Page last updated: 2024-09-04

varespladib and tretinoin

varespladib has been researched along with tretinoin in 2 studies

Compound Research Comparison

Studies
(varespladib)
Trials
(varespladib)
Recent Studies (post-2010)
(varespladib)
Studies
(tretinoin)
Trials
(tretinoin)
Recent Studies (post-2010) (tretinoin)
80114923,6541,0836,085

Protein Interaction Comparison

ProteinTaxonomyvarespladib (IC50)tretinoin (IC50)
Bile salt export pumpHomo sapiens (human)10
Amyloid-beta precursor proteinHomo sapiens (human)0.18
Adenosine receptor A3Homo sapiens (human)5.275
Retinoic acid receptor alphaHomo sapiens (human)2.2542
60 kDa heat shock protein, mitochondrialHomo sapiens (human)5.3
Retinoic acid receptor betaHomo sapiens (human)0.7537
Retinoic acid receptor alphaMus musculus (house mouse)0.0057
Retinoic acid receptor gamma Homo sapiens (human)0.0064
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)5.275
Retinoic acid receptor gammaMus musculus (house mouse)0.004
Retinoic acid receptor betaMus musculus (house mouse)0.005
Mitogen-activated protein kinase 1Homo sapiens (human)0.576
Nuclear receptor ROR-alphaHomo sapiens (human)0.1995
Alpha-synucleinHomo sapiens (human)3
Cellular retinoic acid-binding protein 1Gallus gallus (chicken)0.5233
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.358
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)5.275
Retinoic acid receptor RXR-gammaHomo sapiens (human)0.35
Nuclear receptor ROR-gammaHomo sapiens (human)0.1995
10 kDa heat shock protein, mitochondrialHomo sapiens (human)5.3
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1Homo sapiens (human)0.82
60 kDa chaperonin Escherichia coli6.7
10 kDa chaperonin Escherichia coli6.7
Nuclear receptor ROR-betaHomo sapiens (human)0.1259

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Springer, DM1
Argüeso, P; Gipson, IK; Hori, Y; Russo, CL; Spurr-Michaud, SJ1

Reviews

1 review(s) available for varespladib and tretinoin

ArticleYear
An update on inhibitors of human 14 kDa Type II s-PLA2 in development.
    Current pharmaceutical design, 2001, Volume: 7, Issue:3

    Topics: Acetates; Animals; Anti-Inflammatory Agents, Non-Steroidal; Drug Design; Group II Phospholipases A2; Humans; Indoles; Keto Acids; Molecular Structure; Patents as Topic; Phospholipases A; Phospholipases A2; Sulfonamides; Tretinoin

2001

Other Studies

1 other study(ies) available for varespladib and tretinoin

ArticleYear
Effect of retinoic acid on gene expression in human conjunctival epithelium: secretory phospholipase A2 mediates retinoic acid induction of MUC16.
    Investigative ophthalmology & visual science, 2005, Volume: 46, Issue:11

    Topics: Acetates; Aristolochic Acids; Blotting, Western; CA-125 Antigen; Cell Line; Conjunctiva; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Epithelial Cells; Epithelium; Gene Expression Profiling; Gene Expression Regulation; Humans; Indoles; Keto Acids; Membrane Proteins; Oligonucleotide Array Sequence Analysis; Phospholipases A; Phospholipases A2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tretinoin; Up-Regulation

2005