verapamil and gallopamil

verapamil has been researched along with gallopamil in 302 studies

Research

Studies (302)

TimeframeStudies, this research(%)All Research%
pre-1990250 (82.78)18.7374
1990's40 (13.25)18.2507
2000's9 (2.98)29.6817
2010's3 (0.99)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dietel, M; Höllt, V; Kouba, M; Vogt, G1
Giacomini, JC; Giacomini, KM; Nelson, WL; Theodore, LJ; Zobrist, RH1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Janis, RA; Triggle, DJ1
Campillo, NE; Guerra, A; Páez, JA1
Fijorek, K; Glinka, A; Mendyk, A; Polak, S; Wiśniowska, B1
Brouillette, WJ; Brown, GB; Zha, C1
Emrich, HM; Reich, R1
Bristow, MR; Green, RD1
Duncan, CJ; Publicover, SJ1
Robinson, IC; Russell, JT; Thorn, NA1
Godfraind, T; Morel, N1
Dretchen, KL; Morgenroth, VH; Skirboll, LR; Standaert, FG1
Kin, M; Kubota, K; Uruno, T1
Carchman, RA; Warner, W1
Hiwatari, M; Taira, N1
Dörrscheidt-Käfer, M1
Gotgil'f, NM; Magazanik, LG1
Chapman, RA; Ellis, D1
Blaustein, MP; Nachshen, DA1
Catterall, WA; Galper, JB2
Coburn, RF1
El-Sherif, N; Lazzara, R1
Galkin, AA; Khodorov, BI1
Aguirre, J; Falutz, J; Pinto, JE; Trifaró, JM1
Powell, T; Rowles, PM; Steen, E; Woolf, N1
Babskaia, NE; Kafengauz, BIu; Poskonova, MA1
Engberg, I; Flatman, JA; Lambert, JD1
McGee, R; Schneider, JE1
Göthert, M; Nawroth, P; Neumeyer, H1
Crankshaw, DJ; Daniel, EE; Janis, RA1
Götz von Olenhusen, K; Wohlfarth-Bottermann, KE1
Schümann, HJ; Wagner, J1
Golenhofen, K2
Campbell, AK; Siddle, K1
Beck, OA; Hochrein, H; Lehmann, HU; Witt, E1
Adcock, RC; Templeton, GH; Wheelan, S; Wildenthal, K; Willerson, JT1
Rossner, KL; Sachs, HG1
Low, JC1
Kecskeméti, V; Kelemen, K; Knoll, J1
Fry, WJ; Hester, RK; Weiss, GB1
Devis, G; Malaisse, WJ; Pipeleers, DG; Somers, G1
Kaumann, AJ; Uchitel, OD1
Leder, O1
Ludwig, C; Nawrath, H1
Eick, RE; McDonald, TF; Nawrath, H; Trautwein, W1
Ferris, RK; Gordon, EE1
Robinson, RB; Sleator, WW1
Aguirre, J; Pinto, JE; Trifaró, JM1
Bristow, MR; Daniels, JR; Harrison, DC; Kernoff, RS1
Freynik, P; Reinhardt, D; Schümann, HJ1
Kuroda, T1
Jetley, M; Weston, AH2
Hoffmann, A; Siegers, CP; Sierra-Callejas, JL; Strubelt, O1
Bassingthwaighte, JB; Fry, CH; McGuigan, JA1
Ignat'eva, VB; Khodorov, BI; Kitaĭgorodskaia, GM; Mukumov, MR; Vornovitskiĭ, EG1
Fleckenstein, A2
Bianchi, CP; Kroeger, EA; Marshall, JM1
Fleckenstein, A; Haastert, HP1
Görlitz, BD; Schümann, HJ; Wagner, J2
Marshall, JM; Reiner, O1
Bayer, R; Hennekes, R; Kaufmann, R; Mannhold, R1
Bayer, R; Kaufmann, R; Mannhold, R1
Bayer, R; Kalusche, D; Kaufmann, R; Mannhold, R1
Hurwitz, L; Tomiyama, A1
Kohlhardt, M1
Fleckenstein, A; Tritthart, H; Volkmann, R; Weiss, R1
Fleckenstein, A; Janke, J; Sigel, H1
Gerlach, E; Zimmer, HG1
Bogoliubov, VM; Gribkova, IN; Kruglova, ZG; Lyskova, MN1
Danilenko, AM; Fialko, VA; Rodionov, VM; Siianov, VS1
Pinto, JE; Trifaró, JM1
Galbani, P; Limbruno, U; Mariani, M; Ronca, G; Ronca-Testoni, S; Yu, G; Zucchi, R1
Finkel, MS; Oddis, CV; Romeo, RC; Salama, G1
Ferrari, R; Pasini, E; Poli, E; Raddino, R1
Czejka, MJ; Podesser, B; Zwoelfer, N1
Blaschke, G; Fieger, H1
Isenberg, G; Klöckner, U1
Beech, DJ; Bolton, TB; Christen, MO; MacKenzie, I1
DeCoursey, TE; Jacobs, ER1
Köbler, W; Möller, P; Neumann, FJ; Parekh, N; Steinhausen, M; Tillmanns, H; Waas, W; Zimmermann, R1
Endo, T; Hayakawa, H; Maroko, PR; Sato, N1
Haass, M; Richardt, G; Schömig, A1
Ibel, H; Suchner, U; Zimmer, HG1
Beil, W; Bersimbaev, RJ; Hannemann, H; Sewing, KF1
Peers, C1
Mutlib, AE; Nelson, WL1
Dorigo, O; Kübler, W; Neumann, FJ; Parekh, N; Steinhausen, M; Tiefenbacher, C; Tillmanns, H; Zimmermann, R1
Coghlan, JP; Denton, DA; Hardy, KJ; Johnson, EI; McDougall, JG; Scoggins, BA; Wright, RD1
Natochin, IuV1
Horackova, M1
Gallant, EM; Goettl, VM1
Ducreux, C; Gola, M1
Frank, GB2
Affolter, H; Coronado, R1
Froldi, M; Leggieri, E; Lorini, M; Miadonna, A; Tedeschi, A; Zanussi, C1
Höllt, V; Kley, N; Loeffler, JP; Pittius, CW1
Bodewei, R; Hering, S; Schubert, B; Wollenberger, A1
Van Dyke, K; Ye, ZG1
Bielenberg, GW; Krieglstein, J; Weber, J1
Reiterer, W1
Greenidge, E; Wali, FA1
Bustamante, JO1
Graser, T; Kurella, GA; Sukhova, GS; Udel'nov, MG1
Czogalla, W; Dilger, C; Jaeger, H; Otto, R; Salama, ZB1
Ishikawa, T; Murakami, H; Watanabe, H1
Edeson, RO; Madsen, BW; Milne, RK1
Boero, R; Deabate, MC; Forneris, G; Guarena, C; Piccoli, G; Quarello, F; Rosati, C1
Fosset, M; Galizzi, JP; Lazdunski, M1
Ilias, W; Steinbereithner, K1
Ambrosini, F; Bertoni, T; Finzi, A; Foresti, A; Lotto, A; Massari, FM; Matta, F; Valentini, R1
Hester, RK; Satake, N; Shibata, S; Tomiyama, A; Ueda, S; Wakabayashi, S1
Fukuda, H; Ishida, Y; Iwamoto, T; Kanaya, J; Maeshiba, Y; Moritoki, H1
Affolter, H; Burkard, WP; Pletscher, A1
Lim, SL; May, PB; Sutter, MC1
Bracchetti, D; Fulvi, M; Rubboli, A; Sangiorgio, P1
van Amsterdam, FT; Zaagsma, J1
Cartheuser, CF1
Abraham, WM; Ahmed, T; Carpenter, N; D'Brot, J; Kim, CS1
Catalano, I; Davì, G; Mattina, A; Novo, S; Strano, A1
Pang, PK; Sham, JS1
Carmeliet, E; Mubagwa, K1
Bengtsson, B; Khan, AR; Weiber, R1
Auguet, M; Clostre, F; DeFeudis, FV; Delaflotte, S1
Antônio, A; Calixto, JB1
Smedley, MJ; Stanisstreet, M; Veltkamp, CJ1
Cai, HR; Stieve, H1
Bradford, HF; White, EJ1
Kobayashi, H; Mochida, S1
Akiyama, S; Kuwano, M; Tomita, K1
Jackson, GL; Liu, TC1
Akiyama, S1
Liron, Z; Roberts, E; Wong, E1
Kanai, R; Ohashi, M; Takayanagi, I1
Abel, MH; Hollingsworth, M1
Barry, WH; Horowitz, JD; Smith, TW1
Krieglstein, J; Weber, J1
Pang, CC; Sutter, MC2
Akerström, G; Gylfe, E; Johansson, H; Larsson, R; Ljunghall, S; Rastad, J; Wallfelt, C1
Lehmann, HD1
Ishida, A; Yoneda, T1
Bender, F2
McDonald, TF; Pelzer, D; Trautwein, W5
Clay, JR; Shrier, A1
Hertle, L; Nawrath, H1
Callanan, KM; Keenan, AK1
Schlepper, M2
Hisayama, T; Suzuki, S; Takayanagi, I1
Miledi, R; Parker, I1
Bregestovski, PD; Miledi, R; Parker, I1
Adler, M; Atlas, D1
Ohizumi, Y; Shibata, S1
Charles, S; Henquin, JC; Mathot, F; Nenquin, M; Tamagawa, T1
Akaike, N; Ito, H; Nishi, K; Oyama, Y1
Ohashi, M; Takayanagi, I1
Beckeringh, JJ; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Elger, CE; Speckmann, EJ; Walden, J; Witte, OW1
Bertaccini, G; Poli, E; Raddino, R1
Beckeringh, JJ; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Vila, E1
Drzewiecki, G; Middleton, E; Triggle, D1
Rimele, TJ; Vanhoutte, PM1
Eichelberg, D; Peters, R; Schmutzler, W1
Ehlert, FJ; Fairhurst, AS; Whittaker, ML1
Demers, JM; Payet, MD; Ruiz-Ceretti, E; Schanne, OF1
Swamy, VC; Triggle, DJ2
Glossmann, H; Hornung, R1
Payet, MD; Ruiz-Ceretti, E; Schanne, OF1
Carpenter, CA; Saggerson, ED1
Erlichman, J; Fleckman, A; Fleischer, N; Schubart, UK1
Jarrott, B; Nayler, WG; Thompson, JE1
Zong, XG1
Hescheler, J; Pelzer, D; Trautwein, W; Trube, G1
De Schepper, J; Van Bogaert, A1
Haeusler, G; Holck, M; Thorens, S1
Lee, KS; Tsien, RW1
Moger, WH1
Hannemann, H; Sewing, KF1
Baker, JE; Hearse, DJ1
Kojima, M; Sperelakis, N1
Godin, DV; Moore, MM1
Carpenter, DO; Haas, HL; Slater, NT1
Lalanne, C; Lavie, JL; Mironneau, C; Mironneau, J; Savineau, JP1
Bristow, MR; Ginsburg, R; Laser, JA; McAuley, BJ; Minobe, W1
Brown, B; Churchill, P1
Conn, PM; Rogers, DC; Seay, SG1
Peng, HB1
Bowles, MJ; Khurmi, NS; O'Hara, MJ; Raftery, EB; Subramanian, VB1
Drews, H; Hopf, R; Kaltenbach, M1
Brasseur, R; Deleers, M; Malaisse, WJ2
Burch, RM; Halushka, PV1
Kroesen, P1
Bette, L; Rettig, G; Schieffer, H; Sen, S1
Pelto, DJ; Rapoport, SI; Suarez-Isla, BA; Thompson, JM1
Hager, WD; Katz, AM; Messineo, FC; Pappano, AJ1
Mitchelson, F; Ziegler, A1
Hume, JR; Uehara, A1
Defeudis, FV; Taylor, JE1
Schiemann, J; Sućić, M1
Eisenberg, RS; McCarthy, RT; Milton, RL1
Eisenberg, RS; Hui, CS; Milton, RL1
Dannies, PS; Scammell, JG1
Hepler, PK; Saunders, MJ1
Beneit, J; Hidalgo, A; Lorenzo, P1
DeFeudis, FV; Deghenghi, R; Hertz, F; Ranson, M1
Mukai, T; Takagi, K2
Deierkauf, M; Elferink, JG1
Golling, FR; Kindler, M; Neuss, H; Schlepper, M; Thormann, J; Weissmüller, P1
Brown, BL; Merritt, JE1
Dóra, E; Kovách, AG1
Chaudhry, A; Vohra, MM1
Ross, WE; Yalowich, JC1
Babcock, DF; Lardy, HA; Singh, JP1
Pento, JT1
Tritthart, HA1
Dóra, E; Koller, A; Kovách, AG; Szedlacsek, S1
Blinks, JR; Hess, P; Morgan, JP; Wier, WG1
Corcoran, JJ; Kirshner, N1
Engelmann, K; Raschack, M1
Andersson, A; Drakenberg, T; Forsén, S; Thulin, E1
Marwaha, J; Treffers, RC1
Churchill, PC1
Baumbach, L; Skøtt, O1
Nghiem, C; Swamy, VC; Triggle, DJ2
Canga, L; Gimeno, AL; Sterin-Broda, L1
Ehlert, FJ; Itoga, E; Roeske, WR; Yamamura, HI1
Cheung, W; Maroko, PR; Ribeiro, LG1
Asai, F; Nishimura, M; Satoh, E; Urakawa, N1
Buss, J; Horn, HG; Mitrović, V; Neuss, H; Schlepper, M1
Hester, RK; Weiss, GB1
Harmony, JA; Jackson, RJ; Ranganathan, S1
Pert, CB; Quirion, R1
Auguet, M; DeFeudis, FV1
Koidl, B; Tritthart, HA1
Daly, JW; Ebstein, RP1
Webb, RC1
Cheung, WM; Faria, DB; Maroko, PR; Ribeiro, LG1
Harris, A; Jim, K; Rosenberger, LB; Triggle, DJ1
Gross, GJ; Jolly, SR; Menahan, LA1
McNeill, JH; Siegl, PK2
Van Nueten, JM; Vanhoutte, PM1
Chudakov, LI; Kafengauz, BIu; Poskonova, MA1
Brandon, TA; Kim, HS; Maroko, PR; Miller, RR; Ribeiro, LG; Spadaro, J; Titus, JL1
Israel, JM; Meunier, JM1
Lin, CS; Nwako, N; Swamy, VC1
Kubota, K; Mukai, T1
Diamond, J; Shaikh, MI1
Lin, CS; Swamy, VC1
Adams, HR; Durrett, LR1
Mileva, S; Spassov, G1
Abendroth, RR; Breithardt, G; Seipel, L; Wiebringhaus, E1
Bregestovski, PD; Iljin, VI1
Bradley, MP; Forrester, IT1
Kirchengast, M; Lehmann, HD; Rübsamen, K1
Beitlová, D; Bures, P; Fisar, Z; Fuksová, K; Krulík, R; Sikora, J1
Bosse, E; Flockerzi, V; Hofmann, F; Lacinová, L; Ludwig, A1
Bolton, TB; Zhang, H1
Arita, M; Hisatome, I1
Allegra, A; Aloisi, C; Baldari, S; Buemi, M; Imbesi, D; Laganà, A; Morabito, N; Palella, S; Privitera, M; Villari, C1
Ananthanarayanan, VS; Zhorov, BS1
Auriemma, F; Ceriello, A; Macciocchi, B; Papa, A; Scaletta Romeo di Santillo, M; Simonelli, P; Vetrano, A1
Abraham, WM; Ahmed, T; Chapman, GA; Jackowski, J1
Nawrath, H; Wegener, JW2
Degtiar, VE; Döring, F; Glossman, H; Grabner, M; Hering, S; Striessnig, J1
Hartmann, A; Hopf, R; Kneissl, G; Schnell, J1
Feher, J; Juhasz, I; Monos, E; Nadasy, GL; Szekacs, B; Vajo, Z1
Catterall, WA; Hockerman, GH; Johnson, BD; Scheuer, T1
Piñeros, M; Tester, M1
Peterlik, M; Pietschmann, P; Redlich, K; Stulc, T1
Antoine, MH; Cosgrove, KE; Dunne, MJ; Herchuelz, A; Kane, C; Lebrun, P; Ouedraogo, R; Pirotte, B1
Higuchi, S; Kaneko, K; Masumiya, H; Noguchi, K; Shigenobu, K; Takahashi, K; Tanaka, H1
Bonini, W; Botto, GL; Broffoni, T1
Bean, L; Cheng, YF; Neue, UD1
Ferioli, V; Gamberini, G; Gamberini, MC; Rustichelli, C1
Catacuzzeno, L; Franciolini, F; Petris, A; Trequattrini, C1
Jones, SE; McDonald, TF; Missan, S; Zhabyeyev, P1
Catacuzzeno, L; Franciolini, F; Harper, AA; Petris, A; Trequattrini, C1
Dietz, A; Geiger, H; Gossmann, J; Kachel, HG; Kramer, W; Mondorf, U; Scheuermann, EH1
Borlak, J; Levsen, K; Mullett, WM; Pawliszyn, J; Walles, M1
Dierkes, PW; Hochstrate, P; Schlue, WR; Wende, V1
Hoda, JC; Huber, IG; Sinnegger-Brauns, MJ; Striessnig, J; Walter-Bastl, D; Wappl-Kornherr, E1
Awasthi, A; Yadav, A1
Engel, J; Lacinova, L; Tarabova, B1
Cheng, RCK; Tikhonov, DB; Zhorov, BS1

