verapamil and quercetin

verapamil has been researched along with quercetin in 40 studies

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-19903 (7.50)18.7374
1990's5 (12.50)18.2507
2000's14 (35.00)29.6817
2010's15 (37.50)24.3611
2020's3 (7.50)2.80

Authors

AuthorsStudies
Back, DJ; Eagling, VA; Profit, L1
Bacsó, Z; Cianfriglia, M; Fenyvesi, F; Goda, K; Kappelmayer, J; Lustyik, G; Nagy, H; Szabó, G; Szilasi, M1
Choi, CH; Kim, JH; Kim, SH1
Lombardo, F; Obach, RS; Waters, NJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Chan, KF; Chan, TH; Chow, LM; Lam, CY; Tsang, KH; Wong, IL; Zhao, Y1
Ghosh, I; Manoharlal, R; Prakash, O; Prasad, R; Puri, N; Sharma, M1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Bönisch, H; Haenisch, B; Mayer, R; Müller, CE; Müller, H; Pajeva, IK; Pick, A; Weigt, M; Wiese, M1
Freiwald, S; Jiang, Y; Jones, JP; Kaspera, R; Katayama, J; Lee, CA; Smith, E; Totah, RA; Walker, GS1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Chow, LM; Jiang, T; Liu, T; Wan Sheng, B; Wang, SW; Wen, BJ; Wong, IL; Yuan, J1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chong, Y; Choo, H; Kim, MK; Kim, Y1
Dong, S; Gao, JM; He, QR; Huang, LF; Tang, JJ; Wang, MR1
Chan, CF; Chan, KF; Chan, TH; Chong, TC; Chow, LMC; Chow, TS; Cui, J; Law, MC; Liu, Z; Wong, ILK; Zhu, X1
Kurose, M1
Drzewiecki, G; Middleton, E; Triggle, D1
Martz, E; Parker, WL1
Critchfield, JW; Phang, JM; Welsh, CJ; Yeh, GC1
Chen, ZW; Fang, M; Ma, CG; Xu, SY1
Leng, XF; Wu, YJ1
Banan, A; Deshpande, Y; Kokoska, ER; Miller, TA; Rieckenberg, CL; Smith, GS; Wolff, AB1
Duarte, J; Galisteo, M; García-Saura, MF; Jiménez, R; Vargas, F; Villar, IC; Wangensteen, R; Zarzuelo, A1
Duarte, J; Galisteo, M; García-Saura, MF; Jiménez, R; Vargas, F; Villar, IC; Zarzuelo, A1
Borrelli, F; Capasso, F; Capasso, R; Izzo, AA; Mascolo, N1
Choi, JS; Han, HK1
Annaert, PP; Brouwer, KL1
Chen, W; Gong, M; Hu, CY; Huang, B; Huang, PH; Jiang, QY; Lu, M; Lu, ZG; Qiao, CP; Wang, MH; Zhu, F1
Tian, X; Wang, K; Yang, X1
Chen, YC; Lin, T; Nagpal, ML; Stocco, DM1
Bera, T; Bhuyan, NR; Chakraborty, B; Lakshman, K; Roy, AK; Sen, SS1
Gilani, AH; Khan, AU1
Duan, JA; Guo, JM; Qian, DW; Shu, Y; Xue, CF1
Chong, Y; Choo, H; Kim, MK1
Chong, Y; Choo, H; Kim, MK; Park, KS1
Dively, GP; Evans, JD; Guseman, AJ; Hawthorne, DJ; Kunkle, G; Miller, K; Pettis, JS; vanEngelsdorp, D1
Behrens, C; Choe, JY; Dean, JV; Theccanat, T; Vaca, E1
Basir, SF; Khan, LA; Wani, SA1

Other Studies

40 other study(ies) available for verapamil and quercetin

ArticleYear
Inhibition of the CYP3A4-mediated metabolism and P-glycoprotein-mediated transport of the HIV-1 protease inhibitor saquinavir by grapefruit juice components.
    British journal of clinical pharmacology, 1999, Volume: 48, Issue:4

