verapamil has been researched along with gallopamil in 302 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 250 (82.78) | 18.7374 |
1990's | 40 (13.25) | 18.2507 |
2000's | 9 (2.98) | 29.6817 |
2010's | 3 (0.99) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Dietel, M; Höllt, V; Kouba, M; Vogt, G | 1 |
Giacomini, JC; Giacomini, KM; Nelson, WL; Theodore, LJ; Zobrist, RH | 1 |
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Janis, RA; Triggle, DJ | 1 |
Campillo, NE; Guerra, A; Páez, JA | 1 |
Fijorek, K; Glinka, A; Mendyk, A; Polak, S; Wiśniowska, B | 1 |
Brouillette, WJ; Brown, GB; Zha, C | 1 |
Emrich, HM; Reich, R | 1 |
Bristow, MR; Green, RD | 1 |
Duncan, CJ; Publicover, SJ | 1 |
Robinson, IC; Russell, JT; Thorn, NA | 1 |
Godfraind, T; Morel, N | 1 |
Dretchen, KL; Morgenroth, VH; Skirboll, LR; Standaert, FG | 1 |
Kin, M; Kubota, K; Uruno, T | 1 |
Carchman, RA; Warner, W | 1 |
Hiwatari, M; Taira, N | 1 |
Dörrscheidt-Käfer, M | 1 |
Gotgil'f, NM; Magazanik, LG | 1 |
Chapman, RA; Ellis, D | 1 |
Blaustein, MP; Nachshen, DA | 1 |
Catterall, WA; Galper, JB | 2 |
Coburn, RF | 1 |
El-Sherif, N; Lazzara, R | 1 |
Galkin, AA; Khodorov, BI | 1 |
Aguirre, J; Falutz, J; Pinto, JE; Trifaró, JM | 1 |
Powell, T; Rowles, PM; Steen, E; Woolf, N | 1 |
Babskaia, NE; Kafengauz, BIu; Poskonova, MA | 1 |
Engberg, I; Flatman, JA; Lambert, JD | 1 |
McGee, R; Schneider, JE | 1 |
Göthert, M; Nawroth, P; Neumeyer, H | 1 |
Crankshaw, DJ; Daniel, EE; Janis, RA | 1 |
Götz von Olenhusen, K; Wohlfarth-Bottermann, KE | 1 |
Schümann, HJ; Wagner, J | 1 |
Golenhofen, K | 2 |
Campbell, AK; Siddle, K | 1 |
Beck, OA; Hochrein, H; Lehmann, HU; Witt, E | 1 |
Adcock, RC; Templeton, GH; Wheelan, S; Wildenthal, K; Willerson, JT | 1 |
Rossner, KL; Sachs, HG | 1 |
Low, JC | 1 |
Kecskeméti, V; Kelemen, K; Knoll, J | 1 |
Fry, WJ; Hester, RK; Weiss, GB | 1 |
Devis, G; Malaisse, WJ; Pipeleers, DG; Somers, G | 1 |
Kaumann, AJ; Uchitel, OD | 1 |
Leder, O | 1 |
Ludwig, C; Nawrath, H | 1 |
Eick, RE; McDonald, TF; Nawrath, H; Trautwein, W | 1 |
Ferris, RK; Gordon, EE | 1 |
Robinson, RB; Sleator, WW | 1 |
Aguirre, J; Pinto, JE; Trifaró, JM | 1 |
Bristow, MR; Daniels, JR; Harrison, DC; Kernoff, RS | 1 |
Freynik, P; Reinhardt, D; Schümann, HJ | 1 |
Kuroda, T | 1 |
Jetley, M; Weston, AH | 2 |
Hoffmann, A; Siegers, CP; Sierra-Callejas, JL; Strubelt, O | 1 |
Bassingthwaighte, JB; Fry, CH; McGuigan, JA | 1 |
Ignat'eva, VB; Khodorov, BI; Kitaĭgorodskaia, GM; Mukumov, MR; Vornovitskiĭ, EG | 1 |
Fleckenstein, A | 2 |
Bianchi, CP; Kroeger, EA; Marshall, JM | 1 |
Fleckenstein, A; Haastert, HP | 1 |
Görlitz, BD; Schümann, HJ; Wagner, J | 2 |
Marshall, JM; Reiner, O | 1 |
Bayer, R; Hennekes, R; Kaufmann, R; Mannhold, R | 1 |
Bayer, R; Kaufmann, R; Mannhold, R | 1 |
Bayer, R; Kalusche, D; Kaufmann, R; Mannhold, R | 1 |
Hurwitz, L; Tomiyama, A | 1 |
Kohlhardt, M | 1 |
Fleckenstein, A; Tritthart, H; Volkmann, R; Weiss, R | 1 |
Fleckenstein, A; Janke, J; Sigel, H | 1 |
Gerlach, E; Zimmer, HG | 1 |
Bogoliubov, VM; Gribkova, IN; Kruglova, ZG; Lyskova, MN | 1 |
Danilenko, AM; Fialko, VA; Rodionov, VM; Siianov, VS | 1 |
Pinto, JE; Trifaró, JM | 1 |
Galbani, P; Limbruno, U; Mariani, M; Ronca, G; Ronca-Testoni, S; Yu, G; Zucchi, R | 1 |
Finkel, MS; Oddis, CV; Romeo, RC; Salama, G | 1 |
Ferrari, R; Pasini, E; Poli, E; Raddino, R | 1 |
Czejka, MJ; Podesser, B; Zwoelfer, N | 1 |
Blaschke, G; Fieger, H | 1 |
Isenberg, G; Klöckner, U | 1 |
Beech, DJ; Bolton, TB; Christen, MO; MacKenzie, I | 1 |
DeCoursey, TE; Jacobs, ER | 1 |
Köbler, W; Möller, P; Neumann, FJ; Parekh, N; Steinhausen, M; Tillmanns, H; Waas, W; Zimmermann, R | 1 |
Endo, T; Hayakawa, H; Maroko, PR; Sato, N | 1 |
Haass, M; Richardt, G; Schömig, A | 1 |
Ibel, H; Suchner, U; Zimmer, HG | 1 |
Beil, W; Bersimbaev, RJ; Hannemann, H; Sewing, KF | 1 |
Peers, C | 1 |
Mutlib, AE; Nelson, WL | 1 |
Dorigo, O; Kübler, W; Neumann, FJ; Parekh, N; Steinhausen, M; Tiefenbacher, C; Tillmanns, H; Zimmermann, R | 1 |
Coghlan, JP; Denton, DA; Hardy, KJ; Johnson, EI; McDougall, JG; Scoggins, BA; Wright, RD | 1 |
Natochin, IuV | 1 |
Horackova, M | 1 |
Gallant, EM; Goettl, VM | 1 |
Ducreux, C; Gola, M | 1 |
Frank, GB | 2 |
Affolter, H; Coronado, R | 1 |
Froldi, M; Leggieri, E; Lorini, M; Miadonna, A; Tedeschi, A; Zanussi, C | 1 |
Höllt, V; Kley, N; Loeffler, JP; Pittius, CW | 1 |
Bodewei, R; Hering, S; Schubert, B; Wollenberger, A | 1 |
Van Dyke, K; Ye, ZG | 1 |
Bielenberg, GW; Krieglstein, J; Weber, J | 1 |
Reiterer, W | 1 |
Greenidge, E; Wali, FA | 1 |
Bustamante, JO | 1 |
Graser, T; Kurella, GA; Sukhova, GS; Udel'nov, MG | 1 |
Czogalla, W; Dilger, C; Jaeger, H; Otto, R; Salama, ZB | 1 |
Ishikawa, T; Murakami, H; Watanabe, H | 1 |
Edeson, RO; Madsen, BW; Milne, RK | 1 |
Boero, R; Deabate, MC; Forneris, G; Guarena, C; Piccoli, G; Quarello, F; Rosati, C | 1 |
Fosset, M; Galizzi, JP; Lazdunski, M | 1 |
Ilias, W; Steinbereithner, K | 1 |
Ambrosini, F; Bertoni, T; Finzi, A; Foresti, A; Lotto, A; Massari, FM; Matta, F; Valentini, R | 1 |
Hester, RK; Satake, N; Shibata, S; Tomiyama, A; Ueda, S; Wakabayashi, S | 1 |
Fukuda, H; Ishida, Y; Iwamoto, T; Kanaya, J; Maeshiba, Y; Moritoki, H | 1 |
Affolter, H; Burkard, WP; Pletscher, A | 1 |
Lim, SL; May, PB; Sutter, MC | 1 |
Bracchetti, D; Fulvi, M; Rubboli, A; Sangiorgio, P | 1 |
van Amsterdam, FT; Zaagsma, J | 1 |
Cartheuser, CF | 1 |
Abraham, WM; Ahmed, T; Carpenter, N; D'Brot, J; Kim, CS | 1 |
Catalano, I; Davì, G; Mattina, A; Novo, S; Strano, A | 1 |
Pang, PK; Sham, JS | 1 |
Carmeliet, E; Mubagwa, K | 1 |
Bengtsson, B; Khan, AR; Weiber, R | 1 |
Auguet, M; Clostre, F; DeFeudis, FV; Delaflotte, S | 1 |
Antônio, A; Calixto, JB | 1 |
Smedley, MJ; Stanisstreet, M; Veltkamp, CJ | 1 |
Cai, HR; Stieve, H | 1 |
Bradford, HF; White, EJ | 1 |
Kobayashi, H; Mochida, S | 1 |
Akiyama, S; Kuwano, M; Tomita, K | 1 |
Jackson, GL; Liu, TC | 1 |
Akiyama, S | 1 |
Liron, Z; Roberts, E; Wong, E | 1 |
Kanai, R; Ohashi, M; Takayanagi, I | 1 |
Abel, MH; Hollingsworth, M | 1 |
Barry, WH; Horowitz, JD; Smith, TW | 1 |
Krieglstein, J; Weber, J | 1 |
Pang, CC; Sutter, MC | 2 |
Akerström, G; Gylfe, E; Johansson, H; Larsson, R; Ljunghall, S; Rastad, J; Wallfelt, C | 1 |
Lehmann, HD | 1 |
Ishida, A; Yoneda, T | 1 |
Bender, F | 2 |
McDonald, TF; Pelzer, D; Trautwein, W | 5 |
Clay, JR; Shrier, A | 1 |
Hertle, L; Nawrath, H | 1 |
Callanan, KM; Keenan, AK | 1 |
Schlepper, M | 2 |
Hisayama, T; Suzuki, S; Takayanagi, I | 1 |
Miledi, R; Parker, I | 1 |
Bregestovski, PD; Miledi, R; Parker, I | 1 |
Adler, M; Atlas, D | 1 |
Ohizumi, Y; Shibata, S | 1 |
Charles, S; Henquin, JC; Mathot, F; Nenquin, M; Tamagawa, T | 1 |
Akaike, N; Ito, H; Nishi, K; Oyama, Y | 1 |
Ohashi, M; Takayanagi, I | 1 |
Beckeringh, JJ; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
Elger, CE; Speckmann, EJ; Walden, J; Witte, OW | 1 |
Bertaccini, G; Poli, E; Raddino, R | 1 |
Beckeringh, JJ; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Vila, E | 1 |
Drzewiecki, G; Middleton, E; Triggle, D | 1 |
Rimele, TJ; Vanhoutte, PM | 1 |
Eichelberg, D; Peters, R; Schmutzler, W | 1 |
Ehlert, FJ; Fairhurst, AS; Whittaker, ML | 1 |
Demers, JM; Payet, MD; Ruiz-Ceretti, E; Schanne, OF | 1 |
Swamy, VC; Triggle, DJ | 2 |
Glossmann, H; Hornung, R | 1 |
Payet, MD; Ruiz-Ceretti, E; Schanne, OF | 1 |
Carpenter, CA; Saggerson, ED | 1 |
Erlichman, J; Fleckman, A; Fleischer, N; Schubart, UK | 1 |
Jarrott, B; Nayler, WG; Thompson, JE | 1 |
Zong, XG | 1 |
Hescheler, J; Pelzer, D; Trautwein, W; Trube, G | 1 |
De Schepper, J; Van Bogaert, A | 1 |
Haeusler, G; Holck, M; Thorens, S | 1 |
Lee, KS; Tsien, RW | 1 |
Moger, WH | 1 |
Hannemann, H; Sewing, KF | 1 |
Baker, JE; Hearse, DJ | 1 |
Kojima, M; Sperelakis, N | 1 |
Godin, DV; Moore, MM | 1 |
Carpenter, DO; Haas, HL; Slater, NT | 1 |
Lalanne, C; Lavie, JL; Mironneau, C; Mironneau, J; Savineau, JP | 1 |
Bristow, MR; Ginsburg, R; Laser, JA; McAuley, BJ; Minobe, W | 1 |
Brown, B; Churchill, P | 1 |
Conn, PM; Rogers, DC; Seay, SG | 1 |
Peng, HB | 1 |
Bowles, MJ; Khurmi, NS; O'Hara, MJ; Raftery, EB; Subramanian, VB | 1 |
Drews, H; Hopf, R; Kaltenbach, M | 1 |
Brasseur, R; Deleers, M; Malaisse, WJ | 2 |
Burch, RM; Halushka, PV | 1 |
Kroesen, P | 1 |
Bette, L; Rettig, G; Schieffer, H; Sen, S | 1 |
Pelto, DJ; Rapoport, SI; Suarez-Isla, BA; Thompson, JM | 1 |
Hager, WD; Katz, AM; Messineo, FC; Pappano, AJ | 1 |
Mitchelson, F; Ziegler, A | 1 |
Hume, JR; Uehara, A | 1 |
Defeudis, FV; Taylor, JE | 1 |
Schiemann, J; Sućić, M | 1 |
Eisenberg, RS; McCarthy, RT; Milton, RL | 1 |
Eisenberg, RS; Hui, CS; Milton, RL | 1 |
Dannies, PS; Scammell, JG | 1 |
Hepler, PK; Saunders, MJ | 1 |
Beneit, J; Hidalgo, A; Lorenzo, P | 1 |
DeFeudis, FV; Deghenghi, R; Hertz, F; Ranson, M | 1 |
Mukai, T; Takagi, K | 2 |
Deierkauf, M; Elferink, JG | 1 |
Golling, FR; Kindler, M; Neuss, H; Schlepper, M; Thormann, J; Weissmüller, P | 1 |
Brown, BL; Merritt, JE | 1 |
Dóra, E; Kovách, AG | 1 |
Chaudhry, A; Vohra, MM | 1 |
Ross, WE; Yalowich, JC | 1 |
Babcock, DF; Lardy, HA; Singh, JP | 1 |
Pento, JT | 1 |
Tritthart, HA | 1 |
Dóra, E; Koller, A; Kovách, AG; Szedlacsek, S | 1 |
Blinks, JR; Hess, P; Morgan, JP; Wier, WG | 1 |
Corcoran, JJ; Kirshner, N | 1 |
Engelmann, K; Raschack, M | 1 |
Andersson, A; Drakenberg, T; Forsén, S; Thulin, E | 1 |
Marwaha, J; Treffers, RC | 1 |
Churchill, PC | 1 |
Baumbach, L; Skøtt, O | 1 |
Nghiem, C; Swamy, VC; Triggle, DJ | 2 |
Canga, L; Gimeno, AL; Sterin-Broda, L | 1 |
Ehlert, FJ; Itoga, E; Roeske, WR; Yamamura, HI | 1 |
Cheung, W; Maroko, PR; Ribeiro, LG | 1 |
Asai, F; Nishimura, M; Satoh, E; Urakawa, N | 1 |
Buss, J; Horn, HG; Mitrović, V; Neuss, H; Schlepper, M | 1 |
Hester, RK; Weiss, GB | 1 |
Harmony, JA; Jackson, RJ; Ranganathan, S | 1 |
Pert, CB; Quirion, R | 1 |
Auguet, M; DeFeudis, FV | 1 |
Koidl, B; Tritthart, HA | 1 |
Daly, JW; Ebstein, RP | 1 |
Webb, RC | 1 |
Cheung, WM; Faria, DB; Maroko, PR; Ribeiro, LG | 1 |
Harris, A; Jim, K; Rosenberger, LB; Triggle, DJ | 1 |
Gross, GJ; Jolly, SR; Menahan, LA | 1 |
McNeill, JH; Siegl, PK | 2 |
Van Nueten, JM; Vanhoutte, PM | 1 |
Chudakov, LI; Kafengauz, BIu; Poskonova, MA | 1 |
Brandon, TA; Kim, HS; Maroko, PR; Miller, RR; Ribeiro, LG; Spadaro, J; Titus, JL | 1 |
Israel, JM; Meunier, JM | 1 |
Lin, CS; Nwako, N; Swamy, VC | 1 |
Kubota, K; Mukai, T | 1 |
Diamond, J; Shaikh, MI | 1 |
Lin, CS; Swamy, VC | 1 |
Adams, HR; Durrett, LR | 1 |
Mileva, S; Spassov, G | 1 |
Abendroth, RR; Breithardt, G; Seipel, L; Wiebringhaus, E | 1 |
Bregestovski, PD; Iljin, VI | 1 |
Bradley, MP; Forrester, IT | 1 |
Kirchengast, M; Lehmann, HD; Rübsamen, K | 1 |
Beitlová, D; Bures, P; Fisar, Z; Fuksová, K; Krulík, R; Sikora, J | 1 |
