valine and oxadiazoles

valine has been researched along with oxadiazoles in 55 studies

Research

Studies (55)

TimeframeStudies, this research(%)All Research%
pre-199041 (74.55)18.7374
1990's2 (3.64)18.2507
2000's2 (3.64)29.6817
2010's10 (18.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brugger, F; Fagg, GE; Olpe, HR; Pozza, MF1
Aanonsen, LM; Wilcox, GL1
Fischbach, GD; O'Brien, RJ1
Cherubini, E; King, AE; Nistri, A1
Christensen, BN; O'Dell, TJ1
Buckley, KS; Collins, GG1
Brugger, F; Olpe, HR; Pozza, MF; Steinmann, MW1
Chapman, B; Miller, KD; Stryker, MP1
Akoev, GN; Andrianov, IuN; Bromm, B; Sabo, T; Sherman, NO1
Miyachi, E; Murakami, M1
King, AE; Nistri, A; Rovira, C1
Lodge, D; Martin, D1
Hablitz, JJ1
Martin, MR1
Baudry, M; Cummins, JT; Kessler, M; Lynch, G; Way, S1
Curry, K; Magnuson, DS; McLennan, H; Peet, MJ1
Gregersen, H; McLennan, H; Peet, MJ1
Koerner, JF; Marks, RL; Robinson, MB; Whittemore, ER1
King, AE; Nistri, A1
Costa, E; Nicoletti, F; Wroblewski, JT1
Ballanyi, K; Endres, W; Grafe, P; Serve, G1
Cherniack, NS; Mitra, J; Overholt, JL; Prabhakar, NR1
Crepel, F; Dupont, JL; Gardette, R1
Drejer, J; Honoré, T; Schousboe, A1
Bockaert, J; Kemp, DE; Schmidt, BH; Sebben, M; Sladeczek, F; Weiss, S1
Choi, DW; Koh, JY; Peters, S1
Chang, HS; Kano, M; Kato, M1
Kihara, M; Kubo, T1
Carter, CJ; L'Heureux, R; Scatton, B1
Nishizaki, T; Okada, Y1
Dingledine, R; Verdoorn, TA1
King, AE; Thompson, SW; Urban, L; Woolf, CJ1
Astier, H; Tapia-Arancibia, L1
Raigorodsky, G; Urca, G1
Lovinger, DM; Weight, FF1
Lauritzen, M; Nicholson, C; Okada, Y; Rice, ME1
McLennan, H2
Collingridge, GL; Kehl, SJ; McLennan, H1
Crunelli, V; Forda, S; Kelly, JS1
Joëls, M; Urban, IJ1
Mayer, ML; Westbrook, GL1
Jin, D; Miyahara, T; Murofushi, S; Nagakura, K; Toyo'oka, T1
Crump, CE; Hayden, FG; Kaiser, L1
Turner, RB1
Bakris, GL; Cao, C; Kupfer, S; Perez, A; Sica, D; Weber, MA; White, WB1
Bakris, GL; Cao, C; Handley, A; Kupfer, S; Perez, A; Sica, D; Weber, MA; White, WB1
Chono, K; Katsumata, K; Kontani, T; Shimizu, Y; Sudo, K; Suzuki, H1
Ho, C; Kajiya, T; Kurtz, TW; Vilardi, R; Wang, J1
Dhadda, S; Rorig, R; Takenouchi, K; Tyring, S; Wald, A; Zadeikis, N1
Arnold, ME; Aubry, AF; Bifano, M; Burrell, R; Dockens, R; Easter, J; Gu, H; Jiang, H; Wang, J; Wang, JS; Zeng, J1
Haruki, T; Inoue, Y; Kandori, M; Miyazaki, D; Sasaki, S; Suzuki, H; Yakura, K; Yamamoto, Y1
Aguayo, E; Birkus, G; Cihlar, T; Jordan, R; Lee, G; Mello, C; Rodriguez, M1
Honda, M; Imafuku, S; Kato, T; Katsuramaki, T; Kawashima, M; Nakayama, J; Nemoto, O; Watanabe, D1
Lv, W; Wang, Y; Zhang, M; Zhang, Y1

