verapamil and verlukast

verapamil has been researched along with verlukast in 45 studies

Research

Studies (45)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's24 (53.33)29.6817
2010's21 (46.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Berardi, F; Carotti, A; Cellamare, S; Colabufo, NA; Leonetti, F; Nicolotti, O; Niso, M; Pellicani, RZ; Perrone, R; Stefanachi, A1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cory, AH; Cory, JG1
Bates, SE; Dietel, M; Hohenberger, P; Jordan, A; Lage, H; Litman, T; Stein, U; Walther, W1
Taylor, EM; Yan, R1
Buesen, R; Jacob, J; Lampen, A; Mock, M; Nau, H; Seidel, A1
Bacchelli, B; Boraldi, F; Croce, MA; Garcia Fernandez, MI; Gheduzzi, D; Pasquali Ronchetti, I; Quaglino, D; Tiozzo, R1
Candussio, L; Crivellato, E; Damiani, D; Decorti, G; Giraldi, T; Klugmann, FB; Michelutti, A; Rosati, A1
Honkakoski, P; Urtti, A; Vellonen, KS1
Garnier-Suillerot, A; Loechariyakul, P; Saengkhae, C; Salerno, M1
Honda, Y; Koyabu, N; Kuwano, M; Morimoto, S; Ohtani, H; Sawada, Y; Shoyama, Y; Uchiumi, T; Ushigome, F1
Kobayashi, S; Konishi, Y1
Hanada, M; Iwamoto, Y; Li, X; Matsunobu, T; Nakamura, T; Nakatani, F; Oda, Y; Okada, T; Sakimura, R; Tanaka, K; Tsuneyoshi, M1
Leader, JP; O'Donnell, MJ1
Foth, H; Glahn, F; Stehfest, E; Torky, A1
Bertelsen, KM; Greenblatt, DJ; von Moltke, LL1
Cole, B; Epel, D; Hamdoun, A; Thurber, RV1
Chiou, WL; Yao, HM1
Tian, X; Wang, K; Yang, X1
Guo, QM; Tian, L; Tian, XJ; Wang, Y; Xu, W; Yang, XW1
Chen, X; Chowbay, B; Duan, W; Li, CG; Liang, J; Lin, SG; Liu, PQ; Wen, JY; Yu, XY; Zhou, SF; Zhou, ZW1
Jani, M; Kovács, B; Krajcsi, P; Lin, G; Zhang, L; Zuo, Z1
Abdel-Tawab, M; Fricker, G; Hummel, J; Kanzer, J; Krüger, P; Schubert-Zsilavecz, M1
Balimane, PV; Chong, S; Marino, A1
Kamiyama, E; Miura, S; Nakai, D; Okazaki, O; Sugiyama, D1
Barata, C; Faria, M; Luckenbach, T; Navarro, A; Piña, B1
Ahn, SH; Bae, MA; Cheon, HG; Jeon, DJ; Kim, MS; Kwon, KI; Lee, BH; Park, JS; Rho, HJ; Seo, JW; Song, JS1
Gao, C; Jiang, J; Qiu, F; Tan, Y; Zhang, X1
Jakob, I; Molinas, A; Sicard, G1
Deng, ZY; Hu, JN; Li, HY; Li, W; Liu, XR; Luo, T; Ye, H; Zhang, B; Zheng, YN; Zhu, XM1
de Araújo Leite, JC; Marques-Santos, LF; Santi-Gadelha, T; Silva-Neta, HL; Torrezan, E1
Gao, S; Hu, M; Liu, W; Liu, Z; Wang, F; Yang, X; Yang, Z; Ye, L; Yin, T1
Li, X; Liu, D; Rong, Z; Xiang, D; Xu, Y; Zhang, C1
Li, Z; Liu, F; Ruan, J; Yang, C; Zhang, T; Zhang, Z1
Adkins, CE; Bohn, KA; Lockman, PR; Manda, VK; Mittapalli, RK1
Chen, Z; Han, J; Hu, T; Huang, C; Li, J; Ma, T; Zhang, L; Zhong, J1
Chen, Y; Gao, X; Liu, C; Qu, D; Wang, Y; Zhou, J1
Kukkonen, JV; Vehniäinen, ER1
Berginc, K; Kristl, A; Lušin, TT; Mrhar, A; Stieger, B; Trontelj, J1
Altenburger, R; Barata, C; Burkhardt-Medicke, K; Faria, M; Luckenbach, T; Pavlichenko, V; Soares, AM1
Chen, KC; Chen, YL; Hsu, SL; Hsueh, CM; Wu, CL; Yang, TY1
Cao, L; Fang, P; Guo, Z; Hou, Z; Li, Z; Yan, M; Zhang, B1
Khangembam, R; Rath, SS; Singh, H; Singh, NK1
Fukuchi, K; Kawai, K; Kobayashi, M; Mizutani, A; Nakanishi, T; Nishi, K; Nishii, R; Okui, Y; Tamai, I; Tsujiuchi, T1