Bosse, E; Flockerzi, V; Hofmann, F; Lacinová, L; Ludwig, A | 1 |
Bolton, TB; Zhang, H | 1 |
Arita, M; Hisatome, I | 1 |
Allegra, A; Aloisi, C; Baldari, S; Buemi, M; Imbesi, D; Laganà, A; Morabito, N; Palella, S; Privitera, M; Villari, C | 1 |
Ananthanarayanan, VS; Zhorov, BS | 1 |
Auriemma, F; Ceriello, A; Macciocchi, B; Papa, A; Scaletta Romeo di Santillo, M; Simonelli, P; Vetrano, A | 1 |
Abraham, WM; Ahmed, T; Chapman, GA; Jackowski, J | 1 |
Nawrath, H; Wegener, JW | 2 |
Degtiar, VE; Döring, F; Glossman, H; Grabner, M; Hering, S; Striessnig, J | 1 |
Hartmann, A; Hopf, R; Kneissl, G; Schnell, J | 1 |
Feher, J; Juhasz, I; Monos, E; Nadasy, GL; Szekacs, B; Vajo, Z | 1 |
Catterall, WA; Hockerman, GH; Johnson, BD; Scheuer, T | 1 |
Piñeros, M; Tester, M | 1 |
Peterlik, M; Pietschmann, P; Redlich, K; Stulc, T | 1 |
Antoine, MH; Cosgrove, KE; Dunne, MJ; Herchuelz, A; Kane, C; Lebrun, P; Ouedraogo, R; Pirotte, B | 1 |
Higuchi, S; Kaneko, K; Masumiya, H; Noguchi, K; Shigenobu, K; Takahashi, K; Tanaka, H | 1 |
Bonini, W; Botto, GL; Broffoni, T | 1 |
Bean, L; Cheng, YF; Neue, UD | 1 |
Ferioli, V; Gamberini, G; Gamberini, MC; Rustichelli, C | 1 |
Catacuzzeno, L; Franciolini, F; Petris, A; Trequattrini, C | 1 |
Jones, SE; McDonald, TF; Missan, S; Zhabyeyev, P | 1 |
Catacuzzeno, L; Franciolini, F; Harper, AA; Petris, A; Trequattrini, C | 1 |
Dietz, A; Geiger, H; Gossmann, J; Kachel, HG; Kramer, W; Mondorf, U; Scheuermann, EH | 1 |
Borlak, J; Levsen, K; Mullett, WM; Pawliszyn, J; Walles, M | 1 |
Dierkes, PW; Hochstrate, P; Schlue, WR; Wende, V | 1 |
Hoda, JC; Huber, IG; Sinnegger-Brauns, MJ; Striessnig, J; Walter-Bastl, D; Wappl-Kornherr, E | 1 |
Awasthi, A; Yadav, A | 1 |
Engel, J; Lacinova, L; Tarabova, B | 1 |
Cheng, RCK; Tikhonov, DB; Zhorov, BS | 1 |
7 review(s) available for verapamil and gallopamil
Article | Year |
---|---|
New developments in Ca2+ channel antagonists.
Topics: Animals; Binding Sites; Calcium; Calcium Channel Blockers; Calmodulin; Electrophysiology; Heart; Humans; Ion Channels; Muscle Relaxation; Muscle, Smooth; Potassium; Sodium; Structure-Activity Relationship; Substrate Specificity | 1983 |
[Fundamental cardiac and vascular effects of Ca++-antagonistic coronary drugs].
Topics: Action Potentials; Adenosine Triphosphate; Animals; Biological Transport; Calcium; Cats; Chemical Phenomena; Chemistry; Coronary Vessels; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Myocardial Contraction; Myocardium; Nifedipine; Oxygen Consumption; Phenethylamines; Prenylamine; Rabbits; Swine; Verapamil | 1975 |
Calcium antagonists and myocardial microperfusion.
Topics: Animals; Calcium Channel Blockers; Coronary Circulation; Coronary Disease; Gallopamil; Guinea Pigs; Humans; Myocardium; Nifedipine; Rats; Ventricular Function, Left; Verapamil | 1991 |
[Calcium antagonists in acute myocardial infarction].
Topics: Calcium Channel Blockers; Diltiazem; Gallopamil; Hemodynamics; Humans; Myocardial Infarction; Nifedipine; Verapamil | 1988 |
Calcium and alpha-adrenoceptors in activation of vascular smooth muscle.
Topics: Animals; Calcium; Diltiazem; Gallopamil; Humans; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Verapamil | 1982 |
Calcium antagonists. Some chemical-pharmacologic aspects.
Topics: Animals; Calcium; Calcium Channel Blockers; Gallopamil; Heart; Humans; Ion Channels; Muscle, Smooth; Potassium; Stereoisomerism; Structure-Activity Relationship; Verapamil | 1983 |
History of calcium antagonists.
Topics: Aniline Compounds; Animals; Calcium; Calcium Channel Blockers; Cardiovascular Diseases; Gallopamil; Heart; Heart Conduction System; Humans; In Vitro Techniques; Magnesium; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Nifedipine; Verapamil | 1983 |
11 trial(s) available for verapamil and gallopamil
Article | Year |
---|---|
Randomized double-blind comparison of gallopamil and propranolol in stable angina pectoris.
Topics: Aged; Angina Pectoris; Clinical Trials as Topic; Double-Blind Method; Electrocardiography; Exercise Test; Female; Gallopamil; Heart Rate; Humans; Male; Middle Aged; Propranolol; Random Allocation; Verapamil | 1984 |
[Anti-angina effect of gallopamil in comparison with another calcium antagonist and a placebo].
Topics: Adult; Aged; Angina Pectoris; Blood Pressure; Clinical Trials as Topic; Coronary Disease; Double-Blind Method; Electrocardiography; Exercise Test; Gallopamil; Heart Rate; Humans; Kinetics; Male; Middle Aged; Myocardial Infarction; Nifedipine; Verapamil | 1984 |
[Comparison of the anti-angina effectiveness of gallopamil to isosorbide dinitrate in long-term medication].
Topics: Angina Pectoris; Clinical Trials as Topic; Female; Gallopamil; Humans; Isosorbide Dinitrate; Long-Term Care; Male; Middle Aged; Verapamil | 1983 |
[Acute and long-term effects of gallopamil (D 600) in stable angina pectoris--a randomized double-blind study].
Topics: Adult; Aged; Angina Pectoris; Clinical Trials as Topic; Double-Blind Method; Electrocardiography; Female; Gallopamil; Humans; Long-Term Care; Male; Middle Aged; Random Allocation; Verapamil | 1983 |
Clinical uses of calcium ion antagonists in arrhythmias.
Topics: Adult; Aged; Alprenolol; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calcium; Child, Preschool; Clinical Trials as Topic; Female; Gallopamil; Humans; Male; Propylamines; Quinidine; Tachycardia, Paroxysmal; Tiapamil Hydrochloride; Verapamil | 1980 |
Hemodynamic effects in patients with cardiac arrhythmias.
Topics: Arrhythmias, Cardiac; Blood Pressure; Clinical Trials as Topic; Digitalis Glycosides; Gallopamil; Heart Rate; Humans; Propranolol; Tachycardia; Verapamil | 1980 |
[The electrophysiological effects of the Ca-antagonists gallopamil (D 600), dimeditiapramine (Ro 11-1781) and verapamil in man (author's transl)].
Topics: Blood Pressure; Bundle of His; Calcium; Electrophysiology; Gallopamil; Heart Block; Humans; Verapamil | 1980 |
Is erythropoietin-induced hypertension a phenomenon due to the intracellular Ca++ mobilisation?
Topics: Adult; Blood Circulation; Calcium; Erythropoietin; Gallopamil; Humans; Ketanserin; Male; Nifedipine; Recombinant Proteins; Vasoconstrictor Agents; Verapamil | 1994 |
[Treatment of ischemic heart disease in the elderly. Comparison of diltiazem, verapamil and gallopamil].
Topics: Age Factors; Aged; Angina Pectoris; Coronary Angiography; Coronary Disease; Diltiazem; Drug Evaluation; Exercise Test; Female; Gallopamil; Humans; Male; Middle Aged; Myocardial Ischemia; Verapamil | 1993 |
Modulation of ventricular rate in permanent atrial fibrillation: randomized, crossover study of the effects of slow-release formulations of gallopamil, diltiazem, or verapamil.
Topics: Administration, Oral; Aged; Anti-Arrhythmia Agents; Atrial Fibrillation; Calcium Channel Blockers; Cardiotonic Agents; Cross-Over Studies; Delayed-Action Preparations; Digoxin; Diltiazem; Electrocardiography, Ambulatory; Female; Gallopamil; Heart Rate; Humans; Male; Middle Aged; Verapamil | 1998 |
A randomized prospective double-blind placebo-controlled study of gallopamil, calcium antagonist of the verapamil type, in stable cyclosporine-treated renal transplant recipients.
Topics: Adult; Blood Pressure; Calcium Channel Blockers; Creatinine; Cyclosporine; Double-Blind Method; Gallopamil; Humans; Immunosuppressive Agents; Kidney Transplantation; Placebos; Prospective Studies; Urea; Uric Acid; Verapamil | 2002 |
284 other study(ies) available for verapamil and gallopamil
Article | Year |
---|---|
Stereoisomers of calcium antagonists which differ markedly in their potencies as calcium blockers are equally effective in modulating drug transport by P-glycoprotein.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Biological Transport; Calcium Channel Blockers; Cell Line; Dihydropyridines; Drug Resistance; Haplorhini; Immunoblotting; Membrane Glycoproteins; Mice; RNA, Messenger; Stereoisomerism; Verapamil; Vinblastine | 1992 |
Studies on Ca2+ channel antagonists. 5-[(3,4-Dimethoxyphenethyl)methylamino]-2-(3,4-dimethoxyphenyl)-2- isopropylpentyl isothiocyanate, a chemoaffinity ligand derived from verapamil.
Topics: Affinity Labels; Animals; Calcium; Calcium Channel Blockers; Chemical Phenomena; Chemistry; Depression, Chemical; Gallopamil; Ion Channels; Myocardial Contraction; Myocardium; Rats; Verapamil | 1986 |
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical | 2010 |
Predictive model for L-type channel inhibition: multichannel block in QT prolongation risk assessment.
Topics: Artificial Intelligence; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Computational Biology; Computer Simulation; Drugs, Investigational; Ether-A-Go-Go Potassium Channels; Expert Systems; Heart Rate; Humans; Models, Biological; Myocytes, Cardiac; NAV1.5 Voltage-Gated Sodium Channel; Potassium Channel Blockers; Quantitative Structure-Activity Relationship; Risk Assessment; Shaker Superfamily of Potassium Channels; Torsades de Pointes; Voltage-Gated Sodium Channel Blockers | 2012 |
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels | 2014 |
The effect of Ca2+ on the metarhodopsin I-II transition. I. Experiments.
Topics: Animals; Calcium; Cations, Monovalent; Cattle; Gallopamil; Hydrogen-Ion Concentration; Kinetics; Models, Biological; Photolysis; Protons; Retinal Pigments; Rhodopsin; Verapamil | 1976 |
Effect of diazoxide, verapamil and compound D600 on isoproterenol and calcium-mediated dose-response relationships in isolated rabbit atrium.
Topics: Adrenergic beta-Antagonists; Animals; Calcium; Diazoxide; Dose-Response Relationship, Drug; Drug Interactions; Female; Gallopamil; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Rabbits; Verapamil | 1977 |
The action of verapamil on the rate of spontaneous release of transmitter at the frog neuromuscular junction.
Topics: Action Potentials; Animals; Anura; Calcium; Dantrolene; Female; Gallopamil; In Vitro Techniques; Male; Motor Endplate; Neuromuscular Junction; Neurotransmitter Agents; Rana pipiens; Temperature; Theophylline; Verapamil | 1979 |
Calcium and stimulus secretion coupling in the neurohypophysis. V. The effects of the Ca2+ ionophores A23187 and X537 A on vasopressin release and 45Ca2+ efflux; interactions with sodium and a verapamil analogue (D600).
Topics: Animals; Anti-Bacterial Agents; Calcimycin; Calcium; Cattle; Culture Media; Drug Interactions; Gallopamil; Gramicidin; L-Lactate Dehydrogenase; Lasalocid; Leucyl Aminopeptidase; Mitochondria; Neurophysins; Pituitary Gland, Posterior; Secretory Rate; Sodium; Vasopressins; Verapamil | 1976 |
Action of calcium antagonists on microsomal calcium activated ATPase of rat aorta.
