verapamil and s 9788

verapamil has been researched along with s 9788 in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's25 (96.15)18.2507
2000's1 (3.85)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Atassi, G; Dhainaut, A; Kraus-Berthier, L; Léonce, S; Pierré, A; Prost, JF; Régnier, G1
Atassi, G; Dhainaut, A; Guilbaud, N; Kraus-Berthier, L; Leonce, S; Pierre, A; Regnier, G; Tizot, A1
Faussat, AM; Kühnel, JM; Marie, JP; Perrot, JY; Schwaller, MA1
Collett, A; Hallifax, D; Tanianis-Hughes, J; Warhurst, G1
Anstett, M; Atassi, G; Bizzari, JP; Genton, A; Léonce, S; Pérez, V; Pierré, A1
Berlion, M; Dieterlen, A; Lucas, C; Marchal, S; Merlin, JL; Poullain, MG; Ramacci, C; Schultz, G1
Bennis, S; Robert, J1
Lucas, C; Marchal, S; Merlin, JL; Paraire, M; Poullain, MG; Ramacci, C1
Gibassier, J; Leclech, G; Lucas, C; Massart, C; Pourquier, P; Raoul, M; Robert, J1
Berlion, M; Bizzari, JP; Calvo, F; Haddad, P; Lucas, C; Soudon, J1
Berlion, M; Bizzari, JP; Desplaces, A; Dufer, J; Joly, P; Millot-Broglio, C; Oum'Hamed, Z1
Guerci, A; Guerci, O; Humbert, JC; Marchal, S; Merlin, JL; Missoum, N; Ramacci, C; Tsuruo, T1
Berlion, M; Kernaleguen, D; Le Bot, MA; Riché, C; Robert, J1
de Vries, EG; Hill, BT; Hosking, LK; Mulder, NH; van der Graaf, WT; Whelan, RD1
Anstett, M; Atassi, G; Léonce, S; Pérez, V; Pierré, A; Prost, JF1
Berlion, M; Bizzari, JP; Canal, P; Julia, AM; Lucas, C; Milano, G; Robert, J; Roché, H1
Hill, BT; Hosking, LK1
Berlion, M; Kernaleguen, D; Le Bot, MA; Riché, C; Simon, I1
Chapey, C; Hu, YP; Robert, J1
Atassi, G; Dubois, J; Hanocq, M; Tassin, JP1
Belhoussine, R; Manfait, M; Morjani, H1
Cayre, A; Finat-Duclos, F; Maublant, J; Moins, N; Verrelle, P2
Belhoussine, R; Lahlil, R; Manfait, M; Morjani, H1
Buée-Scherrer, V; Cecchelli, R; Dehouck, MP; Descamps, L; Duhem, C; Fenart, L; Poullain, MG1
Belhoussine, R; Manfait, M; Millot, JM; Morjani, H; Sharonov, S1

Reviews

1 review(s) available for verapamil and s 9788

ArticleYear
[Effect of quinine on the multiple drug resistance and intracellular distribution of pirarubicin in LR73 tumor cells: a comparative study with verapamil and S9788 by confocal laser microspectrofluorometry].
    Bulletin du cancer, 1997, Volume: 84, Issue:4

    Topics: Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cricetinae; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; In Vitro Techniques; Microscopy, Confocal; Piperidines; Quinine; Spectrometry, Fluorescence; Triazines; Tumor Cells, Cultured; Verapamil

1997

Trials

1 trial(s) available for verapamil and s 9788

ArticleYear
In vitro activity of S 9788 on a multidrug-resistant leukemic cell line and on normal hematopoietic cells-reversal of multidrug resistance by sera from phase I-treated patients.
    Cancer chemotherapy and pharmacology, 1995, Volume: 36, Issue:3

    Topics: Antineoplastic Agents; Bone Marrow Cells; Cell Division; Cell Line; Cell Survival; Culture Media; Doxorubicin; Drug Resistance, Multiple; Drug Synergism; Hematopoietic Stem Cells; Humans; Leukemia, T-Cell; Neoplasms; Phenotype; Piperidines; Reference Values; Triazines; Tumor Cells, Cultured; Verapamil; Vinblastine

1995

Other Studies

24 other study(ies) available for verapamil and s 9788

ArticleYear
New triazine derivatives as potent modulators of multidrug resistance.
    Journal of medicinal chemistry, 1992, Jun-26, Volume: 35, Issue:13

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Cell Survival; Cricetinae; Cricetulus; Drug Resistance; Drug Synergism; Leukemia P388; Lung; Membrane Glycoproteins; Structure-Activity Relationship; Triazines; Tumor Cells, Cultured

1992
New purines and purine analogs as modulators of multidrug resistance.
    Journal of medicinal chemistry, 1996, Sep-27, Volume: 39, Issue:20

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channels; Doxorubicin; Drug Resistance, Multiple; Female; Leukemia P388; Leukemia, Experimental; Mice; Molecular Structure; Neoplasm Transplantation; Piperidines; Purines; Structure-Activity Relationship; Triazines; Tumor Cells, Cultured; Vincristine

