verapamil and azidopine

verapamil has been researched along with azidopine in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-19908 (21.05)18.7374
1990's28 (73.68)18.2507
2000's2 (5.26)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Naito, M; Tsuruo, T1
Charuk, JH; Reithmeier, RA1
Bruggemann, EP; Currier, SJ; Gottesman, MM; Pastan, I1
Anstett, M; Atassi, G; Bizzari, JP; Genton, A; Léonce, S; Pérez, V; Pierré, A1
Gottesman, MM; Horio, M; Lovelace, E; Pastan, I1
Suzuki, H; Tatsuta, T; Tomida, A1
Fukazawa, N; Sato, W; Suzuki, T; Tsuruo, T; Yusa, K1
Maeda, H; Miyamoto, Y1
Akiyama, S; Douzono, H; Ikeda, S; Nagata, Y; Sugita, M; Sumizawa, T; Yoshimura, A1
Gindin, E; Greenberger, LM; Horwitz, SB; Yang, CP1
Bindslev, N; Demant, EJ; Friche, E; Jensen, PB; Sehested, M; Skovsgaard, T1
Demant, EJ; Friche, E; Jensen, PB; Nissen, NN; Sehested, M1
Ferry, DR; Glossmann, H; Goll, A; Schober, M; Striessnig, J1
Hofmann, F; Nastainczyk, W; Sieber, M; Wernet, W; Zubor, V1
Glossmann, H; Hymel, L; Schindler, H; Striessnig, J1
Flockerzi, V1
Hudecová, S; Krizanová, O; Orlický, J; Zachar, J1
Arceci, RJ; DePinho, SG; Greenberger, LM; Horwitz, SB; Yang, CP1
Safa, AR; Spearman, T; Van Dyke, K; Ye, ZG1
Glossmann, H; Knaus, HG; Striessnig, J1
Boiocchi, M; Cappelletto, B; Corona, G; Gigante, M; Raschack, M; Simone, F; Toffoli, G1
Bennis, S; Ichas, F; Robert, J1
Eliason, JF; Ishikawa, T; Ramuz, H; Tsuruo, T; Yamamoto, T; Yoshikubo, T1
Bates, SE; Dickstein, B; Fojo, AT; Lee, JS; Spolyar, M1
Ashbourne, KJ; DiDiodato, G; Sharom, FJ; Yu, X1
Senior, AE; Urbatsch, IL1
Koseki, Y; Lothstein, L; Sweatman, TW1
Georges, E; Ling, V; Liu, Z; Zordan-Nudo, T1
Kang, Y; Perry, RR1
Gajdzik, L; Graf, J; Stapf, V; Thalhammer, T1
Abraham, I; Sampson, KE; Wolf, CL1
Bamberger, U; Georges, E; Heckel, A; Lheureux, F; Liu, Z; Pouliot, JF1
Boer, R; Gekeler, V; Grunicke, H; Hofmann, J; Ise, W; Klemm, K; Sanders, KH; Schächtele, C; Schubert, C; Uberall, F; Utz, I1
Chapey, C; Hu, YP; Robert, J1
Chen, G; Dumontet, C; Durán, GE; Jaffrézou, JP; Lacayo, NJ; Sikic, BI; Steger, KA1
Abu Khoudoud, OR; Bikhazi, AB; Bitar, KM; el-Kasti, MM; Ibrahim, MZ; Kreydiyyeh, SI; Saleh, RS1
Chen, KG; Cohen, D; Durán, GE; Lacayo, NJ; Sikic, BI1
Fujita, R; Ishikawa, M; Sasaki, K; Takayanagi, M; Takayanagi, Y1

Other Studies

38 other study(ies) available for verapamil and azidopine

ArticleYear
Functionally active homodimer of P-glycoprotein in multidrug-resistant tumor cells.
    Biochemical and biophysical research communications, 1992, May-29, Volume: 185, Issue:1

    Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Dihydropyridines; Doxorubicin; Drug Resistance; Humans; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Macromolecular Substances; Membrane Glycoproteins; Mitolactol; Mitomycins; Precipitin Tests; Succinimides; Tumor Cells, Cultured; Verapamil; Vincristine

1992
Interaction of P-glycoprotein with a hydrophobic component of rat urine.
    Biochemical and biophysical research communications, 1992, Jul-31, Volume: 186, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; CHO Cells; Cricetinae; Dihydropyridines; Drug Resistance; Female; Kinetics; Male; Membrane Glycoproteins; Rats; Tissue Extracts; Urine; Verapamil; Vinblastine