Topics: Animals; Aorta; Calcium; Calcium-Transporting ATPases; Gallopamil; In Vitro Techniques; Microsomes; Rats; Verapamil | 1978 |
A role of cyclic nucleotides in neuromuscular transmission.
Topics: Adenosine; Alloxan; Animals; Axons; Bucladesine; Cats; Cyclic AMP; Dithionitrobenzoic Acid; Electric Stimulation; Fluorides; Gallopamil; Imidazoles; Muscle Contraction; Muscle Denervation; Muscles; Nerve Endings; Neuromuscular Junction; Prostaglandins E; Synaptic Transmission; Theophylline; Verapamil | 1976 |
[Contractile responses of the guinea pig ileal longitudinal muscle to antispasmodics (author's transl)].
Topics: Acetylcholine; Animals; Benactyzine; Calcium; Cyclic GMP; Drug Synergism; Gallopamil; Guinea Pigs; Ileum; In Vitro Techniques; Male; Manganese; Muscle Contraction; Muscle, Smooth; Papaverine; Verapamil | 1977 |
Effects of ruthenium red, A23187 and D-600 on steroidogenesis in Y-1 cells.
Topics: Adrenocorticotropic Hormone; Anti-Bacterial Agents; Calcimycin; Cell Line; Cyclic AMP; Egtazic Acid; Gallopamil; Pregnenolone; Ruthenium; Ruthenium Red; Steroids; Verapamil | 1978 |
Differential effects of D 600 on release of catecholamines by acetylcholine, histamine, tyramine and by cyclic AMP from canine adrenal medulla.
Topics: Acetylcholine; Adrenal Medulla; Animals; Calcium; Catecholamines; Cyclic AMP; Dogs; Drug Interactions; Female; Gallopamil; Histamine; In Vitro Techniques; Male; Tyramine; Verapamil | 1978 |
The action of D600 on frog skeletal muscle: facilitation of excitation-contraction coupling.
Topics: Action Potentials; Animals; Anura; Calcium; Dose-Response Relationship, Drug; Gallopamil; Hindlimb; Magnesium; Membrane Potentials; Muscle Contraction; Muscles; Physical Stimulation; Rana temporaria; Seasons; Verapamil | 1977 |
[Effect of calcium channel blockaders (verapamil, D-600 and manganese ions) on mediator release from frog muscle motor nerve endings].
Topics: Animals; Anura; Gallopamil; Manganese; Membrane Potentials; Neuromuscular Junction; Rana temporaria; Verapamil | 1977 |
The effects of manganese ions on the contraction of the frog's heart.
Topics: Animals; Anura; Cadmium; Cobalt; Gallopamil; Heart Atria; In Vitro Techniques; Manganese; Membrane Potentials; Myocardial Contraction; Nickel; Rana pipiens; Verapamil | 1977 |
The effects of some organic "calcium antagonists" on calcium influx in presynaptic nerve terminals.
Topics: Animals; Anura; Calcium; Gallopamil; In Vitro Techniques; Nerve Endings; Neuromuscular Junction; Nifedipine; Potassium; Rana pipiens; Rats; Synaptosomes; Verapamil | 1979 |
Inhibition of sodium channels by D600.
Topics: Binding, Competitive; Calcium; Cells, Cultured; Gallopamil; Ion Channels; Myocardium; Neoplasms, Experimental; Neuroblastoma; Sodium; Verapamil; Veratridine | 1979 |
Electromechanical coupling in canine trachealis muscle: acetylcholine contractions.
Topics: Acetylcholine; Animals; Biological Transport, Active; Calcium; Dogs; Gallopamil; In Vitro Techniques; Lanthanum; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Potassium; Trachea; Verapamil | 1979 |
Reentrant ventricular arrhythmias in the late myocardial infarction period. 7. Effect of verapamil and D-600 and the role of the "slow channel".
Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Coronary Disease; Dogs; Electrocardiography; Gallopamil; Heart Conduction System; Heart Ventricles; Myocardial Infarction; Tetrodotoxin; Time Factors; Verapamil | 1979 |
[Comparative analysis of the action of papaverine, novodrin, La3+ and compound D-600 on the guinea pig tenia coli depolarized smooth muscle].
Topics: Animals; Calcium; Colon; Gallopamil; Guinea Pigs; Histamine; History, 20th Century; In Vitro Techniques; Ion Channels; Isoproterenol; Lanthanum; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Papaverine; Time Factors; Verapamil | 1979 |
Effects of methoxyverapamil on the stimulation by Ca2+, Sr2+ and Ba2+ and on the inhibition by Mg2+ of catecholamine release from the adrenal medulla.
Topics: Adrenal Medulla; Animals; Barium; Calcium; Catecholamines; Cations, Divalent; Cattle; Drug Interactions; Gallopamil; In Vitro Techniques; Magnesium; Perfusion; Strontium; Verapamil | 1979 |
The effect of a calcium antagonist (D600) on isoprenaline-induced myocardial necrosis in the rat.
Topics: Animals; Calcium; Cardiomyopathies; Gallopamil; Isoproterenol; Male; Myocardium; Necrosis; Rats; Verapamil | 1979 |
[Effect of verapamil, D-600 and papaverine on the sensitivity of denervated muscle to acetylcholine].
Topics: Acetylcholine; Animals; Calcium; Cell Membrane Permeability; Cobalt; Drug Interactions; Gallopamil; Ion Channels; Manganese; Mice; Muscle Denervation; Muscles; Papaverine; Tubocurarine; Verapamil | 1979 |
The actions and interactions of calcium antagonists and DL-homocysteate on cat spinal motoneurones [proceedings].
Topics: Animals; Cats; Cobalt; Gallopamil; Homocysteine; Motor Neurons; Spinal Cord; Verapamil | 1979 |
Inhibition of high affinity synaptosomal uptake systems by verapamil.
Topics: Animals; Brain; Calcium; Gallopamil; In Vitro Techniques; Kinetics; Male; Rats; Serotonin; Sodium Chloride; Synaptosomes; Time Factors; Verapamil | 1979 |
Inhibitory effects of verapamil, prenylamine and D 600 on Ca2+-dependent noradrenaline release from the sympathetic nerves of isolated rabbit hearts.
Topics: Animals; Calcium; Electric Stimulation; Female; Gallopamil; Heart; In Vitro Techniques; Male; Myocardium; Norepinephrine; Prenylamine; Rabbits; Sodium; Sympathetic Nervous System; Verapamil | 1979 |
The effects of Ca2+ antagonists on Ca2+ accumulation by subcellular fractions of rat myometrium.
Topics: Animals; Biological Transport, Active; Calcium; Cations, Divalent; Chlorpromazine; Female; Gallopamil; Lanthanum; Myometrium; Potassium; Rats; Sodium; Subcellular Fractions; Uterus; Verapamil | 1977 |
Oscillating contractions in protoplasmic strands of Physarum: effects of external Ca++-depletion and Ca++-antagonistic drugs on intrinsic contraction automaticity.
Topics: Calcium; Cytoplasm; Gallopamil; Lanthanum; Manganese; Movement; Myxomycetes; Physarum; Verapamil | 1977 |
Developmental changes in the sensitivity of embryonic heart cells to tetrodotoxin and D600.
Topics: Age Factors; Animals; Biological Transport; Chick Embryo; Culture Techniques; Electric Conductivity; Gallopamil; Heart; Myocardial Contraction; Sodium; Tetrodotoxin; Verapamil; Veratridine | 1978 |
Cardiodepressive and noradrenaline-antagonistic effects of the organic calcium-antagonist D 600 in the spontaneously beating guinea-pig atrium.
Topics: Animals; Depression, Chemical; Electric Stimulation; Gallopamil; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Norepinephrine; Reserpine; Verapamil | 1977 |
Calcium activation systems in vascular smooth muscle.
Topics: Action Potentials; Animals; Blood Vessels; Calcium; Gallopamil; Guinea Pigs; In Vitro Techniques; Muscle, Smooth; Nifedipine; Pyridines; Verapamil | 1977 |
Effect of replacement of extracellular sodium ions and of D-600 on the activation by adrenalin of adenylate cyclase in intact pigeon erythrocytes.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Columbidae; Epinephrine; Erythrocytes; Gallopamil; Kinetics; Lithium; Potassium; Sodium; Verapamil | 1978 |
[Action of the calciumantagonistic compound gallopamile on sinus node, atrioventricular and intraventricular conduction (author's transl)].
Topics: Adult; Aged; Arrhythmia, Sinus; Atrioventricular Node; Bundle of His; Calcium; Cardiac Pacing, Artificial; Electrocardiography; Female; Gallopamil; Heart Block; Heart Conduction System; Heart Rate; Humans; Male; Middle Aged; Myocardial Contraction; Sinoatrial Node; Verapamil | 1978 |
Species differences in responses to hyperosmolality and D600 in cat and rat heart.
Topics: Animals; Cats; Dose-Response Relationship, Drug; Gallopamil; Mannitol; Myocardial Contraction; Osmolar Concentration; Rats; Species Specificity; Stimulation, Chemical; Verapamil | 1978 |
Electrophysiological study of Syrian hamster hereditary cardiomyopathy.
Topics: Action Potentials; Animals; Cardiomyopathies; Cricetinae; Gallopamil; In Vitro Techniques; Membrane Potentials; Mesocricetus; Papillary Muscles; Verapamil | 1978 |
Simplification of retinal photoresponses by D 600 [proceedings].
Topics: Animals; Gallopamil; Membrane Potentials; Photoreceptor Cells; Rats; Verapamil | 1978 |
Effect of verapamil and D 600 on cardiac transmembrane potentials.
Topics: Action Potentials; Animals; Cats; Depression, Chemical; Gallopamil; Guinea Pigs; Heart; Membrane Potentials; Myocardial Contraction; Stimulation, Chemical; Time Factors; Verapamil | 1978 |
Differing actions of nitroprusside and D-600 on tension and 45Ca fluxes in canine renal arteries.
Topics: Animals; Blood Vessels; Calcium; Dogs; Drug Interactions; Female; Ferricyanides; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nitroprusside; Norepinephrine; Potassium; Renal Artery; Time Factors; Verapamil | 1979 |
Calcium-antagonists and islet function. IV. Effect of D600.
Topics: Animals; Biological Transport; Calcium; Gallopamil; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Rats; Theophylline; Verapamil | 1976 |
Reversible Inhibition of Potassium Contractures by optical isomers of verapamil and D 600 on slow muscle fibres of the frog.
Topics: Animals; Calcium; Egtazic Acid; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscles; Potassium; Stereoisomerism; Time Factors; Verapamil | 1976 |
[Microscopic quantification of myocardial necroses in experimental cardiology].
Topics: Animals; Calcitonin; Dose-Response Relationship, Drug; Gallopamil; Histological Techniques; Isoproterenol; Magnesium; Male; Myocardium; Necrosis; Potassium; Prenylamine; Rats; Verapamil | 1976 |
Effects of D-600 and its optical isomers on force of contraction in cat papillary muscles and guinea-pig auricles.
Topics: Animals; Cats; Depression, Chemical; Electric Stimulation; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Stereoisomerism; Time Factors; Verapamil | 1977 |
On the mechanism underlying the action of D-600 on slow inward current and tension in mammalian myocardium.
Topics: Action Potentials; Animals; Calcium; Cats; Dose-Response Relationship, Drug; Gallopamil; Heart; Heart Conduction System; Membrane Potentials; Myocardial Contraction; Papillary Muscles; Verapamil | 1977 |
Stimulation of renal gluconeogenesis by verapamil and D-600.
Topics: Animals; Calcium; Gallopamil; Gluconeogenesis; In Vitro Techniques; Ketoglutaric Acids; Kidney Tubules; Male; Rats; Stimulation, Chemical; Succinates; Verapamil | 1977 |
Effects of Ca2+ and catecholamines on the guinea pig atrium action potential plateau.
Topics: Action Potentials; Animals; Atrial Function; Calcium; Epinephrine; Female; Gallopamil; Guinea Pigs; Heart Atria; In Vitro Techniques; Male; Verapamil | 1977 |
Calcium movements during the release of catecholamines from the adrenal medulla: effects of methoxyverapamil and external cations.
Topics: Adrenal Medulla; Animals; Calcium; Catecholamines; Cattle; Gallopamil; In Vitro Techniques; Magnesium; Sodium; Sorbitol; Verapamil | 1977 |
Effect of D600, practolol, and alterations in magnesium on ionized calcium concentration-response relationships in the intact dog heart.
Topics: Animals; Blood Glucose; Calcium; Cardiac Pacing, Artificial; Cations, Divalent; Dogs; Dose-Response Relationship, Drug; Electrocardiography; Gallopamil; Heart; Heart Conduction System; Magnesium; Practolol; Pressure; Ventricular Function; Verapamil | 1977 |
Effects of D 600 and papaverine on the inotropic response to isoprenaline on left guinea-pig atria under the graded influence of changes of frequency and temperature.
Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Gallopamil; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papaverine; Temperature; Verapamil | 1977 |
The effects of D600 and verapamil on action potential in the X-organ neuron of the crayfish.
Topics: Action Potentials; Animals; Astacoidea; Calcium; Eye; Gallopamil; In Vitro Techniques; Magnesium; Neurons; Verapamil | 1976 |
Some effects of D600, nifedipine and sodium nitroprusside on electrical and mechanical activity in rat portal vein [proceedings].
Topics: Animals; Calcium; Electrophysiology; Ferricyanides; Gallopamil; In Vitro Techniques; Muscle Contraction; Nifedipine; Nitroprusside; Portal Vein; Pyridines; Rats; Verapamil | 1976 |
On the pathogenesis of cardiac necroses induced by theophylline and caffeine.
Topics: Animals; Blood Pressure; Caffeine; Calcium; Gallopamil; Heart; Heart Rate; Isoproterenol; Male; Myocarditis; Myocardium; Necrosis; Oxygen Consumption; Propranolol; Rats; Theophylline; Verapamil | 1976 |
Relationship between internal calcium and outward current in mammalian ventricular muscle; a mechanism for the control of the action potential duration?
Topics: Action Potentials; Animals; Calcium; Cattle; Cyanides; Gallopamil; Heart Ventricles; In Vitro Techniques; Membrane Potentials; Myocardial Contraction; Sheep; Sodium; Ventricular Function; Verapamil | 1976 |
[Mechanism of excitation and contraction uncoupling in frog and guinea pig myocardial fibers during block of slow sodium-calcium channels by compound D-600].
Topics: Action Potentials; Animals; Calcium; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Myocardial Contraction; Rana temporaria; Sodium; Verapamil | 1976 |
Effect of isoproterenol and D-600 on calcium movements in rat myometrium.
