verapamil and sirolimus

verapamil has been researched along with sirolimus in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (13.33)18.2507
2000's9 (60.00)29.6817
2010's4 (26.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bacsó, Z; Cianfriglia, M; Fenyvesi, F; Goda, K; Kappelmayer, J; Lustyik, G; Nagy, H; Szabó, G; Szilasi, M1
Cai, W; Hao, Y; Hu, P; Ma, D; Pan, H; Xie, X; Yu, AD; Yu, J; Yuan, J; Zhang, L; Zhu, H1
Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Lay, RH; Medh, RD; Schmidt, TJ1
Crowe, A; Lemaire, M1
Kato, K; Li, ST; Mikoshiba, K1
Allison, MJ; Beyer, D; Bizot, MN; Jiang, Q; Kovarik, JM; Schmouder, RL1
Anglicheau, D; Beaune, P; Cassinat, B; Legendre, C; Marquet, P; Méria, P; Pallet, N; Rabant, M; Thervet, E1
Ambudkar, SV; Calcagno, AM; Gottesman, MM; Kim, IW; Kimchi-Sarfaty, C; Oh, JM; Sauna, ZE1
Heimberg, H; Ling, Z; Pipeleers, D; Wang, Q1
Rund, D1
Campesi, I; Capobianco, G; Dessole, S; Fois, M; Franconi, F; Montella, A; Occhioni, S1

Reviews

1 review(s) available for verapamil and sirolimus

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for verapamil and sirolimus

ArticleYear
Pharmacokinetic interaction between verapamil and everolimus in healthy subjects.
    British journal of clinical pharmacology, 2005, Volume: 60, Issue:4

    Topics: Analysis of Variance; Calcium Channel Agonists; Cross-Over Studies; Drug Interactions; Enzyme Inhibitors; Everolimus; Humans; Immunosuppressive Agents; Sirolimus; Verapamil

2005

Other Studies

13 other study(ies) available for verapamil and sirolimus

ArticleYear
Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.
    Biochemical and biophysical research communications, 2004, Mar-19, Volume: 315, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Anti-Bacterial Agents; Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Calcium Channel Blockers; Cyclosporine; Detergents; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Humans; Ivermectin; Mice; NIH 3T3 Cells; Substrate Specificity

2004
Small molecule regulators of autophagy identified by an image-based high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Nov-27, Volume: 104, Issue:48

    Topics: Autophagy; Calcium Channel Blockers; Cell Line, Tumor; Drug Evaluation, Preclinical; Fluspirilene; Glioblastoma; Green Fluorescent Proteins; Humans; Intracellular Membranes; Loperamide; Microtubule-Associated Proteins; Mycotoxins; Peptides; Phagosomes; Phosphatidylinositol Phosphates; Pimozide; Protein Kinases; Recombinant Fusion Proteins; Sirolimus; Small Molecule Libraries; TOR Serine-Threonine Kinases; Trifluoperazine; Zinc Fingers

2007
Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
    Nature chemical biology, 2008, Volume: 4, Issue:5

    Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Agonist-specific modulation of glucocorticoid receptor-mediated transcription by immunosuppressants.
    Molecular and cellular endocrinology, 1998, Mar-16, Volume: 138, Issue:1-2

    Topics: Animals; Corticosterone; Cortodoxone; Cyclosporine; Desoxycorticosterone; Dexamethasone; Genes, Reporter; Glucocorticoids; Hydrocortisone; Immunosuppressive Agents; L Cells; Luciferases; Mice; Polyenes; Quinidine; Receptors, Glucocorticoid; Recombinant Fusion Proteins; Sirolimus; Tacrolimus; Transcription, Genetic; Transfection; Triamcinolone Acetonide; Verapamil

1998
In vitro and in situ absorption of SDZ-RAD using a human intestinal cell line (Caco-2) and a single pass perfusion model in rats: comparison with rapamycin.
    Pharmaceutical research, 1998, Volume: 15, Issue:11

    Topics: Animals; Caco-2 Cells; Everolimus; Humans; Immunosuppressive Agents; Intestinal Absorption; Mannitol; Propranolol; Rats; Rats, Wistar; Sirolimus; Verapamil

1998
High Ca(2+)/low Mg(2+) solution induces long-term depression in rat CA1 pyramidal neurons.
    Neuroscience letters, 2000, Apr-07, Volume: 283, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Benzoates; Calcium; Calcium Channel Blockers; Electric Stimulation; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; In Vitro Techniques; Magnesium; Neuronal Plasticity; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Sirolimus; Solutions; Tacrolimus; Verapamil

2000
Role of P-glycoprotein in cyclosporine cytotoxicity in the cyclosporine-sirolimus interaction.
    Kidney international, 2006, Volume: 70, Issue:6

    Topics: Acetanilides; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Culture Techniques; Cell Survival; Cells, Cultured; Cyclosporine; Cyclosporins; Dose-Response Relationship, Drug; Drug Interactions; Epithelial Cells; Fluorescent Dyes; Humans; Immunosuppressive Agents; Kidney; Pyrroles; Quinine; Quinolines; Rhodamines; Sirolimus; Verapamil

2006
A "silent" polymorphism in the MDR1 gene changes substrate specificity.
    Science (New York, N.Y.), 2007, Jan-26, Volume: 315, Issue:5811

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Cell Membrane; Chlorocebus aethiops; Codon; Cyclosporine; Genes, MDR; Haplotypes; HeLa Cells; Humans; Mutagenesis, Site-Directed; Polymorphism, Single Nucleotide; Protein Biosynthesis; Protein Conformation; Protein Folding; Protein Structure, Tertiary; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Sirolimus; Substrate Specificity; Transfection; Verapamil

2007
Glibenclamide activates translation in rat pancreatic beta cells through calcium-dependent mTOR, PKA and MEK signalling pathways.
    Diabetologia, 2008, Volume: 51, Issue:7

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Extracellular Signal-Regulated MAP Kinases; Glyburide; Hypoglycemic Agents; Immunosuppressive Agents; Insulin-Secreting Cells; Male; Mitogen-Activated Protein Kinases; Protein Biosynthesis; Rats; Rats, Wistar; Sirolimus; Transcription Factors; Verapamil

2008
'Rapping' on the door of drug resistance.
    Leukemia & lymphoma, 2009, Volume: 50, Issue:7

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; CHO Cells; Cricetinae; Cricetulus; Drug Resistance, Neoplasm; Humans; Macrolides; Neoplasms; Sirolimus; Verapamil

2009
Sex-specific pharmacological modulation of autophagic process in human umbilical artery smooth muscle cells.
    Pharmacological research, 2016, Volume: 113, Issue:Pt A

    Topics: Autophagy; Beclin-1; Cells, Cultured; Female; Humans; Infant, Newborn; Male; Microtubule-Associated Proteins; Myocytes, Smooth Muscle; Sex Characteristics; Sirolimus; TOR Serine-Threonine Kinases; Umbilical Arteries; Verapamil

2016