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Beverages; Caco-2 Cells; Citrus; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Drug Interactions; Gas Chromatography-Mass Spectrometry; HIV Protease Inhibitors; Humans; In Vitro Techniques; Ketoconazole; Liver; Mixed Function Oxygenases; Plant Extracts; Saquinavir; Time Factors; Verapamil

1999
Distinct groups of multidrug resistance modulating agents are distinguished by competition of P-glycoprotein-specific antibodies.
    Biochemical and biophysical research communications, 2004, Mar-19, Volume: 315, Issue:4

    Topics: Adenosine Triphosphatases; Animals; Anti-Bacterial Agents; Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Calcium Channel Blockers; Cyclosporine; Detergents; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Humans; Ivermectin; Mice; NIH 3T3 Cells; Substrate Specificity

2004
Reversal of P-glycoprotein-mediated MDR by 5,7,3',4',5'-pentamethoxyflavone and SAR.
    Biochemical and biophysical research communications, 2004, Jul-30, Volume: 320, Issue:3

    Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Survival; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Enzyme Activation; Flavonoids; Humans; Leukemia, Myeloid, Acute; Structure-Activity Relationship; Vincristine

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Modulation of multidrug resistance protein 1 (MRP1/ABCC1)-mediated multidrug resistance by bivalent apigenin homodimers and their derivatives.
    Journal of medicinal chemistry, 2009, Sep-10, Volume: 52, Issue:17

    Topics: Apigenin; Binding, Competitive; Cell Line, Tumor; Dimerization; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Multiple; Etoposide; Humans; Hydroxides; Intracellular Space; Multidrug Resistance-Associated Proteins; Structure-Activity Relationship

2009
Analysis of physico-chemical properties of substrates of ABC and MFS multidrug transporters of pathogenic Candida albicans.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Candida albicans; Membrane Transport Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Substrate Specificity

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Structure-activity relationships of flavonoids as inhibitors of breast cancer resistance protein (BCRP).
    Bioorganic & medicinal chemistry, 2011, Mar-15, Volume: 19, Issue:6

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Cell Line, Tumor; Drug Resistance, Neoplasm; Female; Flavonoids; Humans; Hydrogen Bonding; Models, Molecular; Neoplasm Proteins; Quantitative Structure-Activity Relationship

2011
Identifying a selective substrate and inhibitor pair for the evaluation of CYP2J2 activity.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:5

    Topics: Amiodarone; Astemizole; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Danazol; Drug Discovery; Drug Interactions; Enzyme Inhibitors; Humans; Hydroxylation; In Vitro Techniques; Methylation; Microsomes, Liver; Models, Biological; Molecular Structure; Substrate Specificity; Tandem Mass Spectrometry; Terfenadine

2012
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Synthesis of methylated quercetin derivatives and their reversal activities on P-gp- and BCRP-mediated multidrug resistance tumour cells.
    European journal of medicinal chemistry, 2012, Volume: 54

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cell Line, Tumor; Chemistry Techniques, Synthetic; Drug Resistance, Multiple; Humans; Methylation; Mice; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Quercetin

2012
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Quercetin-glutamic acid conjugate with a non-hydrolysable linker; a novel scaffold for multidrug resistance reversal agents through inhibition of P-glycoprotein.
    Bioorganic & medicinal chemistry, 2017, 02-01, Volume: 25, Issue:3

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Glutamic Acid; Humans; Molecular Structure; Quercetin; Structure-Activity Relationship

2017
1,10-Seco-Eudesmane sesquiterpenoids as a new type of anti-neuroinflammatory agents by suppressing TLR4/NF-κB/MAPK pathways.
    European journal of medicinal chemistry, 2021, Nov-15, Volume: 224

    Topics: Anti-Inflammatory Agents; Humans; Models, Molecular; Neuroinflammatory Diseases; NF-kappa B; Sesquiterpenes, Eudesmane; Structure-Activity Relationship; Toll-Like Receptor 4