Reviews

7 review(s) available for verapamil and gallopamil

ArticleYear
New developments in Ca2+ channel antagonists.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:6

    Topics: Animals; Binding Sites; Calcium; Calcium Channel Blockers; Calmodulin; Electrophysiology; Heart; Humans; Ion Channels; Muscle Relaxation; Muscle, Smooth; Potassium; Sodium; Structure-Activity Relationship; Substrate Specificity

1983
[Fundamental cardiac and vascular effects of Ca++-antagonistic coronary drugs].
    Medizinische Klinik, 1975, Oct-17, Volume: 70, Issue:42

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Biological Transport; Calcium; Cats; Chemical Phenomena; Chemistry; Coronary Vessels; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Myocardial Contraction; Myocardium; Nifedipine; Oxygen Consumption; Phenethylamines; Prenylamine; Rabbits; Swine; Verapamil

1975
Calcium antagonists and myocardial microperfusion.
    Drugs, 1991, Volume: 42 Suppl 1

    Topics: Animals; Calcium Channel Blockers; Coronary Circulation; Coronary Disease; Gallopamil; Guinea Pigs; Humans; Myocardium; Nifedipine; Rats; Ventricular Function, Left; Verapamil

1991
[Calcium antagonists in acute myocardial infarction].
    Giornale italiano di cardiologia, 1988, Volume: 18, Issue:11

    Topics: Calcium Channel Blockers; Diltiazem; Gallopamil; Hemodynamics; Humans; Myocardial Infarction; Nifedipine; Verapamil

1988
Calcium and alpha-adrenoceptors in activation of vascular smooth muscle.
    Journal of cardiovascular pharmacology, 1982, Volume: 4 Suppl 3

    Topics: Animals; Calcium; Diltiazem; Gallopamil; Humans; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Verapamil

1982
Calcium antagonists. Some chemical-pharmacologic aspects.
    Circulation research, 1983, Volume: 52, Issue:2 Pt 2

    Topics: Animals; Calcium; Calcium Channel Blockers; Gallopamil; Heart; Humans; Ion Channels; Muscle, Smooth; Potassium; Stereoisomerism; Structure-Activity Relationship; Verapamil

1983
History of calcium antagonists.
    Circulation research, 1983, Volume: 52, Issue:2 Pt 2

    Topics: Aniline Compounds; Animals; Calcium; Calcium Channel Blockers; Cardiovascular Diseases; Gallopamil; Heart; Heart Conduction System; Humans; In Vitro Techniques; Magnesium; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Nifedipine; Verapamil

1983

Trials

11 trial(s) available for verapamil and gallopamil

ArticleYear
Randomized double-blind comparison of gallopamil and propranolol in stable angina pectoris.
    The American journal of cardiology, 1984, Mar-01, Volume: 53, Issue:6

    Topics: Aged; Angina Pectoris; Clinical Trials as Topic; Double-Blind Method; Electrocardiography; Exercise Test; Female; Gallopamil; Heart Rate; Humans; Male; Middle Aged; Propranolol; Random Allocation; Verapamil

1984
[Anti-angina effect of gallopamil in comparison with another calcium antagonist and a placebo].
    Zeitschrift fur Kardiologie, 1984, Volume: 73, Issue:9

    Topics: Adult; Aged; Angina Pectoris; Blood Pressure; Clinical Trials as Topic; Coronary Disease; Double-Blind Method; Electrocardiography; Exercise Test; Gallopamil; Heart Rate; Humans; Kinetics; Male; Middle Aged; Myocardial Infarction; Nifedipine; Verapamil

1984
[Comparison of the anti-angina effectiveness of gallopamil to isosorbide dinitrate in long-term medication].
    Die Medizinische Welt, 1983, Dec-16, Volume: 34, Issue:50

    Topics: Angina Pectoris; Clinical Trials as Topic; Female; Gallopamil; Humans; Isosorbide Dinitrate; Long-Term Care; Male; Middle Aged; Verapamil

1983
[Acute and long-term effects of gallopamil (D 600) in stable angina pectoris--a randomized double-blind study].
    Zeitschrift fur Kardiologie, 1983, Volume: 72, Issue:12

    Topics: Adult; Aged; Angina Pectoris; Clinical Trials as Topic; Double-Blind Method; Electrocardiography; Female; Gallopamil; Humans; Long-Term Care; Male; Middle Aged; Random Allocation; Verapamil

1983
Clinical uses of calcium ion antagonists in arrhythmias.
    Clinical and investigative medicine. Medecine clinique et experimentale, 1980, Volume: 3, Issue:1-2

    Topics: Adult; Aged; Alprenolol; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Calcium; Child, Preschool; Clinical Trials as Topic; Female; Gallopamil; Humans; Male; Propylamines; Quinidine; Tachycardia, Paroxysmal; Tiapamil Hydrochloride; Verapamil

1980
Hemodynamic effects in patients with cardiac arrhythmias.
    Clinical and investigative medicine. Medecine clinique et experimentale, 1980, Volume: 3, Issue:1-2

    Topics: Arrhythmias, Cardiac; Blood Pressure; Clinical Trials as Topic; Digitalis Glycosides; Gallopamil; Heart Rate; Humans; Propranolol; Tachycardia; Verapamil

1980
[The electrophysiological effects of the Ca-antagonists gallopamil (D 600), dimeditiapramine (Ro 11-1781) and verapamil in man (author's transl)].
    Zeitschrift fur Kardiologie, 1980, Volume: 69, Issue:8

    Topics: Blood Pressure; Bundle of His; Calcium; Electrophysiology; Gallopamil; Heart Block; Humans; Verapamil

1980
Is erythropoietin-induced hypertension a phenomenon due to the intracellular Ca++ mobilisation?
    International angiology : a journal of the International Union of Angiology, 1994, Volume: 13, Issue:1

    Topics: Adult; Blood Circulation; Calcium; Erythropoietin; Gallopamil; Humans; Ketanserin; Male; Nifedipine; Recombinant Proteins; Vasoconstrictor Agents; Verapamil

1994
[Treatment of ischemic heart disease in the elderly. Comparison of diltiazem, verapamil and gallopamil].
    Minerva cardioangiologica, 1993, Volume: 41, Issue:5

    Topics: Age Factors; Aged; Angina Pectoris; Coronary Angiography; Coronary Disease; Diltiazem; Drug Evaluation; Exercise Test; Female; Gallopamil; Humans; Male; Middle Aged; Myocardial Ischemia; Verapamil

1993
Modulation of ventricular rate in permanent atrial fibrillation: randomized, crossover study of the effects of slow-release formulations of gallopamil, diltiazem, or verapamil.
    Clinical cardiology, 1998, Volume: 21, Issue:11

    Topics: Administration, Oral; Aged; Anti-Arrhythmia Agents; Atrial Fibrillation; Calcium Channel Blockers; Cardiotonic Agents; Cross-Over Studies; Delayed-Action Preparations; Digoxin; Diltiazem; Electrocardiography, Ambulatory; Female; Gallopamil; Heart Rate; Humans; Male; Middle Aged; Verapamil

1998
A randomized prospective double-blind placebo-controlled study of gallopamil, calcium antagonist of the verapamil type, in stable cyclosporine-treated renal transplant recipients.
    Transplantation proceedings, 2002, Volume: 34, Issue:5

    Topics: Adult; Blood Pressure; Calcium Channel Blockers; Creatinine; Cyclosporine; Double-Blind Method; Gallopamil; Humans; Immunosuppressive Agents; Kidney Transplantation; Placebos; Prospective Studies; Urea; Uric Acid; Verapamil

2002

Other Studies

284 other study(ies) available for verapamil and gallopamil

ArticleYear
Stereoisomers of calcium antagonists which differ markedly in their potencies as calcium blockers are equally effective in modulating drug transport by P-glycoprotein.
    Biochemical pharmacology, 1992, Jun-23, Volume: 43, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding, Competitive; Biological Transport; Calcium Channel Blockers; Cell Line; Dihydropyridines; Drug Resistance; Haplorhini; Immunoblotting; Membrane Glycoproteins; Mice; RNA, Messenger; Stereoisomerism; Verapamil; Vinblastine

1992
Studies on Ca2+ channel antagonists. 5-[(3,4-Dimethoxyphenethyl)methylamino]-2-(3,4-dimethoxyphenyl)-2- isopropylpentyl isothiocyanate, a chemoaffinity ligand derived from verapamil.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:9

    Topics: Affinity Labels; Animals; Calcium; Calcium Channel Blockers; Chemical Phenomena; Chemistry; Depression, Chemical; Gallopamil; Ion Channels; Myocardial Contraction; Myocardium; Rats; Verapamil

1986
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Predictive model for L-type channel inhibition: multichannel block in QT prolongation risk assessment.
    Journal of applied toxicology : JAT, 2012, Volume: 32, Issue:10

    Topics: Artificial Intelligence; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Computational Biology; Computer Simulation; Drugs, Investigational; Ether-A-Go-Go Potassium Channels; Expert Systems; Heart Rate; Humans; Models, Biological; Myocytes, Cardiac; NAV1.5 Voltage-Gated Sodium Channel; Potassium Channel Blockers; Quantitative Structure-Activity Relationship; Risk Assessment; Shaker Superfamily of Potassium Channels; Torsades de Pointes; Voltage-Gated Sodium Channel Blockers

2012
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels

2014
The effect of Ca2+ on the metarhodopsin I-II transition. I. Experiments.
    Pflugers Archiv : European journal of physiology, 1976, Jun-29, Volume: 364, Issue:1

    Topics: Animals; Calcium; Cations, Monovalent; Cattle; Gallopamil; Hydrogen-Ion Concentration; Kinetics; Models, Biological; Photolysis; Protons; Retinal Pigments; Rhodopsin; Verapamil

1976
Effect of diazoxide, verapamil and compound D600 on isoproterenol and calcium-mediated dose-response relationships in isolated rabbit atrium.
    European journal of pharmacology, 1977, Oct-01, Volume: 45, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Calcium; Diazoxide; Dose-Response Relationship, Drug; Drug Interactions; Female; Gallopamil; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Rabbits; Verapamil

1977
The action of verapamil on the rate of spontaneous release of transmitter at the frog neuromuscular junction.
    European journal of pharmacology, 1979, Feb-15, Volume: 54, Issue:1-2

    Topics: Action Potentials; Animals; Anura; Calcium; Dantrolene; Female; Gallopamil; In Vitro Techniques; Male; Motor Endplate; Neuromuscular Junction; Neurotransmitter Agents; Rana pipiens; Temperature; Theophylline; Verapamil

1979
Calcium and stimulus secretion coupling in the neurohypophysis. V. The effects of the Ca2+ ionophores A23187 and X537 A on vasopressin release and 45Ca2+ efflux; interactions with sodium and a verapamil analogue (D600).
    Acta endocrinologica, 1976, Volume: 83, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Calcimycin; Calcium; Cattle; Culture Media; Drug Interactions; Gallopamil; Gramicidin; L-Lactate Dehydrogenase; Lasalocid; Leucyl Aminopeptidase; Mitochondria; Neurophysins; Pituitary Gland, Posterior; Secretory Rate; Sodium; Vasopressins; Verapamil

1976
Action of calcium antagonists on microsomal calcium activated ATPase of rat aorta.
    Archives internationales de pharmacodynamie et de therapie, 1978, Volume: 236, Issue:2

    Topics: Animals; Aorta; Calcium; Calcium-Transporting ATPases; Gallopamil; In Vitro Techniques; Microsomes; Rats; Verapamil

1978
A role of cyclic nucleotides in neuromuscular transmission.
    The Journal of pharmacology and experimental therapeutics, 1976, Volume: 199, Issue:3

    Topics: Adenosine; Alloxan; Animals; Axons; Bucladesine; Cats; Cyclic AMP; Dithionitrobenzoic Acid; Electric Stimulation; Fluorides; Gallopamil; Imidazoles; Muscle Contraction; Muscle Denervation; Muscles; Nerve Endings; Neuromuscular Junction; Prostaglandins E; Synaptic Transmission; Theophylline; Verapamil

1976
[Contractile responses of the guinea pig ileal longitudinal muscle to antispasmodics (author's transl)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1977, Volume: 73, Issue:7

    Topics: Acetylcholine; Animals; Benactyzine; Calcium; Cyclic GMP; Drug Synergism; Gallopamil; Guinea Pigs; Ileum; In Vitro Techniques; Male; Manganese; Muscle Contraction; Muscle, Smooth; Papaverine; Verapamil

1977
Effects of ruthenium red, A23187 and D-600 on steroidogenesis in Y-1 cells.
    Biochimica et biophysica acta, 1978, Mar-30, Volume: 528, Issue:3

    Topics: Adrenocorticotropic Hormone; Anti-Bacterial Agents; Calcimycin; Cell Line; Cyclic AMP; Egtazic Acid; Gallopamil; Pregnenolone; Ruthenium; Ruthenium Red; Steroids; Verapamil

1978
Differential effects of D 600 on release of catecholamines by acetylcholine, histamine, tyramine and by cyclic AMP from canine adrenal medulla.
    Japanese journal of pharmacology, 1978, Volume: 28, Issue:5

    Topics: Acetylcholine; Adrenal Medulla; Animals; Calcium; Catecholamines; Cyclic AMP; Dogs; Drug Interactions; Female; Gallopamil; Histamine; In Vitro Techniques; Male; Tyramine; Verapamil

1978
The action of D600 on frog skeletal muscle: facilitation of excitation-contraction coupling.
    Pflugers Archiv : European journal of physiology, 1977, Jul-19, Volume: 369, Issue:3

    Topics: Action Potentials; Animals; Anura; Calcium; Dose-Response Relationship, Drug; Gallopamil; Hindlimb; Magnesium; Membrane Potentials; Muscle Contraction; Muscles; Physical Stimulation; Rana temporaria; Seasons; Verapamil

1977
[Effect of calcium channel blockaders (verapamil, D-600 and manganese ions) on mediator release from frog muscle motor nerve endings].
    Neirofiziologiia = Neurophysiology, 1977, Volume: 9, Issue:4

    Topics: Animals; Anura; Gallopamil; Manganese; Membrane Potentials; Neuromuscular Junction; Rana temporaria; Verapamil

1977
The effects of manganese ions on the contraction of the frog's heart.
    The Journal of physiology, 1977, Volume: 272, Issue:2

    Topics: Animals; Anura; Cadmium; Cobalt; Gallopamil; Heart Atria; In Vitro Techniques; Manganese; Membrane Potentials; Myocardial Contraction; Nickel; Rana pipiens; Verapamil

1977
The effects of some organic "calcium antagonists" on calcium influx in presynaptic nerve terminals.
    Molecular pharmacology, 1979, Volume: 16, Issue:2

    Topics: Animals; Anura; Calcium; Gallopamil; In Vitro Techniques; Nerve Endings; Neuromuscular Junction; Nifedipine; Potassium; Rana pipiens; Rats; Synaptosomes; Verapamil

1979
Inhibition of sodium channels by D600.
    Molecular pharmacology, 1979, Volume: 15, Issue:1

    Topics: Binding, Competitive; Calcium; Cells, Cultured; Gallopamil; Ion Channels; Myocardium; Neoplasms, Experimental; Neuroblastoma; Sodium; Verapamil; Veratridine

1979
Electromechanical coupling in canine trachealis muscle: acetylcholine contractions.
    The American journal of physiology, 1979, Volume: 236, Issue:3

    Topics: Acetylcholine; Animals; Biological Transport, Active; Calcium; Dogs; Gallopamil; In Vitro Techniques; Lanthanum; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Potassium; Trachea; Verapamil

1979
Reentrant ventricular arrhythmias in the late myocardial infarction period. 7. Effect of verapamil and D-600 and the role of the "slow channel".
    Circulation, 1979, Volume: 60, Issue:3

    Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Coronary Disease; Dogs; Electrocardiography; Gallopamil; Heart Conduction System; Heart Ventricles; Myocardial Infarction; Tetrodotoxin; Time Factors; Verapamil