1992
Characterization of the azidopine and vinblastine binding site of P-glycoprotein.
    The Journal of biological chemistry, 1992, Oct-15, Volume: 267, Issue:29

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line; Cell Membrane; Colchicine; Cyanogen Bromide; Dihydropyridines; Drug Resistance; Humans; KB Cells; Kinetics; Membrane Glycoproteins; Molecular Weight; Peptide Fragments; Transfection; Trypsin; Verapamil; Vinblastine; Vincristine

1992
Effects of a new triazinoaminopiperidine derivative on adriamycin accumulation and retention in cells displaying P-glycoprotein-mediated multidrug resistance.
    Biochemical pharmacology, 1992, Nov-03, Volume: 44, Issue:9

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Carcinoma, Squamous Cell; Cell Cycle; Cell Membrane; Cells, Cultured; Colonic Neoplasms; Cricetinae; Cricetulus; Dihydropyridines; Doxorubicin; Drug Resistance; Flow Cytometry; Fluorescence; Humans; Kinetics; Leukemia P388; Leukemia, Myeloid, Acute; Lung; Membrane Glycoproteins; Mice; Piperidines; Sensitivity and Specificity; Triazines; Tritium; Tumor Cells, Cultured; Verapamil

1992
Agents which reverse multidrug-resistance are inhibitors of [3H]vinblastine transport by isolated vesicles.
    Biochimica et biophysica acta, 1991, Jan-09, Volume: 1061, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Biological Transport, Active; Carcinoma, Squamous Cell; Cell Membrane; Dihydropyridines; Drug Resistance; Humans; Kinetics; Leucine; Membrane Glycoproteins; Phenothiazines; Quinidine; Trifluoperazine; Tumor Cells, Cultured; Verapamil; Vinblastine

1991
Novel mechanism of N-solanesyl-N,N'-bis(3,4-dimethoxybenzyl)ethylenediamine in potentiation of antitumor drug action on multidrug-resistant and sensitive Chinese hamster cells.
    Japanese journal of cancer research : Gann, 1991, Volume: 82, Issue:1

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Membrane; Cricetinae; Cricetulus; Daunorubicin; Dihydropyridines; Doxorubicin; Drug Resistance; Drug Synergism; Ethylenediamines; Membrane Glycoproteins; Terpenes; Verapamil; Vinblastine

1991
Circumvention of multidrug resistance by a newly synthesized quinoline derivative, MS-073.
    Cancer research, 1991, May-01, Volume: 51, Issue:9

    Topics: Affinity Labels; Animals; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Dihydropyridines; Drug Administration Schedule; Drug Resistance; Drug Screening Assays, Antitumor; Drug Synergism; Female; Leukemia P388; Membrane Glycoproteins; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Piperazines; Quinolines; Tumor Cells, Cultured; Verapamil; Vincristine

1991
Enhancement by verapamil of neocarzinostatin action on multidrug-resistant Chinese hamster ovary cells: possible release of nonprotein chromophore in cells.
    Japanese journal of cancer research : Gann, 1991, Volume: 82, Issue:3

    Topics: Animals; Antioxidants; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Division; Cell Line; Cell Membrane; Cell Survival; Cells, Cultured; Cricetinae; Cricetulus; Dihydropyridines; Drug Resistance; Drug Synergism; Female; Kinetics; Membrane Glycoproteins; Ovary; Verapamil; Zinostatin

1991
Aspergillus species strain M39 produces two naphtho-gamma-pyrones that reverse drug resistance in human KB cells.
    International journal of cancer, 1990, Mar-15, Volume: 45, Issue:3

    Topics: Aspergillus; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Chemical Phenomena; Chemistry; Dihydropyridines; Doxorubicin; Drug Resistance; Humans; Membrane Glycoproteins; Naphthols; Pyrans; Pyrones; Verapamil; Vinblastine

1990
Photoaffinity probes for the alpha 1-adrenergic receptor and the calcium channel bind to a common domain in P-glycoprotein.
    The Journal of biological chemistry, 1990, Mar-15, Volume: 265, Issue:8

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Binding, Competitive; Calcium Channels; Cell Line; Cell Membrane; Chymotrypsin; Dihydropyridines; Drug Resistance; Macrophages; Membrane Glycoproteins; Mice; Peptide Mapping; Prazosin; Receptors, Adrenergic, alpha; Sequence Homology, Nucleic Acid; Verapamil

