti, G; Giraldi, T; Klugmann, FB; Michelutti, A; Rosati, A | 1 |
Honkakoski, P; Urtti, A; Vellonen, KS | 1 |
Garnier-Suillerot, A; Loechariyakul, P; Saengkhae, C; Salerno, M | 1 |
Honda, Y; Koyabu, N; Kuwano, M; Morimoto, S; Ohtani, H; Sawada, Y; Shoyama, Y; Uchiumi, T; Ushigome, F | 1 |
Kobayashi, S; Konishi, Y | 1 |
Hanada, M; Iwamoto, Y; Li, X; Matsunobu, T; Nakamura, T; Nakatani, F; Oda, Y; Okada, T; Sakimura, R; Tanaka, K; Tsuneyoshi, M | 1 |
Leader, JP; O'Donnell, MJ | 1 |
Foth, H; Glahn, F; Stehfest, E; Torky, A | 1 |
Bertelsen, KM; Greenblatt, DJ; von Moltke, LL | 1 |
Cole, B; Epel, D; Hamdoun, A; Thurber, RV | 1 |
Chiou, WL; Yao, HM | 1 |
Tian, X; Wang, K; Yang, X | 1 |
Guo, QM; Tian, L; Tian, XJ; Wang, Y; Xu, W; Yang, XW | 1 |
Chen, X; Chowbay, B; Duan, W; Li, CG; Liang, J; Lin, SG; Liu, PQ; Wen, JY; Yu, XY; Zhou, SF; Zhou, ZW | 1 |
Jani, M; Kovács, B; Krajcsi, P; Lin, G; Zhang, L; Zuo, Z | 1 |
Abdel-Tawab, M; Fricker, G; Hummel, J; Kanzer, J; Krüger, P; Schubert-Zsilavecz, M | 1 |
Balimane, PV; Chong, S; Marino, A | 1 |
Kamiyama, E; Miura, S; Nakai, D; Okazaki, O; Sugiyama, D | 1 |
Barata, C; Faria, M; Luckenbach, T; Navarro, A; Piña, B | 1 |
Ahn, SH; Bae, MA; Cheon, HG; Jeon, DJ; Kim, MS; Kwon, KI; Lee, BH; Park, JS; Rho, HJ; Seo, JW; Song, JS | 1 |
Gao, C; Jiang, J; Qiu, F; Tan, Y; Zhang, X | 1 |
Jakob, I; Molinas, A; Sicard, G | 1 |
Deng, ZY; Hu, JN; Li, HY; Li, W; Liu, XR; Luo, T; Ye, H; Zhang, B; Zheng, YN; Zhu, XM | 1 |
de Araújo Leite, JC; Marques-Santos, LF; Santi-Gadelha, T; Silva-Neta, HL; Torrezan, E | 1 |
Gao, S; Hu, M; Liu, W; Liu, Z; Wang, F; Yang, X; Yang, Z; Ye, L; Yin, T | 1 |
Li, X; Liu, D; Rong, Z; Xiang, D; Xu, Y; Zhang, C | 1 |
Li, Z; Liu, F; Ruan, J; Yang, C; Zhang, T; Zhang, Z | 1 |
Adkins, CE; Bohn, KA; Lockman, PR; Manda, VK; Mittapalli, RK | 1 |
Chen, Z; Han, J; Hu, T; Huang, C; Li, J; Ma, T; Zhang, L; Zhong, J | 1 |
Chen, Y; Gao, X; Liu, C; Qu, D; Wang, Y; Zhou, J | 1 |
Kukkonen, JV; Vehniäinen, ER | 1 |
Berginc, K; Kristl, A; Lušin, TT; Mrhar, A; Stieger, B; Trontelj, J | 1 |
Altenburger, R; Barata, C; Burkhardt-Medicke, K; Faria, M; Luckenbach, T; Pavlichenko, V; Soares, AM | 1 |
Chen, KC; Chen, YL; Hsu, SL; Hsueh, CM; Wu, CL; Yang, TY | 1 |
Cao, L; Fang, P; Guo, Z; Hou, Z; Li, Z; Yan, M; Zhang, B | 1 |
Khangembam, R; Rath, SS; Singh, H; Singh, NK | 1 |
Fukuchi, K; Kawai, K; Kobayashi, M; Mizutani, A; Nakanishi, T; Nishi, K; Nishii, R; Okui, Y; Tamai, I; Tsujiuchi, T | 1 |
45 other study(ies) available for verapamil and verlukast
Article | Year |
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Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Potent galloyl-based selective modulators targeting multidrug resistance associated protein 1 and P-glycoprotein.