1979
[Comparative analysis of the action of papaverine, novodrin, La3+ and compound D-600 on the guinea pig tenia coli depolarized smooth muscle].
    Biulleten' eksperimental'noi biologii i meditsiny, 1979, Volume: 87, Issue:6

    Topics: Animals; Calcium; Colon; Gallopamil; Guinea Pigs; Histamine; History, 20th Century; In Vitro Techniques; Ion Channels; Isoproterenol; Lanthanum; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Papaverine; Time Factors; Verapamil

1979
Effects of methoxyverapamil on the stimulation by Ca2+, Sr2+ and Ba2+ and on the inhibition by Mg2+ of catecholamine release from the adrenal medulla.
    British journal of pharmacology, 1979, Volume: 66, Issue:4

    Topics: Adrenal Medulla; Animals; Barium; Calcium; Catecholamines; Cations, Divalent; Cattle; Drug Interactions; Gallopamil; In Vitro Techniques; Magnesium; Perfusion; Strontium; Verapamil

1979
The effect of a calcium antagonist (D600) on isoprenaline-induced myocardial necrosis in the rat.
    British journal of experimental pathology, 1979, Volume: 60, Issue:3

    Topics: Animals; Calcium; Cardiomyopathies; Gallopamil; Isoproterenol; Male; Myocardium; Necrosis; Rats; Verapamil

1979
[Effect of verapamil, D-600 and papaverine on the sensitivity of denervated muscle to acetylcholine].
    Doklady Akademii nauk SSSR, 1979, Volume: 247, Issue:4

    Topics: Acetylcholine; Animals; Calcium; Cell Membrane Permeability; Cobalt; Drug Interactions; Gallopamil; Ion Channels; Manganese; Mice; Muscle Denervation; Muscles; Papaverine; Tubocurarine; Verapamil

1979
The actions and interactions of calcium antagonists and DL-homocysteate on cat spinal motoneurones [proceedings].
    The Journal of physiology, 1979, Volume: 296

    Topics: Animals; Cats; Cobalt; Gallopamil; Homocysteine; Motor Neurons; Spinal Cord; Verapamil

1979
Inhibition of high affinity synaptosomal uptake systems by verapamil.
    Molecular pharmacology, 1979, Volume: 16, Issue:3

    Topics: Animals; Brain; Calcium; Gallopamil; In Vitro Techniques; Kinetics; Male; Rats; Serotonin; Sodium Chloride; Synaptosomes; Time Factors; Verapamil

1979
Inhibitory effects of verapamil, prenylamine and D 600 on Ca2+-dependent noradrenaline release from the sympathetic nerves of isolated rabbit hearts.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 310, Issue:1

    Topics: Animals; Calcium; Electric Stimulation; Female; Gallopamil; Heart; In Vitro Techniques; Male; Myocardium; Norepinephrine; Prenylamine; Rabbits; Sodium; Sympathetic Nervous System; Verapamil

1979
The effects of Ca2+ antagonists on Ca2+ accumulation by subcellular fractions of rat myometrium.
    Canadian journal of physiology and pharmacology, 1977, Volume: 55, Issue:5

    Topics: Animals; Biological Transport, Active; Calcium; Cations, Divalent; Chlorpromazine; Female; Gallopamil; Lanthanum; Myometrium; Potassium; Rats; Sodium; Subcellular Fractions; Uterus; Verapamil

1977
Oscillating contractions in protoplasmic strands of Physarum: effects of external Ca++-depletion and Ca++-antagonistic drugs on intrinsic contraction automaticity.
    Cell biology international reports, 1977, Volume: 1, Issue:3

    Topics: Calcium; Cytoplasm; Gallopamil; Lanthanum; Manganese; Movement; Myxomycetes; Physarum; Verapamil

1977
Developmental changes in the sensitivity of embryonic heart cells to tetrodotoxin and D600.
    Developmental biology, 1978, Volume: 65, Issue:1

    Topics: Age Factors; Animals; Biological Transport; Chick Embryo; Culture Techniques; Electric Conductivity; Gallopamil; Heart; Myocardial Contraction; Sodium; Tetrodotoxin; Verapamil; Veratridine

1978
Cardiodepressive and noradrenaline-antagonistic effects of the organic calcium-antagonist D 600 in the spontaneously beating guinea-pig atrium.
    Archives internationales de pharmacodynamie et de therapie, 1977, Volume: 229, Issue:2

    Topics: Animals; Depression, Chemical; Electric Stimulation; Gallopamil; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Norepinephrine; Reserpine; Verapamil

1977
Calcium activation systems in vascular smooth muscle.
    Bibliotheca anatomica, 1977, Issue:15 Pt 1

    Topics: Action Potentials; Animals; Blood Vessels; Calcium; Gallopamil; Guinea Pigs; In Vitro Techniques; Muscle, Smooth; Nifedipine; Pyridines; Verapamil

1977
Effect of replacement of extracellular sodium ions and of D-600 on the activation by adrenalin of adenylate cyclase in intact pigeon erythrocytes.
    Molecular and cellular endocrinology, 1978, Volume: 11, Issue:1

    Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Columbidae; Epinephrine; Erythrocytes; Gallopamil; Kinetics; Lithium; Potassium; Sodium; Verapamil

1978
[Action of the calciumantagonistic compound gallopamile on sinus node, atrioventricular and intraventricular conduction (author's transl)].
    Zeitschrift fur Kardiologie, 1978, Volume: 67, Issue:8

    Topics: Adult; Aged; Arrhythmia, Sinus; Atrioventricular Node; Bundle of His; Calcium; Cardiac Pacing, Artificial; Electrocardiography; Female; Gallopamil; Heart Block; Heart Conduction System; Heart Rate; Humans; Male; Middle Aged; Myocardial Contraction; Sinoatrial Node; Verapamil

1978
Species differences in responses to hyperosmolality and D600 in cat and rat heart.
    The American journal of physiology, 1978, Volume: 235, Issue:3

    Topics: Animals; Cats; Dose-Response Relationship, Drug; Gallopamil; Mannitol; Myocardial Contraction; Osmolar Concentration; Rats; Species Specificity; Stimulation, Chemical; Verapamil

1978
Electrophysiological study of Syrian hamster hereditary cardiomyopathy.
    Cardiovascular research, 1978, Volume: 12, Issue:7

    Topics: Action Potentials; Animals; Cardiomyopathies; Cricetinae; Gallopamil; In Vitro Techniques; Membrane Potentials; Mesocricetus; Papillary Muscles; Verapamil

1978
Simplification of retinal photoresponses by D 600 [proceedings].
    The Journal of physiology, 1978, Volume: 284

    Topics: Animals; Gallopamil; Membrane Potentials; Photoreceptor Cells; Rats; Verapamil

1978
Effect of verapamil and D 600 on cardiac transmembrane potentials.
    Acta physiologica Academiae Scientiarum Hungaricae, 1978, Volume: 51, Issue:1-2

    Topics: Action Potentials; Animals; Cats; Depression, Chemical; Gallopamil; Guinea Pigs; Heart; Membrane Potentials; Myocardial Contraction; Stimulation, Chemical; Time Factors; Verapamil

1978
Differing actions of nitroprusside and D-600 on tension and 45Ca fluxes in canine renal arteries.
    The Journal of pharmacology and experimental therapeutics, 1979, Volume: 208, Issue:1

    Topics: Animals; Blood Vessels; Calcium; Dogs; Drug Interactions; Female; Ferricyanides; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nitroprusside; Norepinephrine; Potassium; Renal Artery; Time Factors; Verapamil

1979
Calcium-antagonists and islet function. IV. Effect of D600.
    Diabetologia, 1976, Volume: 12, Issue:1

    Topics: Animals; Biological Transport; Calcium; Gallopamil; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Rats; Theophylline; Verapamil

1976
Reversible Inhibition of Potassium Contractures by optical isomers of verapamil and D 600 on slow muscle fibres of the frog.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 292, Issue:1

    Topics: Animals; Calcium; Egtazic Acid; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscles; Potassium; Stereoisomerism; Time Factors; Verapamil

1976
[Microscopic quantification of myocardial necroses in experimental cardiology].
    Acta histochemica. Supplementband, 1976, Volume: 16

    Topics: Animals; Calcitonin; Dose-Response Relationship, Drug; Gallopamil; Histological Techniques; Isoproterenol; Magnesium; Male; Myocardium; Necrosis; Potassium; Prenylamine; Rats; Verapamil

1976
Effects of D-600 and its optical isomers on force of contraction in cat papillary muscles and guinea-pig auricles.
    British journal of pharmacology, 1977, Volume: 59, Issue:3

    Topics: Animals; Cats; Depression, Chemical; Electric Stimulation; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Stereoisomerism; Time Factors; Verapamil

1977
On the mechanism underlying the action of D-600 on slow inward current and tension in mammalian myocardium.
    Circulation research, 1977, Volume: 40, Issue:4

    Topics: Action Potentials; Animals; Calcium; Cats; Dose-Response Relationship, Drug; Gallopamil; Heart; Heart Conduction System; Membrane Potentials; Myocardial Contraction; Papillary Muscles; Verapamil

1977
Stimulation of renal gluconeogenesis by verapamil and D-600.
    Biochemical pharmacology, 1977, Jun-01, Volume: 26, Issue:11

    Topics: Animals; Calcium; Gallopamil; Gluconeogenesis; In Vitro Techniques; Ketoglutaric Acids; Kidney Tubules; Male; Rats; Stimulation, Chemical; Succinates; Verapamil

1977
Effects of Ca2+ and catecholamines on the guinea pig atrium action potential plateau.
    The American journal of physiology, 1977, Volume: 233, Issue:2

    Topics: Action Potentials; Animals; Atrial Function; Calcium; Epinephrine; Female; Gallopamil; Guinea Pigs; Heart Atria; In Vitro Techniques; Male; Verapamil

1977
Calcium movements during the release of catecholamines from the adrenal medulla: effects of methoxyverapamil and external cations.
    The Journal of physiology, 1977, Volume: 269, Issue:2

    Topics: Adrenal Medulla; Animals; Calcium; Catecholamines; Cattle; Gallopamil; In Vitro Techniques; Magnesium; Sodium; Sorbitol; Verapamil

1977
Effect of D600, practolol, and alterations in magnesium on ionized calcium concentration-response relationships in the intact dog heart.
    Circulation research, 1977, Volume: 41, Issue:4

    Topics: Animals; Blood Glucose; Calcium; Cardiac Pacing, Artificial; Cations, Divalent; Dogs; Dose-Response Relationship, Drug; Electrocardiography; Gallopamil; Heart; Heart Conduction System; Magnesium; Practolol; Pressure; Ventricular Function; Verapamil

1977
Effects of D 600 and papaverine on the inotropic response to isoprenaline on left guinea-pig atria under the graded influence of changes of frequency and temperature.
    Archives internationales de pharmacodynamie et de therapie, 1977, Volume: 229, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Gallopamil; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Papaverine; Temperature; Verapamil

1977
The effects of D600 and verapamil on action potential in the X-organ neuron of the crayfish.
    The Japanese journal of physiology, 1976, Volume: 26, Issue:2

    Topics: Action Potentials; Animals; Astacoidea; Calcium; Eye; Gallopamil; In Vitro Techniques; Magnesium; Neurons; Verapamil

1976
Some effects of D600, nifedipine and sodium nitroprusside on electrical and mechanical activity in rat portal vein [proceedings].
    British journal of pharmacology, 1976, Volume: 58, Issue:2

    Topics: Animals; Calcium; Electrophysiology; Ferricyanides; Gallopamil; In Vitro Techniques; Muscle Contraction; Nifedipine; Nitroprusside; Portal Vein; Pyridines; Rats; Verapamil

1976
On the pathogenesis of cardiac necroses induced by theophylline and caffeine.
    Acta pharmacologica et toxicologica, 1976, Volume: 39, Issue:3

    Topics: Animals; Blood Pressure; Caffeine; Calcium; Gallopamil; Heart; Heart Rate; Isoproterenol; Male; Myocarditis; Myocardium; Necrosis; Oxygen Consumption; Propranolol; Rats; Theophylline; Verapamil

1976
Relationship between internal calcium and outward current in mammalian ventricular muscle; a mechanism for the control of the action potential duration?
    The Journal of physiology, 1976, Volume: 262, Issue:1

    Topics: Action Potentials; Animals; Calcium; Cattle; Cyanides; Gallopamil; Heart Ventricles; In Vitro Techniques; Membrane Potentials; Myocardial Contraction; Sheep; Sodium; Ventricular Function; Verapamil

1976
[Mechanism of excitation and contraction uncoupling in frog and guinea pig myocardial fibers during block of slow sodium-calcium channels by compound D-600].
    Biofizika, 1976, Volume: 21, Issue:6

    Topics: Action Potentials; Animals; Calcium; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Myocardial Contraction; Rana temporaria; Sodium; Verapamil

1976
Effect of isoproterenol and D-600 on calcium movements in rat myometrium.
    The Journal of pharmacology and experimental therapeutics, 1975, Volume: 193, Issue:2

    Topics: Animals; Calcium; Calcium Radioisotopes; Depression, Chemical; Female; Gallopamil; In Vitro Techniques; Isoproterenol; Kinetics; Lanthanum; Myometrium; Potassium; Pregnancy; Rats; Sodium; Stimulation, Chemical; Uterus; Verapamil

1975
Proceedings: Ca-dependence of supraventricular pacemaker activity and its responsiveness to Ca-antagonistic compounds (verapamil, D 600, nifedipine).
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 287 Suppl

    Topics: Animals; Calcium; Gallopamil; Nifedipine; Sinoatrial Node; Verapamil

1975
Proceedings: P- and T-blockade in smooth muscle: a new pharmacological principle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 287 Suppl

    Topics: Animals; Calcium; Female; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Verapamil

1975
Functional antagonism between calcium-antagonists and noradrenaline on isolated guinea-pig atria.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 288, Issue:2-3

    Topics: Animals; Atrial Function; Calcium; Depression, Chemical; Electric Stimulation; Gallopamil; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Nifedipine; Norepinephrine; Pyridines; Verapamil

1975
Influence of papaverine, D600, and nifedipine on the effects of noradrenaline and calcium on the isolated aorta and mesenteric artery of the rabbit.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 289, Issue:4

    Topics: Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Calcium; Calcium Chloride; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Papaverine; Pyridines; Rabbits; Verapamil

1975
Action of D-600 on spontaneous and electrically stimulated activity of the parturient rat uterus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 290, Issue:1

    Topics: Action Potentials; Animals; Depression, Chemical; Electric Stimulation; Evoked Potentials; Female; Gallopamil; In Vitro Techniques; Labor, Obstetric; Membrane Potentials; Muscle, Smooth; Myometrium; Postpartum Period; Pregnancy; Rats; Uterine Contraction; Verapamil

1975
Inotropic and electrophysiological actions of verapamil and D 600 in mammalian myocardium. I. Pattern of inotropic effects of the racemic compounds.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 290, Issue:1

    Topics: Action Potentials; Animals; Calcium; Cats; Electric Stimulation; Gallopamil; Lanthanum; Membrane Potentials; Myocardial Contraction; Myocardium; Nickel; Verapamil

1975
Inotropic and electrophysiological actions of verapamil and D 600 in mammalian myocardium. II. Pattern of inotropic effects of the optical isomers.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 290, Issue:1

    Topics: Animals; Calcium; Cats; Depression, Chemical; Electric Stimulation; Gallopamil; Myocardial Contraction; Myocardium; Optical Rotation; Stereoisomerism; Verapamil

1975
Inotropic and electrophysiological actions of verapamil and D 600 in mammalian myocardium. III. Effects of the optical isomers on transmembrane action potentials.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 290, Issue:1

    Topics: Action Potentials; Animals; Calcium; Cats; Electric Stimulation; Gallopamil; Membrane Potentials; Myocardial Contraction; Myocardium; Optical Rotation; Sinoatrial Node; Sodium; Stereoisomerism; Verapamil

1975
Effects of temperature and spasmolytic agents on the rate of relaxation of intestinal smooth muscle.
    Proceedings of the Western Pharmacology Society, 1975, Volume: 18

    Topics: Aminophylline; Animals; Calcium; Cytoplasm; Gallopamil; In Vitro Techniques; Intestines; Manganese; Muscle Contraction; Muscle, Smooth; Papaverine; Parasympatholytics; Rats; Temperature; Verapamil

1975
Functional differentiation of the transmembrane sodium and calcium channels in mammalian cardiac fibers by use of specific inhibitors.
    Recent advances in studies on cardiac structure and metabolism, 1975, Volume: 5

    Topics: Animals; Calcium; Cats; Electric Conductivity; Gallopamil; Heart; In Vitro Techniques; Lidocaine; Membrane Potentials; Metals, Alkaline Earth; Myocardial Contraction; Myocardium; Sodium; Strontium; Verapamil