Topics: Animals; Calcium; Calcium Radioisotopes; Depression, Chemical; Female; Gallopamil; In Vitro Techniques; Isoproterenol; Kinetics; Lanthanum; Myometrium; Potassium; Pregnancy; Rats; Sodium; Stimulation, Chemical; Uterus; Verapamil | 1975 |
Proceedings: Ca-dependence of supraventricular pacemaker activity and its responsiveness to Ca-antagonistic compounds (verapamil, D 600, nifedipine).
Topics: Animals; Calcium; Gallopamil; Nifedipine; Sinoatrial Node; Verapamil | 1975 |
Proceedings: P- and T-blockade in smooth muscle: a new pharmacological principle.
Topics: Animals; Calcium; Female; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Verapamil | 1975 |
Functional antagonism between calcium-antagonists and noradrenaline on isolated guinea-pig atria.
Topics: Animals; Atrial Function; Calcium; Depression, Chemical; Electric Stimulation; Gallopamil; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Nifedipine; Norepinephrine; Pyridines; Verapamil | 1975 |
Influence of papaverine, D600, and nifedipine on the effects of noradrenaline and calcium on the isolated aorta and mesenteric artery of the rabbit.
Topics: Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Calcium; Calcium Chloride; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Papaverine; Pyridines; Rabbits; Verapamil | 1975 |
Action of D-600 on spontaneous and electrically stimulated activity of the parturient rat uterus.
Topics: Action Potentials; Animals; Depression, Chemical; Electric Stimulation; Evoked Potentials; Female; Gallopamil; In Vitro Techniques; Labor, Obstetric; Membrane Potentials; Muscle, Smooth; Myometrium; Postpartum Period; Pregnancy; Rats; Uterine Contraction; Verapamil | 1975 |
Inotropic and electrophysiological actions of verapamil and D 600 in mammalian myocardium. I. Pattern of inotropic effects of the racemic compounds.
Topics: Action Potentials; Animals; Calcium; Cats; Electric Stimulation; Gallopamil; Lanthanum; Membrane Potentials; Myocardial Contraction; Myocardium; Nickel; Verapamil | 1975 |
Inotropic and electrophysiological actions of verapamil and D 600 in mammalian myocardium. II. Pattern of inotropic effects of the optical isomers.
Topics: Animals; Calcium; Cats; Depression, Chemical; Electric Stimulation; Gallopamil; Myocardial Contraction; Myocardium; Optical Rotation; Stereoisomerism; Verapamil | 1975 |
Inotropic and electrophysiological actions of verapamil and D 600 in mammalian myocardium. III. Effects of the optical isomers on transmembrane action potentials.
Topics: Action Potentials; Animals; Calcium; Cats; Electric Stimulation; Gallopamil; Membrane Potentials; Myocardial Contraction; Myocardium; Optical Rotation; Sinoatrial Node; Sodium; Stereoisomerism; Verapamil | 1975 |
Effects of temperature and spasmolytic agents on the rate of relaxation of intestinal smooth muscle.
Topics: Aminophylline; Animals; Calcium; Cytoplasm; Gallopamil; In Vitro Techniques; Intestines; Manganese; Muscle Contraction; Muscle, Smooth; Papaverine; Parasympatholytics; Rats; Temperature; Verapamil | 1975 |
Functional differentiation of the transmembrane sodium and calcium channels in mammalian cardiac fibers by use of specific inhibitors.
Topics: Animals; Calcium; Cats; Electric Conductivity; Gallopamil; Heart; In Vitro Techniques; Lidocaine; Membrane Potentials; Metals, Alkaline Earth; Myocardial Contraction; Myocardium; Sodium; Strontium; Verapamil | 1975 |
Inhibition of calcium-dependent action potentials in mammalian myocardium by specific inhibitors of the transmembrane calcium conductivity (verapamil, D 600).
Topics: Action Potentials; Animals; Calcium; Cats; Electric Conductivity; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Papillary Muscles; Potassium; Sodium; Verapamil | 1975 |
Restriction of isoproterenol-induced myocardial Ca uptake and necrotization in rats by a new Ca-antagonistic compound (ethyl-4-(3,4,5-trimethoxycinnamoyl) piperazinyl acetate (Vascordil)).
Topics: Animals; Biological Transport; Calcium; Cardiomyopathies; Cinnamates; Dose-Response Relationship, Drug; Gallopamil; Isoproterenol; Myocardium; Necrosis; Piperazines; Prenylamine; Rats; Verapamil | 1975 |
Influence of isoproterenol, propranolol, and D 600 on the de novo synthesis of adenine nucleotides in rat hearts.
Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Female; Gallopamil; Heart; Isoproterenol; Myocardium; Propranolol; Rats; Verapamil | 1975 |
[Influence of anti-arrhythmia agents on electrolyte metabolism].
Topics: Adult; Aged; Anti-Arrhythmia Agents; Coronary Disease; Female; Gallopamil; Humans; Hypertension; Male; Middle Aged; Potassium; Propranolol; Quinidine; Sodium; Verapamil | 1976 |
[Use of panangin, obsidan and isoptin in acute rhythm disorders under conditions of cardiological first aid service].
Topics: Acute Disease; Adolescent; Adult; Aged; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Aspartic Acid; Female; First Aid; Gallopamil; Humans; Male; Middle Aged; Propranolol; Verapamil | 1976 |
The different effects of D-600 (methoxyverapamil) on the release of adrenal catecholamines induced by acetylcholine, high potassium or sodium deprivation.
Topics: Acetylcholine; Adrenal Medulla; Animals; Catecholamines; Cattle; Gallopamil; In Vitro Techniques; Potassium; Sodium; Stimulation, Chemical; Time Factors; Verapamil | 1976 |
Effects of verapamil, gallopamil, diltiazem and nifedipine on sarcoplasmic reticulum function in rat heart.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Diltiazem; Gallopamil; Heart; Nifedipine; Rats; Rats, Sprague-Dawley; Ryanodine; Sarcoplasmic Reticulum; Verapamil | 1992 |
Inotropic effects of calcium antagonists in the cardiomyopathic Syrian hamster.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Cardiomyopathies; Cricetinae; Depression, Chemical; Diltiazem; Gallopamil; Mesocricetus; Myocardial Contraction; Nifedipine; Stimulation, Chemical; Verapamil | 1992 |
Effects of the novel calcium channel blocker, anipamil, on the isolated rabbit heart. Comparison with verapamil and gallopamil.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Blood Pressure; Calcium Channel Blockers; Coronary Circulation; Female; Gallopamil; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Propylamines; Rabbits; Verapamil | 1992 |
Red blood cell partitioning of gallopamil, verapamil and norverapamil.
Topics: Biological Availability; Chromatography, High Pressure Liquid; Erythrocytes; Gallopamil; Humans; In Vitro Techniques; Regression Analysis; Verapamil | 1992 |
Direct determination of the enantiomeric ratio of verapamil, its major metabolite norverapamil and gallopamil in plasma by chiral high-performance liquid chromatography.
Topics: Animals; Chromatography, High Pressure Liquid; Gallopamil; Humans; Male; Microsomes, Liver; Rats; Rats, Inbred Strains; Reproducibility of Results; Stereoisomerism; Verapamil | 1992 |
Myocytes isolated from porcine coronary arteries: reduction of currents through L-type Ca-channels by verapamil-type Ca-antagonists.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cell Separation; Coronary Vessels; Electrophysiology; Gallopamil; Kinetics; Muscle, Smooth, Vascular; Swine; Verapamil | 1991 |
Effects of pinaverium on voltage-activated calcium channel currents of single smooth muscle cells isolated from the longitudinal muscle of the rabbit jejunum.
Topics: Animals; Barium; Calcium Channels; Diltiazem; Flunarizine; Gallopamil; In Vitro Techniques; Ion Channels; Jejunum; Membrane Potentials; Morpholines; Muscle, Smooth; Parasympatholytics; Rabbits; Verapamil | 1990 |
Mechanisms of potassium channel block in rat alveolar epithelial cells.
Topics: Animals; Calcium; Calcium Channels; Capsaicin; Cells, Cultured; Charybdotoxin; Chlorpromazine; Epithelium; Gallopamil; Kinetics; Nifedipine; Phencyclidine; Potassium Channels; Pulmonary Alveoli; Quinidine; Rats; Scorpion Venoms; Tacrine; Tetraethylammonium Compounds; Verapamil | 1990 |
Reduction in myocardial hemorrhage and the extent of necrosis by gallopamil (D600) in dogs with coronary artery reperfusion.
Topics: Animals; Autoradiography; Blood Pressure; Coronary Vessels; Dogs; Female; Gallopamil; Heart Diseases; Heart Rate; Hemorrhage; Male; Myocardial Reperfusion; Necrosis; Verapamil | 1991 |
Calcium antagonists and cardiac noradrenaline release in ischemia.
Topics: Animals; Biological Transport; Calcium; Chromatography, High Pressure Liquid; Cyanides; Gallopamil; Heart; Ischemia; Male; Methoxyhydroxyphenylglycol; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains; Verapamil | 1991 |
Beta-adrenergic agonists stimulate the oxidative pentose phosphate pathway in the rat heart.
Topics: Adenine Nucleotides; Adrenergic beta-Agonists; Animals; Cycloheximide; Dactinomycin; Female; Fenoterol; Gallopamil; Glucosephosphate Dehydrogenase; Heart; Isoproterenol; Myocardium; Oxidation-Reduction; Pentose Phosphate Pathway; Rats; Rats, Inbred Strains; Ribose; Stimulation, Chemical; Time Factors; Verapamil | 1990 |
Interaction of calcium channel antagonists with parietal cell acid production, adenylate cyclase, intracellular-free Ca2+ and H+/K+-ATPase.
Topics: Adenosine Triphosphatases; Adenylyl Cyclases; Animals; Calcium; Calcium Channel Blockers; Carbachol; Gallopamil; Guinea Pigs; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrochloric Acid; Membranes; Nifedipine; Parietal Cells, Gastric; Protons; Stomach; Verapamil | 1990 |
Effects of D600 on hypoxic suppression of K+ currents in isolated type I carotid body cells of the neonatal rat.
Topics: Animals; Animals, Newborn; Calcium; Calcium Channels; Carotid Body; Cells, Cultured; Gallopamil; Magnesium; Oxygen; Potassium; Potassium Channels; Rats; Verapamil | 1990 |
Synthesis and identification of the N-glucuronides of norgallopamil and norverapamil, unusual metabolites of gallopamil and verapamil.
Topics: Animals; Chromatography, High Pressure Liquid; Gallopamil; Gas Chromatography-Mass Spectrometry; Glucuronates; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil | 1990 |
Pharmacologic effects on coronary microvessels during myocardial ischaemia.
Topics: Animals; Blood Flow Velocity; Capillary Permeability; Coronary Circulation; Coronary Disease; Coronary Vessels; Erythrocyte Count; Fatty Acids; Gallopamil; Imidazoles; Indomethacin; Microcirculation; Platelet Count; Rats; Thromboxane-A Synthase; Verapamil | 1990 |
Ca antagonists do not alter aldosterone secretion during established Na depletion.
Topics: Adrenal Glands; Aldosterone; Animals; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Edetic Acid; Female; Gallopamil; Hydrocortisone; Indenes; Ion Channels; Lanthanum; Nifedipine; Nisoldipine; Ryanodine; Sheep; Sodium; Verapamil | 1985 |
[Co2+ activation and D-600 inhibition of sodium transport across the apical membrane of skin epithelial cells in the frog].
Topics: Animals; Biological Transport; Cell Membrane; Cobalt; Epithelium; Gallopamil; Ion Channels; Membrane Potentials; Rana temporaria; Skin; Sodium; Verapamil | 1985 |
The effect of D600 on tonic tension, Na+ inward current, and Na+-Ca2+ exchange in frog heart.
Topics: Animals; Calcium; Gallopamil; In Vitro Techniques; Ion Channels; Ion Exchange; Membrane Potentials; Myocardial Contraction; Myocardium; Rana pipiens; Sodium; Tetrodotoxin; Verapamil | 1985 |
Effects of calcium antagonists on mechanical responses of mammalian skeletal muscles.
Topics: Animals; Calcium; Calcium Channel Blockers; Electric Stimulation; Gallopamil; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Mice; Muscle Contraction; Muscles; Rats; Rats, Inbred Strains; Verapamil | 1985 |
D600 as a direct blocker of Ca-dependent K currents in Helix neurons.
Topics: Animals; Cadmium; Calcium Channel Blockers; Diltiazem; Gallopamil; Helix, Snails; In Vitro Techniques; Ion Channels; Membrane Potentials; Neuromuscular Depolarizing Agents; Neurons; Verapamil | 1985 |
A pharmacological explanation of the use-dependency of the verapamil (and D-600) block of slow calcium channels.
Topics: Animals; Calcium; Decerebrate State; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Ion Channels; Muscle Contraction; Potassium; Rana pipiens; Time Factors; Verapamil | 1986 |
Sidedness of reconstituted calcium channels from muscle transverse tubules as determined by D600 and D890 blockade.
Topics: Animals; Calcium; Gallopamil; Ion Channels; Muscles; Rats; Verapamil | 1986 |
Effect of calcium antagonists on histamine release from human basophil leukocytes.
Topics: Adult; Basophils; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Histamine Release; Humans; In Vitro Techniques; Verapamil | 1986 |
Involvement of ion channels in the induction of proenkephalin A gene expression by nicotine and cAMP in bovine chromaffin cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Colforsin; Cyclic AMP; Enkephalins; Gallopamil; Gene Expression Regulation; Ion Channels; Nicotine; Nifedipine; Protein Precursors; RNA, Messenger; Sodium; Tubocurarine; Verapamil | 1987 |
Inhibition of calcium channels in neuroblastoma x glioma hybrid cells by verapamil, D600, diltiazem and nisoldipine.
Topics: Animals; Calcium; Calcium Channel Blockers; Diltiazem; Gallopamil; Glioma; Ion Channels; Neuroblastoma; Neurons; Nifedipine; Nisoldipine; Tumor Cells, Cultured; Verapamil | 1987 |
Reversal of chloroquine resistance in falciparum malaria independent of calcium channels.
Topics: Animals; Calcium; Chloroquine; Drug Interactions; Drug Resistance; Gallopamil; Ion Channels; Malaria; Plasmodium falciparum; Verapamil | 1988 |
Effects of phenylalkylamine calcium entry blockers on postischemic energy metabolism in the isolated perfused rat brain: stereoselective action of emopamil.
Topics: Animals; Brain; Brain Ischemia; Calcium Channel Blockers; Energy Metabolism; Gallopamil; In Vitro Techniques; Ion Channels; Male; Perfusion; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil | 1988 |
[Exercise capacity of coronary heart disease patients in long-term follow-up with gallopamil in comparison with premedication with verapamil].
