verapamil has been researched along with flunarizine in 143 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 62 (43.36) | 18.7374 |
1990's | 62 (43.36) | 18.2507 |
2000's | 10 (6.99) | 29.6817 |
2010's | 9 (6.29) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Barrett, RJ; Johnson, CP; Proakis, AG; Shanklin, JR | 1 |
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Janis, RA; Triggle, DJ | 1 |
Anger, T; Madge, DJ; Mulla, M; Riddall, D | 1 |
Bruno-Blanch, L; Gálvez, J; García-Domenech, R | 1 |
Cai, W; Hao, Y; Hu, P; Ma, D; Pan, H; Xie, X; Yu, AD; Yu, J; Yuan, J; Zhang, L; Zhu, H | 1 |
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ | 1 |
Brouillette, WJ; Brown, GB; Zha, C | 1 |
Furune, Y; Kato, T; Otsu, Y; Yamamoto, T | 1 |
Bertolucci, PH; De Andrade, LA; Ferraz, HB; Pereira, JS | 1 |
Correale, J; Link, H; Mix, E; Olsson, T; Solders, G | 1 |
Dantchev, N; Popov, P; Staneva-Stoytcheva, D | 1 |
Kawamura, M; Murakami, M; Nakamichi, N; Takamura, M; Tou, S; Yamada, K | 1 |
Amano, T; Ishihara, K; Momiyama, T; Renming, X; Sasa, M; Serikawa, T; Todo, N; Yamada, J | 1 |
Akaike, N; Kameda, H; Kataoka, M; Takahashi, K; Ueno, S | 1 |
Montastruc, JL; Senard, JM | 1 |
Berga, P; Bou, J; Cardelús, I; Gristwood, RW; Llenas, J | 1 |
Berga, P; Furman, BL; Gristwood, RW; Jauregui, J; Llenas, J | 1 |
De Sarro, A; De Sarro, GB; Nistico', G; Trimarchi, GR | 1 |
D'Ancona, S; Mazzo, M; Pea, F | 1 |
Benedetti, M; Pezzola, A; Popoli, P; Scotti de Carolis, A | 1 |
Kamei, J; Kasuya, Y | 1 |
Lipton, SA | 1 |
Danchev, N; Popov, P; Staneva-Stoytcheva, D | 1 |
Beech, DJ; Bolton, TB; Christen, MO; MacKenzie, I | 1 |
Gorgels, AP; Havenith, MG; Kriek, E; Leunissen, JD; Smeets, JL; Vos, MA; Wellens, HJ | 1 |
Bleehen, NM; Honess, DJ | 1 |
Almeida, AR; Bunnachak, D; Burke, TJ; Burnier, M; Schrier, RW; Wetzels, JF | 1 |
Ivanova, E; Popova, J; Staneva-Stoytcheva, D; Tosheva, T | 1 |
Fabrègues, E; John, GW; Kamal, M; Massingham, R | 1 |
Pang, CC; Waite, RP; Walker, MJ | 2 |
Amagasa, M; Ogawa, A; Yoshimoto, T | 1 |
Achille, P; Frascella, G; Lastilla, M; Savarese, MA | 1 |
Campisi, D; Cascio Ingurgio, N; Marsala, BA; Martino, SG; Paterna, S | 1 |
Alov, P; Mutafova-Yambolieva, V; Popova, J; Staneva-Stoytcheva, D | 1 |
Locher, R; Sachinidis, A; Steiner, A; Vetter, W | 1 |
Akaike, N; Kanaide, H; Kuga, T; Nakamura, M; Sadoshima, J; Tomoike, H | 1 |
Handa, J; Kidooka, M; Shiino, A | 1 |
Hunter, JB; Pegram, BL; Peters, T; Scheufler, E; Vogelgesang, R; Wermelskirchen, D; Wilffert, B | 1 |
Mutafova, V; Popova, J; Staneva-Stoytcheva, D | 1 |
Peters, T; Scheufler, E | 1 |
Borgers, M; De Clerck, F; Vandewiele, R; Ver Donck, L; Verellen, G | 1 |
Gaggi, R; Gianni, AM | 1 |
Carpenter, CL; Greenberg, DA; Messing, RO | 2 |
Greenberg, DA | 1 |
Traber, J; Van Rooijen, LA | 1 |
Boddeke, HW; Heynis, JB; van Zwieten, PA; Wilffert, B | 1 |
Blanco, I; Brandner, R; Rodriguez, J; Rodriguez, R; Sabrià, J; Toledo, A | 1 |
Pan, M; Scriabine, A | 1 |
De Clerck, F; Janssen, PA; Loots, W; Voeten, J | 1 |
Duhm, J; Engelmann, B | 1 |
Hirst, DG; Wood, PJ | 2 |
Geerts, H; Nuydens, R; Nuyens, R; Ver Donck, L | 1 |
Carvalho, AP; Carvalho, CM; Leysen, JE; Lima, MP; Oliveira, CR | 1 |
Edvinsson, L; Ikomi-Kumm, J; Monti, M | 1 |
Gachev, E; Karadzhaeva, G | 1 |
Janssen, PA; Melis, W; Wauquier, A | 1 |
Christie-Pope, BC; Palmer, GC; Palmer, SJ | 1 |
Carmeliet, E; Tytgat, J; Vereecke, J | 1 |
Bingmann, D; Speckmann, EJ | 1 |
Cruz, LJ; Olivera, BM | 1 |
Dolin, SJ; Little, HJ | 1 |
Schwartzkroin, PA; Taube, JS | 1 |
Hamberger, A; Lazarewicz, JW; Lehmann, A | 1 |
Agnoli, A | 1 |
Marriott, JF | 1 |
Baker, RE; Bingmann, D; de Jong, BM; Ruijter, J; Speckmann, EJ | 1 |
Koch, P; Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wilhelm, D | 1 |
Cartheuser, CF | 1 |
Brockelman, CR; Bunnag, D; Satayavivad, J; Tan-ariya, P; Wongsawatkul, O | 1 |
Metzger, HP; Savas, Y | 1 |
Amoroso, S; Annunzia, L; Canzoniero, L; Di Renzo, G; Maida, P; Nappi, C; Taglialatela, M | 1 |
Fitzpatrick, JM; Leahy, AL; Wait, RB | 1 |
Harrison, GG; Morrell, DF; Wright, IG | 1 |
Monti, E; Paracchini, L; Piccinini, F; Rozza, A; Villani, F | 1 |
Christie-Pope, BC; Palmer, GC | 1 |
Favalli, L; Formelli, F; Lanza, E; Monti, E; Piccinini, F; Poggi, P; Rozza, A; Villani, F | 1 |
Baeyens, JM; Esposito, E; Ossowska, G; Samanin, R | 1 |
Auguet, M; Clostre, F; DeFeudis, FV; Delaflotte, S | 1 |
Clutterbuck, RD; McElwain, TJ; Millar, JL; Robinson, BA | 1 |
Dolin, SJ; Halsey, MJ; Little, HJ | 1 |
Albano, O; Altomare, E; Attolini, E; Campanozzi, F; Centonze, V; Macinagrossa, G; Magrone, D; Tesauro, P; Trizio, T | 1 |
Henry, PD | 1 |
Solomon, GD | 1 |
Chiang, BN; Fong, JC; Hong, CY; Ku, J; Wei, YH | 1 |
Borgers, M; Donck, LV; Pauwels, PJ; Vandeplassche, G | 1 |
Boccuni, M; Cangi, F; Fanciullacci, M; Fusco, BM; Gatto, G; Marabini, S; Pietrini, U | 1 |
DeLong, RE; Phillis, JW; Towner, JK | 1 |
Ginesi, LM; Noble, AR | 1 |
Bishop, CM; Capetola, RJ; Hedli, CC; Levinson, SL; Ritchie, DM; Sierchio, JN | 1 |
Beatty, DA; Colker, JE; Fairhurst, AS; Thayer, SA | 1 |
Fagbemi, O; Kane, KA; McDonald, FM; Parratt, JR; Rothaul, AL | 1 |
Clincke, GH; Wauquier, A | 1 |
Dubinsky, B; Ritchie, DM; Sierchio, JN; Temple, DE | 1 |
Miller, WC; Moore, JB | 1 |
Bolger, GT; Gengo, P; Janis, RA; Klockowski, R; Luchowski, E; Siegel, H; Triggle, AM; Triggle, DJ | 1 |
Karasawa, A; Kumada, Y; Nakamizo, N; Shuto, K; Yamada, K | 1 |
Kasuya, Y; Nakayama, K | 1 |
Van Nueten, JM; Vanhoutte, PM | 1 |
Flaim, SF; Zelis, R | 1 |
Abbe, R; Appel, SH; Bostwick, JR | 1 |
García, AG; Guantes, JM; Michelena, P; Montiel, C; Uceda, G | 1 |