1975
Inhibition of calcium-dependent action potentials in mammalian myocardium by specific inhibitors of the transmembrane calcium conductivity (verapamil, D 600).
    Recent advances in studies on cardiac structure and metabolism, 1975, Volume: 5

    Topics: Action Potentials; Animals; Calcium; Cats; Electric Conductivity; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Papillary Muscles; Potassium; Sodium; Verapamil

1975
Restriction of isoproterenol-induced myocardial Ca uptake and necrotization in rats by a new Ca-antagonistic compound (ethyl-4-(3,4,5-trimethoxycinnamoyl) piperazinyl acetate (Vascordil)).
    Recent advances in studies on cardiac structure and metabolism, 1975, Volume: 6

    Topics: Animals; Biological Transport; Calcium; Cardiomyopathies; Cinnamates; Dose-Response Relationship, Drug; Gallopamil; Isoproterenol; Myocardium; Necrosis; Piperazines; Prenylamine; Rats; Verapamil

1975
Influence of isoproterenol, propranolol, and D 600 on the de novo synthesis of adenine nucleotides in rat hearts.
    Recent advances in studies on cardiac structure and metabolism, 1975, Volume: 7

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Female; Gallopamil; Heart; Isoproterenol; Myocardium; Propranolol; Rats; Verapamil

1975
[Influence of anti-arrhythmia agents on electrolyte metabolism].
    Kardiologiia, 1976, Volume: 16, Issue:1

    Topics: Adult; Aged; Anti-Arrhythmia Agents; Coronary Disease; Female; Gallopamil; Humans; Hypertension; Male; Middle Aged; Potassium; Propranolol; Quinidine; Sodium; Verapamil

1976
[Use of panangin, obsidan and isoptin in acute rhythm disorders under conditions of cardiological first aid service].
    Sovetskaia meditsina, 1976, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Aged; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Aspartic Acid; Female; First Aid; Gallopamil; Humans; Male; Middle Aged; Propranolol; Verapamil

1976
The different effects of D-600 (methoxyverapamil) on the release of adrenal catecholamines induced by acetylcholine, high potassium or sodium deprivation.
    British journal of pharmacology, 1976, Volume: 57, Issue:1

    Topics: Acetylcholine; Adrenal Medulla; Animals; Catecholamines; Cattle; Gallopamil; In Vitro Techniques; Potassium; Sodium; Stimulation, Chemical; Time Factors; Verapamil

1976
Effects of verapamil, gallopamil, diltiazem and nifedipine on sarcoplasmic reticulum function in rat heart.
    Cardioscience, 1992, Volume: 3, Issue:3

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Diltiazem; Gallopamil; Heart; Nifedipine; Rats; Rats, Sprague-Dawley; Ryanodine; Sarcoplasmic Reticulum; Verapamil

1992
Inotropic effects of calcium antagonists in the cardiomyopathic Syrian hamster.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Calcium Channels; Cardiomyopathies; Cricetinae; Depression, Chemical; Diltiazem; Gallopamil; Mesocricetus; Myocardial Contraction; Nifedipine; Stimulation, Chemical; Verapamil

1992
Effects of the novel calcium channel blocker, anipamil, on the isolated rabbit heart. Comparison with verapamil and gallopamil.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Blood Pressure; Calcium Channel Blockers; Coronary Circulation; Female; Gallopamil; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Propylamines; Rabbits; Verapamil

1992
Red blood cell partitioning of gallopamil, verapamil and norverapamil.
    Farmaco (Societa chimica italiana : 1989), 1992, Volume: 47, Issue:3

    Topics: Biological Availability; Chromatography, High Pressure Liquid; Erythrocytes; Gallopamil; Humans; In Vitro Techniques; Regression Analysis; Verapamil

1992
Direct determination of the enantiomeric ratio of verapamil, its major metabolite norverapamil and gallopamil in plasma by chiral high-performance liquid chromatography.
    Journal of chromatography, 1992, Mar-27, Volume: 575, Issue:2

    Topics: Animals; Chromatography, High Pressure Liquid; Gallopamil; Humans; Male; Microsomes, Liver; Rats; Rats, Inbred Strains; Reproducibility of Results; Stereoisomerism; Verapamil

1992
Myocytes isolated from porcine coronary arteries: reduction of currents through L-type Ca-channels by verapamil-type Ca-antagonists.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 1991, Volume: 42, Issue:2

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cell Separation; Coronary Vessels; Electrophysiology; Gallopamil; Kinetics; Muscle, Smooth, Vascular; Swine; Verapamil

1991
Effects of pinaverium on voltage-activated calcium channel currents of single smooth muscle cells isolated from the longitudinal muscle of the rabbit jejunum.
    British journal of pharmacology, 1990, Volume: 99, Issue:2

    Topics: Animals; Barium; Calcium Channels; Diltiazem; Flunarizine; Gallopamil; In Vitro Techniques; Ion Channels; Jejunum; Membrane Potentials; Morpholines; Muscle, Smooth; Parasympatholytics; Rabbits; Verapamil

1990
Mechanisms of potassium channel block in rat alveolar epithelial cells.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:2

    Topics: Animals; Calcium; Calcium Channels; Capsaicin; Cells, Cultured; Charybdotoxin; Chlorpromazine; Epithelium; Gallopamil; Kinetics; Nifedipine; Phencyclidine; Potassium Channels; Pulmonary Alveoli; Quinidine; Rats; Scorpion Venoms; Tacrine; Tetraethylammonium Compounds; Verapamil

1990
Reduction in myocardial hemorrhage and the extent of necrosis by gallopamil (D600) in dogs with coronary artery reperfusion.
    Journal of cardiovascular pharmacology, 1991, Volume: 18, Issue:5

    Topics: Animals; Autoradiography; Blood Pressure; Coronary Vessels; Dogs; Female; Gallopamil; Heart Diseases; Heart Rate; Hemorrhage; Male; Myocardial Reperfusion; Necrosis; Verapamil

1991
Calcium antagonists and cardiac noradrenaline release in ischemia.
    Journal of molecular and cellular cardiology, 1991, Volume: 23, Issue:3

    Topics: Animals; Biological Transport; Calcium; Chromatography, High Pressure Liquid; Cyanides; Gallopamil; Heart; Ischemia; Male; Methoxyhydroxyphenylglycol; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains; Verapamil

1991
Beta-adrenergic agonists stimulate the oxidative pentose phosphate pathway in the rat heart.
    Circulation research, 1990, Volume: 67, Issue:6

    Topics: Adenine Nucleotides; Adrenergic beta-Agonists; Animals; Cycloheximide; Dactinomycin; Female; Fenoterol; Gallopamil; Glucosephosphate Dehydrogenase; Heart; Isoproterenol; Myocardium; Oxidation-Reduction; Pentose Phosphate Pathway; Rats; Rats, Inbred Strains; Ribose; Stimulation, Chemical; Time Factors; Verapamil

1990
Interaction of calcium channel antagonists with parietal cell acid production, adenylate cyclase, intracellular-free Ca2+ and H+/K+-ATPase.
    Pharmacology, 1990, Volume: 40, Issue:1

    Topics: Adenosine Triphosphatases; Adenylyl Cyclases; Animals; Calcium; Calcium Channel Blockers; Carbachol; Gallopamil; Guinea Pigs; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrochloric Acid; Membranes; Nifedipine; Parietal Cells, Gastric; Protons; Stomach; Verapamil

1990
Effects of D600 on hypoxic suppression of K+ currents in isolated type I carotid body cells of the neonatal rat.
    FEBS letters, 1990, Oct-01, Volume: 271, Issue:1-2

    Topics: Animals; Animals, Newborn; Calcium; Calcium Channels; Carotid Body; Cells, Cultured; Gallopamil; Magnesium; Oxygen; Potassium; Potassium Channels; Rats; Verapamil

1990
Synthesis and identification of the N-glucuronides of norgallopamil and norverapamil, unusual metabolites of gallopamil and verapamil.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:2

    Topics: Animals; Chromatography, High Pressure Liquid; Gallopamil; Gas Chromatography-Mass Spectrometry; Glucuronates; Male; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil

1990
Pharmacologic effects on coronary microvessels during myocardial ischaemia.
    European heart journal, 1990, Volume: 11 Suppl B

    Topics: Animals; Blood Flow Velocity; Capillary Permeability; Coronary Circulation; Coronary Disease; Coronary Vessels; Erythrocyte Count; Fatty Acids; Gallopamil; Imidazoles; Indomethacin; Microcirculation; Platelet Count; Rats; Thromboxane-A Synthase; Verapamil

1990
Ca antagonists do not alter aldosterone secretion during established Na depletion.
    The American journal of physiology, 1985, Volume: 248, Issue:6 Pt 1

    Topics: Adrenal Glands; Aldosterone; Animals; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Edetic Acid; Female; Gallopamil; Hydrocortisone; Indenes; Ion Channels; Lanthanum; Nifedipine; Nisoldipine; Ryanodine; Sheep; Sodium; Verapamil

1985
[Co2+ activation and D-600 inhibition of sodium transport across the apical membrane of skin epithelial cells in the frog].
    Doklady Akademii nauk SSSR, 1985, Volume: 281, Issue:5

    Topics: Animals; Biological Transport; Cell Membrane; Cobalt; Epithelium; Gallopamil; Ion Channels; Membrane Potentials; Rana temporaria; Skin; Sodium; Verapamil

1985
The effect of D600 on tonic tension, Na+ inward current, and Na+-Ca2+ exchange in frog heart.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:11

    Topics: Animals; Calcium; Gallopamil; In Vitro Techniques; Ion Channels; Ion Exchange; Membrane Potentials; Myocardial Contraction; Myocardium; Rana pipiens; Sodium; Tetrodotoxin; Verapamil

1985
Effects of calcium antagonists on mechanical responses of mammalian skeletal muscles.
    European journal of pharmacology, 1985, Nov-05, Volume: 117, Issue:2

    Topics: Animals; Calcium; Calcium Channel Blockers; Electric Stimulation; Gallopamil; In Vitro Techniques; Ion Channels; Male; Membrane Potentials; Mice; Muscle Contraction; Muscles; Rats; Rats, Inbred Strains; Verapamil

1985
D600 as a direct blocker of Ca-dependent K currents in Helix neurons.
    European journal of pharmacology, 1985, Nov-19, Volume: 117, Issue:3

    Topics: Animals; Cadmium; Calcium Channel Blockers; Diltiazem; Gallopamil; Helix, Snails; In Vitro Techniques; Ion Channels; Membrane Potentials; Neuromuscular Depolarizing Agents; Neurons; Verapamil

1985
A pharmacological explanation of the use-dependency of the verapamil (and D-600) block of slow calcium channels.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:2

    Topics: Animals; Calcium; Decerebrate State; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Ion Channels; Muscle Contraction; Potassium; Rana pipiens; Time Factors; Verapamil

1986
Sidedness of reconstituted calcium channels from muscle transverse tubules as determined by D600 and D890 blockade.
    Biophysical journal, 1986, Volume: 49, Issue:3

    Topics: Animals; Calcium; Gallopamil; Ion Channels; Muscles; Rats; Verapamil

1986
Effect of calcium antagonists on histamine release from human basophil leukocytes.
    British journal of clinical pharmacology, 1986, Volume: 22, Issue:4

    Topics: Adult; Basophils; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Histamine Release; Humans; In Vitro Techniques; Verapamil

1986
Involvement of ion channels in the induction of proenkephalin A gene expression by nicotine and cAMP in bovine chromaffin cells.
    The Journal of biological chemistry, 1987, Mar-25, Volume: 262, Issue:9

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Colforsin; Cyclic AMP; Enkephalins; Gallopamil; Gene Expression Regulation; Ion Channels; Nicotine; Nifedipine; Protein Precursors; RNA, Messenger; Sodium; Tubocurarine; Verapamil

1987
Inhibition of calcium channels in neuroblastoma x glioma hybrid cells by verapamil, D600, diltiazem and nisoldipine.
    Biomedica biochimica acta, 1987, Volume: 46, Issue:8-9

    Topics: Animals; Calcium; Calcium Channel Blockers; Diltiazem; Gallopamil; Glioma; Ion Channels; Neuroblastoma; Neurons; Nifedipine; Nisoldipine; Tumor Cells, Cultured; Verapamil

1987
Reversal of chloroquine resistance in falciparum malaria independent of calcium channels.
    Biochemical and biophysical research communications, 1988, Aug-30, Volume: 155, Issue:1

    Topics: Animals; Calcium; Chloroquine; Drug Interactions; Drug Resistance; Gallopamil; Ion Channels; Malaria; Plasmodium falciparum; Verapamil

1988
Effects of phenylalkylamine calcium entry blockers on postischemic energy metabolism in the isolated perfused rat brain: stereoselective action of emopamil.
    Pharmacology, 1988, Volume: 37, Issue:1

    Topics: Animals; Brain; Brain Ischemia; Calcium Channel Blockers; Energy Metabolism; Gallopamil; In Vitro Techniques; Ion Channels; Male; Perfusion; Rats; Rats, Inbred Strains; Stereoisomerism; Verapamil

1988
[Exercise capacity of coronary heart disease patients in long-term follow-up with gallopamil in comparison with premedication with verapamil].
    Zeitschrift fur Kardiologie, 1989, Volume: 78 Suppl 5

    Topics: Aged; Angina Pectoris; Arrhythmias, Cardiac; Coronary Disease; Electrocardiography; Exercise Test; Follow-Up Studies; Gallopamil; Humans; Long-Term Care; Middle Aged; Verapamil

1989
Comparative effects of verapamil and D-600 on the contractile responses produced by neurotransmitters and depolarizing agents in the rat isolated seminal vesicle.
    General pharmacology, 1989, Volume: 20, Issue:5

    Topics: Acetylcholine; Animals; Carbachol; Clonidine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Depolarizing Agents; Neurotransmitter Agents; Norepinephrine; Phenylephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Seminal Vesicles; Verapamil

1989
Block of sodium currents by the calcium antagonist D600 in human heart cell segments.
    Pflugers Archiv : European journal of physiology, 1985, Volume: 403, Issue:2

    Topics: Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; Humans; Ion Channels; Middle Aged; Myocardium; Sodium; Verapamil

1985
[Possible participation of slow Na+--Ca++ channels in realizing cholinergic effects on the cardiac pacemaker].
    Fiziologicheskii zhurnal SSSR imeni I. M. Sechenova, 1985, Volume: 71, Issue:4

    Topics: Acetylcholine; Animals; Calcium; Electric Stimulation; Gallopamil; Heart Conduction System; In Vitro Techniques; Ion Channels; Manganese; Rana temporaria; Receptors, Cholinergic; Sodium; Verapamil

1985
Quantitative determination of verapamil and metabolites in human serum by high-performance liquid chromatography and its application to biopharmaceutic investigations.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:2

    Topics: Biopharmaceutics; Biotransformation; Chromatography, High Pressure Liquid; Gallopamil; Humans; Indicators and Reagents; Verapamil

1989
Effects of Ca-antagonists and antispasmodic drugs on contraction by ACh in molluscan smooth muscle.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1985, Volume: 80, Issue:1

    Topics: Acetylcholine; Animals; Bivalvia; Calcium Channel Blockers; Diltiazem; Dimethylphenylpiperazinium Iodide; Drug Interactions; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Papaverine; Parasympatholytics; Piperidines; Verapamil

1985
Verapamil alters the amplitude and time course of miniature endplate current.
    Neuropharmacology, 1985, Volume: 24, Issue:6

    Topics: Animals; Anura; Gallopamil; In Vitro Techniques; Iontophoresis; Motor Endplate; Neuromuscular Junction; Synaptic Transmission; Time Factors; Verapamil

1985
In vitro effects of verapamil and methoxy-verapamil [D 600] on transmembrane sodium and potassium transport in human erythrocytes.
    Bollettino della Societa italiana di biologia sperimentale, 1985, Jun-30, Volume: 61, Issue:6

    Topics: Biological Transport, Active; Bumetanide; Erythrocytes; Gallopamil; Humans; In Vitro Techniques; Ouabain; Potassium; Sodium; Sodium-Potassium-Exchanging ATPase; Verapamil

1985
Characterization of the Ca2+ coordination site regulating binding of Ca2+ channel inhibitors d-cis-diltiazem, (+/-)bepridil and (-)desmethoxyverapamil to their receptor site in skeletal muscle transverse tubule membranes.
    Biochemical and biophysical research communications, 1985, Oct-15, Volume: 132, Issue:1

    Topics: Barium; Benzazepines; Bepridil; Calcium; Calcium Channel Blockers; Calcium Channels; Diltiazem; Gallopamil; Kinetics; Magnesium; Membranes; Microtubules; Muscles; Pyrrolidines; Receptors, Nicotinic; Strontium; Verapamil

1985
Potentiation of pancuronium induced neuromuscular blockade by calcium channel blockers in vitro.
    Journal of neural transmission, 1985, Volume: 64, Issue:3-4