Other Studies

45 other study(ies) available for verapamil and verlukast

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Potent galloyl-based selective modulators targeting multidrug resistance associated protein 1 and P-glycoprotein.
    Journal of medicinal chemistry, 2012, Jan-12, Volume: 55, Issue:1

    Topics: Anilides; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Cell Line; Dogs; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Stability; Ethers; Gallic Acid; Pyrogallol; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship

2012
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Comparison of the properties of human breast cancer cells: MCF-7 and MCF-7 cells selected for resistance to etoposide.
    Advances in enzyme regulation, 2001, Volume: 41

    Topics: Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Chromatography, High Pressure Liquid; Dactinomycin; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Neoplasm; Etoposide; Flow Cytometry; Humans; Leukotriene Antagonists; Propionates; Protein Synthesis Inhibitors; Quinolines; Tumor Cells, Cultured; Vasodilator Agents; Verapamil; Vinblastine

2001
Impact of BCRP/MXR, MRP1 and MDR1/P-Glycoprotein on thermoresistant variants of atypical and classical multidrug resistant cancer cells.
    International journal of cancer, 2002, Feb-20, Volume: 97, Issue:6

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Calcium Channel Blockers; DNA Primers; DNA-Binding Proteins; Doxorubicin; Drug Resistance, Multiple; Fluorescent Dyes; Gastrointestinal Neoplasms; Gene Expression Regulation; Genes, MDR; Hot Temperature; Humans; Indenes; Mitoxantrone; Multidrug Resistance-Associated Proteins; MutS Homolog 3 Protein; Mycotoxins; Neoplasm Proteins; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; RNA, Neoplasm; Stomach Neoplasms; Verapamil

2002
Neotrofin is transported out of brain by a saturable mechanism: possible involvement of multidrug resistance and monocarboxylic acid transporters.
    Drug metabolism and disposition: the biological fate of chemicals, 2002, Volume: 30, Issue:5

    Topics: Aminobenzoates; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Brain; Capillaries; Drug Resistance, Multiple; Endothelium, Vascular; Hypoxanthines; Injections, Intraventricular; Male; Mice; Monocarboxylic Acid Transporters; Nootropic Agents; Organic Anion Transporters; Probenecid; Propionates; Purines; Quinolines; Verapamil

2002
Human intestinal Caco-2 cells display active transport of benzo[a]pyrene metabolites.
    Chemico-biological interactions, 2003, Jan-06, Volume: 142, Issue:3

    Topics: Adenosine Triphosphate; Aryl Hydrocarbon Hydroxylases; ATP-Binding Cassette Transporters; Benzo(a)pyrene; Benzoflavones; Biological Transport, Active; Caco-2 Cells; Cell Polarity; Cyclosporine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1B1; Enterocytes; Gene Expression; Humans; Models, Biological; Probenecid; Propionates; Quinolines; Verapamil; Vinblastine