1990
Transport of the multidrug resistance modulators verapamil and azidopine in wild type and daunorubicin resistant Ehrlich ascites tumour cells.
    British journal of cancer, 1990, Volume: 62, Issue:1

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Carcinoma, Ehrlich Tumor; Cells, Cultured; Daunorubicin; Dihydropyridines; Dose-Response Relationship, Drug; Drug Resistance; Humans; In Vitro Techniques; Membrane Glycoproteins; Verapamil; Vincristine

1990
The solvents cremophor EL and Tween 80 modulate daunorubicin resistance in the multidrug resistant Ehrlich ascites tumor.
    Cancer communications, 1990, Volume: 2, Issue:9

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Carcinoma, Ehrlich Tumor; Cyclosporins; Daunorubicin; Dihydropyridines; Drug Resistance; Drug Synergism; Drug Therapy, Combination; Glycerol; Humans; Intracellular Membranes; Membrane Glycoproteins; Polysorbates; Tritium; Tumor Cells, Cultured; Verapamil

1990
Calcium channels: basic properties as revealed by radioligand binding studies.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: Affinity Labels; Animals; Azides; Binding Sites; Binding, Competitive; Brain; Calcium; Calcium Channel Blockers; Dihydropyridines; Guinea Pigs; Iodobenzenes; Ion Channels; Molecular Weight; Muscles; Neurilemma; Photochemistry; Pyridines; Sarcolemma; Verapamil

1985
The 165-kDa peptide of the purified skeletal muscle dihydropyridine receptor contains the known regulatory sites of the calcium channel.
    European journal of biochemistry, 1987, Aug-17, Volume: 167, Issue:1

    Topics: Affinity Labels; Animals; Azides; Calcium; Calcium Channels; Dihydropyridines; Ion Channels; Isradipine; Kinetics; Molecular Weight; Muscles; Oxadiazoles; Pyridines; Rabbits; Receptors, Nicotinic; Verapamil

1987
Purification and reconstitution of calcium channel drug-receptor sites.
    Annals of the New York Academy of Sciences, 1988, Volume: 522

    Topics: Affinity Labels; Animals; Azides; Calcium; Calcium Channels; Dihydropyridines; Guinea Pigs; Ion Channels; Muscles; Receptors, Drug; Receptors, Nicotinic; Verapamil

1988
Molecular properties of voltage-activated calcium channels.
    Journal of protein chemistry, 1989, Volume: 8, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Affinity Labels; Animals; Azides; Calcium Channels; Cloning, Molecular; Dihydropyridines; DNA; Glycoproteins; Muscles; Phosphorylation; Protein Conformation; Protein Kinases; Receptors, Nicotinic; Verapamil

1989
Is Ca2+ antagonists binding protein from cytosolic fraction the precursor of alpha 1-subunit of Ca2+ channel?
    General physiology and biophysics, 1989, Volume: 8, Issue:2

    Topics: Affinity Labels; Animals; Antibodies; Azides; Binding, Competitive; Calcium Channel Blockers; Calcium Channels; Cytoplasm; Dihydropyridines; In Vitro Techniques; Isradipine; Muscles; Oxadiazoles; Protein Precursors; Rabbits; Radioligand Assay; Receptors, Nicotinic; Ultraviolet Rays; Verapamil

1989
Progesterone interacts with P-glycoprotein in multidrug-resistant cells and in the endometrium of gravid uterus.
    The Journal of biological chemistry, 1989, Jan-15, Volume: 264, Issue:2

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Line; Dihydropyridines; Drug Resistance; Endometrium; Estradiol; Female; Intracellular Membranes; Kinetics; Membrane Glycoproteins; Mice; Mice, Inbred C57BL; Microsomes; Pregnancy; Pregnancy, Animal; Progesterone; Protein Binding; Steroids; Verapamil; Vinblastine

1989
3H-azidopine photoaffinity labeling of high molecular weight proteins in chloroquine resistant falciparum malaria.
    Biochemical and biophysical research communications, 1989, Jul-31, Volume: 162, Issue:2

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Chloroquine; Chlorpromazine; Dihydropyridines; Drug Resistance; Glycoproteins; Molecular Weight; Nicardipine; Photochemistry; Plasmodium falciparum; Proteins; Quinacrine; Reserpine; Trifluoperazine; Verapamil