    Topics: Animals; Calcium Channel Blockers; Depression, Chemical; Diltiazem; Drug Synergism; Gallopamil; Male; Neuromuscular Junction; Nifedipine; Nisoldipine; Pancuronium; Rats; Rats, Inbred Strains; Synaptic Transmission; Verapamil

1985
Mode of vasorelaxing action of 5-[3-[[2-(3,4-dimethoxyphenyl)-ethyl]amino]-1-oxopropyl]-2,3,4,5- tetrahydro-1,5-benzothiazepine fumarate (KT-362), a new intracellular calcium antagonist.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Animals; Caffeine; Calcium Channel Blockers; Diltiazem; Egtazic Acid; Gallopamil; Lanthanum; Male; Methoxamine; Muscle Contraction; Nifedipine; Nitroglycerin; Norepinephrine; Rabbits; Thiazepines; Vasodilation; Verapamil

1987
Verapamil enhances the non-adrenergic twitch response of rat vas deferens.
    European journal of pharmacology, 1987, Aug-04, Volume: 140, Issue:1

    Topics: Animals; Autonomic Nervous System; Electric Stimulation; Gallopamil; Hydroxydopamines; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxidopamine; Prazosin; Rats; Reserpine; Vas Deferens; Verapamil; Yohimbine

1987
Verapamil, an antagonist at 5-hydroxytryptamine receptors of human blood platelets.
    European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2

    Topics: Adenosine Diphosphate; Binding, Competitive; Blood Platelets; Cerebral Cortex; Gallopamil; Humans; In Vitro Techniques; Ketanserin; Membranes; Piperidines; Receptors, Serotonin; Spiperone; Verapamil

1985
Manganese can inhibit or potentiate contractile responses in mesenteric portal vein.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:6

    Topics: Animals; Barium; Calcium; Felodipine; Gallopamil; In Vitro Techniques; Male; Manganese; Mesenteric Veins; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Spectrophotometry, Atomic; Strontium; Tissue Distribution; Verapamil

1988
[Calcium antagonists in angina pectoris].
    Giornale italiano di cardiologia, 1988, Volume: 18, Issue:11

    Topics: Angina Pectoris; Angina Pectoris, Variant; Calcium Channel Blockers; Diltiazem; Gallopamil; Humans; Nifedipine; Physical Exertion; Verapamil

1988
Stereoisomers of calcium antagonists discriminate between coronary vascular and myocardial sites.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 337, Issue:2

    Topics: Animals; Bepridil; Calcium Channel Blockers; Coronary Vessels; Gallopamil; Heart; In Vitro Techniques; Male; Pyrrolidines; Rats; Stereoisomerism; Verapamil

1988
Slow channel inhibitor effects on brain function: tolerance to severe hypoxia in the rat.
    British journal of pharmacology, 1988, Volume: 95, Issue:3

    Topics: Animals; Bencyclane; Bepridil; Brain; Calcium Channel Blockers; Cinnarizine; Diltiazem; Electroencephalography; Fendiline; Flunarizine; Gallopamil; Heart Rate; Hypoxia; Nimodipine; Prenylamine; Pyrrolidines; Rats; Rats, Inbred Strains; Respiration; Verapamil

1988
Effect of gallopamil, a calcium channel blocker, on carbachol- and histamine-induced bronchoconstriction in sheep.
    The Journal of allergy and clinical immunology, 1988, Volume: 81, Issue:5 Pt 1

    Topics: Aerosols; Airway Resistance; Animals; Bronchial Spasm; Carbachol; Female; Gallopamil; Histamine; Infusions, Intravenous; Sheep; Verapamil

1988
In vitro effects of gallopamil on platelet aggregation and thromboxane generation.
    Arzneimittel-Forschung, 1988, Volume: 38, Issue:5

    Topics: Blood Platelets; Gallopamil; Humans; In Vitro Techniques; Platelet Aggregation; Thromboxanes; Verapamil

1988
Calcium-dependent chronotropic action of bovine parathyroid hormone (1-34) in isolated atria of Japanese quail, Coturnix coturnix japonica.
    General and comparative endocrinology, 1986, Volume: 64, Issue:2

    Topics: Animals; Atrial Function; Calcium; Coturnix; Dose-Response Relationship, Drug; Gallopamil; Heart Rate; Male; Parathyroid Hormone; Peptide Fragments; Propranolol; Quail; Stimulation, Chemical; Verapamil

1986
Interaction of AOA 39, D600, verapamil and diltiazem with cardiac cholinergic effects.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 286, Issue:1

    Topics: Animals; Calcium Channel Blockers; Diltiazem; Drug Interactions; Gallopamil; Heart Conduction System; Isoindoles; Nifedipine; Phthalimides; Purkinje Fibers; Quinuclidinyl Benzilate; Rabbits; Radioligand Assay; Receptors, Muscarinic; Tritium; Verapamil

1987
Low potency of Ca antagonists in smooth muscle from different levels of the respiratory tract.
    Acta physiologica Scandinavica, 1987, Volume: 131, Issue:2

    Topics: Animals; Bronchi; Calcium Channel Blockers; Felodipine; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Nitrendipine; Rats; Rats, Inbred Strains; Respiratory Muscles; Trachea; Verapamil

1987
Verapamil as an apparent competitive antagonist of the serotonin receptor of rabbit isolated aorta.
    General pharmacology, 1986, Volume: 17, Issue:2

    Topics: Animals; Aorta, Thoracic; Binding, Competitive; Cinnarizine; Diltiazem; Flunarizine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Receptors, Serotonin; Verapamil

1986
Effects of compound D600 (methoxyverapamil) on drug-induced contractions of isolated dog uterine muscle.
    General pharmacology, 1986, Volume: 17, Issue:2

    Topics: Acetylcholine; Animals; Barium; Calcium Chloride; Dogs; Female; Gallopamil; Histamine; In Vitro Techniques; Oxytocin; Uterine Contraction; Verapamil

1986
Effects of calcium antagonists and calcium-buffered salines on wound healing in Xenopus early embryos.
    Cytobios, 1986, Volume: 46, Issue:184

    Topics: Animals; Buffers; Calcium; Calcium Channel Blockers; Embryo, Nonmammalian; Female; Gallic Acid; Gallopamil; Microscopy, Electron, Scanning; Sodium Chloride; Verapamil; Wound Healing; Xenopus

1986
Effects of some Ca2+ blockers on receptor potentials of crayfish retina.
    Scientia Sinica. Series B, Chemical, biological, agricultural, medical & earth sciences, 1986, Volume: 29, Issue:3

    Topics: Animals; Astacoidea; Calcium; Calcium Channel Blockers; Evoked Potentials, Visual; Gallopamil; In Vitro Techniques; Photoreceptor Cells; Retina; Trifluoperazine; Verapamil

1986
Participation of intracellular sites in the action of Ca2+ channel blockers.
    European journal of pharmacology, 1986, Nov-04, Volume: 130, Issue:3

    Topics: Amino Acids; Animals; Calcium Channel Blockers; Calcium Radioisotopes; Cerebral Cortex; Gallopamil; In Vitro Techniques; Potassium; Rats; Synaptosomes; Verapamil; Veratrine

1986
Effects of Ca antagonists on the action potential and their relationship to the muscarinic ACh actions in isolated sympathetic neurons of rabbits.
    Neuroscience letters, 1986, Dec-12, Volume: 72, Issue:2

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Cells, Cultured; Cobalt; Gallopamil; Ganglia, Sympathetic; Male; Mollusk Venoms; Nifedipine; omega-Conotoxin GVIA; Rabbits; Receptors, Muscarinic; Verapamil

1986
The effect of calcium antagonists on the proteolytic degradation of low-density lipoprotein in HeLa cells.
    Experimental cell research, 1985, Volume: 158, Issue:1

    Topics: Calcium Channel Blockers; Cell Compartmentation; Chloroquine; Cholesterol; Endocytosis; Female; Gallopamil; HeLa Cells; Humans; Kinetics; Lipoproteins, LDL; Lysosomes; Peptide Hydrolases; Verapamil

1985
Synthesis and release of luteinizing hormone in vitro by rat anterior pituitary cells: effects of gallopamil hydrochloride (D600) and pimozide.
    Endocrinology, 1985, Volume: 117, Issue:4

    Topics: Alanine; Animals; Carbohydrate Metabolism; Gallopamil; Glucosamine; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Pimozide; Pituitary Gland, Anterior; Rats; Verapamil

1985
[The effect of calcium antagonists on intracellular transport of epidermal growth factor and the conjugate of epidermal growth factor with pseudomonas exotoxin].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1985, Volume: 12, Issue:3 Pt 2

    Topics: Biological Transport; Calcium Channel Blockers; Cathepsin B; Cathepsins; Cell Line; Cell Survival; Cells, Cultured; Chloroquine; Endotoxins; Enzyme Activation; Epidermal Growth Factor; Gallopamil; Humans; Lysosomes; Neoplasms, Experimental; Nifedipine; Pseudomonas aeruginosa; Verapamil

1985
Verapamil is a competitive inhibitor of gamma-aminobutyric acid and calcium uptakes by mouse brain subcellular particles.
    Life sciences, 1985, Jan-28, Volume: 36, Issue:4

    Topics: Animals; Biological Transport; Brain; Calcium; Gallopamil; gamma-Aminobutyric Acid; Kinetics; Mice; Sodium; Synaptosomes; Verapamil

1985
Do D 600 and diltiazem interact with serotonin receptors in rabbit vascular tissues?
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:3

    Topics: Animals; Aorta; Basilar Artery; Benzazepines; Blood Vessels; Calcium; Dibenzylchlorethamine; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Male; Rabbits; Receptors, Serotonin; Serotonin; Vasoconstriction; Verapamil

1985
The potencies and selectivities of four calcium antagonists as inhibitors of uterine contractions in the rat in vivo.
    British journal of pharmacology, 1985, Volume: 85, Issue:1

    Topics: Albuterol; Animals; Blood Pressure; Calcium Channel Blockers; Castration; Diltiazem; Female; Gallopamil; Heart Rate; Nifedipine; Pregnancy; Rats; Rats, Inbred Strains; Uterine Contraction; Verapamil

1985
Comparison of negative inotropic potency, reversibility, and effects on calcium influx of six calcium channel antagonists in cultured myocardial cells.
    British journal of pharmacology, 1985, Volume: 85, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Cells, Cultured; Chick Embryo; Gallopamil; Half-Life; Lidoflazine; Myocardial Contraction; Myocardium; Nifedipine; Perhexiline; Time Factors; Verapamil

1985
Effect of gallopamil on energy metabolism of the isolated perfused rat brain in the postischemic period.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Adenosine Monophosphate; Adenosine Triphosphate; Animals; Brain; Electroencephalography; Energy Metabolism; Gallopamil; Ischemic Attack, Transient; Male; Mathematics; Perfusion; Phosphocreatine; Rats; Rats, Inbred Strains; Verapamil

1985
Chronic treatment of rats with D-600 causes a compensatory decrease in the calcium requirement for contractility of vascular smooth and cardiac muscles.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:5

    Topics: Animals; Blood Pressure; Calcium; Gallopamil; Heart Rate; Hydralazine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Norepinephrine; Portal Vein; Potassium; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Verapamil

1985
Paradoxical effects of K+ and D-600 on parathyroid hormone secretion and cytoplasmic Ca2+ in normal bovine and pathological human parathyroid cells.
    Biochimica et biophysica acta, 1985, Nov-20, Volume: 847, Issue:2

    Topics: Animals; Calcium; Cattle; Cytoplasm; Drug Antagonism; Gallopamil; Humans; Hyperparathyroidism; Kinetics; Parathyroid Glands; Parathyroid Hormone; Potassium; Verapamil

1985
Pharmacodynamic interaction of gallopamil and propranolol in the conscious dog.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:12

    Topics: Animals; Atropine Derivatives; Blood Pressure; Dogs; Drug Interactions; Female; Gallopamil; Heart Rate; Hemodynamics; Kinetics; Male; Myocardial Contraction; Parasympatholytics; Propranolol; Verapamil

1985
Proceedings: Effects of inhibitors against the uptake of 45Ca at the neurosecretory nerve endings.
    Nihon seirigaku zasshi. Journal of the Physiological Society of Japan, 1974, Sep-01, Volume: 36, Issue:8-9

    Topics: Animals; Calcium; Gallopamil; Nerve Endings; Neurosecretory Systems; Rats; Verapamil

1974
[Treatment of heart arrhythmias with calcium antagonists].
    Zeitschrift fur Kardiologie, 1984, Volume: 73 Suppl 2

    Topics: Arrhythmias, Cardiac; Atrioventricular Node; Calcium Channel Blockers; Cardiac Complexes, Premature; Coronary Circulation; Diltiazem; Drug Therapy, Combination; Electrocardiography; Gallopamil; Heart Conduction System; Heart Rate; Humans; Risk; Sinoatrial Node; Tachycardia; Verapamil

1984
Cat ventricular muscle treated with D600: effects on calcium and potassium currents.
    The Journal of physiology, 1984, Volume: 352

    Topics: Action Potentials; Animals; Calcium; Cats; Electric Conductivity; Gallopamil; In Vitro Techniques; Ion Channels; Muscles; Papillary Muscles; Potassium; Time Factors; Verapamil

1984
Cat ventricular muscle treated with D600: characteristics of calcium channel block and unblock.
    The Journal of physiology, 1984, Volume: 352

    Topics: Action Potentials; Animals; Calcium; Cats; Electric Conductivity; Gallopamil; In Vitro Techniques; Ion Channels; Membrane Potentials; Muscles; Papillary Muscles; Time Factors; Verapamil

1984
Effects of D-600 on sodium current in squid axons.
    The Journal of membrane biology, 1984, Volume: 79, Issue:3

    Topics: Animals; Axons; Decapodiformes; Gallopamil; Ion Channels; Membrane Potentials; Sodium; Verapamil

1984
Calcium channel blockade in smooth muscle of the human upper urinary tract. I. Effects on depolarization-induced activation.
    The Journal of urology, 1984, Volume: 132, Issue:6

    Topics: Action Potentials; Adult; Aged; Calcium; Calcium Channel Blockers; Diltiazem; Gallopamil; Humans; Ion Channels; Kidney Calices; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Papaverine; Potassium; Ureter; Verapamil

1984
Differential effects of D600, nifedipine and dantrolene sodium on excitation-secretion coupling and presynaptic beta-adrenoceptor responses in rat atria.
    British journal of pharmacology, 1984, Volume: 83, Issue:3

    Topics: Animals; Calcium; Calcium Channel Blockers; Dantrolene; Electric Stimulation; Female; Gallopamil; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Manganese; Nifedipine; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Verapamil

1984
Differentiation of calcium ion antagonism and beta-adrenergic blockade.
    Clinical and investigative medicine. Medecine clinique et experimentale, 1980, Volume: 3, Issue:1-2

    Topics: Action Potentials; Adrenergic beta-Antagonists; Blood Pressure; Calcium; Drug Therapy, Combination; Gallopamil; Heart Conduction System; Humans; Myocardial Contraction; Myocardium; Oxygen Consumption; Propranolol; Verapamil

1980
Effects of nonspecific smooth muscle relaxants and Ca-blocker on Ca-release and Ca-binding in microsomal fractions from rabbit taenia coli.
    Japanese journal of pharmacology, 1980, Volume: 30, Issue:5

    Topics: Animals; Calcium; Colon; Gallopamil; In Vitro Techniques; Male; Microsomes; Papaverine; Parasympatholytics; Piperidines; Rabbits; Verapamil

1980
Blocking of acetylcholine-induced channels by extracellular or intracellular application of D600.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1980, Dec-31, Volume: 211, Issue:1182

    Topics: Acetylcholine; Animals; Gallopamil; Ion Channels; Motor Endplate; Neuromuscular Junction; Rana temporaria; Verapamil

1980
Blocking of frog endplate channels by the organic calcium antagonist D600.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1980, Dec-31, Volume: 211, Issue:1182

    Topics: Acetylcholine; Animals; Gallopamil; Ion Channels; Neuromuscular Junction; Potassium; Rana temporaria; Sodium; Verapamil

1980
alpha-adrenergic antagonists as possible calcium channel inhibitors.
    Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Calcium; Cell Line; Cell Membrane; Dioxanes; Dioxins; Gallopamil; Glioma; Ion Channels; Kinetics; Membrane Potentials; Mice; Neuroblastoma; Rats; Verapamil

1981
Nature of anthopleurin-B-induced release of norepinephrine from adrenergic nerves.
    The American journal of physiology, 1982, Volume: 243, Issue:5

    Topics: Adrenergic Fibers; Animals; Cnidaria; Gallopamil; Guanethidine; Guinea Pigs; Intercellular Signaling Peptides and Proteins; Kinetics; Male; Norepinephrine; Ouabain; Peptides; Potassium; Sea Anemones; Tetrodotoxin; Vas Deferens; Verapamil

