vanadates has been researched along with verapamil in 54 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 12 (22.22) | 18.7374 |
1990's | 22 (40.74) | 18.2507 |
2000's | 16 (29.63) | 29.6817 |
2010's | 4 (7.41) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Daniel, JC; Lecerf, JM; Levy, SB; Slapak, CA | 1 |
Hertelendy, F; Molnár, M | 1 |
Casteels, R; Droogmans, G; Himpens, B; Missiaen, L | 1 |
Kasai, M; Muto, S | 1 |
Johnsson, R; Saris, NE | 1 |
Duhm, J; Engelmann, B | 1 |
Dhalla, NS; Tuana, BS | 1 |
Shimada, T; Shimamura, K; Sunano, S; Tsuji, A | 1 |
Ichida, S; Moriyama, K; Shimada, T; Shimamura, K; Sunano, S | 1 |
Kato, S; Moriyama, K; Shimamura, K; Sunano, S | 1 |
Shimada, T; Sunano, S | 1 |
Benabe, JE; Cruz-Soto, M; López-Novoa, JM; Martínez-Maldonado, M | 1 |
Goetz, KL; Hakumäki, MO; Sundet, WD; Wang, BC | 1 |
Benabe, JE; Cruz-Soto, MA; Martínez-Maldonado, M | 1 |
Benabe, JE; Martínez-Maldonado, M | 1 |
Akera, T; Takeda, K; Temma, K | 1 |
Antón, M; Cortijo, J; Morcillo, E; Santamaría, P; Villagrasa, V | 1 |
Futai, M; Manabe, T; Moriyama, Y; Tashiro, Y; Yoshimori, T | 1 |
Bryant, HJ; Iwasa, KH; Kowtha, VC; Krauthamer, V; Stenger, DA | 1 |
Dhalla, NS; Foerster, DR; Matsubara, T; Shah, KR; Xu, YJ | 1 |
Fox, MH; He, L | 1 |
Bakos, E; Goodfellow, HR; Higgins, CF; Müller, M; Sarkadi, B; Szabó, K; Váradi, A; Welker, E | 1 |
Litman, T; Skovsgaard, T; Stein, WD; Zeuthen, T | 1 |
Beck, WT; Dantzig, AH; Hsaio, SC; Pearce, HL; Shepard, RL; Winter, MA | 1 |
Rao, US | 1 |
Ashida, H; Oonishi, T; Uyesaka, N | 1 |
Baysal, F; Ogülener, N; Onder, S; Yaktubay, N | 1 |
Chakrabarti, P; Choudhuri, BS; Sen, S | 1 |
Herrmann, A; Lang, C; Marx, U; Nelson, H; Nelson, N; Polakowski, T; Pomorski, T | 1 |
Cheng, PW; Germann, UA; Gottesman, MM; Hrycyna, CA; Pastan, I; Ramachandra, M | 1 |
Breves, G; Schröder, B; Vössing, S | 1 |
Chen, KG; Cohen, D; Durán, GE; Lacayo, NJ; Sikic, BI | 1 |
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ | 1 |
Alvaro, D; Boyer, JL; Fraioli, F; Gigliozzi, A; Lee, J; Mennone, A; Sundaram, P | 1 |
Ambudkar, SV; Müller, M; Sauna, ZE; Smith, MM | 1 |
Hill, MA; Murphy, TV; Spurrell, BE | 1 |
Cosgrove, DJ; Spalding, EP | 1 |
Belyavskaya, NA; Tsarik, NP | 1 |
Hirsch-Ernst, KI; Kahl, GF; Rustenbeck, I; Ziemann, C | 1 |
Senior, AE; Tombline, G; Tyndall, GA; Urbatsch, IL | 1 |
Ahearn, GA; Chavez-Crooker, P; Garrido, N; Pozo, P | 1 |
Huda, MN; Kuroda, T; Lee, EW; Mizushima, T; Tsuchiya, T | 1 |
Grossmann, A; Hudson, FN; Kavanagh, TJ; Poot, M; Rabinovitch, PS | 1 |
Bartlett, MC; Clarke, DM; Loo, TW | 2 |
Baggetto, LG; Barakat, S; Coleman, AW; Dayan, G; Gayet, L; Labialle, S; Lazar, A; Oleinikov, V | 1 |
Arruebo, MP; Grasa, L; Murillo, MD; Plaza, MA | 1 |
Chattopadhyay, A; Dey, S; Fong, WF; Shen, XL; Wan, CK; Zhu, GY | 1 |
Charman, SA; Katneni, K; Porter, CJ | 1 |
Chen, YC; Lin, T; Nagpal, ML; Stocco, DM | 1 |
Baptista, BB; Farah, LS; Granado e Sá, M; Leite, VP; Zanotto, FP | 1 |
Leite, VP; Zanotto, FP | 1 |
Kaur, P; Li, W; Sharma, M | 1 |
Custódio, MR; Ortega, P; Zanotto, FP | 1 |
54 other study(ies) available for vanadates and verapamil
Article | Year |
---|---|
Energy-dependent accumulation of daunorubicin into subcellular compartments of human leukemia cells and cytoplasts.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Compartmentation; Chloroquine; Daunorubicin; Deoxyglucose; Dinitrophenols; Drug Interactions; Drug Resistance; Energy Metabolism; Ethylmaleimide; Humans; Leukemia; Membrane Glycoproteins; Methylamines; Microscopy, Fluorescence; Monensin; Ouabain; Sodium Azide; Tumor Cells, Cultured; Vanadates; Verapamil | 1992 |
Ca2+ release and InsP3 production in avian uterine cells: effects of PGF2 alpha and AVT.
