verapamil and tetracaine

verapamil has been researched along with tetracaine in 44 studies

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-199030 (68.18)18.7374
1990's2 (4.55)18.2507
2000's7 (15.91)29.6817
2010's5 (11.36)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Alvarez-Pedraglio, A; Colmenarejo, G; Lavandera, JL1
Bacsó, Z; Cianfriglia, M; Fenyvesi, F; Goda, K; Kappelmayer, J; Lustyik, G; Nagy, H; Szabó, G; Szilasi, M1
Johans, C; Kinnunen, PK; Söderlund, T; Suomalainen, P1
Caron, G; Ermondi, G1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Ahman, M; Holmén, AG; Wan, H1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Gozalbes, R; Pineda-Lucena, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Bellman, K; Knegtel, RM; Settimo, L1
Brouillette, WJ; Brown, GB; Zha, C1
Izumi, T; Norton, TR; Seriguchi, DG; Shibata, S1
Papadimituiou, JM; Sforcina, D1
Haslam, RJ; Lynham, JA1
Hirai, M; Kawashima, Y; Shima, S1
Halperin, ML; Hau, L; Taylor, WM1
Freer, RJ1
Davis, BB; Zenser, TV1
García, AG; Horga, JF; Pascual, R; Sánchez-García, P1
Arqueros, L; Daniels, AJ1
Hirai, H; Natori, S; Sekimizu, K1
el Motal, SM; Pian-Smith, MC; Sharp, GW1
Kato, H; Takata, Y2
Enyeart, JJ; Hinkle, PM; Phillips, WJ1
Chen, IJ; Teng, CM; Yeh, HI1
Kontani, H; Koshiura, R1
Lang, CH; McDonough, KH; Spitzer, JJ1
Balzer, H1
Hirai, M; Komoriyama, K; Kouyama, H; Shima, S1
Ehlert, FJ; Fairhurst, AS; Whittaker, ML1
Markosian, RA; Suvorov, AV1
Ohizumi, Y; Takahashi, M; Yasumoto, T1
Paleos, GA; Powers, RD2
Ueda, T1
Aoyama, T; Ono, H; Sato, T1
Kawai, K; Ogata, E1
Boadle-Biber, MC1
Conti, GT; Falkenstein, D; Figueiredo, JF; Ramos, OL; Sigulem, D1
Minakuchi, R; Mori, T; Nishizuka, Y; Takai, Y; Yu, B1
Iwasaki, H; Kawamata, M; Namiki, A; Omote, K; Satoh, O1
Bezstarosti, K; Christoffels, VM; de Boer, PA; Fiolet, JW; Hagoort, J; Lamers, JM; Moorman, AF; Schumacher, CA; van den Hoff, MJ; Wagenaar, GT; Wuytack, F1

Other Studies

44 other study(ies) available for verapamil and tetracaine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Cheminformatic models to predict binding affinities to human serum albumin.
    Journal of medicinal chemistry, 2001, Dec-06, Volume: 44, Issue:25

    Topics: Adrenergic beta-Antagonists; Antidepressive Agents, Tricyclic; Chromatography, Affinity; Cyclooxygenase Inhibitors; Databases, Factual; Humans; Hydrophobic and Hydrophilic Interactions; Penicillins; Pharmaceutical Preparations; Protein Binding; Quantitative Structure-Activity Relationship; Reproducibility of Results; Serum Albumin; Steroids

2001
Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.
    Biochemical and biophysical research communications, 2004, Mar-19, Volume: 315, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Anti-Bacterial Agents; Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Calcium Channel Blockers; Cyclosporine; Detergents; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Humans; Ivermectin; Mice; NIH 3T3 Cells; Substrate Specificity

2004
Surface activity profiling of drugs applied to the prediction of blood-brain barrier permeability.
    Journal of medicinal chemistry, 2004, Mar-25, Volume: 47, Issue:7

    Topics: Blood-Brain Barrier; Lipid Bilayers; Micelles; Permeability; Pharmaceutical Preparations; Structure-Activity Relationship; Surface Properties

2004
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
    Journal of medicinal chemistry, 2009, Mar-26, Volume: 52, Issue:6

    Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
QSAR-based solubility model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2010, Oct-01, Volume: 18, Issue:19

    Topics: Databases, Factual; Models, Molecular; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Solubility; Water

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
Further studies on the positive inotropic effect of the polypeptide anthopleurin-A from a sea anemone.
    The Journal of pharmacology and experimental therapeutics, 1978, Volume: 205, Issue:3

    Topics: Cnidaria; Drug Interactions; Intercellular Signaling Peptides and Proteins; Lanthanum; Myocardial Contraction; Nifedipine; Peptides; Ryanodine; Sea Anemones; Stimulation, Chemical; Tetracaine; Tetrodotoxin; Verapamil