Topics: Anilides; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Cell Line; Dogs; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Stability; Ethers; Gallic Acid; Pyrogallol; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship | 2012 |
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection | 2012 |
Comparison of the properties of human breast cancer cells: MCF-7 and MCF-7 cells selected for resistance to etoposide.
Topics: Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Chromatography, High Pressure Liquid; Dactinomycin; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Neoplasm; Etoposide; Flow Cytometry; Humans; Leukotriene Antagonists; Propionates; Protein Synthesis Inhibitors; Quinolines; Tumor Cells, Cultured; Vasodilator Agents; Verapamil; Vinblastine | 2001 |
Impact of BCRP/MXR, MRP1 and MDR1/P-Glycoprotein on thermoresistant variants of atypical and classical multidrug resistant cancer cells.
Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Calcium Channel Blockers; DNA Primers; DNA-Binding Proteins; Doxorubicin; Drug Resistance, Multiple; Fluorescent Dyes; Gastrointestinal Neoplasms; Gene Expression Regulation; Genes, MDR; Hot Temperature; Humans; Indenes; Mitoxantrone; Multidrug Resistance-Associated Proteins; MutS Homolog 3 Protein; Mycotoxins; Neoplasm Proteins; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; RNA, Neoplasm; Stomach Neoplasms; Verapamil | 2002 |
Neotrofin is transported out of brain by a saturable mechanism: possible involvement of multidrug resistance and monocarboxylic acid transporters.
Topics: Aminobenzoates; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Brain; Capillaries; Drug Resistance, Multiple; Endothelium, Vascular; Hypoxanthines; Injections, Intraventricular; Male; Mice; Monocarboxylic Acid Transporters; Nootropic Agents; Organic Anion Transporters; Probenecid; Propionates; Purines; Quinolines; Verapamil | 2002 |
Human intestinal Caco-2 cells display active transport of benzo[a]pyrene metabolites.
Topics: Adenosine Triphosphate; Aryl Hydrocarbon Hydroxylases; ATP-Binding Cassette Transporters; Benzo(a)pyrene; Benzoflavones; Biological Transport, Active; Caco-2 Cells; Cell Polarity; Cyclosporine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1B1; Enterocytes; Gene Expression; Humans; Models, Biological; Probenecid; Propionates; Quinolines; Verapamil; Vinblastine | 2003 |
Multidrug resistance protein-6 (MRP6) in human dermal fibroblasts. Comparison between cells from normal subjects and from Pseudoxanthoma elasticum patients.
Topics: Adult; Benzbromarone; Cell Count; Cell Division; Chlorambucil; Female; Fibroblasts; Fluoresceins; Fluorescent Dyes; Humans; Indomethacin; Lysosomes; Male; Membrane Transport Proteins; Microscopy, Fluorescence; Middle Aged; Multidrug Resistance-Associated Proteins; Propionates; Pseudoxanthoma Elasticum; Quinolines; Skin; Verapamil; Vinblastine | 2003 |
Bodipy-FL-verapamil: a fluorescent probe for the study of multidrug resistance proteins.
Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Assay; Cell Line, Tumor; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Dyes; Humans; Leukemia; Mice; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Predictive Value of Tests; Probenecid; Propionates; Quinolines; Sus scrofa; Up-Regulation; Verapamil; Vinblastine | 2004 |
Substrates and inhibitors of efflux proteins interfere with the MTT assay in cells and may lead to underestimation of drug toxicity.
Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Cattle; Cell Line; Cell Survival; Drug Screening Assays, Antitumor; Humans; L-Lactate Dehydrogenase; Multidrug Resistance-Associated Proteins; Oxidation-Reduction; Propionates; Quinolines; Tetrahydroisoquinolines; Tetrazolium Salts; Thiazoles; Verapamil | 2004 |
Relation between the ability of some compounds to modulate the MRP1-mediated efflux of glutathione and to inhibit the MRPl-mediated efflux of daunorubicin.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclic P-Oxides; Daunorubicin; Glutathione; Humans; Nicotinic Acids; Propionates; Quinolines; Tumor Cells, Cultured; Verapamil | 2004 |
Effects of grapefruit juice and orange juice components on P-glycoprotein- and MRP2-mediated drug efflux.
Topics: Algorithms; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Beverages; Biological Transport, Active; Caco-2 Cells; Calcium Channel Blockers; Citrus; Cyclosporine; Food-Drug Interactions; HIV Protease Inhibitors; Humans; Immunosuppressive Agents; Membrane Transport Proteins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Plant Extracts; Propionates; Quinolines; Saquinavir; Transfection; Verapamil; Vinblastine | 2004 |
Transepithelial transport of rosmarinic acid in intestinal Caco-2 cell monolayers.
Topics: Caco-2 Cells; Cell Membrane Permeability; Chromatography, High Pressure Liquid; Cinnamates; Depsides; Electrochemistry; Epithelial Cells; Humans; Hydroxybenzoates; Intestinal Mucosa; Propionates; Quinolines; Rosmarinic Acid; Verapamil | 2005 |
Involvement of P-glycoprotein and MRP1 in resistance to cyclic tetrapeptide subfamily of histone deacetylase inhibitors in the drug-resistant osteosarcoma and Ewing's sarcoma cells.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Neoplasms; Calcium Channel Blockers; Depsipeptides; Drug Resistance, Neoplasm; Histone Deacetylase Inhibitors; Humans; Leukotriene Antagonists; Multidrug Resistance-Associated Proteins; Osteosarcoma; Peptides, Cyclic; Propionates; Quinolines; Sarcoma, Ewing; Tumor Cells, Cultured; Verapamil | 2006 |
Transepithelial transport of fluorescent p-glycoprotein and MRP2 substrates by insect Malpighian tubules: confocal microscopic analysis of secreted fluid droplets.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drosophila melanogaster; Epithelium; Fluorescent Dyes; Gryllidae; Malpighian Tubules; Microscopy, Confocal; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinacrine; Quinolines; Tetraethylammonium; Verapamil | 2005 |
Non-destructive micromethod for MRP1 functional assay in human lung tumor cells.
Topics: Acetylcysteine; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Buthionine Sulfoximine; Cell Culture Techniques; Cell Line, Tumor; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Fluorometry; Glutathione; Humans; Immunohistochemistry; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Sensitivity and Specificity; Verapamil | 2006 |
Apparent active transport of MDMA is not mediated by P-glycoprotein: a comparison with MDCK and Caco-2 monolayers.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line; Dogs; Humans; Indomethacin; N-Methyl-3,4-methylenedioxyamphetamine; Probenecid; Progesterone; Propionates; Quinolines; Rhodamine 123; Ritonavir; Verapamil | 2006 |
The sea urchin embryo as a model for studying efflux transporters: roles and energy cost.
