verapamil has been researched along with trifluoperazine in 189 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 110 (58.20) | 18.7374 |
1990's | 55 (29.10) | 18.2507 |
2000's | 18 (9.52) | 29.6817 |
2010's | 6 (3.17) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ | 1 |
Pajeva, IK; Wiese, M | 1 |
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL | 1 |
Dobner, B; Glöde, J; Langner, A; Schmidt, M; Ungvári, J | 1 |
Abraham, MH; Acree, WE; Ibrahim, A | 1 |
Cai, W; Hao, Y; Hu, P; Ma, D; Pan, H; Xie, X; Yu, AD; Yu, J; Yuan, J; Zhang, L; Zhu, H | 1 |
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Chen, X; Lin, X; Skolnik, S; Wang, J | 1 |
Chen, M; Fang, H; Liu, Z; Shi, Q; Tong, W; Vijay, V | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Papadimituiou, JM; Sforcina, D | 1 |
García-Cosmes, P; López-Novoa, JM; Macías-Núñez, JF; Mortezo, A | 1 |
Dantchev, N; Popov, P; Staneva-Stoytcheva, D | 1 |
Goldstein, LJ; Gottesman, MM; Pastan, I | 1 |
Burchés, E; Cortijo, J; Morcillo, EJ; Orón, JD; Ortiz, JL | 1 |
Izutsu, K; Komada, H; Nakabayashi, H; Takanari, H; Yoshida, T | 1 |
Long, P; Yan, CH; Zhang, MS; Zhou, EF | 1 |
Batra, S; Hartley-Asp, B; Popper, LD | 1 |
Danchev, N; Popov, P; Staneva-Stoytcheva, D | 1 |
Gottesman, MM; Horio, M; Lovelace, E; Pastan, I | 1 |
Rice, CD; Weeks, BA | 1 |
Crevel, H; Marthan, R; Savineau, JP | 1 |
Ivanova, E; Popova, J; Staneva-Stoytcheva, D; Tosheva, T | 1 |
Besser, GM; Grossman, A; Rees, LH; Tsagarakis, S | 1 |
Cortijo, J; Foster, RW; Morcillo, EJ; Small, RC | 1 |
Khalbuss, WE; Wondergem, R | 1 |
Johnson, AL; Levorse, JM; Tilly, JL | 1 |
Krishan, A | 1 |
Goodman, HM; Schwartz, Y | 1 |
Anais, D; Arbeit, L; Frei, L; Greif, F; Sorroff, HS | 1 |
Alov, P; Mutafova-Yambolieva, V; Popova, J; Staneva-Stoytcheva, D | 1 |
Gurman, EG | 2 |
Ballard, HS; Haakenson, CM; Johnson, GJ; Moritz, TE; O'Donnell, JF; Ringenberg, QS; Schilsky, RL; Spaulding, MB; Tornyos, K; Zacharski, LR | 1 |
Hahn, EW; Osswald, H; Pommerenke, EW; Volm, M | 1 |
Mutafova, V; Popova, J; Staneva-Stoytcheva, D | 1 |
Alcalde, AI; Barcina, Y; Ilundain, A; Larralde, J | 2 |
Bick, T; Hochberg, Z; Perlman, R | 1 |
Matsumura, Y; Morimoto, S; Sasaki, Y; Shinyama, H; Uriu, T | 1 |
Gautvik, KM; Haug, E; Sletholt, K | 1 |
Bégin-Heick, N; Black, MA; Fournier, LA; Heick, HM | 1 |
Dasarathy, Y; Fanburg, BL | 1 |
Gandhi, VC; Jones, DJ | 1 |
Lee, DB; Misra, BC; Nagineni, CN; Yanagawa, N | 1 |
Blair-West, JR; Nelson, JF; Wright, RD | 1 |
Perchellet, JP; Satyamoorthy, K | 1 |
Das, DK; Jones, RM; Otani, H; Prasad, MR | 1 |
Ganguly, NK; Garg, UC; Goyal, J; Walia, BN | 1 |
Escalante, B; Reyes, JL | 1 |
Jones, HM; Rush, ME; Simpson, WG; Vernon, ME | 1 |
Berger, SG; Hofmann, A; Waser, PG | 1 |
Bos, MP; Herrmann-Erlee, MP; Van Leeuwen, JP | 1 |
Enyeart, JJ; Hinkle, PM; Phillips, WJ | 1 |
Akiyama, S; Ichikawa, M; Ikeda, S; Kuwazuru, Y; Sumizawa, T; Usagawa, T; Yoshimura, A | 1 |
Menditto, A; Silvestroni, L | 1 |
Menditto, A; Modesti, A; Scarpa, S; Silvestroni, L | 1 |
Bindslev, N; Demant, EJ; Friche, E; Jensen, PB; Sehested, M; Skovsgaard, T; Vindeløv, L | 1 |
Safa, AR; Spearman, T; Van Dyke, K; Ye, ZG | 1 |
Khauli, RB; McGraw, BR; Strzelecki, T | 1 |
Bright, EC; Colombani, PM; Hess, AD; Wells, M | 1 |
Cortijo, J; Esplugues, J; Martí-Cabrera, M; Morcillo, E; Sarriá, B | 1 |
Honn, KV; Nelson, KK; Onoda, JM; Taylor, JD | 1 |
Karpov, RS; Larionov, NP; Malyshev, IIu; Meerson, FZ | 2 |
Buffa, M; Della Torre, G; Gambetta, RA; Ingrosso, A; Soranzo, C; Zunino, F | 1 |
Jones, HM; Maley, BE; Rush, ME; Simpson, WG; Vernon, MW | 1 |
Atkinson, MJ; Cade, C; Hesch, RD; Perris, AD; Wadwah, M | 1 |
Diener, M; Knobloch, SF; Rummel, W | 1 |
Cortijo, J; Foster, RW; Small, RC | 1 |
Aguila, MC; McCann, SM | 1 |
Guo, YS; Singh, P; Thompson, JC | 1 |
Fishbaugh, J; Freeman, L; Powers, V; Van Sant, R; Yen, A | 1 |
Düsing, R; Kipnowski, J; Kramer, HJ | 1 |
Mohammad, SF; Nichols, WK; Weber, DR | 1 |
Degnan, KJ; May, SA | 1 |
Barzilai, D; Bick, T; Brandes, JM; Hochberg, Z; Perlman, R | 1 |
Braquet, P; Lauzière, M; Sirois, P | 1 |
Gagliardino, JJ; Rebolledo, OR; Semino, MC | 1 |
Danon, A; Davis, BB; Thomasson, DL; Zenser, TV | 1 |
Karaki, H; Nagase, H; Urakawa, N | 1 |
Anaise, D; Lane, B; Rapaport, FT; Waltzer, WC | 1 |
Filep, J; Rosenkranz, B | 1 |
Ganguly, NK; Garg, UC; Goyal, J; Mahajan, RC; Walia, BN | 2 |
Heidland, A; Kokot, K; Schaefer, RM; Teschner, M | 2 |
Chang, B; Fisher, SE; Karl, PI | 1 |
Dmitrevskaya, TV; Neyfakh, AA; Serpinskaya, AS | 1 |
Cortijo, J; Esplugues, J; Morcillo, EJ; Ortiz, JL; Perpiñá, M; Sanz, C | 1 |
FitzGerald, DJ; Pastan, I; Pirker, R; Willingham, MC | 1 |
Butt, KM; Hong, J; Jaffe, BM; McMillen, MA; Tesi, RJ | 1 |
Anaise, D; Asari, H; Aso, K; Ishii, K; Masaki, Y; Rapaport, FT; Sato, K; Uchida, H; Waltzer, W; Yoda, K | 1 |
Borish, L; Rocklin, R; Rosenbaum, R | 1 |
Matthijs, G; Peeters, TL; Vantrappen, G | 1 |
Monti, E; Paracchini, L; Piccinini, F; Rozza, A; Villani, F | 1 |
Altan, VM; Karasu, C; Oztürk, Y; Yildizoglu, N | 1 |
Kojo, S; Tsukamoto, I | 1 |
Ilundain, A; Larralde, J; Toval, M | 1 |
Mogami, H; Sakamoto, Y; Shimizu, K; Ushio, Y; Yoshida, T | 1 |
Fujita, T; Hirata, Y; Takata, S; Tomita, M | 1 |
Favalli, L; Formelli, F; Lanza, E; Monti, E; Piccinini, F; Poggi, P; Rozza, A; Villani, F | 1 |
Anaise, D; Lane, B; Ramsammy, L; Rapaport, FT; Waltzer, WC | 1 |
Hagiwara, K; Hamada, H; Nakajima, T; Tsuruo, T | 1 |
Cain, CA; Nguyen, HK; Tompkins, WA | 1 |
Cano-Gauci, DF; Riordan, JR | 1 |
Brostrom, CO; Brostrom, MA; Wolfe, SE | 1 |
Schrier, RW; Schwertschlag, U; Wilson, P | 1 |
Formelli, F; Mariani, M; Parmiani, G; Prosperi, E; Supino, R | 1 |
Cai, HR; Stieve, H | 1 |
Furuya, S; Kido, R; Kusuyama, Y; Masuyama, Y; Minatogawa, Y; Nishio, I; Shima, H; Tamaki, T; Tsuda, K; Ueda, E | 1 |
Baraldi, M; Benelli, A; Sandrini, M | 1 |
Gordon, K; Krishan, A; Sauerteig, A; Swinkin, C | 1 |
Izawa, T; Komabayashi, T; Nakamura, T; Nakano, K; Tsuboi, M | 1 |
Abe, K; Adachi, I; Fujiki, H; Kimura, S; Nagasaki, K; Yamaguchi, K | 1 |
Hardcastle, J; Hardcastle, PT; Noble, JM | 1 |
Bauer, C; Kurtz, A; Pfeilschifter, J | 1 |
Fitchett, D; Pountney, E; Stewart, D | 1 |
Hubel, KA | 1 |
Murakami, H; Ohmura, E; Shizume, K; Tsushima, T; Wakai, K | 1 |
Ashraf, M; Peterson, RN; Russell, LD | 1 |
Foder, B; Scharff, O | 1 |
Foder, B; Scharff, O; Skibsted, U | 2 |
Erlichman, J; Fleckman, A; Fleischer, N; Schubart, UK | 1 |
Balla, T; Hunyady, L; Spät, A | 1 |
Carnegie, JA; Tsang, BK | 1 |
Blakeman, DP; Im, WB; Mendlein, J; Sachs, G | 1 |
Peng, HB | 1 |
Benabe, JE; Cruz-Soto, MA; Martínez-Maldonado, M | 1 |
Ausiello, DA; Zusman, RM | 1 |
Hepler, PK; Saunders, MJ | 1 |
Darnold, JR; Fleschner, CR; Long, JW; Martin, AP; Vorbeck, ML | 1 |
Callanan, D; Hubel, KA | 1 |
Brady, RC; Hilfer, SR | 1 |
Bilozur, M; Powers, RD | 1 |
Chernoff, EA; Hilfer, SR | 1 |
Gold, BI | 1 |
Andersson, A; Drakenberg, T; Forsén, S; Thulin, E | 1 |
Balla, T; Enyedi, P; Spät, A | 1 |
Janjic, D; Kikuchi, M; Sharp, GW; Siegel, EG; Wollheim, CB | 1 |
Harmony, JA; Jackson, RJ; Ranganathan, S | 1 |
Iida, H; Sakurai, Y; Tsukagoshi, S; Tsuruo, T | 1 |
Born, E; Chen, H; Field, FJ; Mathur, SN; Murthy, S | 1 |
Kamboj, KK; Meera, P; Rao, PR; Tripathi, O | 1 |
Bold, RJ; Ishizuka, J; Thompson, JC; Townsend, CM | 1 |
Choe, KJ; Gottesman, MM; Hong, IG; Kim, HS; Kim, WH; Kim, YI; Lee, SK; Lim, KH; Park, JG; Tsuruo, T | 1 |
Dalton, WS; de Giuli, R; Emerson, S; Lehnert, M; Salmon, SE | 1 |
Arruebo, MP; de Pedro, MJ; Murillo, MD; Plaza, MA | 1 |
Hénichart, JP; Hornez, L; Mestdagh, N; Vandewalle, B | 1 |
Carvalho, CM; Lopes, MC; Santos, DL | 1 |
Holfels, E; Mack, D; McAuley, J; McLeod, R; Milhous, WK | 1 |
Huang, XL; Krishan, A; Ramachandran, C; Yuan, ZK | 1 |
Raderer, M; Scheithauer, W | 1 |