2021
Flavonoid Monomers as Potent, Nontoxic, and Selective Modulators of the Breast Cancer Resistance Protein (ABCG2).
    Journal of medicinal chemistry, 2021, 10-14, Volume: 64, Issue:19

    Topics: Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flavonoids; HEK293 Cells; Humans; Mitoxantrone; Neoplasm Proteins; Structure-Activity Relationship; Substrate Specificity

2021
Inhibition of anaphylactic histamine release from heterologously sensitized mast cells: differential effects of drugs which interfere with calcium influx.
    Acta medica Okayama, 1981, Volume: 35, Issue:5

    Topics: Animals; Antigens; Biological Transport; Calcium; Cromolyn Sodium; Histamine Release; Immunization; Immunoglobulin E; Male; Mast Cells; Mice; Mice, Inbred BALB C; Quercetin; Rats; Rats, Inbred Strains; Theophylline; Verapamil

1981
Effects of smooth muscle calcium antagonists on human basophil histamine release.
    Biochemical pharmacology, 1981, Volume: 30, Issue:20

    Topics: Basophils; Calcium; Dantrolene; Gallic Acid; Gallopamil; Histamine Release; Humans; Muscle Contraction; Muscle, Smooth; Nifedipine; Quercetin; Verapamil

1981
Calcium ionophore A23187 as a secretagogue for rat mast cells: does it bypass inhibition by calcium flux blockers?
    Agents and actions, 1982, Volume: 12, Issue:3

    Topics: Animals; Anti-Bacterial Agents; Bucladesine; Calcimycin; Calcium Channel Blockers; Immunoglobulin E; In Vitro Techniques; Mast Cells; Quercetin; Rats; Ruthenium Red; Verapamil

1982
Modulation of adriamycin accumulation and efflux by flavonoids in HCT-15 colon cells. Activation of P-glycoprotein as a putative mechanism.
    Biochemical pharmacology, 1994, Oct-07, Volume: 48, Issue:7

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Butyrates; Butyric Acid; Cell Division; Cell Line; Cell Survival; Diet; Dose-Response Relationship, Drug; Doxorubicin; Drug Interactions; Flavonoids; Humans; Kaempferols; Quercetin; Structure-Activity Relationship; Verapamil; Vinblastine

1994
[The blocking effect of hyperin on the inward flow of calcium ion].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1994, Volume: 29, Issue:1

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Myocardial Contraction; Quercetin; Rabbits; Stimulation, Chemical; Verapamil

1994
Comparison of effects of verapamil and quercetin on delayed polyneuropathy induced by Tri-o-cresyl phosphate in hens.
    Bulletin of environmental contamination and toxicology, 1997, Volume: 58, Issue:4

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Chickens; Enzyme Inhibitors; Female; Peripheral Nervous System Diseases; Quercetin; Tritolyl Phosphates; Verapamil

1997
Role of calcium in adaptive cytoprotection and cell injury induced by deoxycholate in human gastric cells.
    The American journal of physiology, 1998, Volume: 275, Issue:2

    Topics: Acclimatization; Calcium; Cell Membrane; Cell Survival; Deoxycholic Acid; Dose-Response Relationship, Drug; Estrenes; Gastric Mucosa; Humans; Kinetics; Lanthanum; Microscopy, Confocal; Neomycin; Nifedipine; Phosphodiesterase Inhibitors; Pyrrolidinones; Quercetin; Stomach Neoplasms; Tumor Cells, Cultured; Type C Phospholipases; Verapamil

1998
Effects of quercetin treatment on vascular function in deoxycorticosterone acetate-salt hypertensive rats. Comparative study with verapamil.
    Planta medica, 2004, Volume: 70, Issue:4

    Topics: Animals; Antihypertensive Agents; Aorta; Blood Pressure; Desoxycorticosterone; Disease Models, Animal; Hypertension; Male; Muscle Contraction; Phytotherapy; Plants, Medicinal; Potassium Chloride; Quercetin; Rats; Rats, Wistar; Sodium Chloride; Verapamil