1982
Diazoxide and D600 inhibition of insulin release. Distinct mechanisms explain the specificity for different stimuli.
    Diabetes, 1982, Volume: 31, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Arginine; Calcium; Depression, Chemical; Diazoxide; Epinephrine; Gallopamil; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Lysine; Male; Rats; Rats, Inbred Strains; Theophylline; Verapamil

1982
Actions of calcium antagonists on calcium currents in Helix neurons. Specificity and potency.
    Circulation research, 1983, Volume: 52, Issue:2 Pt 2

    Topics: Adrenergic beta-Antagonists; Animals; Calcium; Calcium Channel Blockers; Diltiazem; Gallopamil; Helix, Snails; In Vitro Techniques; Ion Channels; Neurons; Temperature; Verapamil

1983
The actions of D 600, aspaminol and papaverine on calcium-, potassium- and histamine-induced contractions of isolated rabbit basilar artery, aorta, taenia coli and tracheal smooth muscle.
    Japanese journal of pharmacology, 1983, Volume: 33, Issue:6

    Topics: Animals; Calcium; Dose-Response Relationship, Drug; Gallopamil; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Piperidines; Potassium; Rabbits; Verapamil

1983
Differential effects of the calcium entry blocker D 600 on contractions of rat and guinea-pig aortas, elicited by various alpha-1 adrenoceptor agonists.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Vasoconstriction; Verapamil; Yohimbine

1984
Reduction of calcium currents in identified neurons of Helix pomatia: intracellular injection of D890.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1984, Volume: 77, Issue:2

    Topics: Animals; Calcium; Gallopamil; Helix, Snails; In Vitro Techniques; Ion Channels; Membrane Potentials; Neurons; Sodium; Verapamil

1984
Action of oxmetidine on the rabbit aorta: comparison with some calcium entry blockers and nitroglycerin.
    Pharmacological research communications, 1984, Volume: 16, Issue:2

    Topics: Animals; Aorta, Thoracic; Calcium Channel Blockers; Female; Gallopamil; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Male; Nifedipine; Nitroglycerin; Rabbits; Vasoconstriction; Verapamil

1984
Lack of effect of D600 on alpha 1-adrenoceptor-mediated contractions of rat isolated anococcygeus muscle.
    European journal of pharmacology, 1984, Oct-30, Volume: 106, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium Channel Blockers; Dose-Response Relationship, Drug; Electric Stimulation; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Potassium; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Verapamil

1984
Effects of smooth muscle calcium antagonists on human basophil histamine release.
    Biochemical pharmacology, 1981, Volume: 30, Issue:20

    Topics: Basophils; Calcium; Dantrolene; Gallic Acid; Gallopamil; Histamine Release; Humans; Muscle Contraction; Muscle, Smooth; Nifedipine; Quercetin; Verapamil

1981
Recognition of the 'calcium paradox' and the effects of verapamil and gallopamil in human adenoidal mast cells.
    Agents and actions, 1984, Volume: 14, Issue:3-4

    Topics: Adenoids; Calcium; Concanavalin A; Gallopamil; Histamine Release; Humans; Mast Cells; Verapamil

1984
Interactions of D600 (methoxyverapamil) and local anesthetics with rat brain alpha-adrenergic and muscarinic receptors.
    Biochemical pharmacology, 1980, Volume: 29, Issue:2

    Topics: Anesthetics, Local; Animals; Gallopamil; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Lidocaine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Cholinergic; Receptors, Muscarinic; Tetracaine; Verapamil

1980
Inhibitory activity of blockers of the slow inward current in rat myocardium, a study in steady state and of rate of action.
    Journal of molecular and cellular cardiology, 1980, Volume: 12, Issue:2

    Topics: Animals; Gallopamil; Heart; Ion Channels; Manganese; Mathematics; Membrane Potentials; Rats; Verapamil

1980
On the mechanism of slow calcium channel block in heart.
    Pflugers Archiv : European journal of physiology, 1980, Volume: 385, Issue:2

    Topics: Animals; Calcium; Calcium Channel Blockers; Cats; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Myocardial Contraction; Myocardium; Sodium; Verapamil

1980
Pharmacology of agents that affect calcium. Agonists and antagonists.
    Chest, 1980, Volume: 78, Issue:1 Suppl

    Topics: Action Potentials; Animals; Calcium; Cats; Cinnarizine; Electrophysiology; Gallopamil; Guinea Pigs; In Vitro Techniques; Ion Channels; Muscle, Smooth; Muscle, Smooth, Vascular; Nifedipine; Nitroprusside; Rabbits; Rats; Verapamil

1980
Calcium- and potassium-channel blockers interact with alpha-adrenoceptors.
    Molecular and cellular endocrinology, 1980, Volume: 19, Issue:3

    Topics: Aminopyridines; Animals; Brain; Calcium; Clonidine; Gallopamil; Guanidines; Ion Channels; Myocardium; Potassium; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Tetraethylammonium Compounds; Verapamil

1980
Competition for slow channel of Ca2+, Mn2+, Verapamil, and D-600 in rat ventricular muscle?
    Journal of molecular and cellular cardiology, 1980, Volume: 12, Issue:6

    Topics: Animals; Calcium; Dose-Response Relationship, Drug; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Manganese; Membrane Potentials; Myocardium; Rats; Verapamil

1980
Effect of compound D-600 (methoxyverapamil) on gluconeogenesis and on acceleration of the process by alpha-adrenergic stimuli in rat kidney tubules.
    The Biochemical journal, 1980, Aug-15, Volume: 190, Issue:2

    Topics: Angiotensin II; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Gallopamil; Gluconeogenesis; Imidazoles; In Vitro Techniques; Kidney Tubules; Male; Norepinephrine; Oxymetazoline; Phentolamine; Rats; Verapamil

1980
Effect of trifluoperazine, D600, and phenytoin on depolarization- and thyrotropin-releasing hormone-induced thyrotropin release from rat pituitary tissue.
    Endocrinology, 1981, Volume: 108, Issue:6

    Topics: Animals; Calcium; Gallopamil; Ion Channels; Male; Membrane Potentials; Phenytoin; Pituitary Gland, Anterior; Potassium; Rats; Sodium; Thyrotropin; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil; Veratridine

1981
The interaction of calcium antagonists (slow channel blockers) with myocardial alpha adrenoceptors.
    Journal of molecular and cellular cardiology, 1982, Volume: 14, Issue:3

    Topics: Animals; Brain; Calcium Channel Blockers; Clonidine; Diltiazem; Gallopamil; In Vitro Techniques; Male; Myocardium; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Verapamil

1982
[Changes of action potential in human papillary muscles by methoxyverapamil (author's transl)].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1982, Volume: 3, Issue:2

    Topics: Action Potentials; Calcium Channel Blockers; Gallopamil; Humans; In Vitro Techniques; Ion Channels; Papillary Muscles; Verapamil

1982
Does the organic calcium channel blocker D600 act from inside or outside on the cardiac cell membrane?
    Pflugers Archiv : European journal of physiology, 1982, Volume: 393, Issue:4

    Topics: Action Potentials; Animals; Calcium; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Ion Channels; Membrane Potentials; Myocardium; Verapamil

1982
Calcium channel block and recovery from block in mammalian ventricular muscle treated with organic channel inhibitors.
    Pflugers Archiv : European journal of physiology, 1982, Volume: 394, Issue:2

    Topics: Action Potentials; Animals; Calcium; Cardiovascular Agents; Cats; Dose-Response Relationship, Drug; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Isoindoles; Phthalimides; Verapamil

1982
Action of a calcium blocking agent (D600) on electrogenesis in the normal heart and the ischaemic heart in the dog.
    Acta cardiologica, 1982, Volume: 37, Issue:3

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Coronary Disease; Dogs; Electrocardiography; Gallopamil; Heart; Heart Conduction System; Ion Channels; Myocardial Contraction; Verapamil

1982
Characterization of [3H]nifedipine binding sites in rabbit myocardium.
    European journal of pharmacology, 1982, Dec-03, Volume: 85, Issue:3-4

    Topics: Animals; Binding Sites; Calcium; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Ion Channels; Kinetics; Myocardial Contraction; Myocardium; Nifedipine; Pyridines; Rabbits; Stereoisomerism; Tritium; Verapamil

1982
Interval- and voltage-dependent effects of the calcium channel-blocking agents D600 and AQA 39 on mammalian ventricular muscle.
    Circulation research, 1983, Volume: 52, Issue:2 Pt 2

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Cats; Diastole; Electric Stimulation; Gallopamil; Heart; Ion Channels; Isoindoles; Phthalimides; Rabbits; Verapamil

1983
Mechanism of calcium channel blockade by verapamil, D600, diltiazem and nitrendipine in single dialysed heart cells.
    Nature, 1983, Apr-28, Volume: 302, Issue:5911

    Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Cats; Diltiazem; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Verapamil

1983
Effects of the calcium-channel blockers cobalt, verapamil, and D600 on Leydig cell steroidogenesis.
    Biology of reproduction, 1983, Volume: 28, Issue:3

    Topics: Androgens; Animals; Calcium Channel Blockers; Cobalt; Gallopamil; Leydig Cells; Male; Mice; Phosphoprotein Phosphatases; Protein Biosynthesis; Verapamil

1983
Calcium channel antagonists verapamil and gallopamil are powerful inhibitors of acid secretion in isolated and enriched guinea pig parietal cells.
    Pharmacology, 1983, Volume: 27, Issue:1

    Topics: Adenosine Triphosphatases; Animals; Bucladesine; Calcium Channel Blockers; Female; Gallopamil; Gastric Acid; Gastric Mucosa; Guinea Pigs; H(+)-K(+)-Exchanging ATPase; Histamine; In Vitro Techniques; Male; Verapamil

1983
Slow calcium channel blockers and the calcium paradox: comparative studies in the rat with seven drugs.
    Journal of molecular and cellular cardiology, 1983, Volume: 15, Issue:7

    Topics: Animals; Butylamines; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Fendiline; Gallopamil; In Vitro Techniques; Ion Channels; Male; Myocardium; Nifedipine; Prenylamine; Rats; Verapamil

1983
Calcium antagonistic drugs differ in ability to block the slow Na+ channels of young embryonic chick hearts.
    European journal of pharmacology, 1983, Oct-14, Volume: 94, Issue:1-2

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Chick Embryo; Gallopamil; In Vitro Techniques; Ion Channels; Myocardium; Nifedipine; Sodium; Verapamil

1983
The protective effects of D-600 and propranolol on reperfusion injury in the anaesthetized rabbit.
    Canadian journal of physiology and pharmacology, 1984, Volume: 62, Issue:2

    Topics: 4-Nitrophenylphosphatase; Adenosine Triphosphate; Anesthesia; Animals; Coronary Circulation; Gallopamil; Heart; Ions; Male; Membranes; Myocardial Contraction; Myocardium; Propranolol; Rabbits; Sarcolemma; Sodium-Potassium-Exchanging ATPase; Subcellular Fractions; Verapamil

1984
Kinetics of acetylcholine-activated cation channel blockade by the calcium antagonist D-600 in Aplysia neurons.
    Cellular and molecular neurobiology, 1983, Volume: 3, Issue:4

    Topics: Acetylcholine; Animals; Aplysia; Calcium; Dose-Response Relationship, Drug; Gallopamil; Ganglia; Ion Channels; Kinetics; Membrane Potentials; Neurons; Receptors, Cholinergic; Synaptic Transmission; Verapamil

1983
Comparison of pinaverium bromide, manganese chloride and D600 effects on electrical and mechanical activities in rat uterine smooth muscle.
    European journal of pharmacology, 1984, Feb-10, Volume: 98, Issue:1

    Topics: Action Potentials; Animals; Calcium; Chlorides; Egtazic Acid; Female; Gallopamil; In Vitro Techniques; Ion Channels; Manganese; Manganese Compounds; Morpholines; Muscle Contraction; Muscle, Smooth; Myometrium; Pregnancy; Rats; Uterus; Verapamil

1984
Tissue response selectivity of calcium antagonists is not due to heterogeneity of [3H]-nitrendipine binding sites.
    British journal of pharmacology, 1984, Volume: 82, Issue:2

    Topics: Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Channels; Diltiazem; Female; Gallopamil; In Vitro Techniques; Isometric Contraction; Kinetics; Membranes; Muscle, Smooth, Vascular; Myocardium; Nicardipine; Nifedipine; Organ Specificity; Rabbits; Receptors, Nicotinic; Verapamil

1984
Renal effects of methoxyverapamil in anesthetized rats.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:2

    Topics: Anesthesia, Intravenous; Animals; Blood Pressure; Calcium; Gallopamil; Kidney; Male; p-Aminohippuric Acid; Potassium; Rats; Rats, Inbred Strains; Renin; Sodium; Verapamil

1983
Structure-function relationship of calcium ion channel antagonists at the pituitary gonadotrope.
    Endocrinology, 1983, Volume: 113, Issue:5

    Topics: Animals; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Female; Gallopamil; Gonadotropin-Releasing Hormone; Luteinizing Hormone; Pituitary Gland; Rats; Structure-Activity Relationship; Verapamil; Veratridine

1983
Participation of calcium and calmodulin in the formation of acetylcholine receptor clusters.
    The Journal of cell biology, 1984, Volume: 98, Issue:2

    Topics: Animals; Calcium; Calmodulin; Cells, Cultured; Embryo, Nonmammalian; Fluorescent Antibody Technique; Gallopamil; Kinetics; Muscles; Nifedipine; Receptors, Cholinergic; Trifluoperazine; Verapamil; Xenopus

1984
Conformational analysis of the calcium-antagonist gallopamil.
    Biochemical pharmacology, 1983, Feb-01, Volume: 32, Issue:3

    Topics: Calcimycin; Calcium Channel Blockers; Gallopamil; Hydrogen-Ion Concentration; Models, Molecular; Molecular Conformation; Verapamil

1983
Verapamil inhibition of vasopressin-stimulated water flow: possible role of intracellular calcium.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Animals; Arginine Vasopressin; Biological Transport; Bufo marinus; Calcium Channel Blockers; Cell Membrane Permeability; Epithelium; Gallopamil; Osmolar Concentration; Urinary Bladder; Verapamil; Water-Electrolyte Balance

1983
Blockers of calcium permeability inhibit neurite extension and formation of neuromuscular synapses in cell culture.
    Brain research, 1984, Volume: 316, Issue:2

    Topics: Age Factors; Animals; Cadmium; Calcium Channel Blockers; Chick Embryo; Cobalt; Gallopamil; Lanthanum; Manganese; Neuromuscular Junction; Nifedipine; Nitrendipine; Retina; Verapamil

1984
Cellular actions and pharmacology of the calcium channel blocking drugs.
    The American journal of medicine, 1984, Aug-31, Volume: 77, Issue:2B

    Topics: Action Potentials; Biological Transport, Active; Calcium; Calcium Channel Blockers; Cell Membrane; Gallopamil; Heart; Humans; Muscle Contraction; Verapamil

1984
The effect of gallamine, gallopamil and nifedipine on responses to acetylcholine and carbachol in the taenia of the guinea-pig caecum.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Calcium; Carbachol; Cecum; Drug Interactions; Gallamine Triethiodide; Gallopamil; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Paraoxon; Time Factors; Verapamil

1984
Voltage clamp comparison of the organic calcium channel blockers D-600 and nisoldipine.
    Proceedings of the Western Pharmacology Society, 1984, Volume: 27

    Topics: Animals; Anura; Atrial Function; Calcium Channel Blockers; Electrophysiology; Gallopamil; Heart Atria; In Vitro Techniques; Kinetics; Nifedipine; Nisoldipine; Verapamil

1984
Inhibition of [3H]spiperone binding to 5-HT2 receptors of rat cerebral cortex by the calcium antagonists verapamil and D600.
    European journal of pharmacology, 1984, Oct-30, Volume: 106, Issue:1

    Topics: Animals; Binding, Competitive; Butyrophenones; Cerebral Cortex; Gallopamil; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiperone; Verapamil

1984
[Multicenter long-term study of gallopamil in patients with coronary heart disease].
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:11

    Topics: Adult; Aged; Angina Pectoris; Blood Pressure; Coronary Disease; Electrocardiography; Female; Gallopamil; Heart Rate; Humans; Male; Middle Aged; Time Factors; Verapamil

1984
Paralysis of frog skeletal muscle fibres by the calcium antagonist D-600.
    The Journal of physiology, 1983, Volume: 341

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscles; Potassium; Rana temporaria; Temperature; Verapamil

1983
Charge movement in skeletal muscle fibers paralyzed by the calcium-entry blocker D600.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:8

    Topics: Animals; Electric Conductivity; Gallopamil; Membrane Potentials; Muscles; Paralysis; Potassium; Rana temporaria; Verapamil