Bloechle, C; Broelsch, CE; Haller, G; Konrad, T; Kusterer, K; Usadel, KH | 1 |
Köhling, R; Speckmann, EJ; Straub, H | 2 |
Carvalho, CM; Lopes, MC; Santos, DL | 1 |
Calder, L; Clikeman, J; Finnegan, KT; Karler, R; Wei, S | 1 |
Fink-Puches, R; Helige, C; Kerl, H; Smolle, J; Tritthart, HA | 1 |
Hill, BT; Hosking, LK | 1 |
Hair, WM; Hughes, AD; Martin, G; Sever, PS; Sunman, W | 1 |
Floersheim, GL | 1 |
Lo, TM; Thayer, SA | 1 |
Fink-Puches, R; Helige, C; Hofmann-Wellenhof, R; Kerl, H; Smolle, J; Tritthart, HA | 1 |
Baker, RE; Ballantyne, D; Bingmann, D; Jones, D; Widman, G | 1 |
Nilles, R | 1 |
Fukui, M; Ikezaki, K; Matsukado, K; Nomura, T | 1 |
Fauteck, JD; Köhling, R; Lüke, A; Moskopp, D; Oppel, F; Pannek, H; Speckmann, EJ; Straub, H; Tuxhorn, I; Wassmann, H; Wolf, P | 1 |
Hunter, AJ | 1 |
Carvajal, A; Dueñas, A; Fernández de la Gándara, F; Maroto, M; Nieto, A; Velasco, A | 1 |
De Marco, C; Gornati, D; Silvestrini, R; Villa, R; Zaffaroni, N | 1 |
Abiko, Y; Chen, M; Hashizume, H; Xiao, CY | 1 |
Haraguchi, K; Iga, T; Ito, K; Kotaki, H; Sawada, Y | 1 |
Getslev, V; Pankova, IA; Pick, CG; Schrieber, S; Weizman, R | 1 |
Arai, T; Araki, T; Arbab, AS; Koizumi, K; Toyama, K | 1 |
Amorim, SC; Costa, PG; Futuro-Neto, HA; Pires, JG; Ribeiro, CA; Saraiva, FP | 1 |
Bespalov, AY; Dravolina, OA; Medvedev, IO; Sukhotina, IA | 1 |
Mediratta, PK; Sharma, KK; Verma, V | 1 |
Araki, T; Arbab, AS; Koizumi, K; Ueki, J | 1 |
Loikkanen, J; Naarala, J; Savolainen, KM; Vähäkangas, KH | 1 |
Armelao, L; Cristoni, S; Gross, S; Seraglia, R; Tondello, E; Traldi, P | 1 |
Breier, A; Dovinová, I; Fiala, R; Gibalová, L; Orlický, J; Seres, M; Sulová, Z; Uhrík, B | 1 |
Phillips, MF; Quinlivan, R | 1 |
Antoons, G; Attevelt, NJ; Beekman, JD; Belardinelli, L; Gomez, AM; Houtman, MJ; Neco, P; Oosterhoff, P; Oros, A; Rajamani, S; Richard, S; van der Heyden, MA; Ver Donck, L; Vos, MA | 1 |
Gieseg, SP; Whiteman, M; Yang, YT | 1 |
Biala, G; Budzynska, B; Polak, P | 1 |
Alfaro-Iznaola, C; Ballesteros-Garcia, MM; Cuadrado-Martin, M; Natera-de Benito, D; Rodriguez-Diaz, R; Taboas-Pereira, MA | 1 |
Bossu, A; van Weperen, VYH; Vos, MA | 1 |
11 review(s) available for verapamil and flunarizine
Article | Year |
---|---|
New developments in Ca2+ channel antagonists.
Topics: Animals; Binding Sites; Calcium; Calcium Channel Blockers; Calmodulin; Electrophysiology; Heart; Humans; Ion Channels; Muscle Relaxation; Muscle, Smooth; Potassium; Sodium; Structure-Activity Relationship; Substrate Specificity | 1983 |
Medicinal chemistry of neuronal voltage-gated sodium channel blockers.
Topics: Amyotrophic Lateral Sclerosis; Analgesics; Anticonvulsants; Epilepsy; Humans; Ion Channel Gating; Models, Molecular; Mutation; Nerve Tissue Proteins; Neuroprotective Agents; Protein Binding; Sodium Channel Blockers; Sodium Channels; Stroke | 2001 |
[Calcium channel blockers and prevention of migraine].
Topics: Adrenergic beta-Antagonists; Clinical Trials as Topic; Diltiazem; Flunarizine; Humans; Migraine Disorders; Nifedipine; Nimodipine; Verapamil | 1992 |
[Ca antagonists in neurosurgical practice].
Topics: Animals; Anticonvulsants; Brain; Calcium Channel Blockers; Cerebral Infarction; Disease Models, Animal; Fatty Acids, Nonesterified; Flunarizine; Humans; Intracranial Aneurysm; Ischemic Attack, Transient; Nimodipine; Piperazines; Verapamil | 1990 |
Calcium channel antagonists and the treatment of migraine.
Topics: Calcium; Calcium Channel Blockers; Cinnarizine; Diltiazem; Flunarizine; Humans; Ion Channels; Kinetics; Migraine Disorders; Nicotinic Acids; Nifedipine; Nimodipine; Verapamil | 1986 |
Atherosclerosis, calcium, and calcium antagonists.
Topics: Animals; Aorta; Arteries; Arteriosclerosis; Calcinosis; Calcium; Calcium Channel Blockers; Cell Survival; Cholesterol, Dietary; Cinnarizine; Diltiazem; Flunarizine; Humans; Membrane Lipids; Muscle, Smooth, Vascular; Nicardipine; Nifedipine; Propranolol; Rabbits; Verapamil | 1985 |
Comparative efficacy of calcium antagonist drugs in the prophylaxis of migraine.
Topics: Calcium Channel Blockers; Cinnarizine; Clinical Trials as Topic; Diltiazem; Double-Blind Method; Flunarizine; Humans; Migraine Disorders; Nicotinic Acids; Nifedipine; Nimodipine; Verapamil | 1985 |
Calcium antagonists: their role in neuroprotection.
Topics: Animals; Brain Ischemia; Calcium Channel Blockers; Calcium Channels; Cerebrovascular Disorders; Dihydropyridines; Flunarizine; Humans; Neuroprotective Agents; Verapamil | 1997 |
Calcium antagonists for Duchenne muscular dystrophy.
Topics: Calcium Channel Blockers; Diltiazem; Flunarizine; Humans; Muscle Strength; Muscle, Skeletal; Muscular Dystrophy, Duchenne; Nifedipine; Randomized Controlled Trials as Topic; Verapamil | 2008 |
[Cluster headache in pediatric population: four case reports and review of the literature].
Topics: Adolescent; Child; Child, Preschool; Cluster Headache; Diagnosis, Differential; Female; Flunarizine; Humans; Male; Tryptamines; Verapamil | 2016 |
Point of View: Electrophysiological Endpoints Differ When Comparing the Mode of Action of Highly Successful Anti-arrhythmic Drugs in the CAVB Dog Model With TdP.
Topics: Action Potentials; Aniline Compounds; Animals; Anti-Arrhythmia Agents; Atrioventricular Block; Chronic Disease; Disease Models, Animal; Dogs; Electrophysiologic Techniques, Cardiac; Endpoint Determination; Flunarizine; Heart Rate; Phenyl Ethers; Pyridines; Time Factors; Torsades de Pointes; Triazoles; Verapamil | 2019 |
4 trial(s) available for verapamil and flunarizine
Article | Year |
---|---|
[Calcium channel blockers and prevention of migraine].