Topics: Aged; Angina Pectoris; Arrhythmias, Cardiac; Coronary Disease; Electrocardiography; Exercise Test; Follow-Up Studies; Gallopamil; Humans; Long-Term Care; Middle Aged; Verapamil | 1989 |
Comparative effects of verapamil and D-600 on the contractile responses produced by neurotransmitters and depolarizing agents in the rat isolated seminal vesicle.
Topics: Acetylcholine; Animals; Carbachol; Clonidine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Depolarizing Agents; Neurotransmitter Agents; Norepinephrine; Phenylephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Seminal Vesicles; Verapamil | 1989 |
Block of sodium currents by the calcium antagonist D600 in human heart cell segments.
Topics: Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; Humans; Ion Channels; Middle Aged; Myocardium; Sodium; Verapamil | 1985 |
[Possible participation of slow Na+--Ca++ channels in realizing cholinergic effects on the cardiac pacemaker].
Topics: Acetylcholine; Animals; Calcium; Electric Stimulation; Gallopamil; Heart Conduction System; In Vitro Techniques; Ion Channels; Manganese; Rana temporaria; Receptors, Cholinergic; Sodium; Verapamil | 1985 |
Quantitative determination of verapamil and metabolites in human serum by high-performance liquid chromatography and its application to biopharmaceutic investigations.
Topics: Biopharmaceutics; Biotransformation; Chromatography, High Pressure Liquid; Gallopamil; Humans; Indicators and Reagents; Verapamil | 1989 |
Effects of Ca-antagonists and antispasmodic drugs on contraction by ACh in molluscan smooth muscle.
Topics: Acetylcholine; Animals; Bivalvia; Calcium Channel Blockers; Diltiazem; Dimethylphenylpiperazinium Iodide; Drug Interactions; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Papaverine; Parasympatholytics; Piperidines; Verapamil | 1985 |
Verapamil alters the amplitude and time course of miniature endplate current.
Topics: Animals; Anura; Gallopamil; In Vitro Techniques; Iontophoresis; Motor Endplate; Neuromuscular Junction; Synaptic Transmission; Time Factors; Verapamil | 1985 |
In vitro effects of verapamil and methoxy-verapamil [D 600] on transmembrane sodium and potassium transport in human erythrocytes.
Topics: Biological Transport, Active; Bumetanide; Erythrocytes; Gallopamil; Humans; In Vitro Techniques; Ouabain; Potassium; Sodium; Sodium-Potassium-Exchanging ATPase; Verapamil | 1985 |
Characterization of the Ca2+ coordination site regulating binding of Ca2+ channel inhibitors d-cis-diltiazem, (+/-)bepridil and (-)desmethoxyverapamil to their receptor site in skeletal muscle transverse tubule membranes.
Topics: Barium; Benzazepines; Bepridil; Calcium; Calcium Channel Blockers; Calcium Channels; Diltiazem; Gallopamil; Kinetics; Magnesium; Membranes; Microtubules; Muscles; Pyrrolidines; Receptors, Nicotinic; Strontium; Verapamil | 1985 |
Potentiation of pancuronium induced neuromuscular blockade by calcium channel blockers in vitro.
Topics: Animals; Calcium Channel Blockers; Depression, Chemical; Diltiazem; Drug Synergism; Gallopamil; Male; Neuromuscular Junction; Nifedipine; Nisoldipine; Pancuronium; Rats; Rats, Inbred Strains; Synaptic Transmission; Verapamil | 1985 |
Mode of vasorelaxing action of 5-[3-[[2-(3,4-dimethoxyphenyl)-ethyl]amino]-1-oxopropyl]-2,3,4,5- tetrahydro-1,5-benzothiazepine fumarate (KT-362), a new intracellular calcium antagonist.
Topics: Animals; Caffeine; Calcium Channel Blockers; Diltiazem; Egtazic Acid; Gallopamil; Lanthanum; Male; Methoxamine; Muscle Contraction; Nifedipine; Nitroglycerin; Norepinephrine; Rabbits; Thiazepines; Vasodilation; Verapamil | 1987 |
Verapamil enhances the non-adrenergic twitch response of rat vas deferens.
Topics: Animals; Autonomic Nervous System; Electric Stimulation; Gallopamil; Hydroxydopamines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxidopamine; Prazosin; Rats; Reserpine; Vas Deferens; Verapamil; Yohimbine | 1987 |
Verapamil, an antagonist at 5-hydroxytryptamine receptors of human blood platelets.
Topics: Adenosine Diphosphate; Binding, Competitive; Blood Platelets; Cerebral Cortex; Gallopamil; Humans; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Receptors, Serotonin; Spiperone; Verapamil | 1985 |
Manganese can inhibit or potentiate contractile responses in mesenteric portal vein.
Topics: Animals; Barium; Calcium; Felodipine; Gallopamil; In Vitro Techniques; Male; Manganese; Mesenteric Veins; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Spectrophotometry, Atomic; Strontium; Tissue Distribution; Verapamil | 1988 |
[Calcium antagonists in angina pectoris].
Topics: Angina Pectoris; Angina Pectoris, Variant; Calcium Channel Blockers; Diltiazem; Gallopamil; Humans; Nifedipine; Physical Exertion; Verapamil | 1988 |
Stereoisomers of calcium antagonists discriminate between coronary vascular and myocardial sites.
Topics: Animals; Bepridil; Calcium Channel Blockers; Coronary Vessels; Gallopamil; Heart; In Vitro Techniques; Male; Pyrrolidines; Rats; Stereoisomerism; Verapamil | 1988 |
Slow channel inhibitor effects on brain function: tolerance to severe hypoxia in the rat.
Topics: Animals; Bencyclane; Bepridil; Brain; Calcium Channel Blockers; Cinnarizine; Diltiazem; Electroencephalography; Fendiline; Flunarizine; Gallopamil; Heart Rate; Hypoxia; Nimodipine; Prenylamine; Pyrrolidines; Rats; Rats, Inbred Strains; Respiration; Verapamil | 1988 |
Effect of gallopamil, a calcium channel blocker, on carbachol- and histamine-induced bronchoconstriction in sheep.
Topics: Aerosols; Airway Resistance; Animals; Bronchial Spasm; Carbachol; Female; Gallopamil; Histamine; Infusions, Intravenous; Sheep; Verapamil | 1988 |
In vitro effects of gallopamil on platelet aggregation and thromboxane generation.
Topics: Blood Platelets; Gallopamil; Humans; In Vitro Techniques; Platelet Aggregation; Thromboxanes; Verapamil | 1988 |
Calcium-dependent chronotropic action of bovine parathyroid hormone (1-34) in isolated atria of Japanese quail, Coturnix coturnix japonica.
Topics: Animals; Atrial Function; Calcium; Coturnix; Dose-Response Relationship, Drug; Gallopamil; Heart Rate; Male; Parathyroid Hormone; Peptide Fragments; Propranolol; Quail; Stimulation, Chemical; Verapamil | 1986 |
Interaction of AOA 39, D600, verapamil and diltiazem with cardiac cholinergic effects.
Topics: Animals; Calcium Channel Blockers; Diltiazem; Drug Interactions; Gallopamil; Heart Conduction System; Isoindoles; Nifedipine; Phthalimides; Purkinje Fibers; Quinuclidinyl Benzilate; Rabbits; Radioligand Assay; Receptors, Muscarinic; Tritium; Verapamil | 1987 |
Low potency of Ca antagonists in smooth muscle from different levels of the respiratory tract.
Topics: Animals; Bronchi; Calcium Channel Blockers; Felodipine; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Respiratory Muscles; Trachea; Verapamil | 1987 |
Verapamil as an apparent competitive antagonist of the serotonin receptor of rabbit isolated aorta.
Topics: Animals; Aorta, Thoracic; Binding, Competitive; Cinnarizine; Diltiazem; Flunarizine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Receptors, Serotonin; Verapamil | 1986 |
Effects of compound D600 (methoxyverapamil) on drug-induced contractions of isolated dog uterine muscle.
Topics: Acetylcholine; Animals; Barium; Calcium Chloride; Dogs; Female; Gallopamil; Histamine; In Vitro Techniques; Oxytocin; Uterine Contraction; Verapamil | 1986 |
Effects of calcium antagonists and calcium-buffered salines on wound healing in Xenopus early embryos.
Topics: Animals; Buffers; Calcium; Calcium Channel Blockers; Embryo, Nonmammalian; Female; Gallic Acid; Gallopamil; Microscopy, Electron, Scanning; Sodium Chloride; Verapamil; Wound Healing; Xenopus | 1986 |
Effects of some Ca2+ blockers on receptor potentials of crayfish retina.
Topics: Animals; Astacoidea; Calcium; Calcium Channel Blockers; Evoked Potentials, Visual; Gallopamil; In Vitro Techniques; Photoreceptor Cells; Retina; Trifluoperazine; Verapamil | 1986 |
Participation of intracellular sites in the action of Ca2+ channel blockers.
Topics: Amino Acids; Animals; Calcium Channel Blockers; Calcium Radioisotopes; Cerebral Cortex; Gallopamil; In Vitro Techniques; Potassium; Rats; Synaptosomes; Verapamil; Veratrine | 1986 |
Effects of Ca antagonists on the action potential and their relationship to the muscarinic ACh actions in isolated sympathetic neurons of rabbits.
Topics: Action Potentials; Animals; Calcium Channel Blockers; Cells, Cultured; Cobalt; Gallopamil; Ganglia, Sympathetic; Male; Mollusk Venoms; Nifedipine; omega-Conotoxin GVIA; Rabbits; Receptors, Muscarinic; Verapamil | 1986 |
The effect of calcium antagonists on the proteolytic degradation of low-density lipoprotein in HeLa cells.
Topics: Calcium Channel Blockers; Cell Compartmentation; Chloroquine; Cholesterol; Endocytosis; Female; Gallopamil; HeLa Cells; Humans; Kinetics; Lipoproteins, LDL; Lysosomes; Peptide Hydrolases; Verapamil | 1985 |
Synthesis and release of luteinizing hormone in vitro by rat anterior pituitary cells: effects of gallopamil hydrochloride (D600) and pimozide.
Topics: Alanine; Animals; Carbohydrate Metabolism; Gallopamil; Glucosamine; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Pimozide; Pituitary Gland, Anterior; Rats; Verapamil | 1985 |
[The effect of calcium antagonists on intracellular transport of epidermal growth factor and the conjugate of epidermal growth factor with pseudomonas exotoxin].
Topics: Biological Transport; Calcium Channel Blockers; Cathepsin B; Cathepsins; Cell Line; Cell Survival; Cells, Cultured; Chloroquine; Endotoxins; Enzyme Activation; Epidermal Growth Factor; Gallopamil; Humans; Lysosomes; Neoplasms, Experimental; Nifedipine; Pseudomonas aeruginosa; Verapamil | 1985 |
Verapamil is a competitive inhibitor of gamma-aminobutyric acid and calcium uptakes by mouse brain subcellular particles.
Topics: Animals; Biological Transport; Brain; Calcium; Gallopamil; gamma-Aminobutyric Acid; Kinetics; Mice; Sodium; Synaptosomes; Verapamil | 1985 |
Do D 600 and diltiazem interact with serotonin receptors in rabbit vascular tissues?
Topics: Animals; Aorta; Basilar Artery; Benzazepines; Blood Vessels; Calcium; Dibenzylchlorethamine; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Male; Rabbits; Receptors, Serotonin; Serotonin; Vasoconstriction; Verapamil | 1985 |
The potencies and selectivities of four calcium antagonists as inhibitors of uterine contractions in the rat in vivo.
Topics: Albuterol; Animals; Blood Pressure; Calcium Channel Blockers; Castration; Diltiazem; Female; Gallopamil; Heart Rate; Nifedipine; Pregnancy; Rats; Rats, Inbred Strains; Uterine Contraction; Verapamil | 1985 |
Comparison of negative inotropic potency, reversibility, and effects on calcium influx of six calcium channel antagonists in cultured myocardial cells.
Topics: Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Chick Embryo; Gallopamil; Half-Life; Lidoflazine; Myocardial Contraction; Myocardium; Nifedipine; Perhexiline; Time Factors; Verapamil | 1985 |
Effect of gallopamil on energy metabolism of the isolated perfused rat brain in the postischemic period.
Topics: Adenosine Monophosphate; Adenosine Triphosphate; Animals; Brain; Electroencephalography; Energy Metabolism; Gallopamil; Ischemic Attack, Transient; Male; Mathematics; Perfusion; Phosphocreatine; Rats; Rats, Inbred Strains; Verapamil | 1985 |
Chronic treatment of rats with D-600 causes a compensatory decrease in the calcium requirement for contractility of vascular smooth and cardiac muscles.
Topics: Animals; Blood Pressure; Calcium; Gallopamil; Heart Rate; Hydralazine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Norepinephrine; Portal Vein; Potassium; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Verapamil | 1985 |
Paradoxical effects of K+ and D-600 on parathyroid hormone secretion and cytoplasmic Ca2+ in normal bovine and pathological human parathyroid cells.
Topics: Animals; Calcium; Cattle; Cytoplasm; Drug Antagonism; Gallopamil; Humans; Hyperparathyroidism; Kinetics; Parathyroid Glands; Parathyroid Hormone; Potassium; Verapamil | 1985 |
Pharmacodynamic interaction of gallopamil and propranolol in the conscious dog.
Topics: Animals; Atropine Derivatives; Blood Pressure; Dogs; Drug Interactions; Female; Gallopamil; Heart Rate; Hemodynamics; Kinetics; Male; Myocardial Contraction; Parasympatholytics; Propranolol; Verapamil | 1985 |
Proceedings: Effects of inhibitors against the uptake of 45Ca at the neurosecretory nerve endings.
Topics: Animals; Calcium; Gallopamil; Nerve Endings; Neurosecretory Systems; Rats; Verapamil | 1974 |
[Treatment of heart arrhythmias with calcium antagonists].
Topics: Arrhythmias, Cardiac; Atrioventricular Node; Calcium Channel Blockers; Cardiac Complexes, Premature; Coronary Circulation; Diltiazem; Drug Therapy, Combination; Electrocardiography; Gallopamil; Heart Conduction System; Heart Rate; Humans; Risk; Sinoatrial Node; Tachycardia; Verapamil | 1984 |
Cat ventricular muscle treated with D600: effects on calcium and potassium currents.
Topics: Action Potentials; Animals; Calcium; Cats; Electric Conductivity; Gallopamil; In Vitro Techniques; Ion Channels; Muscles; Papillary Muscles; Potassium; Time Factors; Verapamil | 1984 |
Cat ventricular muscle treated with D600: characteristics of calcium channel block and unblock.
Topics: Action Potentials; Animals; Calcium; Cats; Electric Conductivity; Gallopamil; In Vitro Techniques; Ion Channels; Membrane Potentials; Muscles; Papillary Muscles; Time Factors; Verapamil | 1984 |
Effects of D-600 on sodium current in squid axons.