2003
Multidrug resistance protein-6 (MRP6) in human dermal fibroblasts. Comparison between cells from normal subjects and from Pseudoxanthoma elasticum patients.
    Matrix biology : journal of the International Society for Matrix Biology, 2003, Volume: 22, Issue:6

    Topics: Adult; Benzbromarone; Cell Count; Cell Division; Chlorambucil; Female; Fibroblasts; Fluoresceins; Fluorescent Dyes; Humans; Indomethacin; Lysosomes; Male; Membrane Transport Proteins; Microscopy, Fluorescence; Middle Aged; Multidrug Resistance-Associated Proteins; Propionates; Pseudoxanthoma Elasticum; Quinolines; Skin; Verapamil; Vinblastine

2003
Bodipy-FL-verapamil: a fluorescent probe for the study of multidrug resistance proteins.
    Cellular oncology : the official journal of the International Society for Cellular Oncology, 2004, Volume: 26, Issue:1-2

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Assay; Cell Line, Tumor; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Dyes; Humans; Leukemia; Mice; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Predictive Value of Tests; Probenecid; Propionates; Quinolines; Sus scrofa; Up-Regulation; Verapamil; Vinblastine

2004
Substrates and inhibitors of efflux proteins interfere with the MTT assay in cells and may lead to underestimation of drug toxicity.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2004, Volume: 23, Issue:2

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Cattle; Cell Line; Cell Survival; Drug Screening Assays, Antitumor; Humans; L-Lactate Dehydrogenase; Multidrug Resistance-Associated Proteins; Oxidation-Reduction; Propionates; Quinolines; Tetrahydroisoquinolines; Tetrazolium Salts; Thiazoles; Verapamil

2004
Relation between the ability of some compounds to modulate the MRP1-mediated efflux of glutathione and to inhibit the MRPl-mediated efflux of daunorubicin.
    Biochemical pharmacology, 2004, Dec-01, Volume: 68, Issue:11

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclic P-Oxides; Daunorubicin; Glutathione; Humans; Nicotinic Acids; Propionates; Quinolines; Tumor Cells, Cultured; Verapamil

2004
Effects of grapefruit juice and orange juice components on P-glycoprotein- and MRP2-mediated drug efflux.
    British journal of pharmacology, 2004, Volume: 143, Issue:7

    Topics: Algorithms; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Beverages; Biological Transport, Active; Caco-2 Cells; Calcium Channel Blockers; Citrus; Cyclosporine; Food-Drug Interactions; HIV Protease Inhibitors; Humans; Immunosuppressive Agents; Membrane Transport Proteins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Plant Extracts; Propionates; Quinolines; Saquinavir; Transfection; Verapamil; Vinblastine

2004
Transepithelial transport of rosmarinic acid in intestinal Caco-2 cell monolayers.
    Bioscience, biotechnology, and biochemistry, 2005, Volume: 69, Issue:3

    Topics: Caco-2 Cells; Cell Membrane Permeability; Chromatography, High Pressure Liquid; Cinnamates; Depsides; Electrochemistry; Epithelial Cells; Humans; Hydroxybenzoates; Intestinal Mucosa; Propionates; Quinolines; Rosmarinic Acid; Verapamil

2005
Involvement of P-glycoprotein and MRP1 in resistance to cyclic tetrapeptide subfamily of histone deacetylase inhibitors in the drug-resistant osteosarcoma and Ewing's sarcoma cells.
    International journal of cancer, 2006, Jan-01, Volume: 118, Issue:1

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Neoplasms; Calcium Channel Blockers; Depsipeptides; Drug Resistance, Neoplasm; Histone Deacetylase Inhibitors; Humans; Leukotriene Antagonists; Multidrug Resistance-Associated Proteins; Osteosarcoma; Peptides, Cyclic; Propionates; Quinolines; Sarcoma, Ewing; Tumor Cells, Cultured; Verapamil