1996
Functional assay of multidrug resistant cells using JC-1, a carbocyanine fluorescent probe.
    Leukemia, 1997, Volume: 11, Issue:7

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Carbocyanines; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Humans; Rhodamine 123; Rhodamines; Spectrometry, Fluorescence; Tumor Cells, Cultured

1997
Predicting P-glycoprotein effects on oral absorption: correlation of transport in Caco-2 with drug pharmacokinetics in wild-type and mdr1a(-/-) mice in vivo.
    Pharmaceutical research, 2004, Volume: 21, Issue:5

    Topics: Administration, Oral; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport, Active; Caco-2 Cells; Cell Membrane Permeability; Humans; Intestinal Absorption; Mice; Mice, Knockout; Pharmacokinetics; Spectrometry, Mass, Electrospray Ionization

2004
Effects of a new triazinoaminopiperidine derivative on adriamycin accumulation and retention in cells displaying P-glycoprotein-mediated multidrug resistance.
    Biochemical pharmacology, 1992, Nov-03, Volume: 44, Issue:9

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Carcinoma, Squamous Cell; Cell Cycle; Cell Membrane; Cells, Cultured; Colonic Neoplasms; Cricetinae; Cricetulus; Dihydropyridines; Doxorubicin; Drug Resistance; Flow Cytometry; Fluorescence; Humans; Kinetics; Leukemia P388; Leukemia, Myeloid, Acute; Lung; Membrane Glycoproteins; Mice; Piperidines; Sensitivity and Specificity; Triazines; Tritium; Tumor Cells, Cultured; Verapamil

1992
Influence of S9788, a new modulator of multidrug resistance, on the cellular accumulation and subcellular distribution of daunorubicin in P-glycoprotein-expressing MCF7 human breast adenocarcinoma cells.
    Cytometry, 1995, Aug-01, Volume: 20, Issue:4

    Topics: Adenocarcinoma; ATP Binding Cassette Transporter, Subfamily B, Member 1; Breast Neoplasms; Cell Nucleus; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Female; Flow Cytometry; Humans; Neoplasm Proteins; Piperidines; Subcellular Fractions; Triazines; Tumor Cells, Cultured; Verapamil

1995
[Difference between the effects of S9788, verapamil and quinine on the reversion of multidrug resistance in two human tumor cell lines].
    Bulletin du cancer, 1994, Volume: 81, Issue:10

    Topics: Antineoplastic Agents; Breast Neoplasms; Cell Death; Doxorubicin; Drug Resistance, Multiple; Humans; Leukemia, Erythroblastic, Acute; Piperidines; Quinine; Triazines; Tumor Cells, Cultured; Verapamil

1994
[Effect of the modality of exposure on the action of S9788 on the modulation of multidrug resistance of human tumor cell lines].
    Bulletin du cancer, 1994, Volume: 81, Issue:10

    Topics: Adenocarcinoma; Antineoplastic Agents; Breast Neoplasms; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Humans; Leukemia; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1994
Cyclosporin A, verapamil and S9788 reverse doxorubicin resistance in a human medullary thyroid carcinoma cell line.
    Anti-cancer drugs, 1995, Volume: 6, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carcinoma, Medullary; Cyclosporine; Doxorubicin; Drug Resistance, Multiple; Drug Synergism; Glutathione; Glutathione Transferase; Humans; Neoplasm Proteins; Piperidines; Polymerase Chain Reaction; RNA, Messenger; RNA, Neoplasm; Thyroid Neoplasms; Triazines; Verapamil

1995
[Quantitative cytological study of the activity of a new resistance modulator, S 9788, on human leukemic cells using multiparametric image analysis].
    Bulletin du cancer, 1994, Volume: 81, Issue:3

    Topics: Animals; Antineoplastic Agents; Cytophotometry; DNA, Neoplasm; Drug Resistance, Multiple; Humans; Image Processing, Computer-Assisted; In Vitro Techniques; Mice; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil; Vinblastine

1994
Comparative evaluation of S9788, verapamil, and cyclosporine A in K562 human leukemia cell lines and in P-glycoprotein-expressing samples from patients with hematologic malignancies.
    Blood, 1994, Jul-01, Volume: 84, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cyclosporine; Doxorubicin; Drug Resistance; Female; Humans; Leukemia; Male; Membrane Glycoproteins; Middle Aged; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1994
Modulation of anthracycline accumulation and metabolism in rat hepatocytes in culture by three revertants of multidrug resistance.
    Cancer chemotherapy and pharmacology, 1994, Volume: 35, Issue:1

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cells, Cultured; Cyclosporine; Drug Resistance, Multiple; Liver; Male; Piperidines; Rats; Rats, Sprague-Dawley; Triazines; Up-Regulation; Verapamil

1994
Evaluation of S9788 as a potential modulator of drug resistance against human tumour sublines expressing differing resistance mechanisms in vitro.
    International journal of cancer, 1993, Sep-09, Volume: 55, Issue:2

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Doxorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Membrane Glycoproteins; Molecular Structure; Neoplasms; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil; Vinblastine; Vincristine

1993
[In vitro characterization of S9788, a new modulator of multidrug resistance].
    Bulletin du cancer, 1993, Volume: 80, Issue:4