Reviews

1 review(s) available for valine and oxadiazoles

ArticleYear
The treatment of rhinovirus infections: progress and potential.
    Antiviral research, 2001, Volume: 49, Issue:1

    Topics: 3C Viral Proteases; Antiviral Agents; Clinical Trials as Topic; Combined Modality Therapy; Common Cold; Cysteine Endopeptidases; Dietary Supplements; Drug Therapy, Combination; Echinacea; Enzyme Inhibitors; Histamine H1 Antagonists; Humans; Intercellular Adhesion Molecule-1; Isoxazoles; Oxadiazoles; Oxazoles; Phenylalanine; Phytotherapy; Picornaviridae Infections; Plant Extracts; Plants, Medicinal; Pyrrolidinones; Receptors, Virus; Rhinovirus; Valine; Viral Proteins; Zinc

2001

Trials

4 trial(s) available for valine and oxadiazoles

ArticleYear
Effects of the angiotensin receptor blocker azilsartan medoxomil versus olmesartan and valsartan on ambulatory and clinic blood pressure in patients with stages 1 and 2 hypertension.
    Hypertension (Dallas, Tex. : 1979), 2011, Volume: 57, Issue:3

    Topics: Adult; Aged; Analysis of Variance; Angiotensin II Type 1 Receptor Blockers; Antihypertensive Agents; Benzimidazoles; Blood Pressure; Blood Pressure Monitoring, Ambulatory; Double-Blind Method; Female; Humans; Hypertension; Imidazoles; Male; Middle Aged; Oxadiazoles; Tetrazoles; Treatment Outcome; Valine; Valsartan

2011
Comparison of the novel angiotensin II receptor blocker azilsartan medoxomil vs valsartan by ambulatory blood pressure monitoring.
    Journal of clinical hypertension (Greenwich, Conn.), 2011, Volume: 13, Issue:7

    Topics: Age Factors; Aged; Antihypertensive Agents; Benzimidazoles; Biological Availability; Blood Pressure; Blood Pressure Monitoring, Ambulatory; Dose-Response Relationship, Drug; Double-Blind Method; Drug Monitoring; Drug-Related Side Effects and Adverse Reactions; Female; Humans; Hypertension; Male; Middle Aged; Oxadiazoles; Sex Factors; Tetrazoles; Treatment Outcome; Valine; Valsartan

2011
ASP2151 for the treatment of genital herpes: a randomized, double-blind, placebo- and valacyclovir-controlled, dose-finding study.
    The Journal of infectious diseases, 2012, Apr-01, Volume: 205, Issue:7

    Topics: Acyclovir; Adult; Antiviral Agents; Double-Blind Method; Female; Herpes Genitalis; Humans; Male; Middle Aged; Oxadiazoles; Placebos; Treatment Outcome; Valacyclovir; Valine

2012
Amenamevir, a novel helicase-primase inhibitor, for treatment of herpes zoster: A randomized, double-blind, valaciclovir-controlled phase 3 study.
    The Journal of dermatology, 2017, Volume: 44, Issue:11

    Topics: Acyclovir; Aged; Antiviral Agents; Double-Blind Method; Female; Herpes Zoster; Humans; Male; Middle Aged; Oxadiazoles; Treatment Outcome; Valacyclovir; Valine

2017

Other Studies

50 other study(ies) available for valine and oxadiazoles

ArticleYear
Electrophysiological characterization of a novel potent and orally active NMDA receptor antagonist: CGP 37849 and its ethylester CGP 39551.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Behavior, Animal; Electrophysiology; Hippocampus; Iontophoresis; Male; Oxadiazoles; Piperazines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spinal Cord; Substantia Nigra; Valine

1990
Phencyclidine selectively blocks a spinal action of N-methyl-D-aspartate in mice.
    Neuroscience letters, 1986, Jun-18, Volume: 67, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Dipeptides; Drug Interactions; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Glutamates; Glutamic Acid; Injections, Spinal; Kainic Acid; Male; Mice; N-Methylaspartate; Norepinephrine; Oxadiazoles; Phencyclidine; Quisqualic Acid; Spinal Cord; Substance P; Tetrazoles; Valine