Topics: Animals; Axons; Decapodiformes; Gallopamil; Ion Channels; Membrane Potentials; Sodium; Verapamil | 1984 |
Calcium channel blockade in smooth muscle of the human upper urinary tract. I. Effects on depolarization-induced activation.
Topics: Action Potentials; Adult; Aged; Calcium; Calcium Channel Blockers; Diltiazem; Gallopamil; Humans; Ion Channels; Kidney Calices; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Papaverine; Potassium; Ureter; Verapamil | 1984 |
Differential effects of D600, nifedipine and dantrolene sodium on excitation-secretion coupling and presynaptic beta-adrenoceptor responses in rat atria.
Topics: Animals; Calcium; Calcium Channel Blockers; Dantrolene; Electric Stimulation; Female; Gallopamil; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Manganese; Nifedipine; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Verapamil | 1984 |
Differentiation of calcium ion antagonism and beta-adrenergic blockade.
Topics: Action Potentials; Adrenergic beta-Antagonists; Blood Pressure; Calcium; Drug Therapy, Combination; Gallopamil; Heart Conduction System; Humans; Myocardial Contraction; Myocardium; Oxygen Consumption; Propranolol; Verapamil | 1980 |
Effects of nonspecific smooth muscle relaxants and Ca-blocker on Ca-release and Ca-binding in microsomal fractions from rabbit taenia coli.
Topics: Animals; Calcium; Colon; Gallopamil; In Vitro Techniques; Male; Microsomes; Papaverine; Parasympatholytics; Piperidines; Rabbits; Verapamil | 1980 |
Blocking of acetylcholine-induced channels by extracellular or intracellular application of D600.
Topics: Acetylcholine; Animals; Gallopamil; Ion Channels; Motor Endplate; Neuromuscular Junction; Rana temporaria; Verapamil | 1980 |
Blocking of frog endplate channels by the organic calcium antagonist D600.
Topics: Acetylcholine; Animals; Gallopamil; Ion Channels; Neuromuscular Junction; Potassium; Rana temporaria; Sodium; Verapamil | 1980 |
alpha-adrenergic antagonists as possible calcium channel inhibitors.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Calcium; Cell Line; Cell Membrane; Dioxanes; Dioxins; Gallopamil; Glioma; Ion Channels; Kinetics; Membrane Potentials; Mice; Neuroblastoma; Rats; Verapamil | 1981 |
Nature of anthopleurin-B-induced release of norepinephrine from adrenergic nerves.
Topics: Adrenergic Fibers; Animals; Cnidaria; Gallopamil; Guanethidine; Guinea Pigs; Intercellular Signaling Peptides and Proteins; Kinetics; Male; Norepinephrine; Ouabain; Peptides; Potassium; Sea Anemones; Tetrodotoxin; Vas Deferens; Verapamil | 1982 |
Diazoxide and D600 inhibition of insulin release. Distinct mechanisms explain the specificity for different stimuli.
Topics: Adrenergic alpha-Antagonists; Animals; Arginine; Calcium; Depression, Chemical; Diazoxide; Epinephrine; Gallopamil; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Lysine; Male; Rats; Rats, Inbred Strains; Theophylline; Verapamil | 1982 |
Actions of calcium antagonists on calcium currents in Helix neurons. Specificity and potency.
Topics: Adrenergic beta-Antagonists; Animals; Calcium; Calcium Channel Blockers; Diltiazem; Gallopamil; Helix, Snails; In Vitro Techniques; Ion Channels; Neurons; Temperature; Verapamil | 1983 |
The actions of D 600, aspaminol and papaverine on calcium-, potassium- and histamine-induced contractions of isolated rabbit basilar artery, aorta, taenia coli and tracheal smooth muscle.
Topics: Animals; Calcium; Dose-Response Relationship, Drug; Gallopamil; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Piperidines; Potassium; Rabbits; Verapamil | 1983 |
Differential effects of the calcium entry blocker D 600 on contractions of rat and guinea-pig aortas, elicited by various alpha-1 adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Vasoconstriction; Verapamil; Yohimbine | 1984 |
Reduction of calcium currents in identified neurons of Helix pomatia: intracellular injection of D890.
Topics: Animals; Calcium; Gallopamil; Helix, Snails; In Vitro Techniques; Ion Channels; Membrane Potentials; Neurons; Sodium; Verapamil | 1984 |
Action of oxmetidine on the rabbit aorta: comparison with some calcium entry blockers and nitroglycerin.
Topics: Animals; Aorta, Thoracic; Calcium Channel Blockers; Female; Gallopamil; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Male; Nifedipine; Nitroglycerin; Rabbits; Vasoconstriction; Verapamil | 1984 |
Lack of effect of D600 on alpha 1-adrenoceptor-mediated contractions of rat isolated anococcygeus muscle.
Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium Channel Blockers; Dose-Response Relationship, Drug; Electric Stimulation; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Potassium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Verapamil | 1984 |
Effects of smooth muscle calcium antagonists on human basophil histamine release.
Topics: Basophils; Calcium; Dantrolene; Gallic Acid; Gallopamil; Histamine Release; Humans; Muscle Contraction; Muscle, Smooth; Nifedipine; Quercetin; Verapamil | 1981 |
Recognition of the 'calcium paradox' and the effects of verapamil and gallopamil in human adenoidal mast cells.
Topics: Adenoids; Calcium; Concanavalin A; Gallopamil; Histamine Release; Humans; Mast Cells; Verapamil | 1984 |
Interactions of D600 (methoxyverapamil) and local anesthetics with rat brain alpha-adrenergic and muscarinic receptors.
Topics: Anesthetics, Local; Animals; Gallopamil; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Lidocaine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Muscarinic; Tetracaine; Verapamil | 1980 |
Inhibitory activity of blockers of the slow inward current in rat myocardium, a study in steady state and of rate of action.
Topics: Animals; Gallopamil; Heart; Ion Channels; Manganese; Mathematics; Membrane Potentials; Rats; Verapamil | 1980 |
On the mechanism of slow calcium channel block in heart.
Topics: Animals; Calcium; Calcium Channel Blockers; Cats; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Myocardial Contraction; Myocardium; Sodium; Verapamil | 1980 |
Pharmacology of agents that affect calcium. Agonists and antagonists.
Topics: Action Potentials; Animals; Calcium; Cats; Cinnarizine; Electrophysiology; Gallopamil; Guinea Pigs; In Vitro Techniques; Ion Channels; Muscle, Smooth; Muscle, Smooth, Vascular; Nifedipine; Nitroprusside; Rabbits; Rats; Verapamil | 1980 |
Calcium- and potassium-channel blockers interact with alpha-adrenoceptors.
Topics: Aminopyridines; Animals; Brain; Calcium; Clonidine; Gallopamil; Guanidines; Ion Channels; Myocardium; Potassium; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Tetraethylammonium Compounds; Verapamil | 1980 |
Competition for slow channel of Ca2+, Mn2+, Verapamil, and D-600 in rat ventricular muscle?
Topics: Animals; Calcium; Dose-Response Relationship, Drug; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Manganese; Membrane Potentials; Myocardium; Rats; Verapamil | 1980 |
Effect of compound D-600 (methoxyverapamil) on gluconeogenesis and on acceleration of the process by alpha-adrenergic stimuli in rat kidney tubules.
Topics: Angiotensin II; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Gallopamil; Gluconeogenesis; Imidazoles; In Vitro Techniques; Kidney Tubules; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Verapamil | 1980 |
Effect of trifluoperazine, D600, and phenytoin on depolarization- and thyrotropin-releasing hormone-induced thyrotropin release from rat pituitary tissue.
Topics: Animals; Calcium; Gallopamil; Ion Channels; Male; Membrane Potentials; Phenytoin; Pituitary Gland, Anterior; Potassium; Rats; Sodium; Thyrotropin; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil; Veratridine | 1981 |
The interaction of calcium antagonists (slow channel blockers) with myocardial alpha adrenoceptors.
Topics: Animals; Brain; Calcium Channel Blockers; Clonidine; Diltiazem; Gallopamil; In Vitro Techniques; Male; Myocardium; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Verapamil | 1982 |
[Changes of action potential in human papillary muscles by methoxyverapamil (author's transl)].
Topics: Action Potentials; Calcium Channel Blockers; Gallopamil; Humans; In Vitro Techniques; Ion Channels; Papillary Muscles; Verapamil | 1982 |
Does the organic calcium channel blocker D600 act from inside or outside on the cardiac cell membrane?
Topics: Action Potentials; Animals; Calcium; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Membrane Potentials; Myocardium; Verapamil | 1982 |
Calcium channel block and recovery from block in mammalian ventricular muscle treated with organic channel inhibitors.
Topics: Action Potentials; Animals; Calcium; Cardiovascular Agents; Cats; Dose-Response Relationship, Drug; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Isoindoles; Phthalimides; Verapamil | 1982 |
Action of a calcium blocking agent (D600) on electrogenesis in the normal heart and the ischaemic heart in the dog.
Topics: Action Potentials; Animals; Calcium Channel Blockers; Coronary Disease; Dogs; Electrocardiography; Gallopamil; Heart; Heart Conduction System; Ion Channels; Myocardial Contraction; Verapamil | 1982 |
Characterization of [3H]nifedipine binding sites in rabbit myocardium.
Topics: Animals; Binding Sites; Calcium; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Ion Channels; Kinetics; Myocardial Contraction; Myocardium; Nifedipine; Pyridines; Rabbits; Stereoisomerism; Tritium; Verapamil | 1982 |
Interval- and voltage-dependent effects of the calcium channel-blocking agents D600 and AQA 39 on mammalian ventricular muscle.
Topics: Action Potentials; Animals; Calcium Channel Blockers; Cats; Diastole; Electric Stimulation; Gallopamil; Heart; Ion Channels; Isoindoles; Phthalimides; Rabbits; Verapamil | 1983 |
Mechanism of calcium channel blockade by verapamil, D600, diltiazem and nitrendipine in single dialysed heart cells.
Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Cats; Diltiazem; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Verapamil | 1983 |
Effects of the calcium-channel blockers cobalt, verapamil, and D600 on Leydig cell steroidogenesis.
Topics: Androgens; Animals; Calcium Channel Blockers; Cobalt; Gallopamil; Leydig Cells; Male; Mice; Phosphoprotein Phosphatases; Protein Biosynthesis; Verapamil | 1983 |
Calcium channel antagonists verapamil and gallopamil are powerful inhibitors of acid secretion in isolated and enriched guinea pig parietal cells.
Topics: Adenosine Triphosphatases; Animals; Bucladesine; Calcium Channel Blockers; Female; Gallopamil; Gastric Acid; Gastric Mucosa; Guinea Pigs; H(+)-K(+)-Exchanging ATPase; Histamine; In Vitro Techniques; Male; Verapamil | 1983 |
Slow calcium channel blockers and the calcium paradox: comparative studies in the rat with seven drugs.
Topics: Animals; Butylamines; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Fendiline; Gallopamil; In Vitro Techniques; Ion Channels; Male; Myocardium; Nifedipine; Prenylamine; Rats; Verapamil | 1983 |
Calcium antagonistic drugs differ in ability to block the slow Na+ channels of young embryonic chick hearts.
Topics: Action Potentials; Animals; Calcium Channel Blockers; Chick Embryo; Gallopamil; In Vitro Techniques; Ion Channels; Myocardium; Nifedipine; Sodium; Verapamil | 1983 |
The protective effects of D-600 and propranolol on reperfusion injury in the anaesthetized rabbit.
Topics: 4-Nitrophenylphosphatase; Adenosine Triphosphate; Anesthesia; Animals; Coronary Circulation; Gallopamil; Heart; Ions; Male; Membranes; Myocardial Contraction; Myocardium; Propranolol; Rabbits; Sarcolemma; Sodium-Potassium-Exchanging ATPase; Subcellular Fractions; Verapamil | 1984 |
Kinetics of acetylcholine-activated cation channel blockade by the calcium antagonist D-600 in Aplysia neurons.
Topics: Acetylcholine; Animals; Aplysia; Calcium; Dose-Response Relationship, Drug; Gallopamil; Ganglia; Ion Channels; Kinetics; Membrane Potentials; Neurons; Receptors, Cholinergic; Synaptic Transmission; Verapamil | 1983 |
Comparison of pinaverium bromide, manganese chloride and D600 effects on electrical and mechanical activities in rat uterine smooth muscle.
Topics: Action Potentials; Animals; Calcium; Chlorides; Egtazic Acid; Female; Gallopamil; In Vitro Techniques; Ion Channels; Manganese; Manganese Compounds; Morpholines; Muscle Contraction; Muscle, Smooth; Myometrium; Pregnancy; Rats; Uterus; Verapamil | 1984 |
Tissue response selectivity of calcium antagonists is not due to heterogeneity of [3H]-nitrendipine binding sites.
Topics: Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Channels; Diltiazem; Female; Gallopamil; In Vitro Techniques; Isometric Contraction; Kinetics; Membranes; Muscle, Smooth, Vascular; Myocardium; Nicardipine; Nifedipine; Organ Specificity; Rabbits; Receptors, Nicotinic; Verapamil | 1984 |
Renal effects of methoxyverapamil in anesthetized rats.
Topics: Anesthesia, Intravenous; Animals; Blood Pressure; Calcium; Gallopamil; Kidney; Male; p-Aminohippuric Acid; Potassium; Rats; Rats, Inbred Strains; Renin; Sodium; Verapamil | 1983 |
Structure-function relationship of calcium ion channel antagonists at the pituitary gonadotrope.
Topics: Animals; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Female; Gallopamil; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Pituitary Gland; Rats; Structure-Activity Relationship; Verapamil; Veratridine | 1983 |
Participation of calcium and calmodulin in the formation of acetylcholine receptor clusters.
Topics: Animals; Calcium; Calmodulin; Cells, Cultured; Embryo, Nonmammalian; Fluorescent Antibody Technique; Gallopamil; Kinetics; Muscles; Nifedipine; Receptors, Cholinergic; Trifluoperazine; Verapamil; Xenopus | 1984 |
Conformational analysis of the calcium-antagonist gallopamil.
Topics: Calcimycin; Calcium Channel Blockers; Gallopamil; Hydrogen-Ion Concentration; Models, Molecular; Molecular Conformation; Verapamil | 1983 |
Verapamil inhibition of vasopressin-stimulated water flow: possible role of intracellular calcium.
Topics: Animals; Arginine Vasopressin; Biological Transport; Bufo marinus; Calcium Channel Blockers; Cell Membrane Permeability; Epithelium; Gallopamil; Osmolar Concentration; Urinary Bladder; Verapamil; Water-Electrolyte Balance | 1983 |
Blockers of calcium permeability inhibit neurite extension and formation of neuromuscular synapses in cell culture.
Topics: Age Factors; Animals; Cadmium; Calcium Channel Blockers; Chick Embryo; Cobalt; Gallopamil; Lanthanum; Manganese; Neuromuscular Junction; Nifedipine; Nitrendipine; Retina; Verapamil | 1984 |
Cellular actions and pharmacology of the calcium channel blocking drugs.