De Jonckheere, S; McCaig, D | 1 |
Barlow, JW; Kolliniatis, E; Scholz, GH; Stockigt, JR; Topliss, DJ | 1 |
Dassylva, B | 1 |
Enigbokan, MA; Preston, J; Thompson, JO; West, D | 1 |
Aleksanian, IuT; Davtian, TK; Gambarov, SS; Giul'khandanian, AV; Ignatova, TN; Nagapetian, KG | 1 |
Dimova, S; Koleva, M; Rangelova, D; Stoythchev, T | 1 |
Dazy, AC; Diogène, G; Marano, F; Venant, A | 1 |
Elías, MM; Ochoa, JE; Weinschelbaum-Jairala, S | 1 |
Alexanyan, YT; Avanessian, LA; Davtyan, TK; Gambarov, SS; Gyulkhandanyan, AV | 1 |
Chang, TS; Cheon, AJ; Khil, LY; Moon, CK | 1 |
Masui, H; Sakamoto, K; Wakabayashi, I; Yoshimoto, S | 1 |
Balossier, G; Bonhomme, A; Bonhomme, P; Bouchot, A; Burlet, H; Klein, C; Pezzella, N; Pingret, L; Pinon, JM | 1 |
Camoirano, A; Cartiglia, C; De Flora, S; Ferguson, L | 1 |
Bhattacharyya, D; Sen, PC | 1 |
Canchola-Martínez, E; Mercado-Sánchez, G; Rodríguez-Medina, MA; Vergara-Onofre, M | 1 |
Bernard, A; Lermioglu, F | 1 |
Biswas, S; Ghosh, R; Sen, PC | 1 |
Hafner, M; Pey, R; Schatten, G; Vial, C | 1 |
Arrington, B; Hardy, MA; Kinkhabwala, M; Polyak, MM; Stubenbord, WT | 1 |
Balint, GA | 1 |
Dimova, S; Koleva, M | 1 |
de Almeida, OM; de Mello, FG; de Mello, MC; Gardino, PF; Kubrusly, RC; Loureiro-Dos-Santos, NE; Reis, RA | 1 |
Epple, HJ; Fromm, M; Riecken, EO; Schulzke, JD | 1 |
Landwojtowicz, E; Nervi, P; Seelig, A | 1 |
Maia, RC; Marques-Santos, LF; Oliveira, JG; Rumjanek, VM | 1 |
Liang, JH; Lu, Y; Ye, XF; Zhang, P | 1 |
Ambu, R; Garau, L; Olianas, MC; Onali, P | 1 |
Gao, YD; Peng, H; Shao, XF; Xiong, DS; Xu, YF; Yang, CZ; Zhu, ZP | 1 |
Bordovsky, MJ; Easterling, WJ; Fitch, WP; Mosier, M; Talbert, RL | 1 |
Levine, L | 1 |
Devecí, E | 1 |
Lange, AB; Orchard, I; Ruiz-Sanchez, E | 1 |
3 review(s) available for verapamil and trifluoperazine
Article | Year |
---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Multidrug resistance in human cancer.
Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Drug Resistance; Feasibility Studies; Gene Expression Regulation, Neoplastic; Humans; Membrane Glycoproteins; Mice; Mice, Transgenic; Neoplasm Proteins; Neoplasms; Neoplasms, Experimental; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1992 |
Clinical trials of agents that reverse multidrug resistance. A literature review.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Clinical Trials as Topic; Cyclosporins; Drug Resistance; Humans; Phenotype; Quinidine; Tamoxifen; Trifluoperazine; Verapamil | 1993 |
2 trial(s) available for verapamil and trifluoperazine
Article | Year |
---|---|
The state of renal preservation for transplantation in New York.
Topics: Alprostadil; Calcium; Humans; Kidney; Kidney Transplantation; New York; Organ Preservation; Perfusion; Pulsatile Flow; Trifluoperazine; Verapamil | 1999 |
Topical verapamil HCl, topical trifluoperazine, and topical magnesium sulfate for the treatment of Peyronie's disease--a placebo-controlled pilot study.
Topics: Administration, Topical; Adult; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Humans; Magnesium Sulfate; Male; Middle Aged; Penile Erection; Penile Induration; Quality of Life; Research Design; Treatment Outcome; Trifluoperazine; Verapamil | 2007 |
184 other study(ies) available for verapamil and trifluoperazine
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Active transport of fluorescent P-glycoprotein substrates: evaluation as markers and interaction with inhibitors.
Topics: 3T3 Cells; Adrenergic Uptake Inhibitors; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Biological Transport, Active; Cell Line; Cell Separation; Cell Survival; Flow Cytometry; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Mice; Protein Binding; Reserpine; Spectrometry, Fluorescence; Substrate Specificity; Time Factors | 2001 |
Pharmacophore model of drugs involved in P-glycoprotein multidrug resistance: explanation of structural variety (hypothesis).
Topics: Adenosine Triphosphatases; Algorithms; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Binding, Competitive; Caco-2 Cells; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship; Radioligand Assay; Rhodamine 123; Stereoisomerism; Verapamil; Vinblastine | 2002 |
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration | 2004 |
New 1,3-dioxolane and 1,3-dioxane derivatives as effective modulators to overcome multidrug resistance.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cell Proliferation; Dioxanes; Dioxolanes; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Structure-Activity Relationship | 2007 |
Air to lung partition coefficients for volatile organic compounds and blood to lung partition coefficients for volatile organic compounds and drugs.
Topics: Air; Animals; Humans; Lung; Organic Chemicals; Probability; Rats; Tissue Distribution; Volatilization | 2008 |
Small molecule regulators of autophagy identified by an image-based high-throughput screen.
Topics: Autophagy; Calcium Channel Blockers; Cell Line, Tumor; Drug Evaluation, Preclinical; Fluspirilene; Glioblastoma; Green Fluorescent Proteins; Humans; Intracellular Membranes; Loperamide; Microtubule-Associated Proteins; Mycotoxins; Peptides; Phagosomes; Phosphatidylinositol Phosphates; Pimozide; Protein Kinases; Recombinant Fusion Proteins; Sirolimus; Small Molecule Libraries; TOR Serine-Threonine Kinases; Trifluoperazine; Zinc Fingers | 2007 |
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase | 2008 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Attenuation of intestinal absorption by major efflux transporters: quantitative tools and strategies using a Caco-2 model.
Topics: Adenosine; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Sub-Family B Member 4; ATP-Binding Cassette Transporters; Biological Transport; Caco-2 Cells; Chromatography, Liquid; Dibenzocycloheptenes; Diketopiperazines; Drug Discovery; Heterocyclic Compounds, 4 or More Rings; Humans; Intestinal Absorption; Mass Spectrometry; Models, Biological; Neoplasm Proteins; Pharmaceutical Preparations; Predictive Value of Tests; Propionates; Quinolines; Substrate Specificity | 2011 |
FDA-approved drug labeling for the study of drug-induced liver injury.
Topics: Animals; Benchmarking; Biomarkers, Pharmacological; Chemical and Drug Induced Liver Injury; Drug Design; Drug Labeling; Drug-Related Side Effects and Adverse Reactions; Humans; Pharmaceutical Preparations; Reproducibility of Results; United States; United States Food and Drug Administration | 2011 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
The effects of drugs on monocytic fusion in vivo.
Topics: Adenosine Triphosphatases; Animals; Calcium; Cell Fusion; Cell Membrane; Cortisone; Cyclic AMP; Diphenhydramine; Edetic Acid; Glucagon; Insulin; Isoproterenol; Lidocaine; Lysosomes; Male; Mice; Mice, Inbred C57BL; Monocytes; Ouabain; Pyrilamine; Tetracaine; Trifluoperazine; Verapamil | 1975 |
Is renal protection with calcium antagonists possible?
Topics: Adenosine; Animals; Blood Pressure; Cells, Cultured; Dogs; Endothelins; Female; Glomerular Filtration Rate; Male; Renal Circulation; Trifluoperazine; Verapamil | 1992 |
Long-term treatment with different calcium- and calmodulin-antagonists induces changes in rat brain alpha-adrenoceptors.
Topics: Administration, Oral; Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Dioxanes; Flunarizine; Male; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Regression Analysis; Trifluoperazine; Verapamil | 1992 |
Effects of calcium antagonists on rat normal and skinned fundus.
Topics: Animals; Calcium Channel Blockers; Cinnarizine; Dantrolene; Female; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1992 |
Lymphocyte calmodulin and its participation in the stimulation of T lymphocytes by mitogenic lectins.