Topics: Animals; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Cyclosporins; Cytotoxins; Embryo, Nonmammalian; Energy Metabolism; Etoposide; Fluoresceins; Membrane Transport Proteins; Models, Animal; Propionates; Quinolines; Sea Urchins; Verapamil; Vinblastine | 2006 |
The complexity of intestinal absorption and exsorption of digoxin in rats.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Digoxin; Ileum; In Vitro Techniques; Intestinal Absorption; Jejunum; Male; Microvilli; Organic Anion Transporters; Propionates; Quinidine; Quinolines; Rats; Rats, Sprague-Dawley; Sulfobromophthalein; Tetrahydroisoquinolines; Verapamil | 2006 |
The efflux of flavonoids morin, isorhamnetin-3-O-rutinoside and diosmetin-7-O-beta-D-xylopyranosyl-(1-6) -beta-D-glucopyranoside in the human intestinal cell line caco-2.
Topics: Adenosine Triphosphate; Antioxidants; Biological Transport, Active; Caco-2 Cells; Chromatography, High Pressure Liquid; Disaccharides; Enzyme Inhibitors; Flavonoids; Humans; Intestinal Mucosa; Iodoacetamide; Probenecid; Propionates; Quercetin; Quinolines; Verapamil | 2006 |
Intestinal permeability of antivirus constituents from the fruits of Eucalyptus globulus Labill. in Caco-2 Cell Model.
Topics: Alkylating Agents; Antiviral Agents; Biological Availability; Caco-2 Cells; Calcium Channel Blockers; Cell Membrane; Chemical Phenomena; Chemistry, Physical; Chromatography, High Pressure Liquid; Eucalyptus; Fruit; Humans; Intestinal Absorption; Iodoacetamide; Phloroglucinol; Propionates; Quinolines; Sesquiterpenes; Verapamil | 2007 |
Role of P-glycoprotein in the intestinal absorption of tanshinone IIA, a major active ingredient in the root of Salvia miltiorrhiza Bunge.
Topics: Abietanes; Adenosine Triphosphate; Administration, Oral; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Availability; Caco-2 Cells; Digoxin; Dogs; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Microsomes, Liver; Multidrug Resistance-Associated Proteins; Phenanthrenes; Plant Roots; Probenecid; Propionates; Quinidine; Quinolines; Rats; Rats, Sprague-Dawley; Salvia miltiorrhiza; Temperature; Transfection; Verapamil | 2007 |
Mechanistic study on the intestinal absorption and disposition of baicalein.
Topics: Animals; ATP-Binding Cassette Transporters; Biological Transport, Active; Caco-2 Cells; Egtazic Acid; Enzyme Inhibitors; Estradiol; Flavanones; Glucuronides; Humans; Intestinal Absorption; Kinetics; Leukotriene C4; Multidrug Resistance-Associated Proteins; Permeability; Probenecid; Propionates; Quinolines; Spectrophotometry, Ultraviolet; Spodoptera; Sulfuric Acid Esters; Tandem Mass Spectrometry; Verapamil | 2007 |
Permeation of Boswellia extract in the Caco-2 model and possible interactions of its constituents KBA and AKBA with OATP1B3 and MRP2.
Topics: Aniline Compounds; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Boswellia; Caco-2 Cells; Cell Line; Dogs; Electric Impedance; Fluoresceins; Fluorescent Dyes; Humans; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Organic Anion Transporters, Sodium-Independent; Permeability; Plant Extracts; Propionates; Quinolines; Solubility; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfobromophthalein; Tight Junctions; Transfection; Triterpenes; Verapamil; Xanthenes | 2009 |
P-gp inhibition potential in cell-based models: which "calculation" method is the most accurate?
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line, Tumor; Cell Membrane Permeability; Digoxin; Drug Evaluation, Preclinical; HIV Protease Inhibitors; Humans; Indinavir; Kinetics; Propionates; Quinolines; Saquinavir; Verapamil | 2008 |
Culture period-dependent change of function and expression of ATP-binding cassette transporters in Caco-2 cells.