1986
Characterization of excitatory amino acid receptors expressed by embryonic chick motoneurons in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Cells, Cultured; Chick Embryo; Dose-Response Relationship, Drug; Electrophysiology; Excitatory Amino Acid Antagonists; Glutamates; In Vitro Techniques; Ion Channels; Kainic Acid; Membrane Potentials; Motor Neurons; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Receptors, Glutamate; Receptors, Neurotransmitter; Spinal Cord; Valine

1986
A study of amino acid-activated currents recorded from frog motoneurones in vitro.
    Neuroscience letters, 1987, May-06, Volume: 76, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anterior Horn Cells; Aspartic Acid; Glutamates; Glutamic Acid; In Vitro Techniques; Ion Channels; Membrane Potentials; Motor Neurons; N-Methylaspartate; Neural Conduction; Oxadiazoles; Quisqualic Acid; Rana temporaria; Valine

1987
Horizontal cells isolated from catfish retina contain two types of excitatory amino acid receptors.
    Journal of neurophysiology, 1989, Volume: 61, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Calcium; Cations, Divalent; Cell Membrane Permeability; Cells, Cultured; Concanavalin A; Convulsants; Glutamates; Ibotenic Acid; Ictaluridae; Ion Channels; Kainic Acid; Membrane Potentials; Oxadiazoles; Quisqualic Acid; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Retina; Valine; Zinc

1989
Antagonism of monosynaptic excitations in the mouse olfactory cortex slice by 6,7-dinitroquinoxaline-2,3-dione.
    Neuropharmacology, 1989, Volume: 28, Issue:10

    Topics: Animals; Aspartic Acid; Cerebral Cortex; In Vitro Techniques; Male; Mice; N-Methylaspartate; Oxadiazoles; Pyramidal Tracts; Quinoxalines; Quisqualic Acid; Receptors, AMPA; Receptors, Kainic Acid; Receptors, Neurotransmitter; Reflex, Monosynaptic; Synapses; Synaptic Transmission; Valine

1989
Excitatory amino acid receptors in rat locus coeruleus. An extracellular in vitro study.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Aspartic Acid; Glutamates; In Vitro Techniques; Kainic Acid; Locus Coeruleus; Magnesium; Male; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Amino Acid; Receptors, Cell Surface; Valine

1989
Visual responses in adult cat visual cortex depend on N-methyl-D-aspartate receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1989, Volume: 86, Issue:13

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Aspartic Acid; Cats; Electric Conductivity; Kainic Acid; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Valine; Visual Cortex; Visual Perception

1989
[Analysis of the effect of quisqualate, N-methyl-D- aspartate and several blockers of amino acid receptors on synaptic transmission in the ampullae of Lorenzini].
    Neirofiziologiia = Neurophysiology, 1989, Volume: 21, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Aminobutyrates; Animals; Aspartic Acid; Electric Fish; Evoked Potentials; Magnesium; Membrane Potentials; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Sensory Receptor Cells; Skates, Fish; Synapses; Synaptic Transmission; Valine

1989
Coexistence of NMDA and non-NMDA receptors on turtle horizontal cells revealed using isolated retina preparations.
    Vision research, 1989, Volume: 29, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Evoked Potentials, Visual; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Neuromuscular Depolarizing Agents; Oxadiazoles; Quisqualic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Retina; Turtles; Valine

1989
The excitation of frog motoneurones in vitro by the glutamate analogue, DI-alpha-amino-3-hydroxy-5-methyl-4-isoxazole-propionic acid (AMPA), and the effect of amino acid antagonists.
    Neuroscience letters, 1985, Mar-22, Volume: 55, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids, Dicarboxylic; Animals; Glutamates; Glutamic Acid; Ibotenic Acid; Membrane Potentials; Motor Neurons; Oxadiazoles; Oxazoles; Quisqualic Acid; Rana temporaria; Receptors, AMPA; Receptors, Drug; Spinal Cord; Synapses; Synaptic Transmission; Valine

1985
Ketamine acts as a non-competitive N-methyl-D-aspartate antagonist on frog spinal cord in vitro.
    Neuropharmacology, 1985, Volume: 24, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Kainic Acid; Ketamine; Magnesium; Motor Neurons; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rana pipiens; Rana temporaria; Spinal Cord; Valine

