verapamil and pk 11195

verapamil has been researched along with pk 11195 in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19902 (28.57)18.7374
1990's1 (14.29)18.2507
2000's3 (42.86)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Botta, M; Bruni, G; Budriesi, R; Campiani, G; Chiarini, A; Ciani, SM; De Filippis, MP; Fiorini, I; Garofalo, A; Giorgi, G; Manzoni, C; Mennini, T; Nacci, V; Romeo, MR; Sega, A1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Benavides, J; Bertrand, P; Burgevin, MC; Doble, A; Ferris, O; Gueremy, C; Le Fur, G; Menager, J; Uzan, A; Vaucher, N1
Belin, C; Carriot, T; Doble, A; Dubroeucq, MC; Guérémy, C; Le Fur, G; Mestre, M; Renault, C; Uzan, A1
Chugun, A; Futamura, K; Hara, Y; Kobayashi, H; Kondo, H; Nishino, T; Ooshiro, S; Temma, K1
Cattaneo, S; Cosentino, M; Di Grazia, L; Fietta, AM; Frigo, G; Lecchini, S; Marino, F; Rasini, E1
Boellaard, R; Lammertsma, AA; Lubberink, M; Mourik, JE; Schuitemaker, A; Tolboom, N; van Berckel, BN1

Other Studies

7 other study(ies) available for verapamil and pk 11195

ArticleYear
Cardiovascular characterization of pyrrolo[2,1-d][1,5]benzothiazepine derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): from dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blocker
    Journal of medicinal chemistry, 1996, Jul-19, Volume: 39, Issue:15

    Topics: Animals; Atrial Function; Binding, Competitive; Calcium Channel Blockers; Calcium Channels; Cardiovascular System; Cerebral Cortex; Depression, Chemical; Female; Guinea Pigs; Heart Rate; Male; Models, Molecular; Myocardial Contraction; Myocardium; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship; Thiazepines

1996
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Dihydropyridine and peripheral type benzodiazepine binding sites: subcellular distribution and molecular size determination.
    European journal of pharmacology, 1985, Dec-17, Volume: 119, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Fractionation; Dogs; Ion Channels; Isoquinolines; Isradipine; Male; Molecular Weight; Myocardium; Nifedipine; Nitrendipine; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Nicotinic; Sarcolemma; Sarcoplasmic Reticulum; Verapamil

1985
Electrophysiological and pharmacological evidence that peripheral type benzodiazepine receptors are coupled to calcium channels in the heart.
    Life sciences, 1985, Jan-28, Volume: 36, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium; Calcium Channel Blockers; Diltiazem; Female; Guinea Pigs; Heart; Ion Channels; Isoquinolines; Male; Myocardial Contraction; Nifedipine; Nitrendipine; Receptors, GABA-A; Tetraethylammonium Compounds; Verapamil

1985
Negative inotropic effect of diazepam in isolated guinea pig heart.
    The Journal of veterinary medical science, 2001, Volume: 63, Issue:2

    Topics: Adjuvants, Anesthesia; Animals; Anti-Arrhythmia Agents; Calcium Channels; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Myocardial Contraction; Patch-Clamp Techniques; Verapamil

2001
Diazepam stimulates migration and phagocytosis of human neutrophils: possible contribution of peripheral-type benzodiazepine receptors and intracellular calcium.
    Pharmacology, 2001, Volume: 63, Issue:1

    Topics: Calcium; Calcium Channel Blockers; Cells, Cultured; Chemotaxis, Leukocyte; Diazepam; Flow Cytometry; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; In Vitro Techniques; Isoquinolines; Neutrophils; Phagocytosis; Receptors, GABA-A; Verapamil

2001
Image-derived input functions for PET brain studies.
    European journal of nuclear medicine and molecular imaging, 2009, Volume: 36, Issue:3

    Topics: Aniline Compounds; Benzothiazoles; Brain; Carbon Radioisotopes; Humans; Image Processing, Computer-Assisted; Isoquinolines; Positron-Emission Tomography; Radiopharmaceuticals; Thiazoles; Verapamil

2009