1978
The effects of drugs on monocytic fusion in vivo.
    Experimental cell research, 1975, Mar-15, Volume: 91, Issue:2

    Topics: Adenosine Triphosphatases; Animals; Calcium; Cell Fusion; Cell Membrane; Cortisone; Cyclic AMP; Diphenhydramine; Edetic Acid; Glucagon; Insulin; Isoproterenol; Lidocaine; Lysosomes; Male; Mice; Mice, Inbred C57BL; Monocytes; Ouabain; Pyrilamine; Tetracaine; Trifluoperazine; Verapamil

1975
Relationship between phosphorylation of blood platelet proteins and secretion of platelet granule constituents II. Effects of different inhibitors.
    Thrombosis research, 1978, Volume: 12, Issue:4

    Topics: Blood Platelets; Blood Proteins; Bucladesine; Collagen; Cytochalasin B; Ethylmaleimide; Humans; In Vitro Techniques; Indomethacin; Prostaglandins E; Tetracaine; Verapamil

1978
Studies on cyclic nucleotides in the adrenal gland. IX. Effects of ACTH on cyclic AMP and steroid production by the zona fasciculata-reticularis of the adrenal cortex.
    Acta endocrinologica, 1979, Volume: 90, Issue:1

    Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Animals; Calcium; Corticosterone; Cyclic AMP; Lanthanum; Male; Rats; Tetracaine; Verapamil

1979
Stimulation of glucose transport in rat adipocytes by calcium.
    Canadian journal of biochemistry, 1979, Volume: 57, Issue:6

    Topics: Adipose Tissue; Animals; Biological Transport, Active; Calcium; Cobalt; Cyclic AMP; Glucose; Male; Methylphenazonium Methosulfate; Nickel; Procaine; Rats; Stimulation, Chemical; Tetracaine; Verapamil

1979
Calcium and angiotensin tachyphylaxis in rat uterine smooth muscle.
    The American journal of physiology, 1975, Volume: 228, Issue:5

    Topics: Acetylcholine; Angiotensin II; Animals; Aorta; Calcium; Diethylstilbestrol; Dose-Response Relationship, Drug; Edetic Acid; Female; Hydrogen-Ion Concentration; Ileum; In Vitro Techniques; Lanthanum; Manganese; Mice; Models, Biological; Muscle Contraction; Muscle, Smooth; Myometrium; Norepinephrine; Proadifen; Rabbits; Rats; Tachyphylaxis; Tetracaine; Uterus; Verapamil

1975
Effects of calcium on prostaglandin E2 synthesis by rat inner medullary slices.
    The American journal of physiology, 1978, Volume: 235, Issue:3

    Topics: Animals; Calcimycin; Calcium; In Vitro Techniques; Kidney Medulla; Magnesium; Perfusion; Prostaglandins E; Rats; Tetracaine; Verapamil

1978
Release of noradrenaline by the ionophore X537A from normal and reserpinized guinea-pig atrium.
    Naunyn-Schmiedeberg's archives of pharmacology, 1977, Volume: 301, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Calcium; Drug Interactions; Guinea Pigs; In Vitro Techniques; Lasalocid; Male; Myocardium; Norepinephrine; Perfusion; Reserpine; Ruthenium Red; Ryanodine; Tetracaine; Time Factors; Verapamil

1977
Analysis of the inhibitory effect of verapamil on adrenal medullary secretion.
    Life sciences, 1978, Dec-11, Volume: 23, Issue:24

    Topics: Acetylcholine; Adrenal Medulla; Animals; Barium; Calcium; Catecholamines; Cattle; Depression, Chemical; Drug Interactions; In Vitro Techniques; Tetracaine; Verapamil

1978
Inhibitory action of phospholipid-interacting drugs on transcription initiation in a nuclear extract of Ehrlich ascites tumor cells.
    Biochimica et biophysica acta, 1991, Feb-16, Volume: 1088, Issue:2

    Topics: Adenoviruses, Human; Animals; Carcinoma, Ehrlich Tumor; Cell Nucleus; Chlorpromazine; HeLa Cells; Humans; Imipramine; Kinetics; Mice; Phospholipases A; Phospholipases A2; Phospholipids; Promoter Regions, Genetic; RNA Polymerase II; Tetracaine; Transcription Factors; Transcription, Genetic; Verapamil

1991
Effects of tetracaine on insulin release and calcium handling by rat pancreatic islets.
    The American journal of physiology, 1987, Volume: 252, Issue:6 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium; Drug Synergism; Gallic Acid; Glucose; Insulin; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Tetracaine; Verapamil

