verapamil and carbamates

verapamil has been researched along with carbamates in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19905 (22.73)18.7374
1990's5 (22.73)18.2507
2000's4 (18.18)29.6817
2010's7 (31.82)24.3611
2020's1 (4.55)2.80

Authors

AuthorsStudies
Hoffman, BF; Mary-Rabine, L; Rosen, MR1
Danilo, P; Davies, M; Hordof, AJ; Reder, RF; Rosen, MR1
Kobayashi, DV; Moriya, K; Numano, F; Shimamoto, T; Takahashi, T1
Misík, V; Ondrias, K; Reguli, J; Stasko, A; Svajdlenka, E1
Danilo, P; Rosen, MR1
Danilo, P; Hordof, AJ; Malm, JR; Mary-Rabine, L; Rosen, MR1
Stolc, S1
Clark, AH; Garland, CJ1
Dissing, S; Frøkjaer-Jensen, J; Gromada, J; Kofod, H1
Bridgers, A; Coffin, M; Long, S; Polli, J; Roy, A; Vickers, A; Winnike, R; Yu, L1
Daily, JP; Fahey, JM; Greenblatt, DJ; Perloff, MD; von Moltke, LL1
Blom-Roosemalen, MC; Breimer, DD; de Boer, AG; Nabulsi, L; van der Sandt, IC; Voorwinden, HH; Vos, CM1
Bhugra, P; Dhalla, NS; Rathi, S; Xu, YJ1
Bui, T; Ho, RJ; Hsiao, P; Unadkat, JD1
Annaert, P; Augustijns, P; Brouwers, J; Mols, R1
Ahmad-Molaei, L; Eslahkar, S; Mazar-Atabaki, A; Motiei-Langroudi, SM; Naderi, N; Ronaghi, A; Shirazi-zand, Z1
Brueggemann, LI; Byron, KL; Cribbs, LL; Dowell, ML; Kakad, PP; Love, RB; Solway, J1
Cao, Y; Jusko, WJ1
Dively, GP; Evans, JD; Guseman, AJ; Hawthorne, DJ; Kunkle, G; Miller, K; Pettis, JS; vanEngelsdorp, D1
Aunes, M; Cullberg, M; Edvardsson, N; Frison, L; Johansson, S; Löfberg, B; Lunde, H1
Bergenholm, L; Chappell, MJ; Collins, T; Evans, ND; Mettetal, J; Parkinson, J1
Ito, S; Iwamoto, K; Kamimura, H; Mizunaga, M; Nakayama, K; Negoro, T; Nishiwaki, M; Nomura, Y; Suemizu, H; Yamazaki, H; Yoneda, N1

Trials

2 trial(s) available for verapamil and carbamates

ArticleYear
In Silico Predictions and In Vivo Results of Drug-Drug Interactions by Ketoconazole and Verapamil on AZD1305, a Combined Ion Channel Blocker and a Sensitive CYP3A4 Substrate.
    Clinical pharmacology in drug development, 2016, Volume: 5, Issue:5

    Topics: Adult; Anti-Arrhythmia Agents; Area Under Curve; Azabicyclo Compounds; Carbamates; Computer Simulation; Cross-Over Studies; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Humans; Ketoconazole; Male; Middle Aged; Verapamil; Young Adult

2016
Predicting QRS and PR interval prolongations in humans using nonclinical data.
    British journal of pharmacology, 2017, Volume: 174, Issue:19

    Topics: Animals; Anti-Arrhythmia Agents; Azabicyclo Compounds; Carbamates; Dogs; Drug Evaluation, Preclinical; Electrocardiography; Flecainide; Guinea Pigs; Heart; Heart Rate; Humans; Long QT Syndrome; Male; Models, Biological; Quinidine; Verapamil

2017

Other Studies

20 other study(ies) available for verapamil and carbamates

ArticleYear
Participation of slow inward current in the Purkinje fiber action potential overshoot.
    The American journal of physiology, 1979, Volume: 237, Issue:2

    Topics: Action Potentials; Animals; Calcium; Carbamates; Dogs; Heart Conduction System; Membrane Potentials; Purkinje Fibers; Pyrrolidines; Tetrodotoxin; Verapamil

1979
Age-related changes in Purkinje fiber action potentials of adult dogs.
    Circulation research, 1978, Volume: 43, Issue:6

    Topics: Action Potentials; Aging; Animals; Carbamates; Dogs; Electrocardiography; Female; Heart Conduction System; Male; Microelectrodes; Purkinje Fibers; Pyrrolidines; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1978
Hyperreactive arterial endothelial cells in atherogenesis. Effect of smooth muscle relaxants.
    Advances in experimental medicine and biology, 1977, Volume: 82