Topics: Calcium; Calmodulin; Humans; In Vitro Techniques; Lectins; Lymphocyte Activation; Lymphocytes; T-Lymphocytes; Trifluoperazine; Verapamil | 1992 |
[Effects of methylflavonolamine hydrochloride on contractility of isolated rabbit ileum].
Topics: Animals; Female; Flavonoids; Flavonols; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rabbits; Trifluoperazine; Verapamil | 1992 |
Effect of calcium and calcium antagonists on 45Ca influx and cellular growth of human prostatic tumor cells.
Topics: Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Radioisotopes; Calmodulin; Cell Division; Extracellular Space; Fibroblasts; Humans; Kinetics; Lanthanum; Male; Potassium; Prostatic Neoplasms; Tamoxifen; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1991 |
Changes in benzodiazepine receptors of rat brain after long-term treatment with the Ca(2+)-antagonists nifedipine, verapamil, flunarizine and with the calmodulin antagonist trifluoperazine.
Topics: Animals; Brain Chemistry; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Flunarizine; Flunitrazepam; Hippocampus; Kinetics; Male; Nifedipine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Trifluoperazine; Verapamil | 1991 |
Agents which reverse multidrug-resistance are inhibitors of [3H]vinblastine transport by isolated vesicles.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Biological Transport, Active; Carcinoma, Squamous Cell; Cell Membrane; Dihydropyridines; Drug Resistance; Humans; Kinetics; Leucine; Membrane Glycoproteins; Phenothiazines; Quinidine; Trifluoperazine; Tumor Cells, Cultured; Verapamil; Vinblastine | 1991 |
Tributyltin stimulates reactive oxygen formation in toadfish macrophages.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Benzoates; Benzoic Acid; Calcimycin; Calcium; Calcium Channels; Fishes; Free Radical Scavengers; Free Radicals; Indomethacin; Luminescent Measurements; Macrophage Activation; Macrophages; Masoprocol; Oxygen; Superoxide Dismutase; Tetradecanoylphorbol Acetate; Trialkyltin Compounds; Trifluoperazine; Verapamil | 1991 |
Contraction of vascular smooth muscle induced by phorbol 12,13 dibutyrate in human and rat pulmonary arteries.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Atropine; Calcium; Humans; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Phentolamine; Phorbol 12,13-Dibutyrate; Potassium; Propranolol; Protein Kinase C; Pulmonary Artery; Rats; Tetrodotoxin; Trifluoperazine; Verapamil | 1991 |
The long-term treatment with the Ca(2+)-antagonists nifedipine, verapamil, flunarizine and with the calmodulin antagonist trifluoperazine decreases the activity of 5-HT1 receptors in rat cerebral cortex and hippocampus.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Flunarizine; Hippocampus; In Vitro Techniques; Kinetics; Male; Nifedipine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Trifluoperazine; Verapamil | 1991 |
Involvement of calmodulin in depolarization-induced release of corticotrophin-releasing hormone-41 from the rat hypothalamus in vitro.
Topics: Animals; Calcimycin; Calcium; Calmodulin; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Hypothalamus; In Vitro Techniques; Membrane Potentials; Phenytoin; Potassium Chloride; Radioimmunoassay; Rats; Trifluoperazine; Verapamil; Veratridine | 1991 |
Calcium antagonist properties of cinnarizine, trifluoperazine and verapamil in guinea-pig normal and skinned trachealis muscle.
Topics: Animals; Calcium Channel Blockers; Cinnarizine; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Trachea; Trifluoperazine; Verapamil | 1990 |
Involvement of cell calcium and transmembrane potential in control of hepatocyte volume.
Topics: Animals; Calcium; Calmodulin; Colchicine; Culture Techniques; Cytochalasin B; Cytoskeleton; Dose-Response Relationship, Drug; Liver; Male; Membrane Potentials; Mice; Mice, Inbred ICR; Microelectrodes; Osmolar Concentration; Osmotic Pressure; Promethazine; Trifluoperazine; Verapamil | 1991 |
Role of calcium in the regulation of theca cell androstenedione production in the domestic hen.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Androstenedione; Animals; Calcimycin; Calcium; Calmodulin; Chickens; Colforsin; Dose-Response Relationship, Drug; Female; Imidazoles; Luteinizing Hormone; Theca Cells; Trifluoperazine; Verapamil | 1991 |
Rapid determination of cellular resistance-related drug efflux in tumor cells.
Topics: Animals; Antibiotics, Antineoplastic; Biological Transport; Chlorpromazine; Doxorubicin; Drug Resistance; Flow Cytometry; Humans; Leukemia P388; Mice; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1990 |
Refractoriness to the insulin-like effects of growth hormone depends upon calcium.
Topics: Adipose Tissue; Animals; Calcimycin; Calcium; Calmodulin; Egtazic Acid; Glucose; Growth Hormone; Imidazoles; Insulin; Male; Rats; Signal Transduction; Trifluoperazine; Verapamil | 1990 |
Blocking the calcium cascade in experimental acute renal failure.
Topics: Acute Kidney Injury; Animals; Calcium; Calmodulin; Etidronic Acid; Male; Rats; Rats, Inbred Strains; Renal Artery Obstruction; Survival Rate; Trifluoperazine; Verapamil | 1990 |
Influence of long-term treatment with the Ca2(+)-antagonists nifedipine, verapamil, flunarizine and with the calmodulin antagonist trifluoperazine on beta-adrenoceptors in rat cerebral cortex.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Dihydroalprenolol; Flunarizine; Male; Membrane Fluidity; Membranes; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Synaptosomes; Trifluoperazine; Verapamil | 1990 |
[The characteristics of the action of calcium antagonists on glucose transport in the rat small intestine].
Topics: Animals; Biological Transport; Calcium Channel Blockers; Calmodulin; Chlorpromazine; Depression, Chemical; Glucose; In Vitro Techniques; Intestinal Absorption; Intestine, Small; Male; Perfusion; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1990 |
Chronic calcium antagonist use in carcinoma of the lung and colon: a retrospective cohort observational study.
Topics: Calcium; Carcinoma, Small Cell; Cohort Studies; Colonic Neoplasms; Diltiazem; Humans; Lung Neoplasms; Nifedipine; Retrospective Studies; Survival Analysis; Trifluoperazine; Verapamil | 1990 |
Activity of various amphiphilic agents in reversing multidrug resistance of L 1210 cells.
Topics: Animals; Drug Resistance; Ethylamines; Hycanthone; Leukemia L1210; Phenotype; Piperidines; Quinidine; Quinine; Tamoxifen; Trifluoperazine; Verapamil | 1990 |
Effects of the Ca2(+)-antagonists nifedipine, verapamil, flunarizine and of the calmodulin antagonist trifluoperazine on muscarinic cholinergic receptors in rat cerebral cortex.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Flunarizine; Kinetics; Male; Nifedipine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Trifluoperazine; Verapamil | 1990 |
Role of calcium in the phloretin effects on sugar transport in rat small intestine.
Topics: Animals; Biological Transport; Calcium; Calmodulin; Galactose; Imines; Intestine, Small; Ion Channels; Male; Phloretin; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1986 |
Interrelated calcium ion and cyclic AMP inhibition of placental lactogen secretion by cultured human term trophoblast.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Bucladesine; Calcimycin; Calcium; Calcium Channel Blockers; Cells, Cultured; Cyclic AMP; Female; Humans; Ion Channels; Placental Lactogen; Pregnancy; Trifluoperazine; Trophoblasts; Verapamil | 1987 |
Inhibitory effects of calcium channel agonists on renin release from rat kidney cortical slices.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dose-Response Relationship, Drug; Imidazoles; Ion Channels; Kidney Cortex; Male; Nifedipine; Pyridines; Rats; Rats, Inbred Strains; Renin; Trifluoperazine; Verapamil | 1987 |
On the involvement of cyclic AMP and extracellular Ca2+ in the regulation of hormone release from rat pituitary tumour (GH3) cells in culture.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Calcimycin; Calcium; Cell Line; Cobalt; Cyclic AMP; Egtazic Acid; Extracellular Space; Growth Hormone; Pituitary Neoplasms; Prolactin; Rats; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil | 1987 |
Different insulin-secretory responses to calcium-channel blockers in islets of lean and obese (ob/ob) mice.
Topics: Animals; Colforsin; Dantrolene; Glucose; Insulin; Insulin Secretion; Ion Channels; Islets of Langerhans; Male; Mice; Mice, Obese; Nifedipine; Obesity; Stimulation, Chemical; Trifluoperazine; Verapamil | 1988 |
Elevation of angiotensin converting enzyme by 3-isobutyl-1-methylxanthine in cultured endothelial cells: a possible role for calmodulin.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Calmodulin; Cattle; Cells, Cultured; Cyclic AMP; Cycloheximide; Dose-Response Relationship, Drug; Egtazic Acid; Endothelium, Vascular; Imidazoles; Indomethacin; Peptidyl-Dipeptidase A; Propranolol; Theophylline; Trifluoperazine; Verapamil; Xanthines | 1988 |
Identification and characterization of [3H]nitrendipine binding sites in rat spinal cord.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Kinetics; Male; Nifedipine; Nitrendipine; Quinacrine; Rats; Rats, Inbred Strains; Spinal Cord; Trifluoperazine; Verapamil | 1988 |
Cyclosporine-A transport in isolated renal proximal tubular cells: inhibition by calcium channel blockers.
Topics: Animals; Biological Transport; Calcimycin; Calcium Channel Blockers; Cyclosporins; Diltiazem; Kidney Tubules, Proximal; Kinetics; Rabbits; Ruthenium Red; Trifluoperazine; Verapamil | 1988 |
On the relation of calcium to ovine parotid secretion.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Blood Flow Velocity; Calcimycin; Calcium; Egtazic Acid; Infusions, Parenteral; Parotid Gland; Saliva; Sheep; Trifluoperazine; Verapamil | 1989 |
Modulation by adriamycin, daunomycin, verapamil, and trifluoperazine of the biochemical processes linked to mouse skin tumor promotion by 12-O-tetradecanoylphorbol-13-acetate.