Topics: Adrenergic beta-Antagonists; Clinical Trials as Topic; Diltiazem; Flunarizine; Humans; Migraine Disorders; Nifedipine; Nimodipine; Verapamil | 1992 |
[Verapamil versus flunarizine in the preventive therapy of hemicrania].
Topics: Adolescent; Adult; Drug Evaluation; Female; Flunarizine; Humans; Male; Middle Aged; Migraine Disorders; Time Factors; Verapamil | 1990 |
[Evaluation of the effects of verapamil, flunarizine, diltiazem, nimodipine and placebo in the prevention of hemicrania. A double-blind randomized cross-over study].
Topics: Adolescent; Adult; Diltiazem; Double-Blind Method; Female; Flunarizine; Humans; Male; Middle Aged; Migraine Disorders; Nimodipine; Placebos; Verapamil | 1990 |
Comparative efficacy of calcium antagonist drugs in the prophylaxis of migraine.
Topics: Calcium Channel Blockers; Cinnarizine; Clinical Trials as Topic; Diltiazem; Double-Blind Method; Flunarizine; Humans; Migraine Disorders; Nicotinic Acids; Nifedipine; Nimodipine; Verapamil | 1985 |
130 other study(ies) available for verapamil and flunarizine
Article | Year |
---|---|
Synthesis, calcium-channel-blocking activity, and antihypertensive activity of 4-(diarylmethyl)-1-[3-(aryloxy)propyl]piperidines and structurally related compounds.
Topics: Animals; Antihypertensive Agents; Aorta; Calcium; Calcium Channel Blockers; Hypertension; Male; Molecular Structure; Muscle Contraction; Piperidines; Rabbits; Rats; Rats, Inbred SHR; Structure-Activity Relationship | 1991 |
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Topological virtual screening: a way to find new anticonvulsant drugs from chemical diversity.
Topics: Anticonvulsants; Computer Simulation; Databases, Factual; Discriminant Analysis; Drug Design; Molecular Structure; Quantitative Structure-Activity Relationship | 2003 |
Small molecule regulators of autophagy identified by an image-based high-throughput screen.
Topics: Autophagy; Calcium Channel Blockers; Cell Line, Tumor; Drug Evaluation, Preclinical; Fluspirilene; Glioblastoma; Green Fluorescent Proteins; Humans; Intracellular Membranes; Loperamide; Microtubule-Associated Proteins; Mycotoxins; Peptides; Phagosomes; Phosphatidylinositol Phosphates; Pimozide; Protein Kinases; Recombinant Fusion Proteins; Sirolimus; Small Molecule Libraries; TOR Serine-Threonine Kinases; Trifluoperazine; Zinc Fingers | 2007 |
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase | 2008 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity | 2013 |
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels | 2014 |
Different effects of L-, N- and T-type calcium channel blockers on striatal dopamine release measured by microdialysis in freely moving rats.
Topics: Animals; Calcium Channel Blockers; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Flunarizine; Male; Mollusk Venoms; Motor Activity; Nicardipine; omega-Conotoxins; Peptides, Cyclic; Rats; Rats, Wistar; Verapamil | 1992 |
A study on the action of two calcium channel blockers (verapamil and flunarizine) upon an experimental model of tardive dyskinesia in rats.
Topics: Animals; Apomorphine; Drug Evaluation, Preclinical; Dyskinesia, Drug-Induced; Flunarizine; Haloperidol; Male; Rats; Rats, Wistar; Stereotyped Behavior; Verapamil | 1992 |
Calcium antagonists suppress experimental allergic neuritis (EAN).
Topics: Action Potentials; Animals; Dose-Response Relationship, Drug; Flunarizine; Lymphocyte Activation; Neuritis, Autoimmune, Experimental; Peripheral Nervous System Diseases; Rats; Rats, Inbred Lew; Sciatic Nerve; T-Lymphocytes; Verapamil | 1992 |
Long-term treatment with different calcium- and calmodulin-antagonists induces changes in rat brain alpha-adrenoceptors.
Topics: Administration, Oral; Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Dioxanes; Flunarizine; Male; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Regression Analysis; Trifluoperazine; Verapamil | 1992 |
[Effect of Ca(2+)-channel antagonists on the corticoidogenesis in primary cultured bovine adrenocortical cells].
Topics: Adrenal Cortex; Adrenal Cortex Hormones; Adrenocorticotropic Hormone; Animals; Calcium Channel Blockers; Cattle; Cells, Cultured; Flunarizine; Nicardipine; Verapamil | 1992 |
Abnormal calcium current in hippocampal CA3 pyramidal cells of the spontaneously epileptic rat (SER).
Topics: Action Potentials; Animals; Calcium Channels; Electric Stimulation; Epilepsy; Flunarizine; Hippocampus; Rats; Rats, Mutant Strains; Verapamil | 1992 |
Effects of Ca2+ antagonists and antiepileptics on tetrodotoxin-sensitive Ca(2+)-conducting channels in isolated rat hippocampal CA1 neurons.
Topics: Animals; Anticonvulsants; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Diltiazem; Dizocilpine Maleate; Dose-Response Relationship, Drug; Flunarizine; Hippocampus; Kinetics; Neurons; Nicardipine; Phenobarbital; Phenytoin; Pyramidal Tracts; Rats; Rats, Wistar; Sodium; Tetrodotoxin; Valproic Acid; Verapamil | 1992 |
Cardiovascular effects of LAS 30538, a new vascular selective Ca(2+)-channel blocker.
Topics: Animals; Blood Pressure; Calcium Channel Blockers; Diltiazem; Electrophysiology; Flunarizine; Guinea Pigs; Heart; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Papillary Muscles; Perfusion; Piperidines; Rabbits; Rats; Rats, Inbred SHR; Rats, Wistar; Vasoconstrictor Agents; Vasodilator Agents; Verapamil | 1992 |
The calcium channel blocker LAS 30538, unlike nifedipine, verapamil, diltiazem or flunarizine, potently inhibits insulin secretion in-vivo in rats and dogs.
Topics: Administration, Oral; Animals; Blood Glucose; Calcium Channel Blockers; Diltiazem; Dogs; Female; Flunarizine; Glucose Tolerance Test; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Piperidines; Rats; Rats, Sprague-Dawley; Verapamil | 1992 |
Effects of some calcium antagonists upon the activity of common antiepileptic compounds on sound-induced seizures in DBA/2 mice.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anticonvulsants; Body Temperature; Calcium Channel Blockers; Diltiazem; Drug Synergism; Flunarizine; Mice; Mice, Inbred DBA; Nimodipine; Phenobarbital; Phenytoin; Seizures; Valproic Acid; Verapamil | 1992 |
Increased spontaneous cell detachment of F10 cells induced in vitro by some calcium-channel blockers.
Topics: Animals; Calcium Channel Blockers; Cell Adhesion; Culture Media; Flunarizine; Growth Inhibitors; Melanoma, Experimental; Nifedipine; Tumor Cells, Cultured; Tumor Stem Cell Assay; Verapamil | 1992 |
Verapamil and flunarizine inhibit phencyclidine-induced effects: an EEG and behavioural study in rats.
Topics: Animals; Behavior, Animal; Electroencephalography; Flunarizine; Injections, Intraventricular; Male; Nimodipine; Phencyclidine; Rats; Rats, Wistar; Verapamil | 1992 |
Antitussive effects of Ca2+ channel antagonists.
Topics: Animals; Antitussive Agents; Calcium Channel Blockers; Capsaicin; Codeine; Cough; Dextromethorphan; Drug Interactions; Drug Synergism; Flunarizine; Guinea Pigs; Male; Morphine; Nifedipine; Verapamil | 1992 |
Calcium channel antagonists and human immunodeficiency virus coat protein-mediated neuronal injury.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Survival; Cells, Cultured; Dihydropyridines; Diltiazem; Flunarizine; HIV Envelope Protein gp120; HIV-1; Peptide Fragments; Rats; Recombinant Fusion Proteins; Retinal Ganglion Cells; Verapamil | 1991 |
Changes in benzodiazepine receptors of rat brain after long-term treatment with the Ca(2+)-antagonists nifedipine, verapamil, flunarizine and with the calmodulin antagonist trifluoperazine.