1985
Action of excitatory amino acids and their antagonists on hippocampal neurons.
    Cellular and molecular neurobiology, 1985, Volume: 5, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Amino Acids; Aminobutyrates; Animals; Aspartic Acid; Excitatory Amino Acid Antagonists; Glutamic Acid; Guinea Pigs; Hippocampus; Iontophoresis; Manganese; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Tetrodotoxin; Valine

1985
Evidence for an excitatory amino acid as the transmitter of the auditory nerve in the in vitro mouse cochlear nucleus.
    Hearing research, 1985, Volume: 20, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Action Potentials; Amino Acids; Animals; Aspartic Acid; Cochlear Nerve; Dose-Response Relationship, Drug; Evoked Potentials; Female; Kainic Acid; Male; Mice; Mice, Inbred C3H; N-Methylaspartate; Neurotransmitter Agents; Oxadiazoles; Pipecolic Acids; Quisqualic Acid; Receptors, Neurotransmitter; Valine; Vestibulocochlear Nerve

1985
Induction of glutamate binding sites in hippocampal membranes by transient exposure to high concentrations of glutamate or glutamate analogs.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1986, Volume: 6, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Aminobutyrates; Animals; Aspartic Acid; Binding Sites; Chlorides; Chromatography, High Pressure Liquid; Glutamates; Glutamic Acid; Hippocampus; Homocysteine; Kainic Acid; Kinetics; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rats; Receptors, Glutamate; Receptors, Neurotransmitter; Saponins; Sodium; Valine

1986
Ca2+-dependent depolarization and burst firing of rat CA1 pyramidal neurones induced by N-methyl-D-aspartic acid and quinolinic acid: antagonism by 2-amino-5-phosphonovaleric and kynurenic acids.
    Canadian journal of physiology and pharmacology, 1986, Volume: 64, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Aspartic Acid; Calcium; Convulsants; Electric Conductivity; Electric Stimulation; Evoked Potentials; Hippocampus; In Vitro Techniques; Kynurenic Acid; N-Methylaspartate; Neurons; Oxadiazoles; Pyramidal Tracts; Pyridines; Quinolinic Acid; Quinolinic Acids; Quisqualic Acid; Rats; Valine

1986
2-Amino-5-phosphonovalerate and Co2+ selectively block depolarization and burst firing of rat hippocampal CA1 pyramidal neurones by N-methyl-D-aspartate.
    Neuroscience, 1986, Volume: 17, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Aspartic Acid; Cobalt; Evoked Potentials; Hippocampus; Iontophoresis; N-Methylaspartate; Neurons; Oxadiazoles; Pyramidal Tracts; Quisqualic Acid; Rats; Tetrodotoxin; Valine

1986
Exposure of hippocampal slices to quisqualate sensitizes synaptic responses to phosphonate-containing analogues of glutamate.
    Brain research, 1986, Aug-27, Volume: 381, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Aminobutyrates; Animals; Evoked Potentials; Glutamates; Hippocampus; In Vitro Techniques; Male; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Stereoisomerism; Synapses; Valine

1986
Blockade by D-aminophosphonovalerate or Mg2+ of excitatory amino acid-induced responses on spinal motoneurons in vitro.
    Advances in experimental medicine and biology, 1986, Volume: 203

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Electric Conductivity; Excitatory Amino Acid Antagonists; In Vitro Techniques; Magnesium; Membrane Potentials; Motor Neurons; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rana temporaria; Synaptic Transmission; Valine

1986
Magnesium ions inhibit the stimulation of inositol phospholipid hydrolysis by endogenous excitatory amino acids in primary cultures of cerebellar granule cells.
    Journal of neurochemistry, 1987, Volume: 48, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Cells, Cultured; Cerebellum; Drug Synergism; Glutamates; Glutamic Acid; Hydrolysis; Inositol Phosphates; Kainic Acid; Magnesium; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rats; Sugar Phosphates; Valine; Veratridine

1987
Excitatory amino acids and intracellular pH in motoneurons of the isolated frog spinal cord.
    Neuroscience letters, 1986, Dec-03, Volume: 72, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anterior Horn Cells; Anura; Aspartic Acid; Hydrogen-Ion Concentration; In Vitro Techniques; Kainic Acid; Motor Neurons; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Valine