1984
Blockade of Ca2+ channels inhibits K+ contractures but not twitches in skeletal muscle.
    Canadian journal of physiology and pharmacology, 1984, Volume: 62, Issue:4

    Topics: Animals; Calcium Channel Blockers; Gallopamil; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Potassium; Rana pipiens; Verapamil

1984
Veratridine and ouabain stimulate calcium-dependent prolactin release.
    Endocrinology, 1983, Volume: 113, Issue:4

    Topics: Animals; Bromocriptine; Calcium; Cells, Cultured; Gallopamil; Male; Ouabain; Pituitary Gland, Anterior; Prolactin; Rats; Sodium; Tetrodotoxin; Verapamil; Veratridine; Veratrine

1983
Calcium antagonists and calmodulin inhibitors block cytokinin-induced bud formation in Funaria.
    Developmental biology, 1983, Volume: 99, Issue:1

    Topics: Calcium; Calmodulin; Cell Division; Cells, Cultured; Chlorpromazine; Cytokinins; Gallic Acid; Gallopamil; Lanthanum; Plant Growth Regulators; Plants; Trifluoperazine; Verapamil

1983
[Effect of calcium antagonists on the response of the rat vas deferens to noradrenaline and field stimulation].
    Revista espanola de fisiologia, 1983, Volume: 39, Issue:2

    Topics: Animals; Calcium Channel Blockers; Electric Stimulation; Gallopamil; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Inbred Strains; Vas Deferens; Verapamil

1983
Effects of calcium-antagonists on passive cutaneous anaphylaxis in the rat.
    International journal of immunopharmacology, 1983, Volume: 5, Issue:5

    Topics: Animals; Calcium Channel Blockers; Diltiazem; Gallopamil; Male; Nifedipine; Passive Cutaneous Anaphylaxis; Rats; Verapamil

1983
[Ba-induced contraction of the guinea pig ileal longitudinal muscle and its inhibition by D-600, benactyzine, and papaverine].
    Nihon Heikatsukin Gakkai zasshi, 1983, Volume: 19, Issue:2

    Topics: Animals; Barium; Benactyzine; Calcium; Gallopamil; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Papaverine; Verapamil

1983
[Histamine-induced contraction of the guinea pig taenia coli and its inhibition by D-600, papaverine, and benactyzine].
    Nihon Heikatsukin Gakkai zasshi, 1983, Volume: 19, Issue:2

    Topics: Animals; Benactyzine; Calcium; Colon; Gallopamil; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nitroprusside; Papaverine; Verapamil

1983
The effect of verapamil and other calcium antagonists on chemotaxis of polymorphonuclear leukocytes.
    Biochemical pharmacology, 1984, Jan-01, Volume: 33, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Cell Survival; Chemotaxis, Leukocyte; Diltiazem; Gallopamil; Magnesium; Neutrophils; Perhexiline; Prenylamine; Rabbits; Verapamil

1984
[Regularization of ventricular intervals in atrial fibrillation--electrophysiologic findings on the underlying mechanism].
    Zeitschrift fur Kardiologie, 1984, Volume: 73, Issue:2

    Topics: Adult; Aged; Atrial Fibrillation; Atrioventricular Node; Cardiac Pacing, Artificial; Electrocardiography; Female; Gallopamil; Heart Conduction System; Heart Rate; Humans; Male; Middle Aged; Verapamil

1984
An investigation of the involvement of calcium in the control of prolactin secretion: studies with low calcium, methoxyverapamil, cobalt and manganese.
    The Journal of endocrinology, 1984, Volume: 101, Issue:3

    Topics: Animals; Calcium; Cells, Cultured; Cobalt; Dose-Response Relationship, Drug; Gallopamil; Male; Manganese; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Verapamil

1984
Contribution of adenosine to the regulation of cerebral blood flow: the role of calcium ions in the adenosine-induced cerebrocortical vasodilatation.
    Advances in experimental medicine and biology, 1984, Volume: 169

    Topics: Adenosine; Animals; Calcium; Calcium Channel Blockers; Cats; Cerebral Cortex; Cerebrovascular Circulation; Gallopamil; Hypoxia; NAD; Oxidation-Reduction; Seizures; Vasodilation; Verapamil

1984
Depletion of cardiac noradrenaline stores by the calcium-channel blocker D-600.
    Canadian journal of physiology and pharmacology, 1984, Volume: 62, Issue:6

    Topics: Animals; Gallopamil; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Time Factors; Verapamil

1984
Potentiation of etoposide-induced DNA damage by calcium antagonists in L1210 cells in vitro.
    Cancer research, 1984, Volume: 44, Issue:8

    Topics: Animals; Cell Division; Cell Nucleus; Cell Survival; DNA Replication; DNA, Neoplasm; Drug Synergism; Etoposide; Gallopamil; Kinetics; Leukemia L1210; Mice; Podophyllotoxin; Verapamil

1984
Induction of accelerated acrosome reaction in guinea pig sperm.
    Biology of reproduction, 1980, Volume: 22, Issue:3

    Topics: Acrosome; Animals; Biological Transport, Active; Calcium; Egtazic Acid; Gallopamil; Guinea Pigs; Kinetics; Male; Sperm Capacitation; Spermatozoa; Verapamil

1980
The inhibitory effects of D-600 and cobalt on theophylline-mediated calcitonin secretion and calcium distribution in porcine thyroid slices.
    Research communications in chemical pathology and pharmacology, 1980, Volume: 30, Issue:2

    Topics: Animals; Calcitonin; Calcium; Cobalt; Gallopamil; In Vitro Techniques; Mannitol; Swine; Theophylline; Thyroid Gland; Verapamil

1980
Pharmacology and electrophysiology of calcium ion antagonists.
    Clinical and investigative medicine. Medecine clinique et experimentale, 1980, Volume: 3, Issue:1-2

    Topics: Calcium; Cardiovascular Diseases; Gallopamil; Heart; Humans; Myocardial Contraction; Nitroglycerin; Verapamil

1980
Effect of the organic calcium antagonist D-600 on cerebrocortical vascular and redox responses evoked by adenosine, anoxia, and epilepsy.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1983, Volume: 3, Issue:1

    Topics: Adenosine; Animals; Blood Volume; Cats; Cerebral Cortex; Cerebrovascular Circulation; Electrocardiography; Gallopamil; Hypoxia; Male; NAD; Oxidation-Reduction; Seizures; Verapamil

1983
Influence of Ca++-channel blocking agents on calcium transients and tension development in isolated mammalian heart muscle.
    Circulation research, 1983, Volume: 52, Issue:2 Pt 2

    Topics: Animals; Calcium; Calcium Channel Blockers; Cats; Dogs; Gallopamil; In Vitro Techniques; Myocardial Contraction; Myocardium; Papillary Muscles; Verapamil

1983
Inhibition of calcium uptake, sodium uptake, and catecholamine secretion by methoxyverapamil (D600) in primary cultures of adrenal medulla cells.
    Journal of neurochemistry, 1983, Volume: 40, Issue:4

    Topics: Adrenal Medulla; Animals; Biological Transport, Active; Calcium; Catecholamines; Cattle; Cells, Cultured; Gallopamil; Kinetics; Nicotine; Sodium; Tetrodotoxin; Verapamil; Veratridine

1983
Calcium antagonistic activity and myocardial ischemic protection by both stereoisomers of verapamil.
    Advances in myocardiology, 1983, Volume: 4

    Topics: Animals; Aorta; Calcium; Coronary Disease; Dose-Response Relationship, Drug; Gallopamil; Heart; Rabbits; Stereoisomerism; Swine; Verapamil

1983
A 113Cd and 1H NMR study of the interaction of calmodulin with D600, trifluoperazine and some other hydrophobic drugs.
    European journal of biochemistry, 1983, Aug-15, Volume: 134, Issue:3

    Topics: Animals; Binding Sites; Calcium; Calcium-Binding Proteins; Calmodulin; Cattle; Chemical Phenomena; Chemistry; Gallopamil; Magnetic Resonance Spectroscopy; Male; Protein Binding; Testis; Trifluoperazine; Verapamil

1983
Actions of a calium antagonist, the D-600, on electrical and mechanical properties of frog skeletal muscle.
    Progress in neuro-psychopharmacology, 1980, Volume: 4, Issue:2

    Topics: Animals; Anura; Calcium; Electric Stimulation; Gallopamil; Membrane Potentials; Muscle Contraction; Muscles; Neuromuscular Junction; Rana pipiens; Verapamil

1980
Effect of D-600 on inhibition of in vitro renin release in the rat by high extracellular potassium and angiotensin II.
    The Journal of physiology, 1980, Volume: 304

    Topics: Angiotensin II; Animals; Calcium; Gallopamil; In Vitro Techniques; Kidney Cortex; Potassium; Rats; Renin; Secretory Rate; Verapamil

1980
Renin release from isolated rat glomeruli: seasonal variations and effects of D600 on the response to calcium deprivation.
    The Journal of physiology, 1981, Volume: 310

    Topics: Animals; Calcium; Gallopamil; In Vitro Techniques; Kidney Glomerulus; Male; Rats; Renin; Seasons; Secretory Rate; Verapamil

1981
Inhibition by D 600 of norepinephrine- and clonidine-induced responses of the aortae from normotensive (WKY) and spontaneously hypertensive rats (SHR).
    Life sciences, 1982, Jan-04, Volume: 30, Issue:1

    Topics: Animals; Aorta; Calcium Channel Blockers; Clonidine; Gallopamil; Hypertension; In Vitro Techniques; Norepinephrine; Rats; Rats, Inbred Strains; Vasoconstriction; Verapamil

1982
Extracellular calcium concentration and calcium blocking agents on the action of ouabain on isolated rat atrium.
    Pharmacological research communications, 1982, Volume: 14, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Diltiazem; Electric Stimulation; Gallopamil; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Ouabain; Rats; Rats, Inbred Strains; Verapamil

1982
The interaction of [3H]nitrendipine with receptors for calcium antagonists in the cerebral cortex and heart of rats.
    Biochemical and biophysical research communications, 1982, Feb-11, Volume: 104, Issue:3

    Topics: Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Chloride; Cerebral Cortex; Diltiazem; Gallopamil; Kinetics; Lanthanum; Male; Myocardium; Nifedipine; Nitrendipine; Pyridines; Rats; Rats, Inbred Strains; Receptors, Drug; Verapamil

1982
Inhibition by methoxyverapamil of the responses of smooth muscle from spontaneously hypertensive and normotensive rats.
    Blood vessels, 1982, Volume: 19, Issue:4

    Topics: Animals; Blood Pressure; Calcium; Calcium Channel Blockers; Drug Interactions; Gallopamil; Hypertension; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rats; Rats, Inbred Strains; Verapamil

1982
Influence of the extent of the zone at risk on the effectiveness of drugs in reducing infarct size.
    Circulation, 1982, Volume: 66, Issue:1

    Topics: Animals; Autoradiography; Calcium Channel Blockers; Collateral Circulation; Coronary Circulation; Disease Models, Animal; Dogs; Gallopamil; Myocardial Infarction; Myocardium; Verapamil

1982
Potentiation of indirectly induced muscle twitches by organic calcium antagonists in phrenic nerve-diaphragm muscle preparations of mice.
    Japanese journal of pharmacology, 1982, Volume: 32, Issue:1

    Topics: Animals; Calcium Channel Blockers; Diltiazem; Gallopamil; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Stimulation, Chemical; Verapamil

1982
[Heart rate reduction in atrial fibrillation with a rapid ventricular response by Gallopamil, a Ca-antagonist (author's transl)].
    Zeitschrift fur Kardiologie, 1982, Volume: 71, Issue:5

    Topics: Administration, Oral; Adult; Aged; Atrial Fibrillation; Atrioventricular Node; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; Heart Rate; Heart Ventricles; Humans; Middle Aged; Monitoring, Physiologic; Verapamil

1982
Effects of nitroprusside and D600 on norepinephrine and KCl activating systems in canine renal vein.
    Proceedings of the Western Pharmacology Society, 1982, Volume: 25

    Topics: Animals; Calcium Radioisotopes; Dogs; Ferricyanides; Gallopamil; In Vitro Techniques; Muscle, Smooth, Vascular; Nitroprusside; Norepinephrine; Potassium Chloride; Renal Veins; Verapamil

1982
Effect of Ca2+ blocking agents on the metabolism of low density lipoproteins in human skin fibroblasts.
    Biochemical and biophysical research communications, 1982, Jul-16, Volume: 107, Issue:1

    Topics: Benzazepines; Calcium Channel Blockers; Dibucaine; Diltiazem; Fendiline; Fibroblasts; Gallopamil; Humans; Kinetics; Lipoproteins, LDL; Nifedipine; Phenethylamines; Prenylamine; Pyridines; Skin; Trifluoperazine; Verapamil

1982
Certain calcium antagonists are potent displacers of [3H]phencyclidine (PCP) binding in rat brain.
    European journal of pharmacology, 1982, Sep-10, Volume: 83, Issue:1-2

    Topics: Animals; Binding, Competitive; Brain; Calcium Channel Blockers; Gallopamil; In Vitro Techniques; Nifedipine; Nitrendipine; Olfactory Bulb; Phencyclidine; Rats; Verapamil

1982
Actions of D 600 on isolated rabbit aorta.
    General pharmacology, 1982, Volume: 13, Issue:4

    Topics: Animals; Aorta; Calcium; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Rabbits; Verapamil

1982
D-600 blocks spontaneous discharge, excitability and contraction of cultured embryonic chick heart cells.
    Journal of molecular and cellular cardiology, 1982, Volume: 14, Issue:5

    Topics: Action Potentials; Animals; Cells, Cultured; Chick Embryo; Electrophysiology; Gallopamil; Heart; Myocardial Contraction; Verapamil

1982
Release of norepinephrine and dopamine from brain vesicular preparations: effects of calcium antagonists.
    Cellular and molecular neurobiology, 1982, Volume: 2, Issue:3

    Topics: Animals; Benzazepines; Calcium; Cerebral Cortex; Corpus Striatum; Diltiazem; Dopamine; Gallopamil; Guinea Pigs; Kinetics; Male; Norepinephrine; Potassium; Verapamil

1982
D-600 and the membrane stabilizing effect of calcium in vascular smooth muscle.
    Pharmacology, 1982, Volume: 25, Issue:5

    Topics: Animals; Caffeine; Calcium; Gallopamil; Male; Membranes; Methoxamine; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Verapamil

1982
Conformation analysis of the neutral and protonated forms of gallopamil (D600).
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 259, Issue:2

    Topics: Calcium Channel Blockers; Chemical Phenomena; Chemistry, Physical; Gallopamil; Molecular Conformation; Verapamil

1982
[Importance of the size of the ischemic area on the beneficial effects of drugs capable of protecting the ischemic myocardium].
    Arquivos brasileiros de cardiologia, 1982, Volume: 39, Issue:5

    Topics: Animals; Blood Pressure; Dogs; Gallopamil; Heart Rate; Myocardial Infarction; Myocardium; Verapamil

1982
Stereoselective and non-stereoselective effects of D 600 (methoxyverapamil) in smooth muscle preparations.
    European journal of pharmacology, 1981, Nov-19, Volume: 76, Issue:1

    Topics: Animals; Calcium; Gallopamil; Guinea Pigs; Ileum; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Portal Vein; Potassium; Rats; Receptors, Adrenergic; Stereoisomerism; Vas Deferens; Verapamil

1981
Effects of several calcium antagonists and dipyridamole in the isolated perfused guinea pig heart.
    Life sciences, 1980, Dec-15, Volume: 27, Issue:24

    Topics: Animals; Calcium; Coronary Circulation; Dipyridamole; Gallopamil; Guinea Pigs; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Nifedipine; Oxygen Consumption; Perfusion; Pyridines; Verapamil

1980
Differential effects of D 600 on contractile response of aorta and portal vein from spontaneously hypertensive rats.
    Blood vessels, 1981, Volume: 18, Issue:3

    Topics: Animals; Aorta; Blood Pressure; Calcium; Gallopamil; Hypertension; Muscle Contraction; Portal Vein; Rats; Verapamil

1981
The negative inotropic potency of compound D 600 in rat, guinea pig, and rabbit cardiac preparations.
    Canadian journal of physiology and pharmacology, 1980, Volume: 58, Issue:12

    Topics: Animals; Calcium; Depression, Chemical; Dose-Response Relationship, Drug; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Rabbits; Rats; Species Specificity; Verapamil

1980
Calcium entry blockers and vascular smooth muscle heterogeneity.
    Federation proceedings, 1981, Volume: 40, Issue:14

    Topics: Animals; Calcium; Calcium Channel Blockers; Cinnarizine; Flunarizine; Gallopamil; Lidoflazine; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Verapamil