Topics: 9,10-Dimethyl-1,2-benzanthracene; Administration, Topical; Animals; Daunorubicin; DNA; Doxorubicin; Female; Mice; Neoplasms, Experimental; Ornithine Decarboxylase; RNA; Skin Neoplasms; Tetradecanoylphorbol Acetate; Time Factors; Trifluoperazine; Verapamil | 1989 |
Mechanism of membrane phospholipid degradation in ischemic-reperfused rat hearts.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcium; Coronary Disease; Fatty Acids, Nonesterified; Glycerol; Male; Membrane Lipids; Myocardial Reperfusion; Myocardium; Phospholipids; Quinacrine; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1989 |
Calcium calmodulin in altered NaCl transport by heat-labile enterotoxin of Escherichia coli.
Topics: Animals; Bacterial Toxins; Biological Transport, Active; Calcimycin; Calmodulin; Chlorides; Enterotoxins; Escherichia coli; Escherichia coli Proteins; Mice; Rabbits; Sodium; Trifluoperazine; Verapamil | 1989 |
[Ca2+-dependent mechanisms of membrane carbohydrate hydrolysis and of the transport of the monosaccharides being formed in the small intestine].
Topics: Animals; Biological Transport; Calcium; Dietary Carbohydrates; Edetic Acid; Hydrolysis; Intestinal Absorption; Intestinal Mucosa; Intestine, Small; Male; Monosaccharides; Perfusion; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1989 |
Intracellular mechanisms of the effect of thromboxane A2 on water transport.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Body Water; Calcium; Cell Line; Colchicine; Kidney; Kinetics; Prostaglandin Endoperoxides, Synthetic; Thromboxane A2; Trifluoperazine; Verapamil | 1989 |
The role of calcium in gonadotropin-releasing hormone induction of follicle-stimulating hormone release by the pituitary gonadotrope.
Topics: Animals; Calcimycin; Calcium; Cyclic AMP; Cyclic GMP; Dantrolene; Female; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; Kinetics; Organ Culture Techniques; Ovariectomy; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1989 |
Effects of new 4-aminopyridine derivatives on neuromuscular transmission and on smooth muscle contractility.
Topics: Aminopyridines; Animals; Botulinum Toxins; Chemical Phenomena; Chemistry, Physical; Dantrolene; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Phrenic Nerve; Respiratory Muscles; Synaptic Transmission; Trifluoperazine; Verapamil | 1989 |
Parathyroid hormone-induced ornithine decarboxylase activity in fetal rat osteoblasts.
Topics: Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Enzyme Induction; Gestational Age; Kinetics; Ornithine Decarboxylase; Ornithine Decarboxylase Inhibitors; Osteoblasts; Parathyroid Hormone; Rats; Second Messenger Systems; Trifluoperazine; Verapamil | 1989 |
Pituitary thyrotropin-releasing hormone receptors: local anesthetic effects on binding and responses.
Topics: Anesthetics, Local; Animals; Benzocaine; Chlordiazepoxide; Chlorpromazine; Dibucaine; Hydrogen-Ion Concentration; Imipramine; Lidocaine; Pituitary Gland; Procaine; Prolactin; Propranolol; Rats; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Tetracaine; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil | 1989 |
Biosynthesis, processing and half-life of P-glycoprotein in a human multidrug-resistant KB cell.
Topics: Antibodies; ATP Binding Cassette Transporter, Subfamily B, Member 1; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Humans; Immunoblotting; KB Cells; Kinetics; Membrane Glycoproteins; Molecular Weight; Protein Processing, Post-Translational; Tetradecanoylphorbol Acetate; Trifluoperazine; Tunicamycin; Verapamil; Vinblastine | 1989 |
Calcium uptake in human spermatozoa: characterization and mechanisms.
Topics: Antimycin A; Biological Transport; Calcium; Dose-Response Relationship, Drug; Humans; Male; Spermatozoa; Sulfhydryl Reagents; Time Factors; Trifluoperazine; Verapamil | 1989 |
Zinc uptake in human seminal spermatozoa: characterization and effects on cell membranes.
Topics: Antimycin A; Biological Transport; Cell Membrane; Dose-Response Relationship, Drug; Humans; Male; Mersalyl; Osmotic Pressure; Spermatozoa; Trifluoperazine; Verapamil; Zinc | 1989 |
Inhibition of vincristine binding to plasma membrane vesicles from daunorubicin-resistant Ehrlich ascites cells by multidrug resistance modulators.
Topics: Animals; Carcinoma, Ehrlich Tumor; Cell Cycle; Cell Membrane; Daunorubicin; Drug Resistance; Polysorbates; Quinidine; Trifluoperazine; Tumor Stem Cell Assay; Verapamil; Vincristine | 1989 |
3H-azidopine photoaffinity labeling of high molecular weight proteins in chloroquine resistant falciparum malaria.
Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Chloroquine; Chlorpromazine; Dihydropyridines; Drug Resistance; Glycoproteins; Molecular Weight; Nicardipine; Photochemistry; Plasmodium falciparum; Proteins; Quinacrine; Reserpine; Trifluoperazine; Verapamil | 1989 |
Comparison of the effect of cyclosporine, verapamil, and trifluoperazine on calcium-induced membrane permeability of mitochondria.
Topics: Animals; Calcium; Cyclosporins; Intracellular Membranes; Kidney Cortex; Kinetics; Mitochondria; Mitochondria, Liver; Mitochondrial Swelling; Rats; Trifluoperazine; Verapamil | 1989 |
Drug-drug interaction between cyclosporine and agents affecting calcium-dependent lymphocyte proliferation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium Channel Blockers; Cells, Cultured; Cyclosporins; Drug Interactions; Humans; Imidazoles; Isoquinolines; Lymphocyte Activation; Piperazines; Protein Kinase C; Sulfonamides; Trifluoperazine; Verapamil | 1989 |
Antagonism of calcium by zinc in guinea-pig isolated taenia caeci and trachealis muscle.
Topics: Acetylcholine; Animals; Cadmium; Calcium; Cecum; Cell Membrane; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Trachea; Trifluoperazine; Verapamil; Zinc | 1989 |
In vivo characterization of combination antitumor chemotherapy with calcium channel blockers and cis-diamminedichloroplatinum(II).
Topics: Animals; Calcium Channel Blockers; Cisplatin; Diltiazem; Drug Evaluation, Preclinical; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Imidazoles; Lung Neoplasms; Melanoma, Experimental; Mice; Nicardipine; Nifedipine; Trifluoperazine; Verapamil | 1989 |
[Prevention of adrenaline-induced arrhythmia by a calmodulin blocker, trifluoroperazine].
Topics: Animals; Arrhythmias, Cardiac; Calmodulin; Epinephrine; Male; Rats; Rats, Inbred Strains; Time Factors; Trifluoperazine; Verapamil | 1989 |
Changes in the three-dimensional organization of LoVo cells associated with resistance to doxorubicin.
Topics: Adenocarcinoma; Cell Aggregation; Cell Division; Colonic Neoplasms; Cyclosporins; Doxorubicin; Drug Resistance; Humans; In Vitro Techniques; Membrane Proteins; Molecular Weight; Organoids; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1989 |
The response of cultured gonadotrophs to inhibin: the role of calcium mobilization.
Topics: Animals; Calcium; Calmodulin; Cells, Cultured; Cyclic GMP; Female; Fluorescent Antibody Technique; Follicle Stimulating Hormone; Inhibins; Luteinizing Hormone; Pituitary Gland, Anterior; Pituitary Hormone-Releasing Hormones; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1987 |
Parathyroid hormone stimulation of mitosis in rat thymic lymphocytes is independent of cyclic AMP.
Topics: Animals; Calcium; Cell Division; Cells, Cultured; Cyclic AMP; Lymphocytes; Male; Parathyroid Hormone; Peptide Fragments; Rats; Rats, Inbred Strains; Teriparatide; Thymus Gland; Trifluoperazine; Verapamil | 1987 |
Action of loperamide on neuronally mediated and Ca2+- or cAMP-mediated secretion in rat colon.
Topics: Animals; Calcium; Carbachol; Colforsin; Colon; Cyclic AMP; Electric Stimulation; In Vitro Techniques; Intestinal Mucosa; Loperamide; Male; Morphine; Neurons; Piperidines; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1988 |
Differentiation of calcium antagonists with respect to their effects in normal and skinned taenia caeci preparations.
Topics: Animals; Calcium; Calcium Channel Blockers; Calmodulin; Cinnarizine; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Intestines; Male; Muscle Contraction; Parasympatholytics; Trifluoperazine; Verapamil | 1987 |
Calmodulin dependence of somatostatin release stimulated by growth hormone-releasing factor.
Topics: Animals; Calmodulin; Drug Synergism; Egtazic Acid; Growth Hormone-Releasing Hormone; In Vitro Techniques; Kinetics; Male; Median Eminence; Nifedipine; Rats; Rats, Inbred Strains; Somatostatin; Trifluoperazine; Verapamil | 1988 |
Role of Ca2+ in bombesin-stimulated release of gastrin and somatostatin from isolated perfused rat stomach.
Topics: Animals; Bombesin; Calcium; Egtazic Acid; Gastric Mucosa; Gastrins; In Vitro Techniques; Male; Nifedipine; Peptides; Rats; Somatostatin; Stimulation, Chemical; Trifluoperazine; Verapamil | 1988 |
Cell cycle dependence of calmodulin levels during HL-60 proliferation and myeloid differentiation. No changes during pre-commitment.
Topics: Calmodulin; Cell Cycle; Cell Differentiation; Cell Division; Cell Line; Humans; Leukemia, Myeloid, Acute; Nifedipine; Nitrendipine; Trifluoperazine; Verapamil | 1986 |
Effects of trifluoperazine and verapamil on the hydro-osmotic response to antidiuretic hormone in the urinary bladder of the toad.
Topics: Animals; Body Water; Bufo marinus; Cyclic AMP; In Vitro Techniques; Kinetics; Osmolar Concentration; Trifluoperazine; Urinary Bladder; Vasopressins; Verapamil | 1985 |
Effect of heparin on platelet aggregation inhibited by PGI2, trifluoperazine and verapamil.
Topics: Blood Platelets; Colforsin; Cyclic AMP; Depression, Chemical; Drug Interactions; Epoprostenol; Heparin; Humans; Platelet Aggregation; Serotonin; Trifluoperazine; Verapamil | 1986 |
Converging adrenergic and cholinergic mechanisms in the inhibition of Cl secretion in fish opercular epithelium.
Topics: Acetylcholine; Animals; Calcium; Chlorine; Clonidine; Cyclic AMP; Dantrolene; Epithelium; Female; Fishes; Killifishes; Male; Receptors, Adrenergic; Receptors, Cholinergic; Trifluoperazine; Verapamil | 1985 |
The dual effect of calcium on aromatization by cultured human trophoblast.
