verapamil and quinazolines

verapamil has been researched along with quinazolines in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19908 (38.10)18.7374
1990's6 (28.57)18.2507
2000's1 (4.76)29.6817
2010's6 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abiko, Y; Ichihara, K; Nasa, Y; Yoshida, R1
Assaraf, YG; Schimke, RT; Sharma, RC1
Assaraf, YG; Molina, A; Schimke, RT; Sherwood, SW1
Assaraf, YG; Molina, A; Schimke, RT1
Arkin, H; Holland, JF; Kamen, BA; Ohnuma, T; Vallabhajosula, S1
Aleixandre, MA; Ayala, LE; García Mora, L1
Chiba, S; Katsuyama, Y; Tada, A; Tsukada, M; Zenda, H1
Gale, GR; Hynes, JB; Smith, AB1
Fairfax, CA; Tanz, RD1
Chen, WZ; Ding, GS; Li, RS; Zhang, YF1
Elliott, HL; McSharry, DR; Meredith, PA; Pasanisi, F; Reid, JL1
Nagatomo, T; Shibata, A; Shimada, K; Tsuchihashi, H; Wakabayashi, H; Watanabe, K1
Adachi, K; Hidaka, T; Muraishi, A; Okamoto, T; Seki, Y; Toshima, H1
Callaghan, R; Ferry, DR; Higgins, CF; Taylor, JC1
Baumert, C; Hilgeroth, A1
Bers, DM; Diecke, S; Gong, T; Knowles, JW; Lan, F; Lee, AS; Liang, P; Nguyen, PK; Robbins, RC; Sallam, K; Sanchez-Freire, V; Wang, PJ; Wang, Y; Wu, JC1
Li, X; Lu, Y; Yin, Z; Yu, Y; Zhao, X1
Böhmer, FD; Kirches, E; Mawrin, C; Pachow, D; Petermann, A; Wallesch, M; Wilisch-Neumann, A1
de Graaf, IA; de Jager, MH; Groothuis, GM; Li, M1
de Graaf, IA; de Jager, MH; Groothuis, GM; Li, M; van de Steeg, E1
Huo, X; Liu, K; Liu, Q; Liu, Z; Ma, X; Meng, Q; Sun, H; Sun, P; Wang, C; Yang, X; Zhang, Y1

Reviews

1 review(s) available for verapamil and quinazolines

ArticleYear
Recent advances in the development of P-gp inhibitors.
    Anti-cancer agents in medicinal chemistry, 2009, Volume: 9, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Coumarins; Drug Design; Drug Resistance, Neoplasm; Flavonoids; Humans; Peptides; Propafenone; Propanolamines; Pyrazoles; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Quinolines; Structure-Activity Relationship; Tamoxifen; Terpenes; Verapamil

2009

Other Studies

20 other study(ies) available for verapamil and quinazolines

ArticleYear
Positive inotropic and negative chronotropic effects of (-)-cis-diltiazem in rat isolated atria.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Atenolol; Calcium; Diltiazem; Endothelium, Vascular; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Potassium Chloride; Quinazolines; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil

1992
A phenotype conferring selective resistance to lipophilic antifolates in Chinese hamster ovary cells.
    Cancer research, 1991, Jun-01, Volume: 51, Issue:11

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Cell Line; Cricetinae; Drug Resistance; Folic Acid Antagonists; Gene Amplification; Membrane Glycoproteins; Methotrexate; Phenotype; Pyrimidines; Quinazolines; RNA, Messenger; Tetrahydrofolate Dehydrogenase; Trimetrexate; Verapamil

1991
Flow cytometric characterization of antifolate resistance in cultured mammalian cells using fluoresceinated methotrexate and daunorubicin.
    Cancer research, 1990, Aug-15, Volume: 50, Issue:16

    Topics: Animals; Cell Line; Colchicine; Cricetinae; Cricetulus; Daunorubicin; Drug Resistance; Female; Flow Cytometry; Folic Acid Antagonists; Kinetics; Methotrexate; Ovary; Quinazolines; Tetrahydrofolate Dehydrogenase; Trimetrexate; Verapamil