Topics: Animals; Brain Chemistry; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Flunarizine; Flunitrazepam; Hippocampus; Kinetics; Male; Nifedipine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Trifluoperazine; Verapamil | 1991 |
Effects of pinaverium on voltage-activated calcium channel currents of single smooth muscle cells isolated from the longitudinal muscle of the rabbit jejunum.
Topics: Animals; Barium; Calcium Channels; Diltiazem; Flunarizine; Gallopamil; In Vitro Techniques; Ion Channels; Jejunum; Membrane Potentials; Morpholines; Muscle, Smooth; Parasympatholytics; Rabbits; Verapamil | 1990 |
Programmed electrical stimulation and drugs identify two subgroups of ventricular tachycardias occurring 16-24 hours after occlusion of the left anterior descending artery.
Topics: Animals; Arterial Occlusive Diseases; Cardiac Pacing, Artificial; Coronary Disease; Dogs; Electrocardiography; Electrophysiology; Female; Flunarizine; Lidocaine; Male; Tachycardia; Time Factors; Verapamil | 1992 |
Effects of calcium channel blockers on renal function in mice.
Topics: Animals; Calcium Channel Blockers; Chromium Radioisotopes; Cinnarizine; Edetic Acid; Female; Flunarizine; Glomerular Filtration Rate; Kidney; Mice; Mice, Inbred C3H; Nifedipine; Verapamil | 1992 |
Time-dependent protective effects of calcium channel blockers on anoxia- and hypoxia-induced proximal tubule injury.
Topics: Animals; Calcium; Cations, Divalent; Flunarizine; In Vitro Techniques; Kidney Tubules, Proximal; L-Lactate Dehydrogenase; Male; Oxygen; Rats; Rats, Inbred Strains; Verapamil | 1992 |
The long-term treatment with the Ca(2+)-antagonists nifedipine, verapamil, flunarizine and with the calmodulin antagonist trifluoperazine decreases the activity of 5-HT1 receptors in rat cerebral cortex and hippocampus.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Flunarizine; Hippocampus; In Vitro Techniques; Kinetics; Male; Nifedipine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Trifluoperazine; Verapamil | 1991 |
Caffeine-induced contractions in rabbit isolated renal artery are differentially inhibited by calcium antagonists.
Topics: Animals; Bepridil; Caffeine; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Fendiline; Flunarizine; Kinetics; Lidoflazine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Renal Artery; Verapamil | 1991 |
Effects of verapamil, nifedipine and flunarizine on haemodynamics and regional blood flows in pentobarbitone-anaesthetized rats.
Topics: Anesthesia; Animals; Calcium Channel Blockers; Cardiac Output; Electrocardiography; Flunarizine; Heart Rate; Hemodynamics; Male; Nifedipine; Pentobarbital; Rats; Rats, Inbred Strains; Regional Blood Flow; Renal Circulation; Verapamil | 1990 |
Effects of calcium and calcium antagonists against deprivation of glucose and oxygen in guinea pig hippocampal slices.
Topics: Action Potentials; Animals; Brain Ischemia; Calcium; Calcium Channel Blockers; Disease Models, Animal; Flunarizine; Glucose; Guinea Pigs; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Male; Nicardipine; Verapamil | 1990 |
Influence of long-term treatment with the Ca2(+)-antagonists nifedipine, verapamil, flunarizine and with the calmodulin antagonist trifluoperazine on beta-adrenoceptors in rat cerebral cortex.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Dihydroalprenolol; Flunarizine; Male; Membrane Fluidity; Membranes; Nifedipine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Synaptosomes; Trifluoperazine; Verapamil | 1990 |
Attenuation of the low-density-lipoprotein-activated phosphoinositide signalling system by calcium blockers in human lymphocytes.
Topics: Calcium Channel Blockers; Cells, Cultured; Cholesterol, LDL; Diglycerides; Diltiazem; Dose-Response Relationship, Drug; Flunarizine; Humans; Lymphocytes; Molsidomine; Nifedipine; Phosphatidylinositols; Protein Kinase C; Verapamil | 1990 |
Actions of Ca2+ antagonists on two types of Ca2+ channels in rat aorta smooth muscle cells in primary culture.
Topics: Animals; Aorta; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Diltiazem; Electric Conductivity; Flunarizine; Kinetics; Male; Membrane Potentials; Muscle, Smooth, Vascular; Nicardipine; Rats; Time Factors; Verapamil | 1990 |
Uptake of catamphiphilic drugs into erythrocytes and muscular tissue correlates to membrane enrichment and to 45Ca displacement from phosphatidylserine monolayers.
Topics: Binding Sites; Calcium; Cell Membrane; Diltiazem; Erythrocytes; Flunarizine; Humans; In Vitro Techniques; Lidocaine; Muscles; Nitrendipine; Phosphatidylserines; Verapamil | 1990 |
Effects of the Ca2(+)-antagonists nifedipine, verapamil, flunarizine and of the calmodulin antagonist trifluoperazine on muscarinic cholinergic receptors in rat cerebral cortex.
Topics: Animals; Calcium Channel Blockers; Calmodulin; Cerebral Cortex; Flunarizine; Kinetics; Male; Nifedipine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Trifluoperazine; Verapamil | 1990 |
Phosphatidylserine monolayers as models for drug uptake into membranes and tissue.
Topics: Animals; Aorta; Benzothiazoles; Cell Membrane; Diltiazem; Erythrocyte Membrane; Flunarizine; Heart Atria; Humans; Lidocaine; Membranes, Artificial; Models, Biological; Nitrendipine; Pharmaceutical Preparations; Pharmacokinetics; Phosphatidylserines; Piperidines; Rats; Thiazoles; Verapamil | 1990 |
Class IV Ca2+ antagonists do not affect lipid peroxidation in singlet oxygen challenged cardiomyocytes.
Topics: Animals; Benzothiazoles; Calcium Channel Blockers; Cell Separation; Cinnarizine; Diltiazem; Flunarizine; Lidoflazine; Lipid Peroxidation; Malondialdehyde; Myocardium; Nicardipine; Oxygen; Piperidines; Rats; Thiazoles; Verapamil | 1990 |
Effects of calcium antagonists on biogenic amines in discrete brain areas.
Topics: Animals; Biogenic Monoamines; Brain Chemistry; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Diltiazem; Electrochemistry; Flunarizine; Male; Nifedipine; Rats; Rats, Inbred Strains; Verapamil | 1990 |
Mechanism of calcium channel inhibition by phenytoin: comparison with classical calcium channel antagonists.
Topics: Adrenal Gland Neoplasms; Animals; Binding Sites; Calcium; Calcium Channel Blockers; Carbachol; Cell Line; Cinnarizine; Diltiazem; Flunarizine; Ion Channels; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Phenytoin; Pheochromocytoma; Potassium; Rats; Sodium; Verapamil | 1985 |
Muscarinic cholinergic enhancement of inositide turnover in cerebral nerve endings is not mediated by calcium uptake.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Calcimycin; Calcium; Carbachol; Cinnarizine; Flunarizine; Male; Nerve Endings; Nicotinic Acids; Nifedipine; Nimodipine; Phosphatidic Acids; Phosphatidylinositols; Rats; Rats, Inbred Strains; Verapamil; Veratridine | 1986 |
Ethanol-induced component of 45Ca2+ uptake in PC12 cells is sensitive to Ca2+ channel modulating drugs.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Cell Line; Diltiazem; Drug Interactions; Ethanol; Flunarizine; Ion Channels; Nifedipine; Verapamil | 1987 |
Investigation of the mechanism of negative inotropic activity of some calcium antagonists.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Arrhythmia Agents; Bepridil; Calcimycin; Calcium Channel Blockers; Depression, Chemical; Diltiazem; Female; Flunarizine; Guinea Pigs; In Vitro Techniques; Lidoflazine; Male; Myocardial Contraction; Pyrrolidines; Verapamil | 1988 |
Histamine stimulated synaptosomal Ca2+ uptake through activation of calcium channels.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Calcium; Cinnarizine; Cyclic AMP; Diltiazem; Flunarizine; Histamine; Ion Channels; Nifedipine; Rats; Synaptosomes; Verapamil | 1988 |
Effects of calcium antagonists on mean circulatory filling pressure in the conscious rat.