2004
Effects of chronic quercetin treatment on antioxidant defence system and oxidative status of deoxycorticosterone acetate-salt-hypertensive rats.
    Molecular and cellular biochemistry, 2004, Volume: 259, Issue:1-2

    Topics: Administration, Oral; Animals; Blood Pressure; Cardiomegaly; Catalase; Desoxycorticosterone; Glutathione; Glutathione Peroxidase; Glutathione Transferase; Hepatomegaly; Hypertension; Kidney; Lipid Peroxidation; Liver; Male; Myocardium; Oxidation-Reduction; Quercetin; Rats; Rats, Wistar; Superoxide Dismutase; Thiobarbituric Acid Reactive Substances; Vasodilator Agents; Verapamil

2004
Inhibitory effect of the antidepressant St. John's wort (hypericum perforatum) on rat bladder contractility in vitro.
    Urology, 2004, Volume: 64, Issue:1

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Anthracenes; Antidepressive Agents; Atropine; Bridged Bicyclo Compounds; Capsaicin; Depression; Electric Stimulation; Female; Haloperidol; Hypericum; Kaempferols; Male; Methysergide; Muscle Contraction; Muscle, Smooth; Naloxone; Perylene; Phentolamine; Phloroglucinol; Piperidines; Plant Extracts; Propranolol; Pyrazoles; Quercetin; Rats; Rats, Wistar; Rimonabant; Rutin; Terpenes; Tetrodotoxin; Urinary Bladder; Urinary Incontinence; Verapamil

2004
The effect of quercetin on the pharmacokinetics of verapamil and its major metabolite, norverapamil, in rabbits.
    The Journal of pharmacy and pharmacology, 2004, Volume: 56, Issue:12

    Topics: Animals; Drug Interactions; Male; Quercetin; Rabbits; Verapamil

2004
Assessment of drug interactions in hepatobiliary transport using rhodamine 123 in sandwich-cultured rat hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 2005, Volume: 33, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Culture Techniques; Cells, Cultured; Collagenases; Digoxin; Drug Interactions; Hepatocytes; Male; Progesterone; Quercetin; Quinidine; Rats; Rats, Wistar; Rhodamine 123; Verapamil

2005
Effects of total flavonoids of Hippophae rhamnoides L. on intracellular free calcium in cultured vascular smooth muscle cells of spontaneously hypertensive rats and Wistar-Kyoto rats.
    Chinese journal of integrative medicine, 2005, Volume: 11, Issue:4

    Topics: Angiotensin II; Animals; Calcium; Cells, Cultured; Flavonoids; Flavonols; Hippophae; Hypertension; Muscle, Smooth, Vascular; Norepinephrine; Quercetin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Verapamil

2005
The efflux of flavonoids morin, isorhamnetin-3-O-rutinoside and diosmetin-7-O-beta-D-xylopyranosyl-(1-6) -beta-D-glucopyranoside in the human intestinal cell line caco-2.
    Pharmaceutical research, 2006, Volume: 23, Issue:8

    Topics: Adenosine Triphosphate; Antioxidants; Biological Transport, Active; Caco-2 Cells; Chromatography, High Pressure Liquid; Disaccharides; Enzyme Inhibitors; Flavonoids; Humans; Intestinal Mucosa; Iodoacetamide; Probenecid; Propionates; Quercetin; Quinolines; Verapamil

2006
Effects of genistein, resveratrol, and quercetin on steroidogenesis and proliferation of MA-10 mouse Leydig tumor cells.
    The Journal of endocrinology, 2007, Volume: 192, Issue:3

    Topics: Adenosine Triphosphatases; Animals; Calcium Channel Blockers; Cell Line, Tumor; Cell Proliferation; Cyclic AMP; Egtazic Acid; Estradiol; Fulvestrant; Genistein; Leydig Cells; Male; Mibefradil; Mice; Phosphoproteins; Phytoestrogens; Progesterone; Quercetin; Receptors, Estrogen; Resveratrol; RNA, Messenger; Stilbenes; Stimulation, Chemical; Vanadates; Verapamil