1986
Respiratory and vasomotor effects of excitatory amino acid on ventral medullary surface.
    Brain research bulletin, 1987, Volume: 18, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Animals; Apnea; Aspartic Acid; Blood Pressure; Carotid Sinus; Cats; Female; Glutamates; Kainic Acid; Male; Medulla Oblongata; N-Methylaspartate; Oxadiazoles; Phrenic Nerve; Quisqualic Acid; Respiration; Vagotomy; Valine; Vasomotor System

1987
Postnatal development of the chemosensitivity of rat cerebellar Purkinje cells to excitatory amino acids. An in vitro study.
    Brain research, 1987, Volume: 431, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Cerebellar Cortex; Glutamates; Glutamic Acid; In Vitro Techniques; N-Methylaspartate; Oxadiazoles; Purkinje Cells; Quisqualic Acid; Rats; Rats, Inbred Strains; Reaction Time; Valine

1987
Excitatory amino acid-induced release of 3H-GABA from cultured mouse cerebral cortex interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:9

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Binding Sites; Cerebral Cortex; gamma-Aminobutyric Acid; Kainic Acid; Mice; N-Methylaspartate; Neurons; Oxadiazoles; Potassium; Quisqualic Acid; Valine

1987
Dual action of excitatory amino acids on the metabolism of inositol phosphates in striatal neurons.
    Molecular pharmacology, 1987, Volume: 32, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Carbachol; Cells, Cultured; Corpus Striatum; Glutamates; Inositol Phosphates; Mice; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Sugar Phosphates; Valine

1987
Pharmacology of glutamate neurotoxicity in cortical cell culture: attenuation by NMDA antagonists.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1988, Volume: 8, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Cells, Cultured; Cerebral Cortex; Glutamates; Glutamic Acid; Isomerism; Kainic Acid; Mice; N-Methylaspartate; Neurons; Neurotoxins; Oxadiazoles; Quisqualic Acid; Valine

1988
The glutamate receptor subtype mediating parallel fibre-Purkinje cell transmission in rabbit cerebellar cortex.
    Neuroscience research, 1988, Volume: 5, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Cerebellar Cortex; Dipeptides; Glutamates; Kynurenic Acid; Oxadiazoles; Purkinje Cells; Quisqualic Acid; Rabbits; Receptors, Glutamate; Receptors, Neurotransmitter; Synaptic Transmission; Valine

1988
Evidence of N-methyl-D-aspartate receptor-mediated modulation of the aortic baroreceptor reflex in the rat nucleus tractus solitarii.
    Neuroscience letters, 1988, Apr-22, Volume: 87, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aorta; Blood Pressure; Glutamates; Glutamic Acid; Heart Rate; Kainic Acid; Male; Medulla Oblongata; Oxadiazoles; Pressoreceptors; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Valine

1988
Differential control by N-methyl-D-aspartate and kainate of striatal dopamine release in vivo: a trans-striatal dialysis study.
    Journal of neurochemistry, 1988, Volume: 51, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Atropine; Carbachol; Corpus Striatum; Dopamine; Kainic Acid; Male; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Tetrodotoxin; Valine

1988
Effects of excitatory amino acids on the oxygen consumption of hippocampal slices from the guinea pig.
    Brain research, 1988, Jun-14, Volume: 452, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Amino Acids; Animals; Aspartic Acid; Glutamates; Guinea Pigs; Hippocampus; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Oxadiazoles; Oxygen Consumption; Quisqualic Acid; Receptors, Amino Acid; Receptors, Cell Surface; Spider Venoms; Valine

1988
Excitatory amino acid receptors expressed in Xenopus oocytes: agonist pharmacology.
    Molecular pharmacology, 1988, Volume: 34, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Aspartic Acid; Chlorides; Female; Ibotenic Acid; Kainic Acid; Membrane Potentials; N-Methylaspartate; Oocytes; Oxadiazoles; Quisqualic Acid; Rats; Receptors, AMPA; Receptors, Drug; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Valine; Xenopus