Topics: Animals; Blood Pressure; Calcium Channel Blockers; Dose-Response Relationship, Drug; Flunarizine; Heart Rate; Hexamethonium Compounds; Male; Muscle Tonus; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Verapamil | 1988 |
Ca2+ antagonists and inhibitory effects of dopamine on isolated rabbit ear artery.
Topics: Animals; Arteries; Blood Pressure; Calcium Channel Blockers; Dihydropyridines; Dopamine; Electric Stimulation; Ethanol; Female; Flunarizine; In Vitro Techniques; Muscle, Smooth, Vascular; Perfusion; Rabbits; Time Factors; Vasoconstriction; Verapamil | 1988 |
Differential effects of verapamil and flunarizine on epinephrine-induced vasoconstriction and on spontaneous vasomotion of arterioles in skeletal muscle in the rat in vivo.
Topics: Animals; Arterioles; Blood Pressure; Calcium; Epinephrine; Flunarizine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Muscles; Rats; Rats, Inbred Strains; Regional Blood Flow; Time Factors; Vasoconstriction; Verapamil | 1989 |
Distinction of two components of passive Ca2+ transport into human erythrocytes by Ca2+ entry blockers.
Topics: Aminoquinolines; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane Permeability; Cobalt; Copper; Diltiazem; Erythrocyte Membrane; Flunarizine; Humans; Nifedipine; Vanadates; Verapamil | 1989 |
Modification of tumour response by calcium antagonists in the SCVII/St tumour implanted at two different sites.
Topics: Animals; Back; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Flunarizine; Hindlimb; Mice; Neoplasm Transplantation; Neoplasms, Experimental; Nifedipine; Radiation Tolerance; Rubidium; Verapamil | 1989 |
The effect of flunarizine on intracellular calcium in isolated rat cardiomyocytes. A digital image processing study.
Topics: Animals; Benzofurans; Calcium; Depression, Chemical; Flunarizine; Fluorescent Dyes; Fura-2; Heart; Image Processing, Computer-Assisted; Isoproterenol; Kinetics; Myocardium; Rats; Verapamil; Veratrine | 1989 |
Calcium antagonists as radiation modifiers: site specificity in relation to tumor response.
Topics: Animals; Calcium Channel Blockers; Combined Modality Therapy; Female; Flunarizine; Mice; Mice, Inbred C3H; Neoplasm Transplantation; Neoplasms, Experimental; Nifedipine; Radiation-Sensitizing Agents; Verapamil | 1989 |
Partition of Ca2+ antagonists in brain plasma membranes.
Topics: Animals; Brain; Calcium Channel Blockers; Flunarizine; Kinetics; Liposomes; Nitrendipine; Sheep; Synaptic Membranes; Verapamil | 1989 |
Effects of calcium entry blockers on human platelet metabolism measured by microcalorimetry.
Topics: Blood Platelets; Calcium Channel Blockers; Calorimetry; Cerebral Arteries; Diltiazem; Flunarizine; Humans; Muscle Relaxation; Nifedipine; Verapamil | 1989 |
[The effect of calcium antagonists nimodipin, verapamil, diltiazem and flunarizin on local cerebral blood flow in rabbits in chronic experiments].
Topics: Animals; Cerebral Cortex; Diltiazem; Female; Flunarizine; Male; Nimodipine; Rabbits; Regional Blood Flow; Verapamil | 1989 |
Long-term neurological assessment of the post-resuscitative effects of flunarizine, verapamil and nimodipine in a new model of global complete ischaemia.
Topics: Anesthesia; Animals; Behavior, Animal; Disease Models, Animal; Electroencephalography; Electromyography; Flunarizine; Injections, Intravenous; Ischemia; Male; Nimodipine; Rats; Reflex; Resuscitation; Verapamil | 1989 |
Protective action of calcium channel blockers on Na+,K+-ATPase in gerbil cerebral cortex following ischemia.
Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; Female; Flunarizine; Gerbillinae; In Vitro Techniques; Ischemic Attack, Transient; Sodium-Potassium-Exchanging ATPase; Verapamil | 1988 |
Differential effects of verapamil and flunarizine on cardiac L-type and T-type Ca channels.
Topics: Animals; Calcium Channels; Flunarizine; Guinea Pigs; Heart; In Vitro Techniques; Myocardium; Potassium Channels; Verapamil | 1988 |
Specific suppression of pentylenetetrazol-induced epileptiform discharges in CA3 neurons (hippocampal slice, guinea pig) by the organic calcium antagonists flunarizine and verapamil.
Topics: Animals; Flunarizine; Guinea Pigs; Hippocampus; In Vitro Techniques; Pentylenetetrazole; Seizures; Verapamil | 1989 |
Calcium channel antagonists. Omega-conotoxin defines a new high affinity site.
Topics: Animals; Binding, Competitive; Brain; Calcium Channel Blockers; Chick Embryo; Cinnarizine; Diltiazem; Flunarizine; Muscles; Nifedipine; Nitrendipine; Prenylamine; Rana pipiens; Synaptosomes; Time Factors; Verapamil | 1986 |
Augmentation by calcium channel antagonists of general anaesthetic potency in mice.
Topics: Anesthesia, General; Animals; Argon; Calcium Channel Blockers; Cinnarizine; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Flunarizine; Male; Mice; Nifedipine; Nitrendipine; Pentobarbital; Time Factors; Verapamil | 1986 |
Ineffectiveness of organic calcium channel blockers in antagonizing long-term potentiation.
Topics: Action Potentials; Animals; Calcium Channel Blockers; Cinnarizine; Diazepam; Flunarizine; Guinea Pigs; Hippocampus; Neurons; Nifedipine; Nitrendipine; Reaction Time; Synaptic Transmission; Verapamil | 1986 |
Effects of Ca2+ entry blockers on kainate-induced changes in extracellular amino acids and Ca2+ in vivo.
Topics: Amino Acids; Animals; Calcium; Calcium Channel Blockers; Cobalt; Flunarizine; Hippocampus; Kainic Acid; Nimodipine; Rabbits; Verapamil | 1987 |
The classification of calcium antagonists by the WHO expert committee: relevance in neurology.
Topics: Brain Diseases; Calcium Channel Blockers; Diltiazem; Flunarizine; Humans; Nifedipine; Verapamil | 1988 |
A comparison of the effects of the calcium entry blockers, verapamil, diltiazem and flunarizine against contractions of the rat isolated aorta and portal vein.
Topics: Animals; Aorta, Thoracic; Calcium Channel Blockers; Diltiazem; Flunarizine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Portal Vein; Rats; Rats, Inbred Strains; Verapamil | 1988 |
Differential antiepileptic effects of the organic calcium antagonists verapamil and flunarizine in neurons of organotypic neocortical explants from newborn rats.
Topics: Animals; Animals, Newborn; Cerebral Cortex; Flunarizine; Membrane Potentials; Neurons; Organ Culture Techniques; Pentylenetetrazole; Rats; Seizures; Verapamil | 1988 |
Different effects of R 56865 and calcium entry blockers on K+- and noradrenaline-induced contractions and 45Ca uptake in rat aorta.
Topics: Animals; Aorta; Benzothiazoles; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Flunarizine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Piperidines; Potassium; Rats; Rats, Inbred Strains; Thiazoles; Verapamil | 1988 |
Slow channel inhibitor effects on brain function: tolerance to severe hypoxia in the rat.
Topics: Animals; Bencyclane; Bepridil; Brain; Calcium Channel Blockers; Cinnarizine; Diltiazem; Electroencephalography; Fendiline; Flunarizine; Gallopamil; Heart Rate; Hypoxia; Nimodipine; Prenylamine; Pyrrolidines; Rats; Rats, Inbred Strains; Respiration; Verapamil | 1988 |
Flunarizine and verapamil inhibit chloroquine-resistant Plasmodium falciparum growth in vitro.
Topics: Animals; Antimalarials; Chloroquine; Chlorpromazine; Drug Resistance; Flunarizine; Mefloquine; Plasmodium falciparum; Quinine; Quinolines; Regression Analysis; Verapamil | 1987 |
The influence of the calcium antagonists flunarizine and verapamil on cerebral blood flow and oxygen tension of anesthetized WFS-rats.