Topics: Action Potentials; Biological Transport, Active; Calcium; Calcium Channel Blockers; Cell Membrane; Gallopamil; Heart; Humans; Muscle Contraction; Verapamil | 1984 |
The effect of gallamine, gallopamil and nifedipine on responses to acetylcholine and carbachol in the taenia of the guinea-pig caecum.
Topics: Acetylcholine; Animals; Atropine; Calcium; Carbachol; Cecum; Drug Interactions; Gallamine Triethiodide; Gallopamil; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Paraoxon; Time Factors; Verapamil | 1984 |
Voltage clamp comparison of the organic calcium channel blockers D-600 and nisoldipine.
Topics: Animals; Anura; Atrial Function; Calcium Channel Blockers; Electrophysiology; Gallopamil; Heart Atria; In Vitro Techniques; Kinetics; Nifedipine; Nisoldipine; Verapamil | 1984 |
Inhibition of [3H]spiperone binding to 5-HT2 receptors of rat cerebral cortex by the calcium antagonists verapamil and D600.
Topics: Animals; Binding, Competitive; Butyrophenones; Cerebral Cortex; Gallopamil; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Verapamil | 1984 |
[Multicenter long-term study of gallopamil in patients with coronary heart disease].
Topics: Adult; Aged; Angina Pectoris; Blood Pressure; Coronary Disease; Electrocardiography; Female; Gallopamil; Heart Rate; Humans; Male; Middle Aged; Time Factors; Verapamil | 1984 |
Paralysis of frog skeletal muscle fibres by the calcium antagonist D-600.
Topics: Action Potentials; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscles; Potassium; Rana temporaria; Temperature; Verapamil | 1983 |
Charge movement in skeletal muscle fibers paralyzed by the calcium-entry blocker D600.
Topics: Animals; Electric Conductivity; Gallopamil; Membrane Potentials; Muscles; Paralysis; Potassium; Rana temporaria; Verapamil | 1984 |
Blockade of Ca2+ channels inhibits K+ contractures but not twitches in skeletal muscle.
Topics: Animals; Calcium Channel Blockers; Gallopamil; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Potassium; Rana pipiens; Verapamil | 1984 |
Veratridine and ouabain stimulate calcium-dependent prolactin release.
Topics: Animals; Bromocriptine; Calcium; Cells, Cultured; Gallopamil; Male; Ouabain; Pituitary Gland, Anterior; Prolactin; Rats; Sodium; Tetrodotoxin; Verapamil; Veratridine; Veratrine | 1983 |
Calcium antagonists and calmodulin inhibitors block cytokinin-induced bud formation in Funaria.
Topics: Calcium; Calmodulin; Cell Division; Cells, Cultured; Chlorpromazine; Cytokinins; Gallic Acid; Gallopamil; Lanthanum; Plant Growth Regulators; Plants; Trifluoperazine; Verapamil | 1983 |
[Effect of calcium antagonists on the response of the rat vas deferens to noradrenaline and field stimulation].
Topics: Animals; Calcium Channel Blockers; Electric Stimulation; Gallopamil; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Inbred Strains; Vas Deferens; Verapamil | 1983 |
Effects of calcium-antagonists on passive cutaneous anaphylaxis in the rat.
Topics: Animals; Calcium Channel Blockers; Diltiazem; Gallopamil; Male; Nifedipine; Passive Cutaneous Anaphylaxis; Rats; Verapamil | 1983 |
[Ba-induced contraction of the guinea pig ileal longitudinal muscle and its inhibition by D-600, benactyzine, and papaverine].
Topics: Animals; Barium; Benactyzine; Calcium; Gallopamil; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Papaverine; Verapamil | 1983 |
[Histamine-induced contraction of the guinea pig taenia coli and its inhibition by D-600, papaverine, and benactyzine].
Topics: Animals; Benactyzine; Calcium; Colon; Gallopamil; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nitroprusside; Papaverine; Verapamil | 1983 |
The effect of verapamil and other calcium antagonists on chemotaxis of polymorphonuclear leukocytes.
Topics: Animals; Calcium; Calcium Channel Blockers; Cell Survival; Chemotaxis, Leukocyte; Diltiazem; Gallopamil; Magnesium; Neutrophils; Perhexiline; Prenylamine; Rabbits; Verapamil | 1984 |
[Regularization of ventricular intervals in atrial fibrillation--electrophysiologic findings on the underlying mechanism].
Topics: Adult; Aged; Atrial Fibrillation; Atrioventricular Node; Cardiac Pacing, Artificial; Electrocardiography; Female; Gallopamil; Heart Conduction System; Heart Rate; Humans; Male; Middle Aged; Verapamil | 1984 |
An investigation of the involvement of calcium in the control of prolactin secretion: studies with low calcium, methoxyverapamil, cobalt and manganese.
Topics: Animals; Calcium; Cells, Cultured; Cobalt; Dose-Response Relationship, Drug; Gallopamil; Male; Manganese; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Verapamil | 1984 |
Contribution of adenosine to the regulation of cerebral blood flow: the role of calcium ions in the adenosine-induced cerebrocortical vasodilatation.
Topics: Adenosine; Animals; Calcium; Calcium Channel Blockers; Cats; Cerebral Cortex; Cerebrovascular Circulation; Gallopamil; Hypoxia; NAD; Oxidation-Reduction; Seizures; Vasodilation; Verapamil | 1984 |
Depletion of cardiac noradrenaline stores by the calcium-channel blocker D-600.
Topics: Animals; Gallopamil; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Time Factors; Verapamil | 1984 |
Potentiation of etoposide-induced DNA damage by calcium antagonists in L1210 cells in vitro.
Topics: Animals; Cell Division; Cell Nucleus; Cell Survival; DNA Replication; DNA, Neoplasm; Drug Synergism; Etoposide; Gallopamil; Kinetics; Leukemia L1210; Mice; Podophyllotoxin; Verapamil | 1984 |
Induction of accelerated acrosome reaction in guinea pig sperm.
Topics: Acrosome; Animals; Biological Transport, Active; Calcium; Egtazic Acid; Gallopamil; Guinea Pigs; Kinetics; Male; Sperm Capacitation; Spermatozoa; Verapamil | 1980 |
The inhibitory effects of D-600 and cobalt on theophylline-mediated calcitonin secretion and calcium distribution in porcine thyroid slices.
Topics: Animals; Calcitonin; Calcium; Cobalt; Gallopamil; In Vitro Techniques; Mannitol; Swine; Theophylline; Thyroid Gland; Verapamil | 1980 |
Pharmacology and electrophysiology of calcium ion antagonists.
Topics: Calcium; Cardiovascular Diseases; Gallopamil; Heart; Humans; Myocardial Contraction; Nitroglycerin; Verapamil | 1980 |
Effect of the organic calcium antagonist D-600 on cerebrocortical vascular and redox responses evoked by adenosine, anoxia, and epilepsy.
Topics: Adenosine; Animals; Blood Volume; Cats; Cerebral Cortex; Cerebrovascular Circulation; Electrocardiography; Gallopamil; Hypoxia; Male; NAD; Oxidation-Reduction; Seizures; Verapamil | 1983 |
Influence of Ca++-channel blocking agents on calcium transients and tension development in isolated mammalian heart muscle.
Topics: Animals; Calcium; Calcium Channel Blockers; Cats; Dogs; Gallopamil; In Vitro Techniques; Myocardial Contraction; Myocardium; Papillary Muscles; Verapamil | 1983 |
Inhibition of calcium uptake, sodium uptake, and catecholamine secretion by methoxyverapamil (D600) in primary cultures of adrenal medulla cells.
Topics: Adrenal Medulla; Animals; Biological Transport, Active; Calcium; Catecholamines; Cattle; Cells, Cultured; Gallopamil; Kinetics; Nicotine; Sodium; Tetrodotoxin; Verapamil; Veratridine | 1983 |
Calcium antagonistic activity and myocardial ischemic protection by both stereoisomers of verapamil.
Topics: Animals; Aorta; Calcium; Coronary Disease; Dose-Response Relationship, Drug; Gallopamil; Heart; Rabbits; Stereoisomerism; Swine; Verapamil | 1983 |
A 113Cd and 1H NMR study of the interaction of calmodulin with D600, trifluoperazine and some other hydrophobic drugs.
Topics: Animals; Binding Sites; Calcium; Calcium-Binding Proteins; Calmodulin; Cattle; Chemical Phenomena; Chemistry; Gallopamil; Magnetic Resonance Spectroscopy; Male; Protein Binding; Testis; Trifluoperazine; Verapamil | 1983 |
Actions of a calium antagonist, the D-600, on electrical and mechanical properties of frog skeletal muscle.
Topics: Animals; Anura; Calcium; Electric Stimulation; Gallopamil; Membrane Potentials; Muscle Contraction; Muscles; Neuromuscular Junction; Rana pipiens; Verapamil | 1980 |
Effect of D-600 on inhibition of in vitro renin release in the rat by high extracellular potassium and angiotensin II.
Topics: Angiotensin II; Animals; Calcium; Gallopamil; In Vitro Techniques; Kidney Cortex; Potassium; Rats; Renin; Secretory Rate; Verapamil | 1980 |
Renin release from isolated rat glomeruli: seasonal variations and effects of D600 on the response to calcium deprivation.
Topics: Animals; Calcium; Gallopamil; In Vitro Techniques; Kidney Glomerulus; Male; Rats; Renin; Seasons; Secretory Rate; Verapamil | 1981 |
Inhibition by D 600 of norepinephrine- and clonidine-induced responses of the aortae from normotensive (WKY) and spontaneously hypertensive rats (SHR).
Topics: Animals; Aorta; Calcium Channel Blockers; Clonidine; Gallopamil; Hypertension; In Vitro Techniques; Norepinephrine; Rats; Rats, Inbred Strains; Vasoconstriction; Verapamil | 1982 |
Extracellular calcium concentration and calcium blocking agents on the action of ouabain on isolated rat atrium.
Topics: Animals; Calcium; Calcium Channel Blockers; Diltiazem; Electric Stimulation; Gallopamil; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Ouabain; Rats; Rats, Inbred Strains; Verapamil | 1982 |
The interaction of [3H]nitrendipine with receptors for calcium antagonists in the cerebral cortex and heart of rats.
Topics: Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Chloride; Cerebral Cortex; Diltiazem; Gallopamil; Kinetics; Lanthanum; Male; Myocardium; Nifedipine; Nitrendipine; Pyridines; Rats; Rats, Inbred Strains; Receptors, Drug; Verapamil | 1982 |
Inhibition by methoxyverapamil of the responses of smooth muscle from spontaneously hypertensive and normotensive rats.
Topics: Animals; Blood Pressure; Calcium; Calcium Channel Blockers; Drug Interactions; Gallopamil; Hypertension; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Verapamil | 1982 |
Influence of the extent of the zone at risk on the effectiveness of drugs in reducing infarct size.
Topics: Animals; Autoradiography; Calcium Channel Blockers; Collateral Circulation; Coronary Circulation; Disease Models, Animal; Dogs; Gallopamil; Myocardial Infarction; Myocardium; Verapamil | 1982 |
Potentiation of indirectly induced muscle twitches by organic calcium antagonists in phrenic nerve-diaphragm muscle preparations of mice.
Topics: Animals; Calcium Channel Blockers; Diltiazem; Gallopamil; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Stimulation, Chemical; Verapamil | 1982 |
[Heart rate reduction in atrial fibrillation with a rapid ventricular response by Gallopamil, a Ca-antagonist (author's transl)].
Topics: Administration, Oral; Adult; Aged; Atrial Fibrillation; Atrioventricular Node; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; Heart Rate; Heart Ventricles; Humans; Middle Aged; Monitoring, Physiologic; Verapamil | 1982 |
Effects of nitroprusside and D600 on norepinephrine and KCl activating systems in canine renal vein.
Topics: Animals; Calcium Radioisotopes; Dogs; Ferricyanides; Gallopamil; In Vitro Techniques; Muscle, Smooth, Vascular; Nitroprusside; Norepinephrine; Potassium Chloride; Renal Veins; Verapamil | 1982 |
Effect of Ca2+ blocking agents on the metabolism of low density lipoproteins in human skin fibroblasts.
Topics: Benzazepines; Calcium Channel Blockers; Dibucaine; Diltiazem; Fendiline; Fibroblasts; Gallopamil; Humans; Kinetics; Lipoproteins, LDL; Nifedipine; Phenethylamines; Prenylamine; Pyridines; Skin; Trifluoperazine; Verapamil | 1982 |
Certain calcium antagonists are potent displacers of [3H]phencyclidine (PCP) binding in rat brain.
Topics: Animals; Binding, Competitive; Brain; Calcium Channel Blockers; Gallopamil; In Vitro Techniques; Nifedipine; Nitrendipine; Olfactory Bulb; Phencyclidine; Rats; Verapamil | 1982 |
Actions of D 600 on isolated rabbit aorta.
Topics: Animals; Aorta; Calcium; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Rabbits; Verapamil | 1982 |
D-600 blocks spontaneous discharge, excitability and contraction of cultured embryonic chick heart cells.
Topics: Action Potentials; Animals; Cells, Cultured; Chick Embryo; Electrophysiology; Gallopamil; Heart; Myocardial Contraction; Verapamil | 1982 |
Release of norepinephrine and dopamine from brain vesicular preparations: effects of calcium antagonists.
Topics: Animals; Benzazepines; Calcium; Cerebral Cortex; Corpus Striatum; Diltiazem; Dopamine; Gallopamil; Guinea Pigs; Kinetics; Male; Norepinephrine; Potassium; Verapamil | 1982 |
D-600 and the membrane stabilizing effect of calcium in vascular smooth muscle.
Topics: Animals; Caffeine; Calcium; Gallopamil; Male; Membranes; Methoxamine; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Verapamil | 1982 |
Conformation analysis of the neutral and protonated forms of gallopamil (D600).
Topics: Calcium Channel Blockers; Chemical Phenomena; Chemistry, Physical; Gallopamil; Molecular Conformation; Verapamil | 1982 |
[Importance of the size of the ischemic area on the beneficial effects of drugs capable of protecting the ischemic myocardium].
Topics: Animals; Blood Pressure; Dogs; Gallopamil; Heart Rate; Myocardial Infarction; Myocardium; Verapamil | 1982 |
Stereoselective and non-stereoselective effects of D 600 (methoxyverapamil) in smooth muscle preparations.
Topics: Animals; Calcium; Gallopamil; Guinea Pigs; Ileum; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Portal Vein; Potassium; Rats; Receptors, Adrenergic; Stereoisomerism; Vas Deferens; Verapamil | 1981 |
Effects of several calcium antagonists and dipyridamole in the isolated perfused guinea pig heart.