Topics: Animals; Calcium; Chickens; Dinoprost; Female; In Vitro Techniques; Inositol; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Kinetics; Muscle, Smooth; Ruthenium Red; Uterus; Vanadates; Vasotocin; Verapamil | 1990 |
AlF4- induces Ca2+ oscillations in guinea-pig ileal smooth muscle.
Topics: Aluminum; Aluminum Compounds; Animals; Biological Transport, Active; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium-Transporting ATPases; Calmodulin; Cell Membrane; Cell Membrane Permeability; Electric Conductivity; Fluorides; Guinea Pigs; Ileum; Imidazoles; Muscle Contraction; Muscle, Smooth; Ryanodine; Vanadates; Verapamil | 1991 |
Ca2+ pump and Ca2+/H+ antiporter in plasma membrane vesicles isolated by aqueous two-phase partitioning from corn leaves.
Topics: Adenosine Triphosphate; Antiporters; Biological Transport, Active; Calcium Channels; Calcium-Binding Proteins; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cation Transport Proteins; Cell Membrane; Hydrogen-Ion Concentration; Lanthanum; Magnesium; Protons; Salts; Vanadates; Verapamil; Zea mays | 1990 |
Ca2+ influx in normal and spherocytic red cells.
Topics: Adult; Calcium; Chlorpromazine; Erythrocytes; Erythrocytes, Abnormal; Female; Humans; Ion Channels; Male; Middle Aged; Spherocytes; Spherocytosis, Hereditary; Splenectomy; Vanadates; Verapamil | 1988 |
Distinction of two components of passive Ca2+ transport into human erythrocytes by Ca2+ entry blockers.
Topics: Aminoquinolines; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane Permeability; Cobalt; Copper; Diltiazem; Erythrocyte Membrane; Flunarizine; Humans; Nifedipine; Vanadates; Verapamil | 1989 |
Solubilization of a divalent cation dependent ATPase from dog heart sarcolemma.
Topics: Adenosine Triphosphatases; Animals; Calcium; Cations, Divalent; Chromatography, Gel; Chromatography, Ion Exchange; Dogs; Heart Ventricles; Kinetics; Magnesium; Myocardium; Oligomycins; Ouabain; Sarcolemma; Solubility; Vanadates; Verapamil | 1987 |
Comparison of contractile effects of sodium vanadate and ouabain in vascular smooth muscles of guinea-pigs and rats.
Topics: Animals; Aorta; Basilar Artery; Guinea Pigs; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Ouabain; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Sodium-Potassium-Exchanging ATPase; Vanadates; Vanadium; Verapamil | 1986 |
Extra- and intracellular calcium in vanadate-induced contraction of vascular smooth muscle.
Topics: Animals; Body Fluids; Calcium; Culture Techniques; Dose-Response Relationship, Drug; Extracellular Space; Female; Guinea Pigs; Intracellular Fluid; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Rabbits; Vanadates; Verapamil | 1988 |
Effects of sodium vanadate on smooth muscles of guinea-pig ureter and their relation to extracellular Ca.
Topics: Animals; Calcium; Guinea Pigs; Humans; In Vitro Techniques; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Potassium; Ureter; Vanadates; Verapamil | 1987 |
Contraction independent of extracellular Ca by sodium vanadate in guinea-pig vas deferens.