Topics: Animals; Brain; Cerebrovascular Circulation; Flunarizine; Kinetics; Oxygen; Oxygen Consumption; Partial Pressure; Rats; Rats, Inbred Strains; Verapamil | 1988 |
Effect of different Ca2+ entry blockers on dopamine-induced inhibition of in vitro prolactin secretion.
Topics: Animals; Calcium Channel Blockers; Diltiazem; Dopamine Antagonists; Flunarizine; In Vitro Techniques; Nimodipine; Prolactin; Rats; Rats, Inbred Strains; Receptors, Dopamine; Verapamil | 1988 |
Variable results of calcium blockade in post-ischaemic renal failure.
Topics: Acute Kidney Injury; Animals; Calcium Channel Blockers; Flunarizine; Ischemia; Kidney; Male; Nifedipine; Rats; Rats, Inbred Strains; Verapamil | 1988 |
The effects of calcium channel blocking drugs on halothane initiation of malignant hyperthermia in MHS swine and on the established syndrome.
Topics: Anesthesia, General; Animals; Calcium Channel Blockers; Diltiazem; Flunarizine; Halothane; Malignant Hyperthermia; Nifedipine; Nisoldipine; Swine; Verapamil | 1988 |
Effect of calcium inhibitors and calcium mobilizers on doxorubicin accumulation in rat myocardial tissue.
Topics: Animals; Calcium; Calcium Channel Blockers; Doxorubicin; Flunarizine; Heart; In Vitro Techniques; Male; Myocardium; Rats; Taurine; Trifluoperazine; Verapamil | 1988 |
Modulation of ischemic-induced damage to cerebral adenylate cyclase in gerbils by calcium channel blockers.
Topics: Adenylyl Cyclases; Animals; Calcium Channel Blockers; Disease Models, Animal; Female; Flunarizine; Gerbillinae; Ischemic Attack, Transient; Manganese; Verapamil | 1986 |
Influence of calcium antagonists on the antitumor activity and the cardiac toxicity of doxorubicin in the rat.
Topics: Animals; Carcinoma 256, Walker; Doxorubicin; Female; Flunarizine; Heart; Myocardium; Rats; Rats, Inbred Strains; Trifluoperazine; Verapamil | 1987 |
Effects of peripheral and central administration of calcium channel blockers in the naloxone-precipitated abstinence syndrome in morphine-dependent rats.
Topics: Animals; Body Weight; Brain; Calcium Channel Blockers; Clonidine; Diarrhea; Flunarizine; Injections, Intraventricular; Male; Morphine Dependence; Naloxone; Rats; Substance Withdrawal Syndrome; Verapamil | 1987 |
Verapamil as an apparent competitive antagonist of the serotonin receptor of rabbit isolated aorta.
Topics: Animals; Aorta, Thoracic; Binding, Competitive; Cinnarizine; Diltiazem; Flunarizine; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Receptors, Serotonin; Verapamil | 1986 |
Effects of verapamil and alcohol on blood flow, melphalan uptake and cytotoxicity, in murine fibrosarcomas and human melanoma xenografts.
Topics: Animals; Cinnarizine; Drug Synergism; Ethanol; Female; Fibrosarcoma; Flunarizine; Humans; Male; Melanoma; Melphalan; Mice; Mice, Inbred CBA; Regional Blood Flow; Verapamil | 1986 |
Calcium channel antagonists decrease the ethanol withdrawal syndrome.
Topics: Animals; Calcium Channel Blockers; Diazepam; Ethanol; Flunarizine; Male; Motor Activity; Nimodipine; Nitrendipine; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Substance Withdrawal Syndrome; Verapamil | 1986 |
[Preventive therapy of migraine: flunarizine versus verapamil].
Topics: Adult; Cinnarizine; Female; Flunarizine; Humans; Male; Middle Aged; Migraine Disorders; Random Allocation; Vasodilator Agents; Verapamil | 1985 |
Calcium antagonists stimulate sperm motility in ejaculated human semen.
Topics: Calcimycin; Calcium; Calcium Channel Blockers; Cinnarizine; Diltiazem; Dose-Response Relationship, Drug; Egtazic Acid; Flunarizine; Humans; Male; Prenylamine; Sperm Motility; Verapamil | 1985 |
Isolated rat cardiac myocytes as an experimental model to study calcium overload: the effect of calcium-entry blockers.
Topics: Animals; Calcium; Calcium Channel Blockers; Cinnarizine; Diltiazem; Flunarizine; Heart; Lidoflazine; Male; Myocardial Contraction; Myocardium; Nicardipine; Nifedipine; Rats; Rats, Inbred Strains; Time Factors; Verapamil; Veratrine | 1986 |
Pupillary and vascular effects of calcium antagonists in migraine.
Topics: Blood Pressure; Calcium Channel Blockers; Cinnarizine; Flunarizine; Humans; Migraine Disorders; Nifedipine; Pupil; Vasoconstriction; Verapamil | 1985 |
The effects of lidoflazine and flunarizine on cerebral reactive hyperemia.
Topics: Animals; Blood Gas Analysis; Cerebrovascular Circulation; Cinnarizine; Extracorporeal Circulation; Flunarizine; Hyperemia; Hypoxia; Lidoflazine; Male; Piperazines; Rats; Rats, Inbred Strains; Verapamil | 1985 |
Secretion of active and inactive renin by rabbit kidney cortex slices: effects of verapamil, flunarizine and A23187.
Topics: Animals; Calcimycin; Calcium; Cinnarizine; Flunarizine; In Vitro Techniques; Ion Channels; Juxtaglomerular Apparatus; Kidney Cortex; Piperazines; Rabbits; Renin; Verapamil | 1984 |
Evaluation of calcium entry blockers in several models of immediate hypersensitivity.
Topics: Animals; Arachidonate Lipoxygenases; Arachidonic Acids; Bronchial Spasm; Calcium Channel Blockers; Cinnarizine; Diltiazem; Flunarizine; Guinea Pigs; Histamine Release; Hydroxyeicosatetraenoic Acids; Hypersensitivity, Immediate; Lipoxygenase; Male; Mast Cells; Nifedipine; Rats; Verapamil | 1984 |
A calcium antagonist drug binding site in skeletal muscle sarcoplasmic reticulum: evidence for a calcium channel.
Topics: Animals; Binding Sites; Calcium; Calcium Channel Blockers; Cinnarizine; Egtazic Acid; Flunarizine; Gallic Acid; Ion Channels; Muscle Contraction; Neuromuscular Junction; Nifedipine; Nitrendipine; Pyridines; Rabbits; Sarcoplasmic Reticulum; Verapamil | 1983 |
The effects of verapamil, prenylamine, flunarizine and cinnarizine on coronary artery occlusion-induced arrhythmias in anaesthetized rats.
Topics: Anesthesia; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Blood Pressure; Calcium Channel Blockers; Cinnarizine; Coronary Disease; Flunarizine; Heart Rate; Male; Prenylamine; Rats; Rats, Inbred Strains; Verapamil | 1984 |
Pharmacological protection against hypoxia-induced effects on medium-term memory in a two-way avoidance paradigm.
Topics: Animals; Avoidance Learning; Calcium Channel Blockers; Cerebral Cortex; Cinnarizine; Dose-Response Relationship, Drug; Flunarizine; Guinea Pigs; Hypoxia, Brain; Male; Memory; Mental Recall; Nicotinic Acids; Nifedipine; Nimodipine; Retention, Psychology; Vasodilation; Verapamil | 1984 |
Flunarizine and verapamil: effects on central nervous system and peripheral consequences of cytotoxic hypoxia in rats.
Topics: Animals; Calcium Channel Blockers; Cinnarizine; Flunarizine; Hyperventilation; Hypoxia; Male; Piperazines; Potassium Cyanide; Rats; Rats, Inbred Strains; Verapamil | 1984 |
High affinity binding sites for [3H]-nitrendipine in rabbit uterine smooth muscle.