    Topics: Actomyosin; Animals; Aorta; Arteriosclerosis; Biological Transport; Carbamates; Carbon; Colchicine; Endothelium; Parasympatholytics; Phthalazines; Pyridazines; Pyridinolcarbamate; Rabbits; Verapamil; Vinblastine

1977
Comparison of perturbation effect of propranolol, verapamil, chlorpromazine and carbisocaine on lecithin liposomes and brain total lipid liposomes. An EPR spectroscopy study.
    Chemico-biological interactions, 1991, Volume: 79, Issue:2

    Topics: Animals; Brain; Carbamates; Chlorpromazine; Dose-Response Relationship, Drug; Electron Spin Resonance Spectroscopy; Liposomes; Molecular Weight; Phosphatidylcholines; Phospholipids; Propranolol; Rats; Verapamil

1991
Effects of tetrodotoxin, lidocaine, verapamil, and AHR-2666 on Ouabain-induced delayed afterdepolarizations in canine Purkinje fibers.
    Circulation research, 1980, Volume: 46, Issue:1

    Topics: Action Potentials; Animals; Carbamates; Diastole; Dogs; Heart Conduction System; Ion Channels; Lidocaine; Ouabain; Purkinje Fibers; Pyrrolidines; Tetrodotoxin; Time Factors; Verapamil

1980
Mechanisms for impulse initiation in isolated human atrial fibers.
    Circulation research, 1980, Volume: 47, Issue:2

    Topics: Acetylcholine; Action Potentials; Adolescent; Adult; Carbamates; Child; Child, Preschool; Electrophysiology; Epinephrine; Heart Atria; Heart Conduction System; Heart Rate; Humans; Infant; Lidocaine; Middle Aged; Myocardial Contraction; Pyrrolidines; Tetrodotoxin; Time Factors; Verapamil

1980
Inhibition of ion currents in membrane of sensory neuron by the antiarrhythmic drug BK 129 and selected Ca2+ entry blockers.
    General physiology and biophysics, 1993, Volume: 12, Issue:6

    Topics: Animals; Anti-Arrhythmia Agents; Azepines; Calcium Channel Blockers; Carbamates; Ganglia, Spinal; Membrane Potentials; Neurons, Afferent; Nifedipine; Piperidines; Rats; Verapamil

1993
Ca2+ channel antagonists and inhibition of protein kinase C each block contraction but not depolarization to 5-hydroxytryptamine in the rabbit basilar artery.
    European journal of pharmacology, 1993, Apr-22, Volume: 235, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Basilar Artery; Calcium Channel Blockers; Carbamates; Female; Isoquinolines; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylcarbamates; Piperazines; Potassium; Protein Kinase C; Rabbits; Serotonin; Type C Phospholipases; Verapamil

1993
Effects of the hypoglycaemic drugs repaglinide and glibenclamide on ATP-sensitive potassium-channels and cytosolic calcium levels in beta TC3 cells and rat pancreatic beta cells.
    Diabetologia, 1995, Volume: 38, Issue:9

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Calcium; Carbamates; Cell Line; Cells, Cultured; Cytosol; Dose-Response Relationship, Drug; Glyburide; Hypoglycemic Agents; Ion Channel Gating; Islets of Langerhans; Kinetics; Membrane Potentials; Mice; Patch-Clamp Techniques; Piperidines; Potassium Channels; Rats; Serum Albumin; Time Factors; Verapamil

1995
Vitamin E-TPGS increases absorption flux of an HIV protease inhibitor by enhancing its solubility and permeability.
    Pharmaceutical research, 1999, Volume: 16, Issue:12

    Topics: Algorithms; Animals; Biological Availability; Caco-2 Cells; Calcium Channel Blockers; Carbamates; Cell Membrane Permeability; Chromatography, High Pressure Liquid; Dogs; Furans; HIV Protease Inhibitors; Humans; Permeability; Polyethylene Glycols; Solubility; Stimulation, Chemical; Sulfonamides; Verapamil; Vitamin E

1999
Induction of P-glycoprotein expression by HIV protease inhibitors in cell culture.
    AIDS (London, England), 2000, Jun-16, Volume: 14, Issue:9

    Topics: Adenocarcinoma; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carbamates; Cell Line, Transformed; Colonic Neoplasms; Drug Resistance, Multiple; Furans; Gene Expression Regulation, Neoplastic; HIV Protease Inhibitors; Humans; Indinavir; Ivermectin; Nelfinavir; Ritonavir; Saquinavir; Sulfonamides; Tumor Cells, Cultured; Verapamil; Vinblastine

2000
Assessment of active transport of HIV protease inhibitors in various cell lines and the in vitro blood--brain barrier.
    AIDS (London, England), 2001, Mar-09, Volume: 15, Issue:4