1988
An intracellular analysis of amino acid induced excitations of deep dorsal horn neurones in the rat spinal cord slice.
    Neuroscience letters, 1988, Jul-08, Volume: 89, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Electrophysiology; Excitatory Amino Acid Antagonists; Glutamates; Glutamic Acid; In Vitro Techniques; Intracellular Membranes; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Rats; Spinal Cord; Tetrodotoxin; Valine

1988
Glutamate stimulates somatostatin release from diencephalic neurons in primary culture.
    Endocrinology, 1988, Volume: 123, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Cells, Cultured; Diencephalon; Glutamates; Glutamic Acid; Kainic Acid; Magnesium; N-Methylaspartate; Neurons; Oxadiazoles; Phencyclidine; Potassium; Quisqualic Acid; Rats; Somatostatin; Tetrodotoxin; Valine; Veratridine

1988
Behavioral classification of excitatory amino acid receptors in mouse spinal cord.
    European journal of pharmacology, 1988, Aug-24, Volume: 153, Issue:2-3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Behavior, Animal; Glutamates; Glutamic Acid; Glutamine; Kainic Acid; Male; Mice; Mice, Inbred ICR; N-Methylaspartate; Oxadiazoles; Quisqualic Acid; Receptors, Amino Acid; Receptors, Cell Surface; Spinal Cord; Valine

1988
Glutamate induces a depolarization of adult rat dorsal root ganglion neurons that is mediated predominantly by NMDA receptors.
    Neuroscience letters, 1988, Dec-05, Volume: 94, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Electrophysiology; Ganglia, Spinal; Glutamates; Glutamic Acid; Glycine; Kainic Acid; Magnesium; Neurons; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Valine

1988
Quisqualate, kainate and NMDA can initiate spreading depression in the turtle cerebellum.
    Brain research, 1988, Dec-20, Volume: 475, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Aspartic Acid; Cerebellum; Electric Stimulation; In Vitro Techniques; Kainic Acid; Magnesium; N-Methylaspartate; Neural Inhibition; Oxadiazoles; Quisqualic Acid; Turtles; Valine

1988
The isomers of 2-amino-5-phosphonovalerate as excitatory amino acid antagonists--a reappraisal.
    European journal of pharmacology, 1982, Apr-08, Volume: 79, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Amino Acids; Animals; Oxadiazoles; Quisqualic Acid; Rats; Spinal Cord; Stereoisomerism; Time Factors; Valine

1982
The antagonism of amino acid-induced excitations of rat hippocampal CA1 neurones in vitro.
    The Journal of physiology, 1983, Volume: 334

    Topics: 2-Amino-5-phosphonovalerate; 2-Aminoadipic Acid; Action Potentials; Amino Acids; Animals; Aspartic Acid; Dipeptides; Hippocampus; In Vitro Techniques; Kainic Acid; Male; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Rats; Valine

1983
Blockade of amino acid-induced depolarizations and inhibition of excitatory post-synaptic potentials in rat dentate gyrus.
    The Journal of physiology, 1983, Volume: 341

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Dipeptides; Evoked Potentials; Hippocampus; In Vitro Techniques; Kainic Acid; Membrane Potentials; N-Methylaspartate; Oxadiazoles; Pipecolic Acids; Quisqualic Acid; Rats; Synapses; Valine

1983
Amino acid neurotransmission between fimbria-fornix fibers and neurons in the lateral septum of the rat: a microiontophoretic study.
    Experimental neurology, 1984, Volume: 84, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Excitatory Amino Acid Antagonists; Glutamates; Hippocampus; Iontophoresis; Male; N-Methylaspartate; Nerve Fibers; Neural Pathways; Neuromuscular Junction; Oxadiazoles; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Amino Acid; Receptors, Cell Surface; Septal Nuclei; Synaptic Transmission; Valine

1984
A comparison of the effects of N-methyl-D-aspartate and quinolinate on central neurones of the rat.
    Neuroscience letters, 1984, May-04, Volume: 46, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Iontophoresis; Microinjections; N-Methylaspartate; Neurons; Oxadiazoles; Pyridines; Quinolinic Acid; Quinolinic Acids; Quisqualic Acid; Rats; Somatosensory Cortex; Spinal Cord; Stimulation, Chemical; Valine

1984
Mixed-agonist action of excitatory amino acids on mouse spinal cord neurones under voltage clamp.
    The Journal of physiology, 1984, Volume: 354