Topics: Animals; Calcium; Calcium Channel Blockers; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium; Vanadates; Vanadium; Vas Deferens; Verapamil | 1985 |
Na+-K+-ATPase inhibitors and renin release: relationship to calcium.
Topics: Animals; Blood Pressure; Calcium; Dogs; Female; Glomerular Filtration Rate; Heart Rate; Ion Channels; Kidney; Kinetics; Male; Natriuresis; Ouabain; Renal Circulation; Renin; Sodium-Potassium-Exchanging ATPase; Vanadates; Vanadium; Verapamil | 1984 |
Cardiovascular and renin responses to vanadate in the conscious dog: attenuation after calcium channel blockade.
Topics: Animals; Blood Pressure; Cardiac Output; Dogs; Hemodynamics; Pulmonary Artery; Renin; Vanadates; Vanadium; Vascular Resistance; Vasopressins; Verapamil | 1984 |
Critical role of extracellular calcium in vanadate-induced renal vasoconstriction.
Topics: Animals; Calcium; Dogs; Drug Combinations; Egtazic Acid; Extracellular Space; Parathyroid Glands; Renal Circulation; Thyroidectomy; Time Factors; Trifluoperazine; Vanadates; Vanadium; Vasoconstriction; Verapamil | 1984 |
Importance of calcium in the renal hemodynamic changes induced by vanadate.
Topics: Animals; Calcium; Dogs; Kidney Function Tests; Parathyroid Glands; Potassium; Renal Circulation; Sodium; Thyroidectomy; Vanadates; Vanadium; Verapamil | 1984 |
Inotropic effects of vanadate in isolated rat and guinea-pig heart under conditions which modify calcium pools involved in contractile activation.
Topics: Animals; Calcium; Calcium Channel Blockers; Electric Stimulation; Male; Membrane Potentials; Myocardial Contraction; Rats; Rats, Inbred Strains; Ryanodine; Vanadates; Vanadium; Verapamil | 1982 |
Effects of vanadate on responses of guinea-pig isolated trachea to spasmogens.
Topics: Acetylcholine; Animals; Caffeine; Calcium; Cell Membrane; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Potassium Chloride; Serotonin; Trachea; Vanadates; Verapamil | 1993 |
ATP-dependent uptake of anti-neoplastic agents by acidic organelles.
Topics: Adenosine Triphosphate; Ammonium Chloride; Animals; Antineoplastic Agents; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cattle; Cells, Cultured; Chromaffin Granules; Daunorubicin; Drug Resistance; Hydrogen-Ion Concentration; Mice; Nigericin; Organelles; Proteolipids; Proton-Translocating ATPases; Quinidine; Reserpine; Valinomycin; Vanadates; Verapamil | 1994 |
Spontaneous firing of NG108-15 cells induced by transient exposure to ammonium chloride.
Topics: Amiloride; Ammonium Chloride; Animals; Cell Differentiation; Cell Membrane; Glioma; Hybrid Cells; Hydrogen-Ion Concentration; Kinetics; Membrane Potentials; Mice; Neuroblastoma; Ouabain; Rats; Tetrodotoxin; Time Factors; Vanadates; Verapamil | 1996 |
Mechanisms of inotropic responses of the isolated rat hearts to vanadate.
Topics: Amiloride; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Diuretics; Enzyme Inhibitors; Male; Myocardial Contraction; Ouabain; Perfusion; Rats; Rats, Sprague-Dawley; Ryanodine; Sodium-Potassium-Exchanging ATPase; Vanadates; Verapamil | 1995 |
Comparison of flow cytometry and western blotting to measure Hsp70.
Topics: Animals; Benzimidazoles; Blotting, Western; Carrier Proteins; Cell Cycle; CHO Cells; Cricetinae; Enzyme Inhibitors; Flow Cytometry; Fluorescent Dyes; Heat-Shock Proteins; Heating; HSC70 Heat-Shock Proteins; HSP70 Heat-Shock Proteins; HSP72 Heat-Shock Proteins; Protein Tyrosine Phosphatases; Vanadates; Verapamil | 1996 |
Phosphorylation site mutations in the human multidrug transporter modulate its drug-stimulated ATPase activity.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Baculoviridae; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Enzyme Activation; Humans; Mutation; Phosphorylation; Recombinant Proteins; Rhodamines; Serine; Spodoptera; Threonine; Vanadates; Verapamil; Vinblastine | 1997 |
Competitive, non-competitive and cooperative interactions between substrates of P-glycoprotein as measured by its ATPase activity.
Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; CHO Cells; Colchicine; Cricetinae; Daunorubicin; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Enzyme Activation; Gramicidin; Kinetics; Microsomes; Progesterone; Vanadates; Verapamil; Vinblastine | 1997 |
Effect of modulators on the ATPase activity and vanadate nucleotide trapping of human P-glycoprotein.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Calcium Channel Blockers; Cell Membrane; Drug Interactions; Drug Resistance, Multiple; Humans; Hydrolysis; Leukemia, Lymphoid; Phosphorus Radioisotopes; Protein Conformation; Stimulation, Chemical; Tumor Cells, Cultured; Vanadates; Verapamil; Vinblastine; Yohimbine | 1998 |
Drug binding and nucleotide hydrolyzability are essential requirements in the vanadate-induced inhibition of the human P-glycoprotein ATPase.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Catalysis; Enzyme Activation; Enzyme Stability; Humans; Hydrolysis; Ligands; Magnesium; Photoaffinity Labels; Receptors, Drug; Vanadates; Verapamil | 1998 |
Kinetic analysis of the mechanism of action of the multidrug transporter.
Topics: Adenosine Triphosphate; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Cell Membrane; Cells; Diffusion; Doxorubicin; Enzyme Activation; Extracellular Space; Humans; Intracellular Fluid; Models, Biological; Vanadates; Verapamil | 1998 |
Possible stimulation of Na+-K+-ATPase by NO produced from sodium nitrite by ultraviolet light in mouse gastric fundal strip.
Topics: Amiloride; Animals; Calcium; Female; Gastric Fundus; In Vitro Techniques; Male; Mice; Muscle Relaxation; Nitric Oxide; Ouabain; Sodium; Sodium Nitrite; Sodium-Potassium-Exchanging ATPase; Ultraviolet Rays; Vanadates; Verapamil | 1999 |
Isoniazid accumulation in Mycobacterium smegmatis is modulated by proton motive force-driven and ATP-dependent extrusion systems.
Topics: Adenosine Triphosphate; Antitubercular Agents; Biological Transport, Active; Calcium Channel Blockers; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Diltiazem; Drug Resistance, Microbial; Hydrogen-Ion Concentration; Ionophores; Isoniazid; Mycobacterium smegmatis; Nifedipine; Nigericin; Proton-Motive Force; Reserpine; Uncoupling Agents; Valinomycin; Vanadates; Verapamil | 1999 |
Rapid transbilayer movement of fluorescent phospholipid analogues in the plasma membrane of endocytosis-deficient yeast cells does not require the Drs2 protein.
Topics: 4-Chloro-7-nitrobenzofurazan; Adenosine Triphosphate; Biological Transport, Active; Calcium-Transporting ATPases; Cell Membrane; Endocytosis; Ethylmaleimide; Fluorescent Dyes; Fungal Proteins; Gene Deletion; Genes, Fungal; Lipid Bilayers; Liposomes; Mutation; Phosphatidylcholines; Phosphatidylserines; Phospholipids; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Vanadates; Verapamil | 1999 |
Both ATP sites of human P-glycoprotein are essential but not symmetric.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Motifs; Amino Acid Substitution; Antibodies, Monoclonal; Asparagine; Aspartic Acid; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Biological Transport; Body Temperature; Cell Membrane; Consensus Sequence; Enzyme Activation; Freezing; HeLa Cells; Humans; Peptide Fragments; Phosphorus Radioisotopes; Photoaffinity Labels; Point Mutation; Prazosin; Protein Conformation; Recombinant Fusion Proteins; Vanadates; Verapamil | 1999 |
In vitro studies on active calcium absorption from ovine rumen.
Topics: Absorption; Amiloride; Animals; Biological Transport; Butyrates; Calcium Channel Blockers; Calcium-Transporting ATPases; Calcium, Dietary; Diuretics; Electrophysiology; Epithelial Cells; Fatty Acids, Volatile; Female; Homeostasis; In Vitro Techniques; Lactation; Male; Prolactin; Rumen; Sheep; Sodium; Vanadates; Verapamil | 1999 |
Loss of cyclosporin and azidopine binding are associated with altered ATPase activity by a mutant P-glycoprotein with deleted phe(335).
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Calcium Channel Blockers; Cyclosporine; Dihydropyridines; Drug Interactions; Enzyme Activation; Humans; Molecular Sequence Data; Phenylalanine; Photoaffinity Labels; Tritium; Tumor Cells, Cultured; Vanadates; Verapamil | 2000 |
In vitro flow cytometry method to quantitatively assess inhibitors of P-glycoprotein.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B; Calcium Channel Blockers; Cell Survival; Cells, Cultured; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Microscopy, Fluorescence; Tumor Cells, Cultured; Vanadates; Verapamil | 2000 |
Molecular identification and functional characterization of Mdr1a in rat cholangiocytes.
Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Bile Ducts; Cell Division; Cell Membrane; Cytosol; Drug Resistance, Multiple; In Vitro Techniques; Isoquinolines; Kinetics; Male; Microscopy, Confocal; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Tetrahydroisoquinolines; Transcription, Genetic; Vanadates; Verapamil | 2000 |
Evidence for the vectorial nature of drug (substrate)-stimulated ATP hydrolysis by human P-glycoprotein.
Topics: Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Baculoviridae; Calcium Channel Blockers; Catalysis; Cell Line; Cell Membrane; Enzyme Inhibitors; Humans; Hydrolysis; Insecta; Kinetics; Models, Chemical; Protein Binding; Protein Conformation; Substrate Specificity; Vanadates; Verapamil | 2001 |
Tyrosine phosphorylation following alterations in arteriolar intraluminal pressure and wall tension.
Topics: Angiotensin II; Animals; Antibody Specificity; Arterioles; Blood Pressure; Calcium; Calcium Channel Blockers; Colforsin; Endothelium, Vascular; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Phosphorylation; Phosphotyrosine; Physical Stimulation; Rats; Rats, Sprague-Dawley; Tyrosine; Tyrphostins; Vanadates; Vasoconstriction; Vasodilator Agents; Verapamil | 2001 |
Mechanism of blue-light-induced plasma-membrane depolarization in etiolated cucumber hypocotyls.
Topics: Adenosine Triphosphate; Cell Membrane; Cucumis sativus; Egtazic Acid; Enzyme Activation; Hypocotyl; Ion Channels; Light; Membrane Potentials; Potassium Channel Blockers; Proton-Translocating ATPases; Tetraethylammonium; Tetraethylammonium Compounds; Vanadates; Verapamil | 1992 |
Calcium balance in pea root statocytes under both clinorotation and Ca2+ channel blockers' influence.
Topics: Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Gravitation; Nicardipine; Organelles; Pisum sativum; Plant Roots; Rotation; Vanadates; Verapamil | 1998 |
Inhibitors of mdr1-dependent transport activity delay accumulation of the mdr1 substrate rhodamine 123 in primary rat hepatocyte cultures.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Calcium Channel Blockers; Cyclosporine; Enzyme Inhibitors; Excipients; Fluorescent Dyes; Hepatocytes; Male; Octoxynol; Rats; Rats, Wistar; Rhodamine 123; Vanadates; Verapamil | 2001 |
P-glycoprotein catalytic mechanism: studies of the ADP-vanadate inhibited state.
Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Amino Acid Substitution; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Transporters; Catalysis; Catalytic Domain; Dimerization; Hydrolysis; Kinetics; Mice; Protein Conformation; Recombinant Proteins; Vanadates; Verapamil | 2003 |
Copper transport by lobster (Homarus americanus) hepatopancreatic lysosomes.
Topics: Animals; Biological Transport; Calcium; Copper; Fluorescence; Hepatopancreas; Lysosomes; Male; Models, Biological; Nephropidae; Vanadates; Verapamil | 2003 |
EfrAB, an ABC multidrug efflux pump in Enterococcus faecalis.
Topics: Acriflavine; Amino Acid Sequence; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Cloning, Molecular; DNA, Bacterial; Enterococcus faecalis; Fluorometry; Microbial Sensitivity Tests; Molecular Sequence Data; Vanadates; Verapamil | 2003 |
Probenicid inhibition of fluorescence extrusion after MCB-staining of rat-1 fibroblasts.
Topics: 3T3 Cells; Animals; Fibroblasts; Flow Cytometry; Glutathione Transferase; Histocytochemistry; Mice; Organic Anion Transporters, ATP-Dependent; Probenecid; Pyrazoles; Rats; Uricosuric Agents; Vanadates; Verapamil | 1996 |
Disulfide cross-linking analysis shows that transmembrane segments 5 and 8 of human P-glycoprotein are close together on the cytoplasmic side of the membrane.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Line; Cell Membrane; Cross-Linking Reagents; Cysteine; Cytoplasm; Disulfides; Electrophoresis, Polyacrylamide Gel; Gene Expression; Humans; Immunoblotting; Models, Molecular; Molecular Structure; Mutagenesis; Oxidation-Reduction; Structure-Activity Relationship; Transfection; Vanadates; Verapamil | 2004 |
Multidrug-resistant cancer cells contain two populations of P-glycoprotein with differently stimulated P-gp ATPase activities: evidence from atomic force microscopy and biochemical analysis.
Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Membrane; Cholesterol; Detergents; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Microscopy, Atomic Force; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Vanadates; Verapamil | 2005 |
Transmembrane segment 7 of human P-glycoprotein forms part of the drug-binding pocket.
Topics: Adenosine Triphosphatases; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Membrane; Cells, Cultured; Cross-Linking Reagents; Cysteine; Disulfides; Enzyme Activation; Humans; Mesylates; Models, Molecular; Molecular Sequence Data; Mutation; Protein Structure, Secondary; Substrate Specificity; Vanadates; Verapamil | 2006 |
The role of tyrosine kinase in prostaglandin E2 and vanadate-evoked contractions in rabbit duodenum in vitro.
Topics: Animals; Calcium; Carbachol; Dinoprostone; Dose-Response Relationship, Drug; Duodenum; Estrenes; Genistein; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle, Smooth; Phosphorylation; Protein-Tyrosine Kinases; Pyrrolidinones; Rabbits; Tyrosine; Tyrphostins; Vanadates; Verapamil | 2006 |
Gomisin A alters substrate interaction and reverses P-glycoprotein-mediated multidrug resistance in HepG2-DR cells.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Anticarcinogenic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Cell Line, Tumor; Cell Survival; Cyclooctanes; Dioxoles; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Humans; Hydrolysis; Lignans; Prazosin; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Vanadates; Verapamil; Vinblastine | 2006 |
Impact of cremophor-EL and polysorbate-80 on digoxin permeability across rat jejunum: delineation of thermodynamic and transporter related events using the reciprocal permeability approach.
Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Digoxin; Glycerol; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Jejunum; Male; Permeability; Polysorbates; Rats; Rats, Sprague-Dawley; Serous Membrane; Surface-Active Agents; Thermodynamics; Vanadates; Verapamil | 2007 |
Effects of genistein, resveratrol, and quercetin on steroidogenesis and proliferation of MA-10 mouse Leydig tumor cells.
Topics: Adenosine Triphosphatases; Animals; Calcium Channel Blockers; Cell Line, Tumor; Cell Proliferation; Cyclic AMP; Egtazic Acid; Estradiol; Fulvestrant; Genistein; Leydig Cells; Male; Mibefradil; Mice; Phosphoproteins; Phytoestrogens; Progesterone; Quercetin; Receptors, Estrogen; Resveratrol; RNA, Messenger; Stilbenes; Stimulation, Chemical; Vanadates; Verapamil | 2007 |
Calcium transport and homeostasis in gill cells of a freshwater crab Dilocarcinus pagei.
Topics: Amiloride; Animals; Biological Transport; Brachyura; Caffeine; Calcium; Calcium Channel Blockers; Cells, Cultured; Epithelial Cells; Gills; Homeostasis; Kinetics; Nifedipine; Ouabain; Sodium; Sodium-Calcium Exchanger; Thiourea; Vanadates; Verapamil | 2010 |
Calcium transport in gill cells of Ucides cordatus, a mangrove crab living in variable salinity environments.
Topics: Animals; Arthropod Proteins; Brachyura; Calcium; Calcium Channel Blockers; Calcium Channels; Gills; Kinetics; Salinity; Salt Tolerance; Vanadates; Verapamil; Wetlands | 2013 |
The DrrAB efflux system of Streptomyces peucetius is a multidrug transporter of broad substrate specificity.
Topics: Amino Acid Sequence; ATP-Binding Cassette Transporters; Bacterial Proteins; Biological Transport; Daunorubicin; Doxorubicin; Kinetics; Molecular Sequence Data; Multidrug Resistance-Associated Proteins; Mutation; Rifampin; Sequence Homology, Amino Acid; Streptomyces; Vanadates; Verapamil; Vinblastine | 2014 |
Characterization of cadmium plasma membrane transport in gills of a mangrove crab Ucides cordatus.
Topics: Animals; Biological Transport; Brachyura; Cadmium; Caffeine; Calcium; Calcium Channel Blockers; Cell Membrane; Cell Survival; Chelating Agents; Egtazic Acid; Fluorescence; Fluorescent Dyes; Gills; Ion Transport; Nimodipine; Vanadates; Verapamil; Water Pollutants, Chemical | 2014 |