2006
Transepithelial transport of fluorescent p-glycoprotein and MRP2 substrates by insect Malpighian tubules: confocal microscopic analysis of secreted fluid droplets.
    The Journal of experimental biology, 2005, Volume: 208, Issue:Pt 23

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drosophila melanogaster; Epithelium; Fluorescent Dyes; Gryllidae; Malpighian Tubules; Microscopy, Confocal; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinacrine; Quinolines; Tetraethylammonium; Verapamil

2005
Non-destructive micromethod for MRP1 functional assay in human lung tumor cells.
    Archives of toxicology, 2006, Volume: 80, Issue:3

    Topics: Acetylcysteine; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Buthionine Sulfoximine; Cell Culture Techniques; Cell Line, Tumor; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Fluorometry; Glutathione; Humans; Immunohistochemistry; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Sensitivity and Specificity; Verapamil

2006
Apparent active transport of MDMA is not mediated by P-glycoprotein: a comparison with MDCK and Caco-2 monolayers.
    Biopharmaceutics & drug disposition, 2006, Volume: 27, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line; Dogs; Humans; Indomethacin; N-Methyl-3,4-methylenedioxyamphetamine; Probenecid; Progesterone; Propionates; Quinolines; Rhodamine 123; Ritonavir; Verapamil

2006
The sea urchin embryo as a model for studying efflux transporters: roles and energy cost.
    Marine environmental research, 2006, Volume: 62 Suppl

    Topics: Animals; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Cyclosporins; Cytotoxins; Embryo, Nonmammalian; Energy Metabolism; Etoposide; Fluoresceins; Membrane Transport Proteins; Models, Animal; Propionates; Quinolines; Sea Urchins; Verapamil; Vinblastine

2006
The complexity of intestinal absorption and exsorption of digoxin in rats.
    International journal of pharmaceutics, 2006, Sep-28, Volume: 322, Issue:1-2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Digoxin; Ileum; In Vitro Techniques; Intestinal Absorption; Jejunum; Male; Microvilli; Organic Anion Transporters; Propionates; Quinidine; Quinolines; Rats; Rats, Sprague-Dawley; Sulfobromophthalein; Tetrahydroisoquinolines; Verapamil

2006
The efflux of flavonoids morin, isorhamnetin-3-O-rutinoside and diosmetin-7-O-beta-D-xylopyranosyl-(1-6) -beta-D-glucopyranoside in the human intestinal cell line caco-2.
    Pharmaceutical research, 2006, Volume: 23, Issue:8

    Topics: Adenosine Triphosphate; Antioxidants; Biological Transport, Active; Caco-2 Cells; Chromatography, High Pressure Liquid; Disaccharides; Enzyme Inhibitors; Flavonoids; Humans; Intestinal Mucosa; Iodoacetamide; Probenecid; Propionates; Quercetin; Quinolines; Verapamil

2006
Intestinal permeability of antivirus constituents from the fruits of Eucalyptus globulus Labill. in Caco-2 Cell Model.
    Bioorganic & medicinal chemistry letters, 2007, Feb-15, Volume: 17, Issue:4

    Topics: Alkylating Agents; Antiviral Agents; Biological Availability; Caco-2 Cells; Calcium Channel Blockers; Cell Membrane; Chemical Phenomena; Chemistry, Physical; Chromatography, High Pressure Liquid; Eucalyptus; Fruit; Humans; Intestinal Absorption; Iodoacetamide; Phloroglucinol; Propionates; Quinolines; Sesquiterpenes; Verapamil

2007
Role of P-glycoprotein in the intestinal absorption of tanshinone IIA, a major active ingredient in the root of Salvia miltiorrhiza Bunge.
    Current drug metabolism, 2007, Volume: 8, Issue:4