Topics: Animals; Calcium; Coronary Circulation; Dipyridamole; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Nifedipine; Oxygen Consumption; Perfusion; Pyridines; Verapamil | 1980 |
Differential effects of D 600 on contractile response of aorta and portal vein from spontaneously hypertensive rats.
Topics: Animals; Aorta; Blood Pressure; Calcium; Gallopamil; Hypertension; Muscle Contraction; Portal Vein; Rats; Verapamil | 1981 |
The negative inotropic potency of compound D 600 in rat, guinea pig, and rabbit cardiac preparations.
Topics: Animals; Calcium; Depression, Chemical; Dose-Response Relationship, Drug; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Rabbits; Rats; Species Specificity; Verapamil | 1980 |
Calcium entry blockers and vascular smooth muscle heterogeneity.
Topics: Animals; Calcium; Calcium Channel Blockers; Cinnarizine; Flunarizine; Gallopamil; Lidoflazine; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Verapamil | 1981 |
[Effect of calcium antagonists on action potentials of muscle fibers in the warm-blooded].
Topics: Action Potentials; Animals; Calcium Channel Blockers; Diaphragm; Gallopamil; In Vitro Techniques; Mice; Muscle Denervation; Muscles; Verapamil | 1981 |
[Effects of D-600 (methoxy-verapamil) on mortality and infarction size after coronary occlusion in rats].
Topics: Animals; Gallopamil; Myocardial Contraction; Myocardial Infarction; Myocardium; Prognosis; Rats; Rats, Inbred Strains; Verapamil | 1981 |
A calcium-dependent acetylcholine depolarization blocked by methoxyverapamil (D600) and procaine in snail neurones.
Topics: Acetylcholine; Animals; Calcium; Cobalt; Gallopamil; Helix, Snails; Membrane Potentials; Neurons; Procaine; Verapamil | 1980 |
Some effects of sodium nitroprusside, methoxyverapamil (D600) and nifedipine on rat portal vein.
Topics: Animals; Calcium; Electrophysiology; Ferricyanides; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitroprusside; Norepinephrine; Phentolamine; Portal Vein; Pyridines; Rats; Verapamil | 1980 |
Interaction of D 600 with phenoxybenzamine-induced adrenergic blockade.
Topics: Animals; Drug Interactions; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phenoxybenzamine; Rats; Sympathetic Nervous System; Time Factors; Vas Deferens; Verapamil | 1980 |
Differences in contractile responses to acetylcholine and serotonin in rat stomach fundus strips.
Topics: Acetylcholine; Animals; Calcium; Gallopamil; In Vitro Techniques; Lanthanum; Muscle Contraction; Muscle, Smooth; Rats; Serotonin; Stomach; Temperature; Verapamil | 1980 |
Influence of frequency and calcium concentration on the inotropic actions of D600 in the rat and guinea pig myocardium.
Topics: Animals; Calcium; Electric Stimulation; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Rats; Species Specificity; Verapamil | 1980 |
Effects of hydralazine and D-600 on KCl induced contraction and phosphorylase activation in rabbit aorta.
Topics: Animals; Aorta; Drug Interactions; Enzyme Activation; Gallopamil; Hydralazine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phosphorylases; Potassium Chloride; Rabbits; Verapamil | 1980 |
Spasmolytic action of verapamil, D600 and cinchocaine on the rat vas deferens.
Topics: Animals; Calcium; Dibucaine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Parasympatholytics; Potassium; Rats; Vas Deferens; Verapamil | 1980 |
A comparison of the influence of La3+, D600 and gentamicin on frequency-force relationships in isolated myocardium.
Topics: Animals; Calcium; Electric Stimulation; Gallopamil; Gentamicins; Guinea Pigs; Heart Rate; In Vitro Techniques; Lanthanum; Male; Myocardial Contraction; Verapamil | 1980 |
Effects of some calcium antagonists on the excitation-contraction coupling in the myocardium under steady-state and nonsteady-state conditions of operation.
Topics: Action Potentials; Animals; Calcium; Electric Stimulation; Gallopamil; Guinea Pigs; In Vitro Techniques; Manganese; Myocardial Contraction; Verapamil | 1980 |
Effect of "calcium antagonist" D-600 on the postsynaptic membrane.
Topics: Acetylcholine; Animals; Calcium; Chlorides; Gallopamil; In Vitro Techniques; Kinetics; Mollusca; Sodium; Synaptic Membranes; Tubocurarine; Verapamil | 1980 |
A sodium-calcium exchange mechanism in plasma membrane vesicles isolated from ram sperm flagella.
Topics: Animals; Biological Transport, Active; Calcium; Carrier Proteins; Cell Membrane; Cell-Free System; Gallopamil; Male; Membrane Proteins; Sheep; Sodium; Sodium-Calcium Exchanger; Sperm Tail; Spermatozoa; Verapamil | 1980 |
Inhibition by the combined Ca2+ and 5-HT2 receptor antagonist nexopamil (LU 49938) of intracoronary thrombus formation in a canine model of arterial stenosis and intimal damage.
Topics: Animals; Calcium; Coronary Circulation; Coronary Thrombosis; Dogs; Female; Gallopamil; Hemodynamics; Injections, Intravenous; Ketanserin; Male; Platelet Aggregation; Platelet Aggregation Inhibitors; Serotonin Antagonists; Verapamil | 1993 |
[Ca(2+)-channel blockers and binding of tricyclic antidepressive agents].
Topics: Animals; Antidepressive Agents, Tricyclic; Blood Platelets; Calcium Channel Blockers; Cattle; Cell Membrane; Desipramine; Gallopamil; Humans; Imipramine; In Vitro Techniques; Lymphocytes; Phosphatidylserines; Synaptic Membranes; Verapamil | 1995 |
The block of the expressed L-type calcium channel is modulated by the beta 3 subunit.
Topics: Animals; Benzimidazoles; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; CHO Cells; Cricetinae; Feedback; Gallopamil; Gene Expression; Intracellular Membranes; Isradipine; Macromolecular Substances; Membrane Potentials; Mibefradil; Microsomes; Myocardium; Rabbits; Recombinant Proteins; Structure-Activity Relationship; Tetrahydronaphthalenes; Transfection; Verapamil | 1995 |
Effect of UK-84149 on voltage-activated calcium currents of single smooth muscle cells from guinea-pig and rabbit jejunum and rabbit coronary artery.
Topics: Animals; Aorta; Arteries; Calcium Channel Blockers; Calcium Channels; Coronary Vessels; Dibenzothiazepines; Dose-Response Relationship, Drug; Evoked Potentials; Gallopamil; Guinea Pigs; Jejunum; Muscle, Smooth, Vascular; Nicardipine; Patch-Clamp Techniques; Rabbits; Time Factors; Verapamil | 1995 |
Effects of catecholamines on the residual sodium channel dependent slow conduction in guinea pig ventricular muscles under normoxia and hypoxia.
Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Calcium Channels; Catecholamines; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Hypoxia; In Vitro Techniques; Isoproterenol; Membrane Potentials; Myocardial Infarction; Myocardium; Norepinephrine; Pindolol; Potassium; Sodium Channels; Verapamil | 1995 |
Conformational analysis of free and Ca(2+)-bound forms of verapamil and methoxyverapamil.
Topics: Binding Sites; Calcium; Computer Simulation; Gallopamil; Models, Molecular; Molecular Conformation; Verapamil | 1993 |
Ovine tracheal muscle contraction in vitro: inhibition by calcium channel blockers gallopamil and verapamil.
Topics: Acetylcholine; Animals; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Sheep; Trachea; Verapamil | 1993 |
Extracellular site of action of phenylalkylamines on L-type calcium current in rat ventricular myocytes.
Topics: Animals; Binding Sites; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Gallopamil; Heart Ventricles; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Verapamil | 1995 |
Transfer of L-type calcium channel IVS6 segment increases phenylalkylamine sensitivity of alpha1A.
Topics: Amino Acid Sequence; Animals; Calcium Channel Blockers; Calcium Channels; Gallopamil; Molecular Sequence Data; Rabbits; Structure-Activity Relationship; Verapamil; Xenopus laevis | 1996 |
Persisting effect of Ca(2+)-channel blockers on left ventricular function in hypertrophic cardiomyopathy after 14 years' treatment.
Topics: Adult; Calcium Channel Blockers; Cardiomyopathy, Hypertrophic; Echocardiography, Doppler, Pulsed; Exercise Test; Female; Gallopamil; Humans; Male; Middle Aged; Time Factors; Treatment Outcome; Ventricular Function, Left; Verapamil | 1996 |
Prostacyclin and thromboxane production of rat and cat arterial tissue is altered independently by several vasoactive substances.
Topics: 6-Ketoprostaglandin F1 alpha; Angiotensin II; Animals; Antihypertensive Agents; Aorta; Bradykinin; Calcium Channel Blockers; Cardiotonic Agents; Cats; Dopamine; Dose-Response Relationship, Drug; Epoprostenol; Gallopamil; Isoproterenol; Norepinephrine; Phentolamine; Propranolol; Rats; Thrombin; Thromboxane B2; Vasoconstrictor Agents; Vasodilator Agents; Vasopressins; Verapamil | 1996 |
Distinct effects of mutations in transmembrane segment IVS6 on block of L-type calcium channels by structurally similar phenylalkylamines.
Topics: Amino Acid Sequence; Aniline Compounds; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Electrophysiology; Gallopamil; Kinetics; Molecular Sequence Data; Mutation; Protein Structure, Secondary; Structure-Activity Relationship; Verapamil | 1996 |
Action of tertiary phenylalkylamines on cardiac transient outward current from outside the cell membrane.
Topics: Animals; Gallopamil; Heart; Hydrogen-Ion Concentration; Rats; Rats, Sprague-Dawley; Verapamil | 1996 |
Characterization of the high-affinity verapamil binding site in a plant plasma membrane Ca2+-selective channel.
Topics: Binding Sites; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Gallopamil; Membrane Potentials; Plant Roots; Triticum; Verapamil | 1997 |
Comparative study on the effect of calcium channel blockers on basal and parathyroid hormone-induced bone resorption in vitro.
Topics: Amlodipine; Animals; Bone Resorption; Calcium Channel Blockers; Gallopamil; Mice; Nifedipine; Organ Culture Techniques; Parathyroid Hormone; Parietal Bone; Specific Pathogen-Free Organisms; Verapamil | 1997 |
Verapamil, a phenylalkylamine Ca2+ channel blocker, inhibits ATP-sensitive K+ channels in insulin-secreting cells from rats.
Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Channel Blockers; Calcium Radioisotopes; Female; Gallopamil; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Potassium Channel Blockers; Potassium Channels; Pyridines; Rats; Rubidium Radioisotopes; Thiadiazines; Verapamil | 1997 |
Comparative effects of gallopamil and verapamil on the mechanical and electrophysiological parameters of isolated guinea-pig myocardium.
Topics: Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Electrophysiology; Gallopamil; Guinea Pigs; Heart; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Ventricular Function, Right; Verapamil | 1997 |
Straightforward solid-phase extraction method for the determination of verapamil and its metabolite in plasma in a 96-well extraction plate.
Topics: Animals; Chromatography, Liquid; Gallopamil; Swine; Verapamil | 1998 |
Properties of the racemic species of verapamil hydrochloride and gallopamil hydrochloride.
Topics: Calcium Channel Blockers; Chemistry Techniques, Analytical; Chromatography, High Pressure Liquid; Crystallization; Gallopamil; Spectrophotometry, Infrared; Spectroscopy, Fourier Transform Infrared; Stereoisomerism; Structure-Activity Relationship; Temperature; Verapamil; X-Ray Diffraction | 1999 |
Mechanism of verapamil block of a neuronal delayed rectifier K channel: active form of the blocker and location of its binding domain.
Topics: Animals; Binding Sites; Binding, Competitive; Biotransformation; Calcium Channel Blockers; Chick Embryo; Electrophysiology; Gallopamil; Ganglia, Spinal; Kinetics; Neurons; Potassium Channel Blockers; Potassium Channels; Tetraethylammonium; Verapamil | 1999 |
Selective phenylalkylamine block of I(Kr) over other K(+) currents in guinea-pig ventricular myocytes.
Topics: Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Heart Ventricles; Male; Membrane Potentials; Phenethylamines; Potassium Channels; Time Factors; Ventricular Function; Verapamil | 2000 |
Verapamil block of large-conductance Ca-activated K channels in rat aortic myocytes.
Topics: Animals; Anti-Arrhythmia Agents; Aorta; Binding Sites; Gallopamil; Kinetics; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Rats; Rats, Wistar; Verapamil | 2001 |
Multidimensional on-line sample preparation of verapamil and its metabolites by a molecularly imprinted polymer coupled to liquid chromatography-mass spectrometry.
Topics: Animals; Cells, Cultured; Chromatography, High Pressure Liquid; Gallopamil; Male; Mass Spectrometry; Polymers; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Specimen Handling; Verapamil | 2004 |
L-type Ca2+ channel antagonists block voltage-dependent Ca2+ channels in identified leech neurons.
Topics: Animals; Caffeine; Calcium Channel Blockers; Calcium Channels, L-Type; Diltiazem; Gallopamil; Leeches; Membrane Potentials; Neurons; Nifedipine; Phosphodiesterase Inhibitors; Verapamil | 2004 |
Opposite effects of a single IIIS5 mutation on phenylalkylamine and dihydropyridine interaction with L-type Ca2+ channels.
Topics: Animals; Brain; Calcium; Calcium Channels; Calcium Channels, L-Type; Carrier Proteins; Cell Membrane; Dihydropyridines; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Gallopamil; Homozygote; In Situ Hybridization; Isradipine; Kinetics; Mice; Mice, Transgenic; Microsomes; Models, Biological; Mutation; Oocytes; Protein Binding; Protein Structure, Tertiary; Recombinant Proteins; RNA, Complementary; Steroid Isomerases; Tyrosine; Verapamil; Xenopus laevis | 2004 |
Pharmacophoric features and Ca2+ ion holding capacity of verapamil.
Topics: Calcium; Calcium Channel Blockers; Gallopamil; Hydrogen Bonding; Models, Molecular; Molecular Conformation; Verapamil | 2005 |
Effects of phenylalkylamines and benzothiazepines on Ca(v)1.3-mediated Ca2+ currents in neonatal mouse inner hair cells.
Topics: Algorithms; Animals; Animals, Newborn; Benzazepines; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Hair Cells, Auditory, Inner; Membrane Potentials; Mice; Mice, Inbred Strains; Phenethylamines; Verapamil | 2007 |
Structural model for phenylalkylamine binding to L-type calcium channels.
Topics: Amino Acid Sequence; Binding Sites; Calcium Channel Blockers; Calcium Channels, L-Type; Computer Simulation; Dihydropyridines; Gallopamil; Models, Molecular; Molecular Sequence Data; Molecular Structure; Monte Carlo Method; Protein Structure, Tertiary; Sequence Alignment; Structure-Activity Relationship; Verapamil | 2009 |