Topics: Androstenedione; Aromatase; Bucladesine; Calcimycin; Calcium; Cells, Cultured; Egtazic Acid; Estradiol; Humans; Trifluoperazine; Trophoblasts; Verapamil | 1986 |
Further studies on the mechanism of action of leukotrienes and histamine on guinea pig lung parenchyma. Role of calcium, phospholipase and methyltransferase.
Topics: Animals; Calcium; Cobalt; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; In Vitro Techniques; Leukotriene B4; Lung; Muscle Contraction; SRS-A; Tetrodotoxin; Trifluoperazine; Tubercidin; Valinomycin; Verapamil | 1986 |
Effect of verapamil and trifluoperazine upon glucose-induced calcium distribution within B cells.
Topics: Animals; Antimony; B-Lymphocytes; Calcium; Female; Glucose; Insulin; Insulin Secretion; Microscopy, Electron; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1988 |
Effect of verapamil on prostaglandin E2 synthesis by hydronephrotic rabbit cortical interstitial cells in primary culture.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bradykinin; Calcimycin; Calcium; Cells, Cultured; Diltiazem; Dinoprostone; Dose-Response Relationship, Drug; Hydronephrosis; Kidney Cortex; Magnesium; Male; Nifedipine; Prostaglandins E; Quinacrine; Rabbits; Trifluoperazine; Verapamil | 1986 |
The inhibitory effects of calmodulin antagonists on the endothelium-dependent relaxation in rabbit aorta.
Topics: Animals; Aorta; Calcimycin; Calmodulin; Carbachol; Endothelium; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Rabbits; Trifluoperazine; Vasodilator Agents; Verapamil | 1986 |
The protective effect of calcium inhibitors and of captopril on the renal microcirculation during reperfusion.
Topics: Angiotensin II; Animals; Calcium; Captopril; Dogs; Heparin; Kidney; Kidney Cortex; Kidney Glomerulus; Kidney Transplantation; Mannitol; Microcirculation; Organ Preservation; Perfusion; Trifluoperazine; Verapamil | 1987 |
Mechanism of vasopressin-induced platelet aggregation.
Topics: Arginine Vasopressin; Calcium; Deamino Arginine Vasopressin; Dose-Response Relationship, Drug; Female; Humans; Lipoxygenase; Platelet Aggregation; Thromboxane B2; Trifluoperazine; Verapamil | 1987 |
Studies on the mechanism of Escherichia coli heat-stable enterotoxin-induced diarrhoea in mice.
Topics: Animals; Bacterial Toxins; Calcimycin; Calcium; Calmodulin; Chlorides; Diarrhea; Enterotoxins; Escherichia coli; Escherichia coli Proteins; Intestinal Absorption; Intestinal Mucosa; Mice; Sodium; Trifluoperazine; Verapamil | 1987 |
Stimulation and inhibition of elastase release from human neutrophil-dependence on the calcium messenger system.
Topics: Adult; Calcimycin; Calcium; Edetic Acid; Enzyme Activation; Humans; Male; Neutrophils; Pancreatic Elastase; Protein Kinase C; Tetradecanoylphorbol Acetate; Trifluoperazine; Verapamil | 1987 |
Stimulation and inhibition of elastase release from human neutrophils dependent on the calcium messenger system.
Topics: Adult; Calcimycin; Calcium; Enzyme Activation; Humans; Male; Neutrophils; Pancreatic Elastase; Protein Kinase C; Trifluoperazine; Verapamil | 1987 |
Calcium-sensitive uptake of amino acids by human placental slices.
Topics: Amino Acids, Branched-Chain; Biological Transport; Calcium; Egtazic Acid; Female; Humans; In Vitro Techniques; Phenylalanine; Placenta; Pregnancy; Protein Synthesis Inhibitors; Trifluoperazine; Verapamil | 1988 |
Role of Ca2+/calmodulin in the regulation of sugar uptake in Escherichia coli heat-stable enterotoxin induced diarrhoea in mice.
Topics: 3-O-Methylglucose; Animals; Bacterial Toxins; Calcimycin; Calcium; Calmodulin; Carbohydrate Metabolism; Diarrhea; Enterotoxins; Escherichia coli Proteins; Intestinal Mucosa; Methylglucosides; Mice; Trifluoperazine; Verapamil | 1987 |
The membrane transport system responsible for multidrug resistance is operating in nonresistant cells.
Topics: Animals; Biological Transport, Active; Cell Line, Transformed; Cell Membrane; Cricetinae; Drug Resistance; Fibroblasts; Fluorescent Dyes; Microscopy, Fluorescence; Mitochondria; Reserpine; Rhodamine 123; Rhodamines; Trifluoperazine; Verapamil | 1988 |
The spasmogenic effect of caffeine in trachealis isolated from control and actively sensitized guinea-pigs.
Topics: Animals; Caffeine; Calcium; Dantrolene; Guinea Pigs; Indomethacin; Male; Muscle Contraction; Muscle, Smooth; Temperature; Trachea; Trifluoperazine; Verapamil | 1988 |
Enhancement of the activity of immunotoxins made with either ricin A chain or Pseudomonas exotoxin in human ovarian and epidermoid carcinoma cell lines.
Topics: ADP Ribose Transferases; Bacterial Toxins; Cadaverine; Calmodulin; Carcinoma, Squamous Cell; Cell Line; Chlorpromazine; Drug Synergism; Exotoxins; Female; Humans; Immunotoxins; Ovarian Neoplasms; Pseudomonas aeruginosa Exotoxin A; Ricin; Trifluoperazine; Verapamil; Virulence Factors | 1988 |
In vivo potentiation of cyclosporine immunosuppression by calcium antagonists.
Topics: Animals; Cyclosporins; Graft Survival; Heart Transplantation; Male; Rats; Rats, Inbred ACI; Rats, Inbred Lew; Transplantation, Heterotopic; Transplantation, Homologous; Trifluoperazine; Verapamil | 1987 |
Usefulness of radionuclide scintiphotography to evaluate preserved kidney viability.
Topics: Animals; Dogs; Female; Hypertonic Solutions; Kidney; Kidney Transplantation; Male; Microspheres; Organ Preservation; Perfusion; Radionuclide Imaging; Technetium; Trifluoperazine; Urokinase-Type Plasminogen Activator; Verapamil | 1987 |
Role of calcium in the activation of neutrophils by leukocyte inhibitory factor (LIF).
Topics: Calcium; Cell Membrane; Colchicine; Fluorescent Dyes; Kinetics; Leukocyte Migration-Inhibitory Factors; Lymphokines; Neutrophils; Trifluoperazine; Verapamil | 1987 |
[Prevention of ischemic and reperfusion arrhythmias using the calmodulin blocker trifluoperazine].
Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calmodulin; Coronary Disease; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1988 |
Effect of different calcium modulators on motilin-induced contractions of the rabbit duodenum. Comparison with acetylcholine.
Topics: Acetylcholine; Animals; Calcium; Calcium Channel Blockers; Diltiazem; Duodenum; Gallic Acid; In Vitro Techniques; Motilin; Muscle Contraction; Muscle, Smooth; Rabbits; Trifluoperazine; Verapamil | 1988 |
Effect of calcium inhibitors and calcium mobilizers on doxorubicin accumulation in rat myocardial tissue.
Topics: Animals; Calcium; Calcium Channel Blockers; Doxorubicin; Flunarizine; Heart; In Vitro Techniques; Male; Myocardium; Rats; Taurine; Trifluoperazine; Verapamil | 1988 |
Altered responses to calcium and trifluoperazine in K+-depolarized duodenum from alloxan diabetic rats.
Topics: Animals; Calcium; Diabetes Mellitus, Experimental; Duodenum; Guinea Pigs; Male; Muscle, Smooth; Neuromuscular Depolarizing Agents; Potassium; Rats; Trifluoperazine; Verapamil | 1987 |
Effect of calcium channel blockers and trifluoperazine on rat liver regeneration.
Topics: Animals; Calcium; Diltiazem; DNA; Hepatectomy; Injections, Intraperitoneal; Liver; Male; Nifedipine; Rats; Rats, Inbred Strains; Thymidine Kinase; Thymidylate Synthase; Trifluoperazine; Verapamil | 1987 |
Iodide transport in rat small intestine: dependence on calcium.
Topics: Animals; Biological Transport; Calcium; In Vitro Techniques; Intestine, Small; Iodides; Male; Rats; Rats, Inbred Strains; Theophylline; Trifluoperazine; Verapamil | 1987 |
[Possibility of overcoming of ACNU resistance in an ACNU-resistant subline of C6 rat glioma].
Topics: Animals; Antineoplastic Agents; Brain Neoplasms; Cell Line; Cells, Cultured; Drug Resistance; Drug Therapy, Combination; Glioma; Male; Nicardipine; Nimustine; Nitrosourea Compounds; Rats; Rats, Inbred Strains; Reserpine; Trifluoperazine; Verapamil | 1986 |
Effects of calcium-antagonists and calmodulin inhibitors on DNA synthesis in cultured rat vascular smooth muscle cells.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cells, Cultured; Diltiazem; DNA Replication; Dose-Response Relationship, Drug; Epidermal Growth Factor; Male; Muscle, Smooth, Vascular; Nicardipine; Platelet-Derived Growth Factor; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine; Verapamil | 1987 |
Influence of calcium antagonists on the antitumor activity and the cardiac toxicity of doxorubicin in the rat.
Topics: Animals; Carcinoma 256, Walker; Doxorubicin; Female; Flunarizine; Heart; Myocardium; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1987 |
The pathophysiology of the no-reflow phenomenon in cold-stored kidneys.
Topics: Animals; Calcium; Captopril; Cold Temperature; Dogs; Kidney; Renal Circulation; Tissue Preservation; Trifluoperazine; Verapamil | 1987 |
Phosphorylation of the Mr 170,000 to 180,000 glycoprotein specific to multidrug-resistant tumor cells: effects of verapamil, trifluoperazine, and phorbol esters.
Topics: Antibodies, Monoclonal; Calmodulin; Drug Resistance; Glycoproteins; Humans; Molecular Weight; Peptide Mapping; Phosphoproteins; Phosphorylation; Phosphoserine; Protein Kinase C; Tetradecanoylphorbol Acetate; Trifluoperazine; Verapamil | 1987 |
Ca2+-calmodulin regulates the induction and expression of macrophage cytotoxicity.