1989
Photoaffinity-labelling of the calcium-channel-associated 1,4-dihydropyridine and phenylalkylamine receptor in guinea-pig hippocampus. A 195 kDa polypeptide carries both drug receptors and has similarities to the alpha 1 subunit of the purified skeletal-m
    The Biochemical journal, 1988, Jul-01, Volume: 253, Issue:1

    Topics: Affinity Labels; Animals; Azides; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Dihydropyridines; Guinea Pigs; Hippocampus; In Vitro Techniques; Kinetics; Muscles; Peptides; Radioimmunoassay; Receptors, Nicotinic; Tritium; Verapamil

1988
Structure-activity relationship of verapamil analogs and reversal of multidrug resistance.
    Biochemical pharmacology, 1995, Oct-12, Volume: 50, Issue:8

    Topics: Animals; Antineoplastic Agents; Aorta; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Calcium; Dihydropyridines; Doxorubicin; Drug Design; Drug Resistance, Microbial; Drug Resistance, Multiple; Drug Synergism; Humans; Male; Rats; Rats, Sprague-Dawley; RNA, Messenger; Structure-Activity Relationship; Tumor Cells, Cultured; Tumor Stem Cell Assay; Verapamil

1995
Differential effects of verapamil and quinine on the reversal of doxorubicin resistance in a human leukemia cell line.
    International journal of cancer, 1995, Jul-28, Volume: 62, Issue:3

    Topics: Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Dihydropyridines; Doxorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Drug Synergism; Humans; Kinetics; Leukemia, Erythroblastic, Acute; Microscopy, Confocal; Microscopy, Fluorescence; Phenotype; Quinine; Subcellular Fractions; Tumor Cells, Cultured; Verapamil

1995
Novel dithiane analogues of tiapamil with high activity to overcome multidrug resistance in vitro.
    Biochemical pharmacology, 1995, Jul-17, Volume: 50, Issue:2

    Topics: Animals; Aorta; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; In Vitro Techniques; Propylamines; Rats; Stereoisomerism; Tiapamil Hydrochloride; Tumor Cells, Cultured; Verapamil; Vincristine

1995
Differential modulation of P-glycoprotein transport by protein kinase inhibition.
    Biochemistry, 1993, Sep-07, Volume: 32, Issue:35

    Topics: Affinity Labels; Alkaloids; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Carrier Proteins; Cyclosporine; Dactinomycin; Dihydropyridines; Drug Resistance; Humans; Isoenzymes; Membrane Glycoproteins; Naphthalenes; Polycyclic Compounds; Protein Kinase C; Rhodamine 123; Rhodamines; Staurosporine; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Verapamil; Vinblastine; Vincristine

1993
Interaction of the P-glycoprotein multidrug transporter with peptides and ionophores.
    The Journal of biological chemistry, 1995, Apr-28, Volume: 270, Issue:17

    Topics: Adenosine Triphosphatases; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cell Membrane; CHO Cells; Cricetinae; Dihydropyridines; Enzyme Activation; Ionophores; Peptides; Photochemistry; Protein Binding; Verapamil

1995
Effects of lipids on ATPase activity of purified Chinese hamster P-glycoprotein.
    Archives of biochemistry and biophysics, 1995, Jan-10, Volume: 316, Issue:1

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Brain Chemistry; Cattle; Cell Membrane; Colchicine; Cricetinae; Cricetulus; Daunorubicin; Dihydropyridines; Escherichia coli; Lipids; Liver; Proteolipids; Sheep; Verapamil; Vinblastine

1995
P-glycoprotein overexpression in mouse cells does not correlate with resistance to N-benzyladriamycin-14-valerate (AD 198).
    Anti-cancer drugs, 1994, Volume: 5, Issue:6

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cells, Cultured; Dihydropyridines; DNA Topoisomerases, Type II; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance; Immunoblotting; Mice; Tumor Cells, Cultured; Verapamil

1994
Effects of nonionic detergents on P-glycoprotein drug binding and reversal of multidrug resistance.
    Cancer research, 1993, Dec-15, Volume: 53, Issue:24

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Carrier Proteins; Cells, Cultured; Cholic Acids; Detergents; Dihydropyridines; Drug Resistance; Humans; Membrane Glycoproteins; Octoxynol; Verapamil

1993
Effect of alpha-interferon on P-glycoprotein expression and function and on verapamil modulation of doxorubicin resistance.
    Cancer research, 1994, Jun-01, Volume: 54, Issue:11