    Topics: Abietanes; Adenosine Triphosphate; Administration, Oral; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Availability; Caco-2 Cells; Digoxin; Dogs; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Microsomes, Liver; Multidrug Resistance-Associated Proteins; Phenanthrenes; Plant Roots; Probenecid; Propionates; Quinidine; Quinolines; Rats; Rats, Sprague-Dawley; Salvia miltiorrhiza; Temperature; Transfection; Verapamil

2007
Mechanistic study on the intestinal absorption and disposition of baicalein.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2007, Volume: 31, Issue:3-4

    Topics: Animals; ATP-Binding Cassette Transporters; Biological Transport, Active; Caco-2 Cells; Egtazic Acid; Enzyme Inhibitors; Estradiol; Flavanones; Glucuronides; Humans; Intestinal Absorption; Kinetics; Leukotriene C4; Multidrug Resistance-Associated Proteins; Permeability; Probenecid; Propionates; Quinolines; Spectrophotometry, Ultraviolet; Spodoptera; Sulfuric Acid Esters; Tandem Mass Spectrometry; Verapamil

2007
Permeation of Boswellia extract in the Caco-2 model and possible interactions of its constituents KBA and AKBA with OATP1B3 and MRP2.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2009, Feb-15, Volume: 36, Issue:2-3

    Topics: Aniline Compounds; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Boswellia; Caco-2 Cells; Cell Line; Dogs; Electric Impedance; Fluoresceins; Fluorescent Dyes; Humans; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Organic Anion Transporters, Sodium-Independent; Permeability; Plant Extracts; Propionates; Quinolines; Solubility; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfobromophthalein; Tight Junctions; Transfection; Triterpenes; Verapamil; Xanthenes

2009
P-gp inhibition potential in cell-based models: which "calculation" method is the most accurate?
    The AAPS journal, 2008, Volume: 10, Issue:4

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line, Tumor; Cell Membrane Permeability; Digoxin; Drug Evaluation, Preclinical; HIV Protease Inhibitors; Humans; Indinavir; Kinetics; Propionates; Quinolines; Saquinavir; Verapamil

2008
Culture period-dependent change of function and expression of ATP-binding cassette transporters in Caco-2 cells.
    Drug metabolism and disposition: the biological fate of chemicals, 2009, Volume: 37, Issue:9

    Topics: Angiotensin II Type 1 Receptor Blockers; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Blotting, Western; Caco-2 Cells; Calcium Channel Blockers; Digoxin; Electric Conductivity; Estrone; Humans; Imidazoles; Leukotriene Antagonists; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Ochratoxins; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazoles; Tight Junctions; Time Factors; Verapamil

2009
Characterization of the multixenobiotic resistance (MXR) mechanism in embryos and larvae of the zebra mussel (Dreissena polymorpha) and studies on its role in tolerance to single and mixture combinations of toxicants.
    Aquatic toxicology (Amsterdam, Netherlands), 2011, Jan-17, Volume: 101, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclosporine; Dreissena; Drug Resistance, Multiple; Drug Tolerance; Embryo, Nonmammalian; Indans; Larva; Oligopeptides; Propionates; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Rhodamines; Risk Assessment; Verapamil; Xenobiotics

2011
Preclinical pharmacokinetics of PDE-310, a novel PDE4 inhibitor.
    Drug metabolism and pharmacokinetics, 2011, Volume: 26, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Availability; Biological Transport; Caco-2 Cells; Cyclic Nucleotide Phosphodiesterases, Type 4; Humans; Male; Microsomes, Liver; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Permeability; Phosphodiesterase 4 Inhibitors; Propionates; Protein Binding; Pyrimidines; Quinolines; Rats; Rats, Sprague-Dawley; Species Specificity; Verapamil

2011
Intestinal absorption mechanisms of berberine, palmatine, jateorhizine, and coptisine: involvement of P-glycoprotein.
    Xenobiotica; the fate of foreign compounds in biological systems, 2011, Volume: 41, Issue:4