Topics: Animals; Binding Sites; Calcium Channel Blockers; Cell Membrane; Cinnarizine; Depression, Chemical; Dose-Response Relationship, Drug; Female; Flunarizine; Muscle, Smooth; Nifedipine; Nitrendipine; Rabbits; Uterus; Verapamil | 1984 |
Characterization of binding of the Ca++ channel antagonist, [3H]nitrendipine, to guinea-pig ileal smooth muscle.
Topics: Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Cinnarizine; Cobalt; Dose-Response Relationship, Drug; Drug Synergism; Flunarizine; Guinea Pigs; Ileum; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Pyridines; Structure-Activity Relationship; Verapamil | 1983 |
Protective effect of flunarizine against cerebral hypoxia-anoxia in mice and rats.
Topics: Animals; Cinnarizine; Flunarizine; Hypoxia, Brain; Male; Mice; Mice, Inbred Strains; Pentobarbital; Piperazines; Rats; Rats, Inbred Strains; Vasodilator Agents; Verapamil | 1982 |
Selective abolition of Ca-dependent responses of smooth and cardiac muscles by flunarizine.
Topics: Animals; Basilar Artery; Calcium; Cinnarizine; Female; Flunarizine; In Vitro Techniques; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Myocardial Contraction; Piperazines; Portal Vein; Potassium; Rabbits; Rats; Uterine Contraction; Vasoconstriction; Verapamil | 1980 |
Calcium entry blockers and vascular smooth muscle heterogeneity.
Topics: Animals; Calcium; Calcium Channel Blockers; Cinnarizine; Flunarizine; Gallopamil; Lidoflazine; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Verapamil | 1981 |
Clinical use of calcium entry blockers.
Topics: Angina Pectoris; Calcium Channel Blockers; Cinnarizine; Coronary Circulation; Coronary Vasospasm; Diltiazem; Flunarizine; Heart Rate; Humans; Lidoflazine; Nifedipine; Perhexiline; Verapamil | 1981 |
Modulation of acetylcholine release in rat hippocampus by amino alcohols and Bay K 8644.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Acetylcholine; Animals; Calcium; Cerebral Cortex; Choline; Corpus Striatum; Diltiazem; Dose-Response Relationship, Drug; Ethanolamine; Ethanolamines; Flunarizine; Hippocampus; In Vitro Techniques; Male; Nifedipine; Osmolar Concentration; Potassium Chloride; Propanolamines; Pyrrolidines; Rats; Rats, Inbred F344; Verapamil | 1993 |
Effects of Ca2+ channel antagonist subtypes on mitochondrial Ca2+ transport.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenal Medulla; Animals; Biological Transport; Calcium; Calcium Channel Blockers; Cattle; Diltiazem; Flunarizine; In Vitro Techniques; Mitochondria; Nitrendipine; Verapamil | 1995 |
Verapamil and flunarizine protect the isolated perfused rat liver against warm ischemia and reperfusion injury.
Topics: Animals; Calcium; Female; Flunarizine; Glutamate Dehydrogenase; Homeostasis; Hot Temperature; Hydrogen-Ion Concentration; Ischemia; L-Lactate Dehydrogenase; Liver; Organ Size; Perfusion; Potassium; Rats; Rats, Wistar; Reperfusion Injury; Verapamil | 1995 |
Picrotoxin-induced epileptic activity in hippocampal and neocortical slices (guinea pig): suppression by organic calcium channel blockers.
Topics: Animals; Cerebral Cortex; Depression, Chemical; Epilepsy; Female; Flunarizine; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Picrotoxin; Receptors, GABA-A; Verapamil | 1994 |
Calcium channel blockers inhibit the (Ca2+ + Mg2+)-ATPase activity and the 125I-calmodulin binding in brain membranes.
Topics: Animals; Autoradiography; Binding Sites; Brain; Ca(2+) Mg(2+)-ATPase; Calcium Channel Blockers; Calmodulin; Cell Membrane; Electrophoresis, Polyacrylamide Gel; Flunarizine; Iodine Radioisotopes; Nitrendipine; Sheep; Stereoisomerism; Synaptic Membranes; Trifluoperazine; Verapamil | 1994 |
Effects of L-type calcium channel antagonists on the serotonin-depleting actions of MDMA in rats.
Topics: 3,4-Methylenedioxyamphetamine; Animals; Brain Chemistry; Calcium Channel Blockers; Cerebral Cortex; Flunarizine; Haloperidol; Hippocampus; Male; Methamphetamine; N-Methyl-3,4-methylenedioxyamphetamine; Nifedipine; Rats; Rats, Sprague-Dawley; Seizures; Serotonin; Stereotyped Behavior; Verapamil | 1993 |
Inhibition of melanoma cell directional migration in vitro via different cellular targets.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Aminoimidazole Carboxamide; Animals; Calcium Channel Blockers; Cell Division; Cell Movement; Dequalinium; Flunarizine; GTP-Binding Proteins; Isoquinolines; Melanoma, Experimental; Mice; Piperazines; Protein Kinase C; Signal Transduction; Tamoxifen; Triazoles; Tumor Cells, Cultured; Verapamil | 1993 |
Differential effectiveness of a range of novel drug-resistance modulators, relative to verapamil, in influencing vinblastine or teniposide cytotoxicity in human lymphoblastoid CCRF-CEM sublines expressing classic or atypical multidrug resistance.
Topics: Cyclosporine; Dihydropyridines; Dose-Response Relationship, Drug; Drug Resistance; Drug Screening Assays, Antitumor; Flunarizine; Humans; Leukemia, T-Cell; Piperidines; Quinidine; Teniposide; Triazines; Tumor Cells, Cultured; Verapamil; Vinblastine | 1994 |
Effect of calcium antagonists on endothelin-induced contraction of isolated human resistance arteries: differences related to site of origin.
Topics: Adipose Tissue; Adult; Aged; Arteries; Calcium Channel Blockers; Calcium Channels; Diltiazem; Endothelins; Flunarizine; Humans; Membrane Potentials; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Myography; Nimodipine; Nisoldipine; Omentum; Vasoconstriction; Verapamil | 1993 |
Radioprotective effects of calcium antagonists used alone or with other types of radioprotectors.
Topics: Animals; Aspartic Acid; Calcium Channel Blockers; Diltiazem; Dimethyl Sulfoxide; Drug Combinations; Female; Flunarizine; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C3H; Mice, Inbred C57BL; Nifedipine; Nimodipine; Nitrendipine; Radiation-Protective Agents; Verapamil; Zinc | 1993 |
Refilling the inositol 1,4,5-trisphosphate-sensitive Ca2+ store in neuroblastoma x glioma hybrid NG108-15 cells.
Topics: Animals; Bradykinin; Calcium; Calcium-Transporting ATPases; Dose-Response Relationship, Drug; Flunarizine; Glioma; Hybrid Cells; Inositol 1,4,5-Trisphosphate; Mice; Neuroblastoma; Nitrendipine; Terpenes; Thapsigargin; Tumor Cells, Cultured; Verapamil | 1993 |
Correlation of melanoma cell motility and invasion in vitro.
Topics: Animals; Calcium Channel Blockers; Cell Movement; Cells, Cultured; Chick Embryo; Cytochalasins; Dequalinium; Female; Flunarizine; Image Processing, Computer-Assisted; Melanoma, Experimental; Mice; Mice, Inbred C3H; Myocardium; Neoplasm Invasiveness; Spheroids, Cellular; Tumor Cells, Cultured; Verapamil | 1995 |
Suppression of rhythmic discharges of medullary neurones in organotypic cultures of new-born rats by calcium antagonists.
Topics: Animals; Animals, Newborn; Calcium Channel Blockers; Flunarizine; Medulla Oblongata; Membrane Potentials; Neurons; Organ Culture Techniques; Rats; Verapamil | 1995 |
[Direct evidence of a protective effect of calcium antagonists on the inner ear. Inhibition of a toxic increase in the calcium level in hair cells of the guinea pig].
Topics: Animals; Calcium; Calcium Channel Blockers; Culture Techniques; Dose-Response Relationship, Drug; Female; Flunarizine; Guinea Pigs; Hair Cells, Auditory; Hair Cells, Auditory, Outer; Male; Membrane Potentials; Nifedipine; Potassium; Second Messenger Systems; Signal Transduction; Verapamil | 1995 |
Effect of calcium antagonists on regional cerebral blood flow in transplanted rat brain tumors.