1987
Differential effects of verapamil, nicardipine and diltiazem on Ca2+-dependent and Ca2+-independent noradrenaline release and contraction in isolated canine saphenous veins.
    Pharmacology, 1988, Volume: 37, Issue:1

    Topics: Animals; Calcium; Diltiazem; Dogs; Female; In Vitro Techniques; Ion Channels; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Norepinephrine; Saphenous Vein; Tetracaine; Tetraethylammonium Compounds; Verapamil

1988
Pituitary thyrotropin-releasing hormone receptors: local anesthetic effects on binding and responses.
    Molecular endocrinology (Baltimore, Md.), 1989, Volume: 3, Issue:9

    Topics: Anesthetics, Local; Animals; Benzocaine; Chlordiazepoxide; Chlorpromazine; Dibucaine; Hydrogen-Ion Concentration; Imipramine; Lidocaine; Pituitary Gland; Procaine; Prolactin; Propranolol; Rats; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Tetracaine; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil

1989
Differential effects of Ca antagonists on the noradrenaline release and contraction evoked by nerve stimulation in the presence of 4-aminopyridine.
    British journal of pharmacology, 1987, Volume: 90, Issue:1

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Calcium Channel Blockers; Diltiazem; Dogs; Electric Stimulation; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Norepinephrine; Salicylates; Salicylic Acid; Stereoisomerism; Tetracaine; Tetrodotoxin; Verapamil

1987
Cyclooxygenase--independent pathway of phospholipase activation in carrageenan--induced platelet aggregation.
    Thrombosis research, 1987, Jan-01, Volume: 45, Issue:1

    Topics: Animals; Calcium; Carrageenan; Chlorpromazine; Drug Synergism; Enzyme Activation; Indomethacin; Nitroprusside; Phospholipases; Platelet Aggregation; Prostaglandin-Endoperoxide Synthases; Rabbits; Tetracaine; Verapamil

1987
The effects of tetrodotoxin, papaverine and verapamil on the increase in the rate of spontaneous afferent discharges induced by local anesthetics from the pulmonary mechanoreceptors of the bullfrog.
    Japanese journal of pharmacology, 1985, Volume: 37, Issue:1

    Topics: Aconitine; Action Potentials; Anesthetics, Local; Animals; Dibucaine; In Vitro Techniques; Lung; Mechanoreceptors; Neurons, Afferent; Papaverine; Procaine; Rana catesbeiana; Tetracaine; Tetrodotoxin; Verapamil

1985
Effect of cardiotropic agents on the myocardial dysfunction of hyperdynamic sepsis.
    Circulatory shock, 1985, Volume: 17, Issue:1

    Topics: Animals; Blood Pressure; Calcium; Cardiac Output; Cardiovascular Agents; Heart; In Vitro Techniques; Male; Myocardial Contraction; Ouabain; Rats; Rats, Inbred Strains; Sepsis; Tetracaine; Verapamil

1985
The effect of quinidine and drugs with quinidine-like action (propranolol, verapamil and tetracaine) on the calcium transport system in isolated sarcoplasmic reticulum vesicles of rabbit skeletal muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1972, Volume: 274, Issue:3

    Topics: Adenosine Triphosphate; Animals; Binding Sites; Biological Transport; Calcium; Membranes; Muscles; Phospholipases; Propranolol; Quinidine; Rabbits; Sarcoplasmic Reticulum; Tetracaine; Verapamil

1972
beta-Adrenergic stimulation of the adenosine 3',5'-monophosphate system regulated by cholinergic stimuli in the prostate.
    Biochemical pharmacology, 1983, Feb-01, Volume: 32, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Animals; Atropine; Calcimycin; Calcium; Cell Membrane; Cyclic AMP; Hexamethonium; Hexamethonium Compounds; Isoproterenol; Male; Parasympathetic Nervous System; Prostate; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Tetracaine; Theophylline; Verapamil

1983
Interactions of D600 (methoxyverapamil) and local anesthetics with rat brain alpha-adrenergic and muscarinic receptors.
    Biochemical pharmacology, 1980, Volume: 29, Issue:2

    Topics: Anesthetics, Local; Animals; Gallopamil; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Lidocaine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Muscarinic; Tetracaine; Verapamil

1980
[Certain mechanisms of the effect of EDTA on thrombocyte aggregation].
    Biulleten' eksperimental'noi biologii i meditsiny, 1981, Volume: 91, Issue:5

    Topics: Blood Platelets; Bucladesine; Calcium; Drug Interactions; Edetic Acid; Egtazic Acid; Humans; Platelet Aggregation; Tetracaine; Theophylline; Verapamil

1981
Maitotoxin, a Ca2+ channel activator candidate.
    The Journal of biological chemistry, 1982, Jul-10, Volume: 257, Issue:13