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Berberine; Berberine Alkaloids; Biological Transport; Caco-2 Cells; Cyclosporine; Drugs, Chinese Herbal; Humans; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Verapamil

2011
Functional evidence of multidrug resistance transporters (MDR) in rodent olfactory epithelium.
    PloS one, 2012, Volume: 7, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Sub-Family B Member 4; Biological Transport; Cyclosporine; Female; Fluoresceins; Gene Expression; Male; Mice; Mice, Inbred BALB C; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Olfactory Mucosa; Olfactory Receptor Neurons; Probenecid; Propionates; Quinolines; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Verapamil

2012
Absorption mechanism of ginsenoside compound K and its butyl and octyl ester prodrugs in Caco-2 cells.
    Journal of agricultural and food chemistry, 2012, Oct-17, Volume: 60, Issue:41

    Topics: Absorption; Acylation; Biological Availability; Biological Transport; Caco-2 Cells; Cell Membrane Permeability; Ginsenosides; Humans; Intestinal Absorption; Panax; Prodrugs; Propionates; Quinolines; Structure-Activity Relationship; Verapamil

2012
Involvement of ABCB1 and ABCC1 transporters in sea urchin Echinometra lucunter fertilization.
    Molecular reproduction and development, 2012, Volume: 79, Issue:12

    Topics: Acrosome; Acrosome Reaction; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Fertilization; Fluoresceins; Leukotriene Antagonists; Male; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Oligopeptides; Organic Anion Transporters; Propionates; Quinolines; Sea Urchins; Spermatozoa; Verapamil

2012
The role of efflux transporters on the transport of highly toxic aconitine, mesaconitine, hypaconitine, and their hydrolysates, as determined in cultured Caco-2 and transfected MDCKII cells.
    Toxicology letters, 2013, Feb-04, Volume: 216, Issue:2-3

    Topics: Aconitine; Adenosine; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Caco-2 Cells; Cyclosporine; Diketopiperazines; Dogs; Heterocyclic Compounds, 4 or More Rings; Humans; Intestinal Absorption; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Propionates; Quinolines; Transfection; Verapamil

2013
Evaluation of intestinal absorption of amtolmetin guacyl in rats: breast cancer resistant protein as a primary barrier of oral bioavailability.
    Life sciences, 2013, Feb-27, Volume: 92, Issue:3

    Topics: Adenosine; Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Availability; Diketopiperazines; Glycine; Heterocyclic Compounds, 4 or More Rings; Intestinal Absorption; Intestinal Mucosa; Leukotriene Antagonists; Male; Mice; Mice, Knockout; Propionates; Pyrroles; Quinolines; Rats; Rats, Sprague-Dawley; Tolmetin; Vasodilator Agents; Verapamil

2013
Transcellular transport of aconitine across human intestinal Caco-2 cells.
    Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association, 2013, Volume: 57

    Topics: Aconitine; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cyclosporine; Dose-Response Relationship, Drug; Glucose; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Sodium; Temperature; Transcytosis; Verapamil

2013
Quantitative fluorescence microscopy provides high resolution imaging of passive diffusion and P-gp mediated efflux at the in vivo blood-brain barrier.
    Journal of neuroscience methods, 2013, Sep-30, Volume: 219, Issue:1

    Topics: Algorithms; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Autoradiography; Blood-Brain Barrier; Calcium Channel Blockers; Cells, Cultured; Data Interpretation, Statistical; Fluorescent Dyes; Green Fluorescent Proteins; Image Processing, Computer-Assisted; Kinetics; Linear Models; Male; Microscopy, Fluorescence; Perfusion; Propionates; Quinolines; Rats; Rats, Inbred F344; Reference Standards; Rhodamine 123; Verapamil; Xanthenes

2013
Efficiency of transcellular transport and efflux of flavonoids with different glycosidic units from flavonoids of Litsea coreana L. in a MDCK epithelial cell monolayer model.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2014, Mar-12, Volume: 53