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Carrier Proteins; Cell Line; Cricetinae; Dihydropyridines; Doxorubicin; Drug Resistance; Drug Synergism; Interferon-alpha; Membrane Glycoproteins; RNA, Messenger; Verapamil

1994
Bile canalicular cationic dye secretion as a model for P-glycoprotein mediated transport.
    European journal of pharmacology, 1994, Apr-04, Volume: 270, Issue:2-3

    Topics: Acridine Orange; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Bile Canaliculi; Blotting, Western; Carrier Proteins; Cell Membrane; Cyclosporine; Dihydropyridines; In Vitro Techniques; Liver; Male; Membrane Glycoproteins; Models, Biological; Perfusion; Precipitin Tests; Rats; Rats, Inbred Strains; Verapamil

1994
Non-glucocorticoid steroid analogues (21-aminosteroids) sensitize multidrug resistant cells to vinblastine.
    Cancer chemotherapy and pharmacology, 1993, Volume: 32, Issue:2

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Survival; Dihydropyridines; Drug Interactions; Drug Resistance; Humans; KB Cells; Membrane Glycoproteins; Pregnatrienes; Structure-Activity Relationship; Verapamil; Vinblastine

1993
BIBW22 BS, potent multidrug resistance-reversing agent, binds directly to P-glycoprotein and accumulates in drug-resistant cells.
    Molecular pharmacology, 1996, Volume: 50, Issue:3

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line; Cell Survival; CHO Cells; Colchicine; Cricetinae; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; Humans; Kinetics; Lymphoma; Morpholines; Peptide Mapping; Protein Binding; Triamterene; Tumor Cells, Cultured; Verapamil; Vinblastine

1996
Effects of the selective bisindolylmaleimide protein kinase C inhibitor GF 109203X on P-glycoprotein-mediated multidrug resistance.
    British journal of cancer, 1996, Volume: 74, Issue:6

    Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Dihydropyridines; Drug Resistance, Multiple; Enzyme Inhibitors; Gene Expression; Humans; Indoles; Maleimides; Mice; Phosphorylation; Protein Kinase C; Verapamil

1996
Relationship between the inhibition of azidopine binding to P-glycoprotein by MDR modulators and their efficiency in restoring doxorubicin intracellular accumulation.
    Cancer letters, 1996, Dec-03, Volume: 109, Issue:1-2

    Topics: Affinity Labels; Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cyclosporine; Cyclosporins; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; Humans; Mice; Nicardipine; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1996
Multidrug-resistant human sarcoma cells with a mutant P-glycoprotein, altered phenotype, and resistance to cyclosporins.
    The Journal of biological chemistry, 1997, Feb-28, Volume: 272, Issue:9

    Topics: Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Cell Survival; Cyclosporins; Dihydropyridines; DNA Topoisomerases, Type II; Doxorubicin; Drug Resistance, Multiple; Humans; Neoplasm Proteins; Phenotype; Polymerase Chain Reaction; Prazosin; Rhodamine 123; Rhodamines; Sarcoma; Vault Ribonucleoprotein Particles; Verapamil

1997
Binding and distribution of three prototype calcium channel blockers in perfused rat liver.
    Molecular and cellular biochemistry, 1997, Volume: 169, Issue:1-2

    Topics: Animals; Azides; Calcium Channel Blockers; Calcium Channels; Carbon Radioisotopes; Dihydropyridines; Inulin; Isradipine; Liver; Models, Biological; Perfusion; Rats; Rats, Sprague-Dawley; Time Factors; Tritium; Urea; Verapamil

1997
Loss of cyclosporin and azidopine binding are associated with altered ATPase activity by a mutant P-glycoprotein with deleted phe(335).
    Molecular pharmacology, 2000, Volume: 57, Issue:4

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Calcium Channel Blockers; Cyclosporine; Dihydropyridines; Drug Interactions; Enzyme Activation; Humans; Molecular Sequence Data; Phenylalanine; Photoaffinity Labels; Tritium; Tumor Cells, Cultured; Vanadates; Verapamil

2000
Enhancement of doxorubicin activity in multidrug-resistant cells by mefloquine.
    Methods and findings in experimental and clinical pharmacology, 2000, Volume: 22, Issue:5

    Topics: Affinity Labels; Antibiotics, Antineoplastic; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Calcium Channel Blockers; Coloring Agents; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Humans; Mefloquine; Phenotype; Rhodamine 123; Tumor Cells, Cultured; Verapamil

2000