Topics: Animals; Calcium; Calmodulin; Cytotoxicity, Immunologic; Female; In Vitro Techniques; Lymphokines; Macrophage Activation; Macrophages; Mice; Sulfonamides; Trifluoperazine; Vaccinia virus; Verapamil | 1987 |
Action of calcium antagonists on multidrug resistant cells. Specific cytotoxicity independent of increased cancer drug accumulation.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Calcium; Calcium Channel Blockers; Cell Line; Cell Survival; Colchicine; Cricetinae; Daunorubicin; Drug Resistance; Humans; Kinetics; Mice; Nifedipine; Trifluoperazine; Verapamil; Vinblastine | 1987 |
Mechanisms of action of inhibitors of prolactin secretion in GH3 pituitary cells. I. Ca2+-dependent inhibition of amino acid incorporation.
Topics: Acetylcholine; Amino Acids; Animals; Bromocriptine; Calcium; Carbachol; Cell Line; Chlorpromazine; Imidazoles; Magnesium; Nifedipine; Pituitary Neoplasms; Prolactin; Protein Processing, Post-Translational; Rats; Trifluoperazine; Verapamil | 1986 |
Beneficial effects of calcium channel blockers and calmodulin binding drugs on in vitro renal cell anoxia.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cell Survival; Cells, Cultured; Hypoxia; Isomerism; Nephrons; Nifedipine; Rabbits; Sulfonamides; Time Factors; Trifluoperazine; Verapamil | 1986 |
Characterization of a doxorubicin-resistant murine melanoma line: studies on cross-resistance and its circumvention.
Topics: Animals; Cell Line; Cell Survival; Clone Cells; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance; Melanins; Melanoma; Mice; Mice, Inbred C57BL; Mitosis; Trifluoperazine; Verapamil; Vincristine | 1986 |
Effects of some Ca2+ blockers on receptor potentials of crayfish retina.
Topics: Animals; Astacoidea; Calcium; Calcium Channel Blockers; Evoked Potentials, Visual; Gallopamil; In Vitro Techniques; Photoreceptor Cells; Retina; Trifluoperazine; Verapamil | 1986 |
Enhanced calcium-sensitivity of erythrocytes in hypertension--calcium-induced changes of erythrocyte osmotic fragility in essential hypertension.
Topics: Adult; Calcium; Calmodulin; Diltiazem; Erythrocytes; Female; Humans; Hypertension; Male; Osmotic Fragility; Trifluoperazine; Verapamil | 1986 |
Regulatory effect of calcium on 3H-dopamine binding to guinea-pig heart membrane preparations.
Topics: Animals; Calcium; Calcium Chloride; Dopamine; Edetic Acid; Guinea Pigs; In Vitro Techniques; Kinetics; Membranes; Myocardium; Potassium; Trifluoperazine; Verapamil | 1985 |
Flow cytometric monitoring of cellular anthracycline accumulation in murine leukemic cells.
Topics: Animals; Biological Transport; Cell Line; Chlorpromazine; Daunorubicin; Doxorubicin; Flow Cytometry; Fluorometry; Leukemia P388; Leukemia, Experimental; Mice; Monitoring, Physiologic; Trifluoperazine; Tumor Stem Cell Assay; Verapamil | 1986 |
Calcium-dependence of sugar transport in rat small intestine.
Topics: Animals; Biological Transport, Active; Calcium; Calmodulin; Galactose; Imines; In Vitro Techniques; Intestinal Mucosa; Intestine, Small; Male; Rats; Rats, Inbred Strains; Theophylline; Trifluoperazine; Verapamil | 1985 |
Effects of Ca2+ and calmodulin antagonists on the oxygen uptake induced by acetylcholine or substance P in rat submandibular gland slices.
Topics: Acetylcholine; Animals; Calcium Channel Blockers; Calmodulin; Chlorpromazine; Diltiazem; In Vitro Techniques; Lanthanum; Male; Oxygen Consumption; Rats; Rats, Inbred Strains; Submandibular Gland; Substance P; Sulfonamides; Trifluoperazine; Vasodilator Agents; Verapamil | 1984 |
Stimulation of hepatic glycogenolysis by 12-O-tetradecanoylphorbol-13-acetate (TPA) via a calcium requiring process.
Topics: Animals; Calcimycin; Calcium Chloride; Cyclic AMP; Cyclic GMP; Diltiazem; Glucose; Kinetics; Liver; Liver Glycogen; Male; Phorbols; Proteins; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Trifluoperazine; Verapamil | 1984 |
The involvement of calcium in the intestinal response to secretagogues in the rat.
Topics: Acetylcholine; Animals; Bucladesine; Calcimycin; Calcium; Chlorides; Dinoprostone; Egtazic Acid; Gallic Acid; In Vitro Techniques; Intestinal Mucosa; Intestinal Secretions; Intestines; Male; Membrane Potentials; Potassium; Prostaglandins E; Rats; Serotonin; Sodium; Theophylline; Trifluoperazine; Verapamil | 1984 |
Is renin secretion governed by the calcium permeability of the juxtaglomerular cell membrane?
Topics: Angiotensin II; Animals; Calcium; Cell Membrane; Cell Membrane Permeability; Cells, Cultured; Colforsin; Cyclic AMP; Diterpenes; Isoproterenol; Juxtaglomerular Apparatus; Kinetics; Rats; Renin; Trifluoperazine; Verapamil | 1984 |
Norepinephrine-stimulated vascular prostacyclin synthesis. Receptor-dependent calcium channels control prostaglandin synthesis.
Topics: 6-Ketoprostaglandin F1 alpha; Animals; Aorta; Epoprostenol; In Vitro Techniques; Ion Channels; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Potassium; Prostaglandins; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1984 |
Chymotrypsin, ileal chloride transport, and neurotransmitters.
Topics: Animals; Chlorides; Chymotrypsin; Dinoprostone; Electric Stimulation; Ileum; Intestinal Mucosa; Ion Channels; Neurotransmitter Agents; Ouabain; Prostaglandins E; Rabbits; Theophylline; Trifluoperazine; Vasoactive Intestinal Peptide; Verapamil | 1984 |
Effect of phorbol esters on the release of growth hormone and prolactin from rat pituitary cells cultured in monolayer.
Topics: Animals; Calcium; Cells, Cultured; Growth Hormone; Hyaluronoglucosaminidase; Indomethacin; Male; Phorbol Esters; Phorbols; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Somatostatin; Trifluoperazine; Verapamil | 1984 |
Effect of calmodulin antagonists on CA2+ uptake by boar spermatozoa.
Topics: Animals; Biological Transport, Active; Calcium; Calcium Channel Blockers; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Cell Membrane; Imidazoles; Kinetics; Male; Spermatozoa; Swine; Trifluoperazine; Verapamil | 1983 |
Effect of trifluoperazine, compound 48/80, TMB-8 and verapamil on the rate of calmodulin binding to erythrocyte Ca2+-ATPase.
Topics: Calcium Channel Blockers; Calcium-Transporting ATPases; Calmodulin; Erythrocyte Membrane; Gallic Acid; Humans; In Vitro Techniques; Kinetics; p-Methoxy-N-methylphenethylamine; Trifluoperazine; Verapamil | 1984 |
Effect of trifluoperazine, compound 48/80, TMB-8 and verapamil on ionophore A23187 induced calcium transients in human red cells.
Topics: Biological Transport, Active; Calcimycin; Calcium; Calcium-Transporting ATPases; Erythrocytes; Gallic Acid; Humans; p-Methoxy-N-methylphenethylamine; Trifluoperazine; Verapamil | 1984 |
Effect of trifluoperazine, D600, and phenytoin on depolarization- and thyrotropin-releasing hormone-induced thyrotropin release from rat pituitary tissue.
Topics: Animals; Calcium; Gallopamil; Ion Channels; Male; Membrane Potentials; Phenytoin; Pituitary Gland, Anterior; Potassium; Rats; Sodium; Thyrotropin; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil; Veratridine | 1981 |
Possible role of calcium uptake and calmodulin in adrenal glomerulosa cells: effects of verapamil and trifluoperazine.
Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Aldosterone; Angiotensin II; Animals; Bucladesine; Calcium; Calcium-Binding Proteins; Calmodulin; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1982 |
Follicle-stimulating hormone--regulated granulosa cell steroidogenesis: involvement of the calcium-calmodulin system.
Topics: Animals; Bucladesine; Calcium; Calcium-Binding Proteins; Calmodulin; Cyclic AMP; Egtazic Acid; Female; Follicle Stimulating Hormone; Granulosa Cells; In Vitro Techniques; Lanthanum; Ovary; Progesterone; Rats; Rats, Inbred Strains; Steroids; Trifluoperazine; Verapamil | 1983 |
Inhibition of (H+ + K+)-ATPase and H+ accumulation in hog gastric membranes by trifluoperazine, verapamil and 8-(N,N-diethylamino)octyl-3,4,5-trimethoxybenzoate.
Topics: Adenosine Triphosphatases; Animals; Gallic Acid; Gastric Mucosa; H(+)-K(+)-Exchanging ATPase; Hydrogen; Kinetics; Rabbits; Swine; Time Factors; Trifluoperazine; Verapamil | 1984 |
Participation of calcium and calmodulin in the formation of acetylcholine receptor clusters.
Topics: Animals; Calcium; Calmodulin; Cells, Cultured; Embryo, Nonmammalian; Fluorescent Antibody Technique; Gallopamil; Kinetics; Muscles; Nifedipine; Receptors, Cholinergic; Trifluoperazine; Verapamil; Xenopus | 1984 |
Critical role of extracellular calcium in vanadate-induced renal vasoconstriction.
Topics: Animals; Calcium; Dogs; Drug Combinations; Egtazic Acid; Extracellular Space; Parathyroid Glands; Renal Circulation; Thyroidectomy; Time Factors; Trifluoperazine; Vanadates; Vanadium; Vasoconstriction; Verapamil | 1984 |
The role of calcium in the stimulation of prostaglandin synthesis by vasopressin in rabbit renal-medullary interstitial cells in tissue culture.
Topics: Angiotensin II; Animals; Arginine Vasopressin; Calcimycin; Calcium; Culture Techniques; Dinoprostone; Kidney Medulla; Prostaglandins E; Rabbits; Stimulation, Chemical; Trifluoperazine; Verapamil | 1984 |
Effect of trifluoperazine, compound 48/80, TMB-8 and verapamil on ionophore A23187 mediated calcium uptake in ATP depleted human red cells.