    Topics: Adrenal Gland Neoplasms; Animals; Calcium; Cell Line; Ion Channels; Kinetics; Manganese; Marine Toxins; Neoplasms, Experimental; Oxocins; Pheochromocytoma; Rats; Tetracaine; Tetrodotoxin; Verapamil

1982
Combined effects of calcium and dibutyryl cyclic AMP on germinal vesicle breakdown in the mouse oocyte.
    Journal of reproduction and fertility, 1982, Volume: 66, Issue:1

    Topics: Animals; Bucladesine; Calcimycin; Calcium; Cells, Cultured; Female; Magnesium; Meiosis; Mice; Mice, Inbred Strains; Oocytes; Ovum; Tetracaine; Verapamil

1982
Na+-Ca2+ exchange activity in rabbit lymphocyte plasma membranes.
    Biochimica et biophysica acta, 1983, Oct-12, Volume: 734, Issue:2

    Topics: Animals; Calcium; Cell Membrane; Kinetics; Lanthanum; Lymphocytes; Rabbits; Sodium; Tetracaine; Time Factors; Verapamil

1983
Mechanisms of slow contracture induced by potassium and caffeine in skeletal muscle of the dog.
    Japanese journal of pharmacology, 1984, Volume: 34, Issue:2

    Topics: Animals; Caffeine; Calcium Chloride; Chlorides; Diltiazem; Dogs; Kinetics; Manganese; Manganese Compounds; Muscle Contraction; Potassium; Potassium Chloride; Tetracaine; Verapamil

1984
The role of Ca++ in sulfation factor activity on embryonic chick cartilage.
    Metabolism: clinical and experimental, 1981, Volume: 30, Issue:8

    Topics: Animals; Blood; Calcimycin; Calcium; Cartilage; Chick Embryo; Dose-Response Relationship, Drug; Humans; Sodium; Somatomedins; Sulfates; Tetracaine; Verapamil

1981
Further studies on the role of calcium in the depolarization-induced activation of tryptophan hydroxylase. Effect of verapamil, Tetracaine, haloperidol and fluphenazine.
    Biochemical pharmacology, 1982, Aug-01, Volume: 31, Issue:15

    Topics: Animals; Brain Stem; Buffers; Calcium; Enzyme Activation; Fluphenazine; Haloperidol; Male; Membrane Potentials; Potassium; Rats; Rats, Inbred Strains; Tetracaine; Tryptophan Hydroxylase; Verapamil

1982
Tetracaine, procaine and verapamil inhibition of fluid absorption in isolated perfused rabbit proximal convoluted tubules.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1982, Volume: 15, Issue:4-5

    Topics: Absorption; Animals; Calcium; Kidney Tubules, Proximal; Male; Perfusion; Procaine; Rabbits; Tetracaine; Verapamil; Water-Electrolyte Balance

1982
The effect of calcium on the first meiotic division of the mammalian oocyte.
    The Journal of experimental zoology, 1981, Volume: 217, Issue:3

    Topics: Animals; Calcium; Culture Media; Female; Hydrogen-Ion Concentration; Lanthanum; Meiosis; Mice; Oocytes; Ovum; Tetracaine; Verapamil

1981
Inhibitory action of chlorpromazine, dibucaine, and other phospholipid-interacting drugs on calcium-activated, phospholipid-dependent protein kinase.
    The Journal of biological chemistry, 1980, Sep-25, Volume: 255, Issue:18

    Topics: Animals; Brain; Calcium; Chlorpromazine; Cytosol; Dibucaine; Enzyme Activation; Imipramine; Kinetics; Phentolamine; Phospholipids; Protein Kinases; Rats; Tetracaine; Verapamil

1980
Effects of verapamil on spinal anesthesia with local anesthetics.
    Anesthesia and analgesia, 1995, Volume: 80, Issue:3

    Topics: Anesthesia, Spinal; Anesthetics, Local; Animals; Dose-Response Relationship, Drug; Drug Synergism; Injections, Spinal; Lidocaine; Male; Motor Activity; Pain Threshold; Rats; Rats, Sprague-Dawley; Reaction Time; Tetracaine; Verapamil

1995
Presence of functional sarcoplasmic reticulum in the developing heart and its confinement to chamber myocardium.
    Developmental biology, 2000, Jul-15, Volume: 223, Issue:2

    Topics: Animals; Calcium Signaling; Calcium-Transporting ATPases; Chick Embryo; Heart; Heart Atria; Heart Ventricles; Humans; Image Processing, Computer-Assisted; Immunohistochemistry; Models, Structural; Morphogenesis; Myocardium; Rats; Ryanodine; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Tetracaine; Tissue Distribution; Verapamil

2000