Topics: Analysis of Variance; Animals; Brain; Brain Neoplasms; Calcium Channel Blockers; Cerebrovascular Circulation; Diltiazem; Flunarizine; Glioma; Male; Neoplasm Transplantation; Nifedipine; Nimodipine; Rats; Rats, Wistar; Verapamil | 1996 |
The effects of verapamil and flunarizine on epileptiform activity induced by bicuculline and low Mg2+ in neocortical tissue of epileptic and primary non-epileptic patients.
Topics: Astrocytoma; Bicuculline; Brain Neoplasms; Cerebral Cortex; Ependymoma; Epilepsy, Frontal Lobe; Epilepsy, Temporal Lobe; Evoked Potentials; Female; Flunarizine; Humans; In Vitro Techniques; Magnesium; Male; Oligodendroglioma; Verapamil | 1996 |
Effect of 4-aminopyridine and 3,4-diaminopyridine on guinea-pig isolated ileum.
Topics: 4-Aminopyridine; Acetylcholine; Amifampridine; Animals; Atropine; Calcium Channel Blockers; Diazoxide; Diltiazem; Dose-Response Relationship, Drug; Drug Interactions; Female; Flunarizine; Guinea Pigs; Ileum; In Vitro Techniques; Lanthanum; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Parasympathetic Nervous System; Parasympatholytics; Potassium Channels; Vasodilator Agents; Verapamil | 1997 |
Modulation of melphalan and cisplatin cytotoxicity in human ovarian cancer cells resistant to alkylating drugs.
Topics: Antineoplastic Agents; Antineoplastic Agents, Alkylating; Blotting, Northern; Calcium Channel Blockers; Cell Survival; Cisplatin; Culture Media; Cystadenoma; Drug Resistance, Neoplasm; Female; Flunarizine; Humans; Melphalan; Nimodipine; Ovarian Neoplasms; RNA Probes; RNA, Neoplasm; Tumor Cells, Cultured; Verapamil | 1997 |
Differential effects of Ca2+ channel blockers on Ca2+ overload induced by lysophosphatidylcholine in cardiomyocytes.
Topics: Animals; Benzofurans; Bepridil; Calcium; Calcium Channel Blockers; Cell Size; Cells, Cultured; Creatine Kinase; Dose-Response Relationship, Drug; Ethers, Cyclic; Flunarizine; Fura-2; Heart; Lysophosphatidylcholines; Male; Rats; Rats, Sprague-Dawley; Sodium; Sodium Channels; Verapamil | 1997 |
Strychnine-induced epileptiform activity in hippocampal and neocortical slice preparations: suppression by the organic calcium antagonists verapamil and flunarizine.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Epilepsy; Evoked Potentials; Female; Flunarizine; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Neocortex; Strychnine; Verapamil | 1997 |
Catalepsy induced by calcium channel blockers in mice.
Topics: Amlodipine; Animals; Binding, Competitive; Calcium Channel Blockers; Catalepsy; Dihydropyridines; Diltiazem; Disease Models, Animal; Flunarizine; Male; Mice; Muscarinic Antagonists; Nitrobenzenes; Piperazines; Predictive Value of Tests; Receptors, Cholinergic; Receptors, Dopamine D1; Receptors, Dopamine D2; Scopolamine; Time Factors; Verapamil | 1998 |
Pharmacological interaction of the calcium channel blockers verapamil and flunarizine with the opioid system.
Topics: Analgesics, Opioid; Animals; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drug Interactions; Flunarizine; Male; Mice; Mice, Inbred ICR; Narcotic Antagonists; Pain Measurement; Receptors, Opioid; Verapamil | 1999 |
Effects of ion channel modulators in the influx and efflux of Tc-99m-MIBI.
Topics: Adrenal Cortex Neoplasms; Amiloride; Calcium; Calcium Channel Blockers; Calcium Channels; Carcinoma, Small Cell; Flunarizine; Humans; Monensin; Sodium; Sodium Channels; Technetium Tc 99m Sestamibi; Tumor Cells, Cultured; Verapamil | 1999 |
Evidence of sex related differences in the effects of calcium channel blockers on neuroleptic-induced catalepsy in mice.
Topics: Animals; Antipsychotic Agents; Basal Ganglia Diseases; Calcium Channel Blockers; Catalepsy; Dose-Response Relationship, Drug; Female; Flunarizine; Haloperidol; Male; Mice; Nimodipine; Sex Factors; Verapamil | 1999 |
Effects of calcium channel blockers on behaviors induced by the N-methyl-D-aspartate receptor antagonist, dizocilpine, in rats.
Topics: Animals; Behavior, Animal; Calcium Channel Blockers; Calcium Channels, P-Type; Discrimination Learning; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Flunarizine; Generalization, Stimulus; Male; Motor Activity; Nimodipine; Rats; Rats, Wistar; Self Stimulation; Verapamil | 1999 |
Potentiation of analgesia and reversal of tolerance to morphine by calcium channel blockers.
Topics: Analgesia; Animals; Calcium Channel Blockers; Diltiazem; Drug Interactions; Drug Tolerance; Female; Flunarizine; Male; Mice; Morphine; Nimodipine; Pain Threshold; Verapamil | 2001 |
Effects of extracellular Na+ and Ca2+ ions and Ca2+ channel modulators on the cell-associated activity of 99mTc-MIBI and 99mTc-tetrofosmin in tumour cells.
Topics: Amiloride; Animals; Antineoplastic Agents; Calcium; Calcium Channels; Carcinoma, Lewis Lung; Cell Survival; Extracellular Space; Flunarizine; Glioma; Humans; Ion Channel Gating; Metabolic Clearance Rate; Mice; Organophosphorus Compounds; Organotechnetium Compounds; Radionuclide Imaging; Radiopharmaceuticals; Sodium; Technetium Tc 99m Sestamibi; Tumor Cells, Cultured; Verapamil | 2003 |
Glutamate increases toxicity of inorganic lead in GT1-7 neurons: partial protection induced by flunarizine.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Cell Death; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Environmental Pollutants; Flunarizine; Glutamic Acid; Glutathione; Hypothalamus; Lead; Mice; Neurons; Oxidative Stress; Reactive Oxygen Species; Receptors, Glutamate; Verapamil | 2003 |
Matrix-assisted laser desorption/ionisation mass spectrometry in the study of polycondensation of Ti(OBun)4 in the presence of Si(OEt)4.
Topics: Algorithms; Biotransformation; Chromatography, High Pressure Liquid; Cisapride; Flunarizine; Humans; In Vitro Techniques; Mass Spectrometry; Microsomes, Liver; Pharmaceutical Preparations; Pharmacokinetics; Propranolol; Verapamil | 2003 |
Expression of P-glycoprotein in L1210 cells is linked with rise in sensitivity to Ca2+.
Topics: Adenosine Triphosphate; Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium; Calcium Channel Blockers; Flunarizine; Leukemia L1210; Mice; Verapamil; Vincristine | 2005 |
Robust anti-arrhythmic efficacy of verapamil and flunarizine against dofetilide-induced TdP arrhythmias is based upon a shared and a different mode of action.
Topics: Animals; Anti-Arrhythmia Agents; Calcium Signaling; Cell Line; Dogs; Flunarizine; Humans; Lidocaine; Mice; Myocytes, Cardiac; Phenethylamines; Sulfonamides; Torsades de Pointes; Verapamil | 2010 |
HOCl causes necrotic cell death in human monocyte derived macrophages through calcium dependent calpain activation.
Topics: Calcimycin; Calcium; Calcium Channel Blockers; Calcium Ionophores; Calpain; Caspase 3; Cyclosporine; Dantrolene; Enzyme Inhibitors; Flunarizine; Humans; Hypochlorous Acid; Lysosomes; Macrophages; Membrane Potential, Mitochondrial; Muscle Relaxants, Central; Necrosis; Nifedipine; Verapamil | 2012 |
Effects of calcium channel antagonists on the motivational effects of nicotine and morphine in conditioned place aversion paradigm.
Topics: Animals; Avoidance Learning; Calcium Channel Blockers; Drug Administration Schedule; Flunarizine; Male; Morphine; Motivation; Nicotine; Nimodipine; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Verapamil | 2012 |