1990
Cross-resistance to the lipid-soluble antifolate trimetrexate in human carcinoma cells with the multidrug-resistant phenotype.
    Journal of the National Cancer Institute, 1989, Feb-15, Volume: 81, Issue:4

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Carcinoma; Cell Line; Drug Resistance; Female; Genes; Humans; Methotrexate; Ovarian Neoplasms; Phenotype; Quinazolines; Quinidine; RNA, Messenger; Trimetrexate; Tumor Cells, Cultured; Verapamil

1989
Multidrug resistance in a human leukemic cell line selected for resistance to trimetrexate.
    Cancer research, 1989, Dec-01, Volume: 49, Issue:23

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Doxorubicin; Drug Resistance; Humans; In Vitro Techniques; Leukemia; Membrane Glycoproteins; Methotrexate; Quinazolines; Tetrahydrofolate Dehydrogenase; Trimetrexate; Tumor Cells, Cultured; Verapamil; Vincristine

1989
Evaluation of different drugs in two models of immediate hypersensitivity.
    The Journal of pharmacy and pharmacology, 1988, Volume: 40, Issue:3

    Topics: Animals; Cromolyn Sodium; Diethylcarbamazine; Diltiazem; Female; Guinea Pigs; Histamine H1 Antagonists; Hypersensitivity, Immediate; In Vitro Techniques; Isometric Contraction; Male; Nicardipine; Ovalbumin; Passive Cutaneous Anaphylaxis; Quinazolines; Trachea; Verapamil

1988
Vasoconstrictor effects of endogenous digitalis-like factors extracted from urine of hypertensive patients.
    Heart and vessels, 1987, Volume: 3, Issue:3

    Topics: Animals; Arteries; Blood Proteins; Cardenolides; Digoxin; Dogs; Ear, External; Epinephrine; Humans; Hypertension; In Vitro Techniques; Mesenteric Arteries; Ouabain; Phentolamine; Potassium Chloride; Quinazolines; Saponins; Vasoconstrictor Agents; Verapamil

1987
Effects of 5,8-dideazaisopteroylglutamate (IAHQ) on L1210 leukemia in mice when given alone and in combination with methotrexate, probenecid, or verapamil.
    Cancer chemotherapy and pharmacology, 1986, Volume: 18, Issue:3

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Folic Acid Antagonists; Leukemia L1210; Male; Methotrexate; Mice; Mice, Inbred DBA; Probenecid; Quinazolines; Time Factors; Verapamil

1986
Insurmountable antagonism of ouabain-induced coronary constriction by prazosin.
    European journal of pharmacology, 1985, May-28, Volume: 112, Issue:1

    Topics: Animals; Coronary Vessels; In Vitro Techniques; Ouabain; Prazosin; Quinazolines; Swine; Vasoconstriction; Verapamil

1985
[Effects of changrolin on contractility and excitability of isolated cat papillary muscle].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1984, Volume: 5, Issue:1

    Topics: Animals; Anti-Arrhythmia Agents; Calcium Chloride; Cats; Female; Male; Myocardial Contraction; Niacinamide; Papillary Muscles; Quinazolines; Verapamil

1984
Combined alpha adrenoceptor antagonism and calcium channel blockade in normal subjects.
    Clinical pharmacology and therapeutics, 1984, Volume: 36, Issue:6

    Topics: Administration, Oral; Adult; Biological Availability; Blood Pressure; Chromatography, High Pressure Liquid; Drug Evaluation; Drug Synergism; Heart Rate; Humans; Hypotension, Orthostatic; Kinetics; Male; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Quinazolines; Random Allocation; Verapamil

1984
Alterations of binding characteristics of alpha 1-,beta 1-adrenoceptors and Ca2+ binding sites in the myocardium of spontaneously hypertensive rats (SHR) by chronically administered bunazosin, atenolol, ketanserin and verapamil.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Atenolol; Binding Sites; Blood Pressure; Calcium Channels; Heart; In Vitro Techniques; Ketanserin; Kinetics; Myocardium; Norepinephrine; Quinazolines; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Verapamil

1993
Induction of DNA breaks in cardiac myoblast cells by norepinephrine.
    Biochemistry and molecular biology international, 1996, Volume: 38, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Calcium Channel Blockers; Captopril; DNA; DNA Damage; DNA, Single-Stranded; Heart; Hydrogen Peroxide; Myocardium; Norepinephrine; Propranolol; Quinazolines; Rats; Stimulation, Chemical; Verapamil