1981
[Effect of calcium antagonists on action potentials of muscle fibers in the warm-blooded].
    Biulleten' eksperimental'noi biologii i meditsiny, 1981, Volume: 92, Issue:11

    Topics: Action Potentials; Animals; Calcium Channel Blockers; Diaphragm; Gallopamil; In Vitro Techniques; Mice; Muscle Denervation; Muscles; Verapamil

1981
[Effects of D-600 (methoxy-verapamil) on mortality and infarction size after coronary occlusion in rats].
    Arquivos brasileiros de cardiologia, 1981, Volume: 37, Issue:2

    Topics: Animals; Gallopamil; Myocardial Contraction; Myocardial Infarction; Myocardium; Prognosis; Rats; Rats, Inbred Strains; Verapamil

1981
A calcium-dependent acetylcholine depolarization blocked by methoxyverapamil (D600) and procaine in snail neurones.
    British journal of pharmacology, 1980, Volume: 68, Issue:2

    Topics: Acetylcholine; Animals; Calcium; Cobalt; Gallopamil; Helix, Snails; Membrane Potentials; Neurons; Procaine; Verapamil

1980
Some effects of sodium nitroprusside, methoxyverapamil (D600) and nifedipine on rat portal vein.
    British journal of pharmacology, 1980, Volume: 68, Issue:2

    Topics: Animals; Calcium; Electrophysiology; Ferricyanides; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Nitroprusside; Norepinephrine; Phentolamine; Portal Vein; Pyridines; Rats; Verapamil

1980
Interaction of D 600 with phenoxybenzamine-induced adrenergic blockade.
    European journal of pharmacology, 1980, Mar-21, Volume: 62, Issue:2-3

    Topics: Animals; Drug Interactions; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phenoxybenzamine; Rats; Sympathetic Nervous System; Time Factors; Vas Deferens; Verapamil

1980
Differences in contractile responses to acetylcholine and serotonin in rat stomach fundus strips.
    European journal of pharmacology, 1980, Jul-25, Volume: 65, Issue:2-3

    Topics: Acetylcholine; Animals; Calcium; Gallopamil; In Vitro Techniques; Lanthanum; Muscle Contraction; Muscle, Smooth; Rats; Serotonin; Stomach; Temperature; Verapamil

1980
Influence of frequency and calcium concentration on the inotropic actions of D600 in the rat and guinea pig myocardium.
    Proceedings of the Western Pharmacology Society, 1980, Volume: 23

    Topics: Animals; Calcium; Electric Stimulation; Female; Gallopamil; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Rats; Species Specificity; Verapamil

1980
Effects of hydralazine and D-600 on KCl induced contraction and phosphorylase activation in rabbit aorta.
    Proceedings of the Western Pharmacology Society, 1980, Volume: 23

    Topics: Animals; Aorta; Drug Interactions; Enzyme Activation; Gallopamil; Hydralazine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phosphorylases; Potassium Chloride; Rabbits; Verapamil

1980
Spasmolytic action of verapamil, D600 and cinchocaine on the rat vas deferens.
    Archives internationales de pharmacodynamie et de therapie, 1980, Volume: 244, Issue:1

    Topics: Animals; Calcium; Dibucaine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Parasympatholytics; Potassium; Rats; Vas Deferens; Verapamil

1980
A comparison of the influence of La3+, D600 and gentamicin on frequency-force relationships in isolated myocardium.
    European journal of pharmacology, 1980, Sep-05, Volume: 66, Issue:4

    Topics: Animals; Calcium; Electric Stimulation; Gallopamil; Gentamicins; Guinea Pigs; Heart Rate; In Vitro Techniques; Lanthanum; Male; Myocardial Contraction; Verapamil

1980
Effects of some calcium antagonists on the excitation-contraction coupling in the myocardium under steady-state and nonsteady-state conditions of operation.
    Acta physiologica et pharmacologica Bulgarica, 1980, Volume: 6, Issue:2

    Topics: Action Potentials; Animals; Calcium; Electric Stimulation; Gallopamil; Guinea Pigs; In Vitro Techniques; Manganese; Myocardial Contraction; Verapamil

1980
Effect of "calcium antagonist" D-600 on the postsynaptic membrane.
    Journal de physiologie, 1980, Volume: 76, Issue:5

    Topics: Acetylcholine; Animals; Calcium; Chlorides; Gallopamil; In Vitro Techniques; Kinetics; Mollusca; Sodium; Synaptic Membranes; Tubocurarine; Verapamil

1980
A sodium-calcium exchange mechanism in plasma membrane vesicles isolated from ram sperm flagella.
    FEBS letters, 1980, Nov-17, Volume: 121, Issue:1

    Topics: Animals; Biological Transport, Active; Calcium; Carrier Proteins; Cell Membrane; Cell-Free System; Gallopamil; Male; Membrane Proteins; Sheep; Sodium; Sodium-Calcium Exchanger; Sperm Tail; Spermatozoa; Verapamil

1980
Inhibition by the combined Ca2+ and 5-HT2 receptor antagonist nexopamil (LU 49938) of intracoronary thrombus formation in a canine model of arterial stenosis and intimal damage.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:5

    Topics: Animals; Calcium; Coronary Circulation; Coronary Thrombosis; Dogs; Female; Gallopamil; Hemodynamics; Injections, Intravenous; Ketanserin; Male; Platelet Aggregation; Platelet Aggregation Inhibitors; Serotonin Antagonists; Verapamil

1993
[Ca(2+)-channel blockers and binding of tricyclic antidepressive agents].
    Ceskoslovenska psychiatrie, 1995, Volume: 91, Issue:3

    Topics: Animals; Antidepressive Agents, Tricyclic; Blood Platelets; Calcium Channel Blockers; Cattle; Cell Membrane; Desipramine; Gallopamil; Humans; Imipramine; In Vitro Techniques; Lymphocytes; Phosphatidylserines; Synaptic Membranes; Verapamil

1995
The block of the expressed L-type calcium channel is modulated by the beta 3 subunit.
    FEBS letters, 1995, Oct-09, Volume: 373, Issue:2

    Topics: Animals; Benzimidazoles; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; CHO Cells; Cricetinae; Feedback; Gallopamil; Gene Expression; Intracellular Membranes; Isradipine; Macromolecular Substances; Membrane Potentials; Mibefradil; Microsomes; Myocardium; Rabbits; Recombinant Proteins; Structure-Activity Relationship; Tetrahydronaphthalenes; Transfection; Verapamil

1995
Effect of UK-84149 on voltage-activated calcium currents of single smooth muscle cells from guinea-pig and rabbit jejunum and rabbit coronary artery.
    British journal of pharmacology, 1995, Volume: 114, Issue:8

    Topics: Animals; Aorta; Arteries; Calcium Channel Blockers; Calcium Channels; Coronary Vessels; Dibenzothiazepines; Dose-Response Relationship, Drug; Evoked Potentials; Gallopamil; Guinea Pigs; Jejunum; Muscle, Smooth, Vascular; Nicardipine; Patch-Clamp Techniques; Rabbits; Time Factors; Verapamil

1995
Effects of catecholamines on the residual sodium channel dependent slow conduction in guinea pig ventricular muscles under normoxia and hypoxia.
    Cardiovascular research, 1995, Volume: 29, Issue:1

    Topics: Action Potentials; Animals; Arrhythmias, Cardiac; Calcium Channels; Catecholamines; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Hypoxia; In Vitro Techniques; Isoproterenol; Membrane Potentials; Myocardial Infarction; Myocardium; Norepinephrine; Pindolol; Potassium; Sodium Channels; Verapamil

1995
Conformational analysis of free and Ca(2+)-bound forms of verapamil and methoxyverapamil.
    Journal of biomolecular structure & dynamics, 1993, Volume: 11, Issue:3

    Topics: Binding Sites; Calcium; Computer Simulation; Gallopamil; Models, Molecular; Molecular Conformation; Verapamil

1993
Ovine tracheal muscle contraction in vitro: inhibition by calcium channel blockers gallopamil and verapamil.
    Respiration; international review of thoracic diseases, 1993, Volume: 60, Issue:1

    Topics: Acetylcholine; Animals; Gallopamil; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Sheep; Trachea; Verapamil

1993
Extracellular site of action of phenylalkylamines on L-type calcium current in rat ventricular myocytes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: Animals; Binding Sites; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Gallopamil; Heart Ventricles; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Verapamil

1995
Transfer of L-type calcium channel IVS6 segment increases phenylalkylamine sensitivity of alpha1A.
    The Journal of biological chemistry, 1996, May-17, Volume: 271, Issue:20

    Topics: Amino Acid Sequence; Animals; Calcium Channel Blockers; Calcium Channels; Gallopamil; Molecular Sequence Data; Rabbits; Structure-Activity Relationship; Verapamil; Xenopus laevis

1996
Persisting effect of Ca(2+)-channel blockers on left ventricular function in hypertrophic cardiomyopathy after 14 years' treatment.
    Angiology, 1996, Volume: 47, Issue:8

    Topics: Adult; Calcium Channel Blockers; Cardiomyopathy, Hypertrophic; Echocardiography, Doppler, Pulsed; Exercise Test; Female; Gallopamil; Humans; Male; Middle Aged; Time Factors; Treatment Outcome; Ventricular Function, Left; Verapamil

1996
Prostacyclin and thromboxane production of rat and cat arterial tissue is altered independently by several vasoactive substances.
    Prostaglandins, 1996, Volume: 52, Issue:3

    Topics: 6-Ketoprostaglandin F1 alpha; Angiotensin II; Animals; Antihypertensive Agents; Aorta; Bradykinin; Calcium Channel Blockers; Cardiotonic Agents; Cats; Dopamine; Dose-Response Relationship, Drug; Epoprostenol; Gallopamil; Isoproterenol; Norepinephrine; Phentolamine; Propranolol; Rats; Thrombin; Thromboxane B2; Vasoconstrictor Agents; Vasodilator Agents; Vasopressins; Verapamil

1996
Distinct effects of mutations in transmembrane segment IVS6 on block of L-type calcium channels by structurally similar phenylalkylamines.
    Molecular pharmacology, 1996, Volume: 50, Issue:5

    Topics: Amino Acid Sequence; Aniline Compounds; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Electrophysiology; Gallopamil; Kinetics; Molecular Sequence Data; Mutation; Protein Structure, Secondary; Structure-Activity Relationship; Verapamil

1996
Action of tertiary phenylalkylamines on cardiac transient outward current from outside the cell membrane.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:6

    Topics: Animals; Gallopamil; Heart; Hydrogen-Ion Concentration; Rats; Rats, Sprague-Dawley; Verapamil

1996
Characterization of the high-affinity verapamil binding site in a plant plasma membrane Ca2+-selective channel.
    The Journal of membrane biology, 1997, May-15, Volume: 157, Issue:2

    Topics: Binding Sites; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Gallopamil; Membrane Potentials; Plant Roots; Triticum; Verapamil

1997
Comparative study on the effect of calcium channel blockers on basal and parathyroid hormone-induced bone resorption in vitro.
    Pharmacology & toxicology, 1997, Volume: 80, Issue:6

    Topics: Amlodipine; Animals; Bone Resorption; Calcium Channel Blockers; Gallopamil; Mice; Nifedipine; Organ Culture Techniques; Parathyroid Hormone; Parietal Bone; Specific Pathogen-Free Organisms; Verapamil

1997
Verapamil, a phenylalkylamine Ca2+ channel blocker, inhibits ATP-sensitive K+ channels in insulin-secreting cells from rats.
    Diabetologia, 1997, Volume: 40, Issue:12

    Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Channel Blockers; Calcium Radioisotopes; Female; Gallopamil; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Potassium Channel Blockers; Potassium Channels; Pyridines; Rats; Rubidium Radioisotopes; Thiadiazines; Verapamil

1997
Comparative effects of gallopamil and verapamil on the mechanical and electrophysiological parameters of isolated guinea-pig myocardium.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:12

    Topics: Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Electrophysiology; Gallopamil; Guinea Pigs; Heart; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Ventricular Function, Right; Verapamil

1997
Straightforward solid-phase extraction method for the determination of verapamil and its metabolite in plasma in a 96-well extraction plate.
    Journal of chromatography. A, 1998, Dec-18, Volume: 828, Issue:1-2

    Topics: Animals; Chromatography, Liquid; Gallopamil; Swine; Verapamil

1998
Properties of the racemic species of verapamil hydrochloride and gallopamil hydrochloride.
    International journal of pharmaceutics, 1999, Feb-01, Volume: 178, Issue:1

    Topics: Calcium Channel Blockers; Chemistry Techniques, Analytical; Chromatography, High Pressure Liquid; Crystallization; Gallopamil; Spectrophotometry, Infrared; Spectroscopy, Fourier Transform Infrared; Stereoisomerism; Structure-Activity Relationship; Temperature; Verapamil; X-Ray Diffraction

1999
Mechanism of verapamil block of a neuronal delayed rectifier K channel: active form of the blocker and location of its binding domain.
    British journal of pharmacology, 1999, Volume: 126, Issue:8

    Topics: Animals; Binding Sites; Binding, Competitive; Biotransformation; Calcium Channel Blockers; Chick Embryo; Electrophysiology; Gallopamil; Ganglia, Spinal; Kinetics; Neurons; Potassium Channel Blockers; Potassium Channels; Tetraethylammonium; Verapamil

1999
Selective phenylalkylamine block of I(Kr) over other K(+) currents in guinea-pig ventricular myocytes.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Gallopamil; Guinea Pigs; Heart Ventricles; Male; Membrane Potentials; Phenethylamines; Potassium Channels; Time Factors; Ventricular Function; Verapamil

2000
Verapamil block of large-conductance Ca-activated K channels in rat aortic myocytes.
    The Journal of membrane biology, 2001, Jan-15, Volume: 179, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; Aorta; Binding Sites; Gallopamil; Kinetics; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Calcium-Activated; Rats; Rats, Wistar; Verapamil

2001
Multidimensional on-line sample preparation of verapamil and its metabolites by a molecularly imprinted polymer coupled to liquid chromatography-mass spectrometry.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2004, Mar-05, Volume: 801, Issue:2

    Topics: Animals; Cells, Cultured; Chromatography, High Pressure Liquid; Gallopamil; Male; Mass Spectrometry; Polymers; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Specimen Handling; Verapamil

2004
L-type Ca2+ channel antagonists block voltage-dependent Ca2+ channels in identified leech neurons.
    Brain research, 2004, Jul-09, Volume: 1013, Issue:2

    Topics: Animals; Caffeine; Calcium Channel Blockers; Calcium Channels, L-Type; Diltiazem; Gallopamil; Leeches; Membrane Potentials; Neurons; Nifedipine; Phosphodiesterase Inhibitors; Verapamil

2004
Opposite effects of a single IIIS5 mutation on phenylalkylamine and dihydropyridine interaction with L-type Ca2+ channels.
    The Journal of biological chemistry, 2004, Dec-31, Volume: 279, Issue:53

    Topics: Animals; Brain; Calcium; Calcium Channels; Calcium Channels, L-Type; Carrier Proteins; Cell Membrane; Dihydropyridines; DNA, Complementary; Dose-Response Relationship, Drug; Electrophysiology; Gallopamil; Homozygote; In Situ Hybridization; Isradipine; Kinetics; Mice; Mice, Transgenic; Microsomes; Models, Biological; Mutation; Oocytes; Protein Binding; Protein Structure, Tertiary; Recombinant Proteins; RNA, Complementary; Steroid Isomerases; Tyrosine; Verapamil; Xenopus laevis

2004
Pharmacophoric features and Ca2+ ion holding capacity of verapamil.
    Bioorganic & medicinal chemistry letters, 2005, Dec-15, Volume: 15, Issue:24

    Topics: Calcium; Calcium Channel Blockers; Gallopamil; Hydrogen Bonding; Models, Molecular; Molecular Conformation; Verapamil

2005
Effects of phenylalkylamines and benzothiazepines on Ca(v)1.3-mediated Ca2+ currents in neonatal mouse inner hair cells.
    European journal of pharmacology, 2007, Nov-14, Volume: 573, Issue:1-3

    Topics: Algorithms; Animals; Animals, Newborn; Benzazepines; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Diltiazem; Dose-Response Relationship, Drug; Gallopamil; Hair Cells, Auditory, Inner; Membrane Potentials; Mice; Mice, Inbred Strains; Phenethylamines; Verapamil

2007
Structural model for phenylalkylamine binding to L-type calcium channels.
    The Journal of biological chemistry, 2009, Oct-09, Volume: 284, Issue:41

    Topics: Amino Acid Sequence; Binding Sites; Calcium Channel Blockers; Calcium Channels, L-Type; Computer Simulation; Dihydropyridines; Gallopamil; Models, Molecular; Molecular Sequence Data; Molecular Structure; Monte Carlo Method; Protein Structure, Tertiary; Sequence Alignment; Structure-Activity Relationship; Verapamil

2009