2007
Membrane bound pyrophosphatase and P-type adenosine triphosphatase of Leishmania donovani as possible chemotherapeutic targets: similarities and differences in inhibitor sensitivities.
    Biochemistry. Biokhimiia, 2009, Volume: 74, Issue:12

    Topics: 4-Chloromercuribenzenesulfonate; Adenosine Triphosphatases; Antiprotozoal Agents; Dicyclohexylcarbodiimide; Drug Design; Enzyme Inhibitors; Leishmania donovani; Maleimides; Pyrophosphatases; Quercetin; Verapamil

2009
Pharmacological studies on Hypericum perforatum fractions and constituents.
    Pharmaceutical biology, 2011, Volume: 49, Issue:1

    Topics: Animals; Anthracenes; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Female; Guinea Pigs; Hypericum; In Vitro Techniques; Male; Perylene; Phloroglucinol; Phosphodiesterase Inhibitors; Plant Extracts; Quercetin; Rabbits; Terpenes; Verapamil

2011
[Absorption of flavonoids from Abelmoschus manihot extract by in situ intestinal perfusion].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2011, Volume: 46, Issue:4

    Topics: Abelmoschus; Animals; ATP Binding Cassette Transporter, Subfamily B; Flavonoids; Flowers; Glucosides; Intestinal Absorption; Male; Perfusion; Plant Extracts; Plants, Medicinal; Quercetin; Rats; Rats, Sprague-Dawley; Verapamil

2011
Water-soluble and cleavable quercetin-amino acid conjugates as safe modulators for P-glycoprotein-based multidrug resistance.
    Journal of medicinal chemistry, 2014, Sep-11, Volume: 57, Issue:17

    Topics: Alanine; Amino Acids; Antineoplastic Agents; Antioxidants; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cell Line, Tumor; Cell Survival; Dactinomycin; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Multiple; Glutamic Acid; Humans; Microscopy, Confocal; Models, Chemical; Molecular Structure; Paclitaxel; Quercetin; Verapamil; Vinblastine

2014
Quercetin-POM (pivaloxymethyl) conjugates: Modulatory activity for P-glycoprotein-based multidrug resistance.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2015, Jul-15, Volume: 22, Issue:7-8

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Binding Sites; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Molecular Structure; Quercetin; Verapamil

2015
Multi-Drug Resistance Transporters and a Mechanism-Based Strategy for Assessing Risks of Pesticide Combinations to Honey Bees.
    PloS one, 2016, Volume: 11, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Bees; Biological Transport; Biphenyl Compounds; Carbamates; Cyclohexanes; Drug Resistance, Multiple; Environmental Exposure; Fatty Acids, Unsaturated; Insecticides; Ivermectin; Membrane Transport Proteins; Neonicotinoids; Niacinamide; Pyrazoles; Pyridines; Quercetin; Rhodamines; Risk Assessment; Sesquiterpenes; Verapamil

2016
Mechanistic differences in the uptake of salicylic acid glucose conjugates by vacuolar membrane-enriched vesicles isolated from Arabidopsis thaliana.
    Physiologia plantarum, 2017, Volume: 161, Issue:3

    Topics: Adenosine Triphosphate; Arabidopsis; Arbutin; ATP-Binding Cassette Transporters; Benzyl Alcohols; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Glucose; Glucosides; Gramicidin; Intracellular Membranes; Kinetics; Metabolome; Protoplasts; Quercetin; Salicylic Acid; Time Factors; Transport Vesicles; Vacuolar Proton-Translocating ATPases; Vacuoles; Verapamil

2017
Quercetin and resveratrol ameliorate nickel-mediated hypercontraction in isolated Wistar rat aorta.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2022, Volume: 58

    Topics: Animals; Aorta; Aorta, Thoracic; Calcium Channels; Dose-Response Relationship, Drug; Endothelial Cells; Endothelium, Vascular; Indomethacin; NG-Nitroarginine Methyl Ester; Nickel; Nitric Oxide; Quercetin; Rats; Rats, Wistar; Reactive Oxygen Species; Resveratrol; Verapamil

2022