Topics: Angiotensin II Type 1 Receptor Blockers; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Blotting, Western; Caco-2 Cells; Calcium Channel Blockers; Digoxin; Electric Conductivity; Estrone; Humans; Imidazoles; Leukotriene Antagonists; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Ochratoxins; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazoles; Tight Junctions; Time Factors; Verapamil | 2009 |
Characterization of the multixenobiotic resistance (MXR) mechanism in embryos and larvae of the zebra mussel (Dreissena polymorpha) and studies on its role in tolerance to single and mixture combinations of toxicants.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclosporine; Dreissena; Drug Resistance, Multiple; Drug Tolerance; Embryo, Nonmammalian; Indans; Larva; Oligopeptides; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Rhodamines; Risk Assessment; Verapamil; Xenobiotics | 2011 |
Preclinical pharmacokinetics of PDE-310, a novel PDE4 inhibitor.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Availability; Biological Transport; Caco-2 Cells; Cyclic Nucleotide Phosphodiesterases, Type 4; Humans; Male; Microsomes, Liver; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Permeability; Phosphodiesterase 4 Inhibitors; Propionates; Protein Binding; Pyrimidines; Quinolines; Rats; Rats, Sprague-Dawley; Species Specificity; Verapamil | 2011 |
Intestinal absorption mechanisms of berberine, palmatine, jateorhizine, and coptisine: involvement of P-glycoprotein.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Berberine; Berberine Alkaloids; Biological Transport; Caco-2 Cells; Cyclosporine; Drugs, Chinese Herbal; Humans; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Verapamil | 2011 |
Functional evidence of multidrug resistance transporters (MDR) in rodent olfactory epithelium.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Sub-Family B Member 4; Biological Transport; Cyclosporine; Female; Fluoresceins; Gene Expression; Male; Mice; Mice, Inbred BALB C; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Olfactory Mucosa; Olfactory Receptor Neurons; Probenecid; Propionates; Quinolines; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Verapamil | 2012 |
Absorption mechanism of ginsenoside compound K and its butyl and octyl ester prodrugs in Caco-2 cells.
Topics: Absorption; Acylation; Biological Availability; Biological Transport; Caco-2 Cells; Cell Membrane Permeability; Ginsenosides; Humans; Intestinal Absorption; Panax; Prodrugs; Propionates; Quinolines; Structure-Activity Relationship; Verapamil | 2012 |
Involvement of ABCB1 and ABCC1 transporters in sea urchin Echinometra lucunter fertilization.
Topics: Acrosome; Acrosome Reaction; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Fertilization; Fluoresceins; Leukotriene Antagonists; Male; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Oligopeptides; Organic Anion Transporters; Propionates; Quinolines; Sea Urchins; Spermatozoa; Verapamil | 2012 |
The role of efflux transporters on the transport of highly toxic aconitine, mesaconitine, hypaconitine, and their hydrolysates, as determined in cultured Caco-2 and transfected MDCKII cells.
Topics: Aconitine; Adenosine; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Caco-2 Cells; Cyclosporine; Diketopiperazines; Dogs; Heterocyclic Compounds, 4 or More Rings; Humans; Intestinal Absorption; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Propionates; Quinolines; Transfection; Verapamil | 2013 |
Evaluation of intestinal absorption of amtolmetin guacyl in rats: breast cancer resistant protein as a primary barrier of oral bioavailability.
Topics: Adenosine; Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Availability; Diketopiperazines; Glycine; Heterocyclic Compounds, 4 or More Rings; Intestinal Absorption; Intestinal Mucosa; Leukotriene Antagonists; Male; Mice; Mice, Knockout; Propionates; Pyrroles; Quinolines; Rats; Rats, Sprague-Dawley; Tolmetin; Vasodilator Agents; Verapamil | 2013 |
Transcellular transport of aconitine across human intestinal Caco-2 cells.
Topics: Aconitine; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cyclosporine; Dose-Response Relationship, Drug; Glucose; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Sodium; Temperature; Transcytosis; Verapamil | 2013 |
Quantitative fluorescence microscopy provides high resolution imaging of passive diffusion and P-gp mediated efflux at the in vivo blood-brain barrier.