    Topics: Animals; Astrocytes; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport, Active; Blood-Brain Barrier; Caco-2 Cells; Carbamates; Cattle; Cell Line, Transformed; Cells, Cultured; Coculture Techniques; Cyclosporins; Dibenzocycloheptenes; Endothelium, Vascular; Furans; HIV Protease Inhibitors; Humans; Indinavir; LLC-PK1 Cells; Multidrug Resistance-Associated Proteins; Probenecid; Quinolines; Rats; Rats, Wistar; Ritonavir; Sulfonamides; Swine; Verapamil

2001
Modification of intracellular free calcium in cultured A10 vascular smooth muscle cells by exogenous phosphatidic acid.
    Biochemical pharmacology, 2003, Jun-15, Volume: 65, Issue:12

    Topics: Animals; Boron Compounds; Calcium; Carbamates; Cells, Cultured; Diltiazem; Drug Interactions; Egtazic Acid; Indoles; Macrocyclic Compounds; Maleimides; Muscle, Smooth, Vascular; Oxazoles; Pertussis Toxin; Phenylcarbamates; Phosphatidic Acids; Rats; Tetradecanoylphorbol Acetate; Thapsigargin; Verapamil

2003
In vitro-to-in vivo prediction of P-glycoprotein-based drug interactions at the human and rodent blood-brain barrier.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Boron Compounds; Carbamates; Carbon Radioisotopes; Cyclosporine; Drug Interactions; Fluorescent Dyes; Furans; Humans; LLC-PK1 Cells; Positron-Emission Tomography; Quinidine; Quinine; Rats; Sulfonamides; Swine; Verapamil

2008
Validation of a differential in situ perfusion method with mesenteric blood sampling in rats for intestinal drug interaction profiling.
    Biopharmaceutics & drug disposition, 2010, Volume: 31, Issue:5-6

    Topics: Adrenergic beta-Antagonists; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carbamates; Drug Interactions; Furans; Intestinal Absorption; Ketoconazole; Male; Perfusion; Polyethylene Glycols; Rats; Rats, Wistar; Splanchnic Circulation; Sulfonamides; Verapamil; Vitamin E

2010
L-type calcium channel mediates anticonvulsant effect of cannabinoids in acute and chronic murine models of seizure.
    Neurochemical research, 2012, Volume: 37, Issue:2

    Topics: Acute Disease; Animals; Anticonvulsants; Benzamides; Benzoxazines; Calcium Channels, L-Type; Cannabinoids; Carbamates; Chronic Disease; Diltiazem; Disease Models, Animal; Kindling, Neurologic; Male; Mice; Morpholines; Naphthalenes; Rats; Rats, Wistar; Seizures; Verapamil

2012
Kv7 potassium channels in airway smooth muscle cells: signal transduction intermediates and pharmacological targets for bronchodilator therapy.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Jan-01, Volume: 302, Issue:1

    Topics: Aminopyridines; Animals; Anthracenes; Bronchoconstriction; Bronchodilator Agents; Calcium Channel Blockers; Carbamates; Celecoxib; Guinea Pigs; Histamine; Humans; KCNQ Potassium Channels; Male; Methacholine Chloride; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Phenylenediamines; Pyrazoles; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Sulfonamides; Verapamil

2012
Applications of minimal physiologically-based pharmacokinetic models.
    Journal of pharmacokinetics and pharmacodynamics, 2012, Volume: 39, Issue:6

    Topics: Anti-Bacterial Agents; Antibodies, Monoclonal; beta-Lactams; Biological Availability; Carbamates; Codeine; Humans; Kinetics; Liver; Midazolam; Models, Biological; Piperidines; Regional Blood Flow; Verapamil

2012
Multi-Drug Resistance Transporters and a Mechanism-Based Strategy for Assessing Risks of Pesticide Combinations to Honey Bees.
    PloS one, 2016, Volume: 11, Issue:2

    Topics: Animals; ATP-Binding Cassette Transporters; Bees; Biological Transport; Biphenyl Compounds; Carbamates; Cyclohexanes; Drug Resistance, Multiple; Environmental Exposure; Fatty Acids, Unsaturated; Insecticides; Ivermectin; Membrane Transport Proteins; Neonicotinoids; Niacinamide; Pyrazoles; Pyridines; Quercetin; Rhodamines; Risk Assessment; Sesquiterpenes; Verapamil

2016
Predicted values for human total clearance of a variety of typical compounds with differently humanized-liver mouse plasma data.
    Drug metabolism and pharmacokinetics, 2020, Volume: 35, Issue:4

    Topics: Acetamides; Albuterol; Animals; Carbamates; Chromatography, Liquid; Diazepam; Diclofenac; Digitoxin; Humans; Itraconazole; Ketoprofen; Liver; Metabolic Clearance Rate; Mice; Mice, Transgenic; Naproxen; Pharmaceutical Preparations; Phenytoin; Piperidines; Pravastatin; Pyrimidines; Quinidine; Tandem Mass Spectrometry; Telmisartan; Terfenadine; Verapamil

2020