Topics: Adenosine Triphosphate; Biological Transport; Calcimycin; Calcium; Erythrocytes; Gallic Acid; Humans; Kinetics; p-Methoxy-N-methylphenethylamine; Trifluoperazine; Verapamil | 1984 |
Calcium antagonists and calmodulin inhibitors block cytokinin-induced bud formation in Funaria.
Topics: Calcium; Calmodulin; Cell Division; Cells, Cultured; Chlorpromazine; Cytokinins; Gallic Acid; Gallopamil; Lanthanum; Plant Growth Regulators; Plants; Trifluoperazine; Verapamil | 1983 |
Ca2+ release from energetically coupled tumor mitochondria.
Topics: Animals; Calcium; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Carcinoma, Ehrlich Tumor; Cell Line; Dibucaine; Male; Mice; Mitochondria; Sodium; Trifluoperazine; Verapamil | 1983 |
Effects of Ca2+ on ileal transport and electrically induced secretion.
Topics: Animals; Biological Transport, Active; Calcium; Chlorides; Egtazic Acid; Electric Stimulation; Ileum; Nifedipine; Rabbits; Sodium; Trifluoperazine; Verapamil | 1980 |
Optic cup formation: a calcium-regulated process.
Topics: Animals; Caffeine; Calcimycin; Calcium; Chick Embryo; Eye; Microscopy, Fluorescence; Organ Culture Techniques; Retina; Theophylline; Trifluoperazine; Verapamil | 1982 |
Two sites for calcium action in compaction of the mouse embryo.
Topics: Animals; Calcimycin; Calcium; Cell Communication; Embryo, Mammalian; Female; In Vitro Techniques; Mice; Mice, Inbred ICR; Trifluoperazine; Verapamil | 1982 |
Calcium dependence and contraction in somite formation.
Topics: Animals; Benzimidazoles; Calcimycin; Calcium; Calcium-Binding Proteins; Calmodulin; Cell Movement; Chick Embryo; Culture Techniques; Mesoderm; Microscopy, Electron, Scanning; Microtubules; Nocodazole; Papaverine; Trifluoperazine; Verapamil | 1982 |
Further studies on the role of calcium in the regulation of glutamate decarboxylase activity in brain slices.
Topics: 2,4-Dinitrophenol; Animals; Antimycin A; Brain; Calcium; Carboxy-Lyases; Corpus Striatum; Dinitrophenols; gamma-Aminobutyric Acid; Glutamate Decarboxylase; In Vitro Techniques; Male; Potassium; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1983 |
A 113Cd and 1H NMR study of the interaction of calmodulin with D600, trifluoperazine and some other hydrophobic drugs.
Topics: Animals; Binding Sites; Calcium; Calcium-Binding Proteins; Calmodulin; Cattle; Chemical Phenomena; Chemistry; Gallopamil; Magnetic Resonance Spectroscopy; Male; Protein Binding; Testis; Trifluoperazine; Verapamil | 1983 |
Role of calcium ions and calmodulin in the aldosterone stimulating action of prostaglandin E2.
Topics: Adrenal Glands; Aldosterone; Animals; Calcium; Calcium-Binding Proteins; Calmodulin; Dinoprostone; Dose-Response Relationship, Drug; Male; Osmolar Concentration; Prostaglandins E; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1982 |
Importance of cellular calcium stores in glucose-stimulated insulin release.
Topics: Animals; Calcium; Calmodulin; Cytosol; Glucose; Insulin; Insulin Secretion; Male; Ouabain; Rats; Rats, Inbred Strains; Secretory Rate; Trifluoperazine; Verapamil | 1981 |
Effect of Ca2+ blocking agents on the metabolism of low density lipoproteins in human skin fibroblasts.
Topics: Benzazepines; Calcium Channel Blockers; Dibucaine; Diltiazem; Fendiline; Fibroblasts; Gallopamil; Humans; Kinetics; Lipoproteins, LDL; Nifedipine; Phenethylamines; Prenylamine; Pyridines; Skin; Trifluoperazine; Verapamil | 1982 |
Increased accumulation of vincristine and adriamycin in drug-resistant P388 tumor cells following incubation with calcium antagonists and calmodulin inhibitors.
Topics: Animals; Calcium Channel Blockers; Calcium-Binding Proteins; Calmodulin; Clomipramine; Doxorubicin; Drug Resistance; Kinetics; Leukemia P388; Leukemia, Experimental; Mice; Prenylamine; Quinoxalines; Trifluoperazine; Verapamil; Vincristine | 1982 |
Esterification of plasma membrane cholesterol and triacylglycerol-rich lipoprotein secretion in CaCo-2 cells: possible role of p-glycoprotein.
Topics: Apolipoproteins B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Membrane; Cholesterol; Cholesterol Esters; Endoplasmic Reticulum; Esterification; Humans; Intestinal Mucosa; Intestines; Lipids; Lipoproteins; Nigericin; Progesterone; Trifluoperazine; Triglycerides; Verapamil | 1995 |
Role of calcium in biphasic immunomodulation by gamma-HCH (lindane) in mice.
Topics: Adjuvants, Immunologic; Animals; Calcium; Calcium Channels; Calmodulin; Cells, Cultured; Female; Hexachlorocyclohexane; Immunosuppressive Agents; Lymphocyte Activation; Lymphocytes; Mice; Trifluoperazine; Verapamil | 1993 |
Role of calcium in the regulation of ornithine decarboxylase enzyme activity in mouse colon cancer cells.
Topics: Animals; Calcium; Calcium Channels; Calmodulin; Colonic Neoplasms; Ion Transport; Mice; Nifedipine; Ornithine Decarboxylase; Potassium Chloride; Sulfonamides; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1995 |
MDR1 gene expression: its effect on drug resistance to doxorubicin in human hepatocellular carcinoma cell lines.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carcinoma, Hepatocellular; Carrier Proteins; Cefoperazone; Ceftriaxone; Doxorubicin; Drug Resistance; Drug Synergism; Gene Expression; Humans; Immunohistochemistry; Liver Neoplasms; Membrane Glycoproteins; Neoplasm Proteins; Quinidine; RNA, Messenger; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1994 |
In vitro evaluation of chemosensitizers for clinical reversal of P-glycoprotein-associated Taxol resistance.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cyclosporine; Drug Resistance; Humans; Membrane Glycoproteins; Multiple Myeloma; Paclitaxel; Quinine; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1993 |
The effect of Ca2+ antagonists on spontaneous motility from sheep duodenum.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Diltiazem; Duodenum; Gallic Acid; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Sheep; Trifluoperazine; Verapamil | 1994 |
Comparative study of intracellular calcium and adenosine 3',5'-cyclic monophosphate levels in human breast carcinoma cells sensitive or resistant to Adriamycin: contribution to reversion of chemoresistance.
Topics: Binding Sites; Breast Neoplasms; Calcium; Cell Line; Cyclic AMP; Doxorubicin; Drug Resistance; Glutathione; Phosphoprotein Phosphatases; Protein Kinases; Second Messenger Systems; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1994 |
Calcium channel blockers inhibit the (Ca2+ + Mg2+)-ATPase activity and the 125I-calmodulin binding in brain membranes.
Topics: Animals; Autoradiography; Binding Sites; Brain; Ca(2+) Mg(2+)-ATPase; Calcium Channel Blockers; Calmodulin; Cell Membrane; Electrophoresis, Polyacrylamide Gel; Flunarizine; Iodine Radioisotopes; Nitrendipine; Sheep; Stereoisomerism; Synaptic Membranes; Trifluoperazine; Verapamil | 1994 |
In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.
Topics: Animals; Artemisinins; Female; Mefloquine; Mice; Primaquine; Proguanil; Quinine; Sesquiterpenes; Sulfadiazine; Toxoplasma; Triazines; Trifluoperazine; Uracil; Verapamil | 1994 |
Doxorubicin resistance in human melanoma cells: MDR-1 and glutathione S-transferase pi gene expression.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Death; Cell Division; Cell Line; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance; Gene Expression; Glutathione Transferase; Humans; Leukemia P388; Melanoma; Membrane Glycoproteins; Mice; RNA, Messenger; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1993 |
Effects of two Ca2+ modulators in normal and albumin-sensitized guinea-pig trachea.
Topics: Acetylcholine; Albumins; Animals; Asthma; Calcium; Disease Models, Animal; Guinea Pigs; Immunization; Male; Muscle, Smooth; Trachea; Trifluoperazine; Vagus Nerve; Verapamil | 1993 |
Influence of calmodulin antagonists and calcium channel blockers on triiodothyronine uptake by rat hepatoma and myoblast cell lines.
Topics: Analysis of Variance; Animals; Cadmium; Calcium; Calcium Channel Blockers; Calmodulin; Cell Line; Diltiazem; Imidazoles; Iodine Radioisotopes; Liver Neoplasms, Experimental; Magnesium; Muscles; Nifedipine; Protein Kinase C; Rats; Sulfonamides; Tetradecanoylphorbol Acetate; Trifluoperazine; Triiodothyronine; Tumor Cells, Cultured; Verapamil | 1993 |
Verapamil may cause depression.
Topics: Bipolar Disorder; Depressive Disorder; Drug Therapy, Combination; Female; Humans; Middle Aged; Phenelzine; Trifluoperazine; Verapamil | 1993 |
Calmodulin inhibitors and calcium channel blockers influence dideoxycytidine renal excretion.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Calmodulin; Kidney Tubules; Loperamide; Male; Metabolic Clearance Rate; Mice; Trifluoperazine; Verapamil; Zalcitabine | 1995 |
[The effect of adriamycin and ethidium bromide on the Ca2(+)-dependent K channel of human erythrocytes].
Topics: Antibiotics, Antineoplastic; Calcimycin; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Doxorubicin; Drug Interactions; Erythrocyte Membrane; Ethidium; Humans; In Vitro Techniques; Ionophores; Oxidation-Reduction; Potassium; Potassium Channels; Propranolol; Trifluoperazine; Verapamil | 1996 |
Effect of nifedipine, verapamil, diltiazem and trifluoperazine on acetaminophen toxicity in mice.
Topics: Acetaminophen; Animals; Aspartate Aminotransferases; Calcium Channel Blockers; Calmodulin; Cytochrome P-450 Enzyme System; Diltiazem; Glutathione; Lipid Peroxidation; Male; Mice; Microsomes, Liver; Nifedipine; Survival Rate; Trifluoperazine; Verapamil | 1995 |
Differential effects of maitotoxin on calcium entry and ciliary beating in the rabbit ciliated tracheal epithelium.