Topics: Algorithms; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Autoradiography; Blood-Brain Barrier; Calcium Channel Blockers; Cells, Cultured; Data Interpretation, Statistical; Fluorescent Dyes; Green Fluorescent Proteins; Image Processing, Computer-Assisted; Kinetics; Linear Models; Male; Microscopy, Fluorescence; Perfusion; Propionates; Quinolines; Rats; Rats, Inbred F344; Reference Standards; Rhodamine 123; Verapamil; Xanthenes | 2013 |
Efficiency of transcellular transport and efflux of flavonoids with different glycosidic units from flavonoids of Litsea coreana L. in a MDCK epithelial cell monolayer model.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Dogs; Flavonoids; Glycosides; Hydrogen-Ion Concentration; Litsea; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Sodium-Glucose Transporter 1; Temperature; Verapamil | 2014 |
Study on the mechanism of intestinal absorption of epimedins a, B and C in the Caco-2 cell model.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Membrane Permeability; Cell Survival; Dipyridamole; Flavonoids; Humans; Intestinal Absorption; Propionates; Quinolines; Verapamil | 2014 |
Multixenobiotic resistance efflux activity in Daphnia magna and Lumbriculus variegatus.
Topics: Animals; Arthropod Proteins; ATP-Binding Cassette Transporters; Daphnia; Environmental Monitoring; Environmental Pollutants; Oligochaeta; Oligopeptides; Propionates; Quinolines; Real-Time Polymerase Chain Reaction; Verapamil | 2015 |
Efflux and uptake transporters involved in the disposition of bazedoxifene.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; Biological Transport, Active; Caco-2 Cells; Cell Line; Cell Line, Tumor; CHO Cells; Cricetulus; Diketopiperazines; Heterocyclic Compounds, 4 or More Rings; Humans; Indoles; Liver-Specific Organic Anion Transporter 1; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Organic Anion Transporters, Sodium-Independent; Permeability; Propionates; Quinolines; Verapamil | 2016 |
Use of a combined effect model approach for discriminating between ABCB1- and ABCC1-type efflux activities in native bivalve gill tissue.
Topics: Animals; ATP-Binding Cassette Transporters; Base Sequence; DNA, Complementary; Dreissena; Gills; Models, Theoretical; Molecular Sequence Data; Oligopeptides; Phylogeny; Propionates; Quinolines; Sequence Analysis, DNA; Verapamil | 2016 |
Hypoxia can impair doxorubicin resistance of non-small cell lung cancer cells by inhibiting MRP1 and P-gp expression and boosting the chemosensitizing effects of MRP1 and P-gp blockers.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Carcinoma, Non-Small-Cell Lung; Cell Hypoxia; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Verapamil | 2016 |
Glycyrrhetinic Acid Accelerates the Clearance of Triptolide through P-gp In Vitro.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Chromatography, High Pressure Liquid; Diterpenes; Epoxy Compounds; Glycyrrhetinic Acid; Humans; Mass Spectrometry; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Phenanthrenes; Plants, Medicinal; Propionates; Quinolines; Tripterygium; Verapamil | 2017 |
Effect of synergists on ivermectin resistance in field populations of Rhipicephalus (Boophilus) microplus from Punjab districts, India.
Topics: Animals; Cyclosporine; India; Insecticide Resistance; Ivermectin; Larva; Propionates; Quinolines; Rhipicephalus; Verapamil | 2018 |
Different Efflux Transporter Affinity and Metabolism of
Topics: Animals; Cell Line, Tumor; Drug Monitoring; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Stability; Female; Humans; Liver; Mice, SCID; Molecular Imaging; Multidrug Resistance-Associated Proteins; Neoplasms; Organophosphorus Compounds; Organotechnetium Compounds; Propionates; Quinolines; Radiopharmaceuticals; Time Factors; Verapamil; Xenograft Model Antitumor Assays | 2018 |