1996
The equilibrium and kinetic drug binding properties of the mouse P-gp1a and P-gp1b P-glycoproteins are similar.
    British journal of cancer, 1999, Volume: 81, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Sub-Family B Member 4; ATP-Binding Cassette Transporters; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Drug Resistance, Multiple; Isoquinolines; Kinetics; Mice; Nicardipine; Progesterone; Protein Binding; Protein Isoforms; Quinazolines; Verapamil; Vinblastine

1999
Drug screening using a library of human induced pluripotent stem cell-derived cardiomyocytes reveals disease-specific patterns of cardiotoxicity.
    Circulation, 2013, Apr-23, Volume: 127, Issue:16

    Topics: Action Potentials; Cardiomyopathy, Dilated; Cardiomyopathy, Hypertrophic, Familial; Cell Differentiation; Cell Line; Cell Size; Cisapride; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Embryoid Bodies; Embryonic Stem Cells; Gene Expression Profiling; Genetic Predisposition to Disease; HEK293 Cells; Humans; In Vitro Techniques; Induced Pluripotent Stem Cells; Ion Channels; Kidney; Long QT Syndrome; Myocytes, Cardiac; Myofibrils; Nicorandil; Patch-Clamp Techniques; Quinazolines; Verapamil

2013
Intestinal absorption of raltitrexed and evaluation of the effects of absorption enhancers.
    Die Pharmazie, 2013, Volume: 68, Issue:9

    Topics: 2-Pyridinylmethylsulfinylbenzimidazoles; Acrylic Resins; Algorithms; Animals; Antimetabolites, Antineoplastic; ATP-Binding Cassette Transporters; Biological Availability; Caco-2 Cells; Decanoic Acids; Deoxycholic Acid; Excipients; Folic Acid; Humans; Intestinal Absorption; Male; Pantoprazole; Probenecid; Quinazolines; Rats; Rats, Wistar; Thiophenes; Verapamil

2013
Re-evaluation of cytostatic therapies for meningiomas in vitro.
    Journal of cancer research and clinical oncology, 2014, Volume: 140, Issue:8

    Topics: Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Dacarbazine; DNA Methylation; DNA Modification Methylases; DNA Repair Enzymes; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Erlotinib Hydrochloride; Humans; Hydroxyurea; Losartan; Meningeal Neoplasms; Meningioma; Metformin; Mifepristone; Neurofibromin 2; Promoter Regions, Genetic; Quinazolines; Radiation Tolerance; Tamoxifen; Temozolomide; Tumor Suppressor Proteins; Verapamil

2014
Rat precision-cut intestinal slices to study P-gp activity and the potency of its inhibitors ex vivo.
    Toxicology in vitro : an international journal published in association with BIBRA, 2015, Volume: 29, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Cyclosporins; In Vitro Techniques; Intestinal Mucosa; Isoquinolines; Ketoconazole; Male; Quinazolines; Quinidine; Rats, Wistar; Rhodamine 123; Verapamil

2015
The consequence of regional gradients of P-gp and CYP3A4 for drug-drug interactions by P-gp inhibitors and the P-gp/CYP3A4 interplay in the human intestine ex vivo.
    Toxicology in vitro : an international journal published in association with BIBRA, 2017, Volume: 40

    Topics: Adult; Aged; Aged, 80 and over; ATP Binding Cassette Transporter, Subfamily B, Member 1; Colon; Cyclosporins; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Female; Humans; Ileum; In Vitro Techniques; Isoquinolines; Jejunum; Ketoconazole; Male; Middle Aged; Quinazolines; Quinidine; Verapamil

2017
P-gp is involved in the intestinal absorption and biliary excretion of afatinib in vitro and in rats.
    Pharmacological reports : PR, 2018, Volume: 70, Issue:2

    Topics: Adenosine Triphosphatases; Afatinib; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bile; Biological Transport; Caco-2 Cells; Cell Line, Tumor; Cyclosporine; Hepatobiliary Elimination; Hepatocytes; Humans; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Quinazolines; Rats; Rats, Wistar; Verapamil

2018