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Dogs; Flavonoids; Glycosides; Hydrogen-Ion Concentration; Litsea; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinolines; Sodium-Glucose Transporter 1; Temperature; Verapamil

2014
Study on the mechanism of intestinal absorption of epimedins a, B and C in the Caco-2 cell model.
    Molecules (Basel, Switzerland), 2014, Jan-07, Volume: 19, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Membrane Permeability; Cell Survival; Dipyridamole; Flavonoids; Humans; Intestinal Absorption; Propionates; Quinolines; Verapamil

2014
Multixenobiotic resistance efflux activity in Daphnia magna and Lumbriculus variegatus.
    Chemosphere, 2015, Volume: 124

    Topics: Animals; Arthropod Proteins; ATP-Binding Cassette Transporters; Daphnia; Environmental Monitoring; Environmental Pollutants; Oligochaeta; Oligopeptides; Propionates; Quinolines; Real-Time Polymerase Chain Reaction; Verapamil

2015
Efflux and uptake transporters involved in the disposition of bazedoxifene.
    European journal of drug metabolism and pharmacokinetics, 2016, Volume: 41, Issue:3

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; Biological Transport, Active; Caco-2 Cells; Cell Line; Cell Line, Tumor; CHO Cells; Cricetulus; Diketopiperazines; Heterocyclic Compounds, 4 or More Rings; Humans; Indoles; Liver-Specific Organic Anion Transporter 1; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Organic Anion Transporters, Sodium-Independent; Permeability; Propionates; Quinolines; Verapamil

2016
Use of a combined effect model approach for discriminating between ABCB1- and ABCC1-type efflux activities in native bivalve gill tissue.
    Toxicology and applied pharmacology, 2016, Apr-15, Volume: 297

    Topics: Animals; ATP-Binding Cassette Transporters; Base Sequence; DNA, Complementary; Dreissena; Gills; Models, Theoretical; Molecular Sequence Data; Oligopeptides; Phylogeny; Propionates; Quinolines; Sequence Analysis, DNA; Verapamil

2016
Hypoxia can impair doxorubicin resistance of non-small cell lung cancer cells by inhibiting MRP1 and P-gp expression and boosting the chemosensitizing effects of MRP1 and P-gp blockers.
    Cellular oncology (Dordrecht), 2016, Volume: 39, Issue:5

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Carcinoma, Non-Small-Cell Lung; Cell Hypoxia; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Verapamil

2016
Glycyrrhetinic Acid Accelerates the Clearance of Triptolide through P-gp In Vitro.
    Phytotherapy research : PTR, 2017, Volume: 31, Issue:7

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Chromatography, High Pressure Liquid; Diterpenes; Epoxy Compounds; Glycyrrhetinic Acid; Humans; Mass Spectrometry; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Phenanthrenes; Plants, Medicinal; Propionates; Quinolines; Tripterygium; Verapamil

2017
Effect of synergists on ivermectin resistance in field populations of Rhipicephalus (Boophilus) microplus from Punjab districts, India.
    Ticks and tick-borne diseases, 2018, Volume: 9, Issue:3

    Topics: Animals; Cyclosporine; India; Insecticide Resistance; Ivermectin; Larva; Propionates; Quinolines; Rhipicephalus; Verapamil

2018
Different Efflux Transporter Affinity and Metabolism of
    Pharmaceutical research, 2018, Nov-29, Volume: 36, Issue:1

    Topics: Animals; Cell Line, Tumor; Drug Monitoring; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Stability; Female; Humans; Liver; Mice, SCID; Molecular Imaging; Multidrug Resistance-Associated Proteins; Neoplasms; Organophosphorus Compounds; Organotechnetium Compounds; Propionates; Quinolines; Radiopharmaceuticals; Time Factors; Verapamil; Xenograft Model Antitumor Assays

2018