Topics: Animals; Arachidonic Acids; Biological Transport, Active; Bradykinin; Calcium; Calcium Channel Blockers; Chelating Agents; Cilia; Cyclic AMP; Cyclooxygenase Inhibitors; Egtazic Acid; Enzyme Inhibitors; Epithelium; Indomethacin; Inositol Phosphates; Ionomycin; Kinetics; Lipoxygenase Inhibitors; Marine Toxins; Masoprocol; Motion; Oxocins; Phospholipases A; Quinacrine; Rabbits; Signal Transduction; Stimulation, Chemical; Terpenes; Thapsigargin; Trachea; Trifluoperazine; Verapamil | 1995 |
Influence of trifluoperazine and verapamil on the isolated perfused rat kidney.
Topics: Animals; Antipsychotic Agents; Biomarkers; Calcium Channel Blockers; In Vitro Techniques; Kidney; Kidney Cortex; Kidney Diseases; L-Lactate Dehydrogenase; Lipid Peroxidation; Male; Perfusion; Rats; Rats, Wistar; Trifluoperazine; Verapamil; Water-Electrolyte Balance | 1996 |
The effects of adriamycin and adriamycin complexes with transitional metals on Ca(2+)-dependent K+ channels of human erythrocytes.
Topics: Calcium; Chromatography, Thin Layer; Doxorubicin; Electrochemistry; Erythrocytes; Ethidium; Humans; Hydrogen-Ion Concentration; Metals, Heavy; Models, Biological; Molecular Structure; Organometallic Compounds; Oxidation-Reduction; Potassium; Potassium Channels; Propranolol; Trifluoperazine; Verapamil | 1996 |
Effects of calcium on brazilin-induced glucose transport in isolated rat epididymal adipocytes.
Topics: Adipocytes; Animals; Benzopyrans; Biological Transport; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Cell Membrane; Dose-Response Relationship, Drug; Epididymis; Glucose; Hypoglycemic Agents; Insulin Antagonists; Male; Nifedipine; Rats; Rats, Sprague-Dawley; Trifluoperazine; Verapamil | 1997 |
Daunorubicin-induced smooth muscle contraction: involvement of Ca2+ entry mechanism.
Topics: Animals; Antibiotics, Antineoplastic; Calcium; Calcium Channel Blockers; Daunorubicin; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Potassium Chloride; Trifluoperazine; Verapamil | 1997 |
Involvement of calcium and calmodulin in Toxoplasma gondii tachyzoite invasion.
Topics: Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Carcinoma, Squamous Cell; Cytosol; Epithelial Cells; Humans; Imidazoles; Ionophores; Toxoplasma; Trifluoperazine; Tumor Cells, Cultured; Verapamil | 1997 |
Modulation of the potency of promutagens and direct acting mutagens in bacteria by inhibitors of the multidrug resistance mechanism.
Topics: Acridines; Aminacrine; Benzo(a)pyrene; Calcium Channel Blockers; Chromates; Cyclophosphamide; Dopamine Antagonists; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Multiple; Fluorenes; Indoles; Mutagenesis; Mutagenicity Tests; Mutagens; Mutation; Nicotine; Nitrogen Mustard Compounds; Quinolines; Salmonella typhimurium; Trifluoperazine; Verapamil | 1997 |
Purification and functional characterization of a low-molecular-mass Ca2+,Mg2+- and Ca2+-ATPase modulator protein from rat brain cytosol.
Topics: Animals; Body Temperature; Brain; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Circular Dichroism; Cytosol; Endoplasmic Reticulum; Enzyme Inhibitors; Goats; Male; Molecular Weight; Nerve Tissue Proteins; Rats; Sarcoplasmic Reticulum; Spectrometry, Fluorescence; Spermatozoa; Sulfhydryl Reagents; Trifluoperazine; Tryptophan; Verapamil | 1998 |
[Inhibitors of calcium-calmodulin system and hypothalamic sex differentiation in rats. Biochemical parameters].
Topics: Animals; Animals, Newborn; Antipsychotic Agents; Calcium Channel Blockers; Calmodulin; DNA; Dopamine Antagonists; Female; Haloperidol; Hypothalamus; Male; Organ Size; Ovary; Penfluridol; Pimozide; Proteins; Rats; RNA; Sex Differentiation; Testis; Trifluoperazine; Verapamil | 1997 |
Effect of calmodulin-inhibitors and verapamil on the nephrotoxicity of cadmium in rat.
Topics: Animals; Cadmium Chloride; Calcium Channel Blockers; Calmodulin; Chlorpromazine; Dopamine Antagonists; Drug Synergism; Enzyme Inhibitors; Female; Injections, Subcutaneous; Kidney Diseases; Kidney Tubules; Proteins; Proteinuria; Rats; Rats, Sprague-Dawley; Trifluoperazine; Uteroglobin; Verapamil | 1998 |
Mimosa pudica apyrase requires polysaccharide and Ca2+ for the activity.
Topics: Amylases; Apoenzymes; Apyrase; Arabinose; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Chelating Agents; Circular Dichroism; Galactans; Galactose; Guanidine; Isoenzymes; Plant Leaves; Polysaccharides; Protein Structure, Secondary; Trifluoperazine; Tryptophan; Verapamil; Xylan Endo-1,3-beta-Xylosidase; Xylosidases | 1998 |
Increase of intracellular Ca2+ and relocation of E-cadherin during experimental decompaction of mouse embryos.
Topics: Animals; Blastocyst; Cadherins; Calcium; Calmodulin; Carrier Proteins; Cell Size; Chorionic Gonadotropin; Cytochalasin D; Cytosol; Egtazic Acid; Embryonic and Fetal Development; Female; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Microfilament Proteins; Microscopy, Confocal; Morphogenesis; Morula; Trifluoperazine; Verapamil; Zona Pellucida | 1998 |
Cytoprotection and intracellular calcium.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calmodulin; Cytoprotection; Diazepam; Epoprostenol; Female; Gastric Fundus; Gastric Mucosa; Models, Biological; Pyloric Antrum; Rats; Rats, Wistar; Trifluoperazine; Verapamil | 1999 |
Effects of nifedipine, verapamil, diltiazem and trifluoperazine on the antinociceptive activity of acetaminophen.
Topics: Acetaminophen; Analgesics; Analgesics, Non-Narcotic; Animals; Calcium Channel Blockers; Cell Fractionation; Diltiazem; Dopamine Antagonists; Drug Synergism; Liver; Male; Mice; Nifedipine; Pain Measurement; Trifluoperazine; Verapamil | 2000 |
Inhibition of choline acetyltransferase by excitatory amino acids as a possible mechanism for cholinergic dysfunction in the central nervous system.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium; Cells, Cultured; Chick Embryo; Choline O-Acetyltransferase; Cycloleucine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Kainic Acid; Neurons; NG-Nitroarginine Methyl Ester; Propionates; Quisqualic Acid; Retina; Signal Transduction; Tetrodotoxin; Trifluoperazine; Verapamil | 2001 |
Antisecretory effect of loperamide in colon epithelial cells by inhibition of basolateral K+ conductance.
Topics: Antidiarrheals; Calcium Channel Blockers; Calmodulin; Carbachol; Chlorides; Cholinergic Agonists; Colforsin; Colon; Drug Evaluation, Preclinical; Enterocytes; HT29 Cells; Humans; Intestinal Mucosa; Loperamide; Naloxone; Narcotic Antagonists; Potassium Channels; Signal Transduction; Time Factors; Trifluoperazine; Verapamil | 2001 |
Real-time monitoring of P-glycoprotein activation in living cells.
Topics: 3T3 Cells; Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biosensing Techniques; Chloride-Bicarbonate Antiporters; Cyclosporine; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Induction; Enzyme Inhibitors; Extracellular Space; Humans; Hydrogen-Ion Concentration; LLC-PK1 Cells; Mice; Sodium-Hydrogen Exchangers; Substrate Specificity; Swine; Transfection; Trifluoperazine; Verapamil | 2002 |
Mitotracker green is a P-glycoprotein substrate.
Topics: Aldehydes; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Cycle; Cell Size; Cyclosporine; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescence; Fluorescent Dyes; Humans; K562 Cells; Mitochondria; Rhodamine 123; Time Factors; Trifluoperazine; Verapamil | 2003 |
Calmodulin inhibitor trifluoperazine attenuates the development and expression of morphine-induced conditioned place preference in rats.
Topics: Animals; Apomorphine; Calcium Channel Blockers; Calmodulin; Conditioning, Psychological; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Morphine; Motor Activity; Narcotics; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Trifluoperazine; Verapamil | 2004 |
Allosteric modulation of GABA(B) receptor function in human frontal cortex.
Topics: Adenylyl Cyclases; Adult; Aged; Aged, 80 and over; Calcium; Calcium Channel Blockers; Cell Membrane; Colforsin; Diphenhydramine; Dopamine Antagonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Histamine H1 Antagonists; Humans; Male; Middle Aged; Phenols; Prefrontal Cortex; Receptors, GABA-B; Trifluoperazine; Verapamil | 2005 |
[Construction and expression of anti-CD3/ anti-Pgp Diabody].
Topics: Animals; Antibodies, Monoclonal; Antibody Specificity; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; CD3 Complex; Chromatography, Gel; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Jurkat Cells; K562 Cells; Mice; Polymerase Chain Reaction; Radioimmunoassay; Trifluoperazine; Verapamil | 2003 |
Comment on 'Topical verapamil HCL, topical trifluoroperazine, and topical magnesium sulfate for the treatment of Peyronie's disease--a placebo-controlled pilot study'.
Topics: Administration, Topical; Adult; Double-Blind Method; Humans; Magnesium Sulfate; Male; Penile Erection; Penile Induration; Research Design; Trifluoperazine; Verapamil | 2007 |
Role of allopurinol, verapamil, dexamethasone and trifluoperazine as prophylactic agents in intestinal ischemia-reperfusion.
Topics: Allopurinol; Animals; Dexamethasone; Intestine, Small; Male; Rats; Rats, Wistar; Reperfusion Injury; Trifluoperazine; Verapamil | 2008 |
Effects of the mycotoxin destruxin A on Locusta migratoria visceral muscles.
Topics: Animals; Calcium Channel Blockers; Calcium Signaling; Cell Membrane; Cobalt; Depsipeptides; Dose-Response Relationship, Drug; Drug Antagonism; Female; Locusta migratoria; Lower Gastrointestinal Tract; Muscle Contraction; Muscle, Smooth; Mycotoxins; Nifedipine; Oviducts; Trifluoperazine; Verapamil | 2010 |