    Topics: Animals; Antineoplastic Agents; Cell Cycle; Drug Resistance; Drug Screening Assays, Antitumor; Humans; In Vitro Techniques; Mice; Neoplasms; Neoplasms, Experimental; Phenotype; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1993
Multidrug resistance circumvention by a new triazinoaminopiperidine derivative S9788 in vitro: definition of the optimal schedule and comparison with verapamil.
    British journal of cancer, 1994, Volume: 69, Issue:5

    Topics: Antineoplastic Agents; Breast Neoplasms; Doxorubicin; Drug Resistance; Female; Humans; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1994
Differential effectiveness of a range of novel drug-resistance modulators, relative to verapamil, in influencing vinblastine or teniposide cytotoxicity in human lymphoblastoid CCRF-CEM sublines expressing classic or atypical multidrug resistance.
    Cancer chemotherapy and pharmacology, 1994, Volume: 33, Issue:4

    Topics: Cyclosporine; Dihydropyridines; Dose-Response Relationship, Drug; Drug Resistance; Drug Screening Assays, Antitumor; Flunarizine; Humans; Leukemia, T-Cell; Piperidines; Quinidine; Teniposide; Triazines; Tumor Cells, Cultured; Verapamil; Vinblastine

1994
[Effect of S9788, cyclosporin A and verapamil on intracellular accumulation of doxorubicin, daunorubicin and daunorubicinol in primary rat hepatocyte culture].
    Annales de biologie clinique, 1996, Volume: 54, Issue:1

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Cyclosporine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Liver; Piperidines; Rats; Rats, Sprague-Dawley; Triazines; Verapamil

1996
Relationship between the inhibition of azidopine binding to P-glycoprotein by MDR modulators and their efficiency in restoring doxorubicin intracellular accumulation.
    Cancer letters, 1996, Dec-03, Volume: 109, Issue:1-2

    Topics: Affinity Labels; Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cyclosporine; Cyclosporins; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; Humans; Mice; Nicardipine; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1996
Simultaneous determination of cytotoxic (adriamycin, vincristine) and modulator of resistance (verapamil, S 9788) drugs in human cells by high-performance liquid chromatography and ultraviolet detection.
    Journal of chromatography. B, Biomedical sciences and applications, 1997, Apr-11, Volume: 691, Issue:2

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Chromatography, High Pressure Liquid; Doxorubicin; Drug Interactions; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; KB Cells; Piperidines; Reproducibility of Results; Sensitivity and Specificity; Spectrophotometry, Ultraviolet; Triazines; Verapamil; Vincristine

1997
Comparison between technetium-99m-sestamibi and hydrogen-3-daunomycin myocardial cellular retention in vitro.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1997, Volume: 38, Issue:11

    Topics: Animals; Animals, Newborn; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Cyclosporins; Daunorubicin; Drug Resistance, Neoplasm; Genes, MDR; Heart; In Vitro Techniques; Myocardium; Piperidines; Radionuclide Imaging; Rats; Rats, Wistar; Technetium Tc 99m Sestamibi; Triazines; Tritium; Verapamil

1997
Evidence for reversal of multidrug resistance by quinine in LR73 cells without alteration of nuclear pirarubicin uptake and down-regulation of mdr1 gene expression.
    International journal of cancer, 1997, Nov-14, Volume: 73, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Nucleus; CHO Cells; Cricetinae; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Gene Expression Regulation; Genes, MDR; Piperidines; Quinine; Triazines; Verapamil

1997
Inhibition of P-glycoprotein: rapid assessment of its implication in blood-brain barrier integrity and drug transport to the brain by an in vitro model of the blood-brain barrier.
    Pharmaceutical research, 1998, Volume: 15, Issue:7

    Topics: Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Astrocytes; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blood-Brain Barrier; Brain; Calcium Channel Blockers; Cattle; Coculture Techniques; Cyclosporine; Doxorubicin; Endothelium, Vascular; Immunosuppressive Agents; Piperidines; Predictive Value of Tests; Rats; Triazines; Verapamil; Vincristine

1998
Confocal scanning microspectrofluorometry reveals specific anthracyline accumulation in cytoplasmic organelles of multidrug-resistant cancer cells.
    The journal of histochemistry and cytochemistry : official journal of the Histochemistry Society, 1998, Volume: 46, Issue:12

    Topics: Animals; Antibiotics, Antineoplastic; Cell Nucleus; CHO Cells; Cricetinae; Cytoplasm; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Golgi Apparatus; Humans; Microspectrophotometry; Piperidines; Quinine; Triazines; Tumor Cells, Cultured; Verapamil

1998
Comparative 99mTc-sestamibi and 3H-daunomycin uptake in human carcinoma cells: relation to the MDR phenotype and effects of reversing agents.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1999, Volume: 40, Issue:4

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Cyclosporins; Daunorubicin; Drug Resistance, Multiple; Humans; Piperidines; Radiopharmaceuticals; Reverse Transcriptase Polymerase Chain Reaction; Technetium Tc 99m Sestamibi; Triazines; Tritium; Tumor Cells, Cultured; Verapamil

1999