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Aspartic Acid; Culture Techniques; Electric Conductivity; Glutamates; Glutamic Acid; Homocysteine; Kainic Acid; Membrane Potentials; Mice; Mice, Inbred C57BL; N-Methylaspartate; Neurons; Oxadiazoles; Quisqualic Acid; Spinal Cord; Valine

1984
Total resolution of 17 DL-amino acids labelled with a fluorescent chiral reagent, R(-)-4-(3-isothiocyanatopyrrolidin-1-y1)-7-(N,N-dimethylaminosulfonyl)- 2,1,3-benzoxadiazole, by high-performance liquid chromatography.
    Journal of chromatography. A, 1998, Oct-02, Volume: 822, Issue:2

    Topics: Amino Acids; Chromatography, High Pressure Liquid; Fluorescent Dyes; Isothiocyanates; Mass Spectrometry; Oxadiazoles; Stereoisomerism; Valine; Yogurt

1998
In vitro activity of pleconaril and AG7088 against selected serotypes and clinical isolates of human rhinoviruses.
    Antiviral research, 2000, Volume: 47, Issue:3

    Topics: Antiviral Agents; Cell Survival; Cells, Cultured; Common Cold; Humans; Isoxazoles; Oxadiazoles; Oxazoles; Phenylalanine; Pyrrolidinones; Reverse Transcriptase Polymerase Chain Reaction; Rhinovirus; Spectrophotometry; Valine

2000
Effect of ASP2151, a herpesvirus helicase-primase inhibitor, in a guinea pig model of genital herpes.
    Molecules (Basel, Switzerland), 2011, Aug-25, Volume: 16, Issue:9

    Topics: Acyclovir; Animals; Antiviral Agents; Area Under Curve; DNA Helicases; DNA Primase; Drug Evaluation, Preclinical; Female; Guinea Pigs; Herpes Genitalis; Herpesvirus 1, Human; Herpesvirus 2, Human; Oxadiazoles; Valacyclovir; Valine; Viral Load; Viral Plaque Assay; Viral Proteins; Virus Shedding

2011
Molecular and cellular effects of azilsartan: a new generation angiotensin II receptor blocker.
    Journal of hypertension, 2011, Volume: 29, Issue:12

    Topics: 3T3 Cells; Adipocytes; Adipogenesis; Adiponectin; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Biomarkers; Cell Differentiation; Cell Proliferation; Complement Factor D; Gene Expression; Leptin; Mice; Oxadiazoles; PPAR alpha; PPAR delta; Tetrazoles; Valine; Valsartan

2011
Calculation and mitigation of isotopic interferences in liquid chromatography-mass spectrometry/mass spectrometry assays and its application in supporting microdose absolute bioavailability studies.
    Analytical chemistry, 2012, Jun-05, Volume: 84, Issue:11

    Topics: Biological Availability; Carbamates; Carbon Isotopes; Chromatography, Liquid; Flow Injection Analysis; Humans; Imidazoles; Nitrogen Isotopes; Oxadiazoles; Pyrrolidines; Reference Standards; Sulfonamides; Tandem Mass Spectrometry; Valine

2012
Efficacy of herpes virus helicase-primase inhibitor, ASP2151, for treating herpes simplex keratitis in mouse model.
    The British journal of ophthalmology, 2013, Volume: 97, Issue:4

    Topics: Acyclovir; Administration, Oral; Administration, Topical; Animals; Disease Models, Animal; DNA Helicases; DNA Primase; DNA, Viral; Herpesvirus 1, Human; Keratitis, Herpetic; Mice; Mice, Inbred BALB C; Oxadiazoles; Real-Time Polymerase Chain Reaction; Tears; Treatment Outcome; Valacyclovir; Valine; Viral Proteins

2013
Multiple classes of antiviral agents exhibit in vitro activity against human rhinovirus type C.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:3

    Topics: Antiviral Agents; Common Cold; Dose-Response Relationship, Drug; HeLa Cells; Humans; In Vitro Techniques; Isoxazoles; Oxadiazoles; Oxazoles; Phenylalanine; Piperidines; Pyridazines; Pyrrolidinones; Replicon; Rhinovirus; RNA, Viral; Tubercidin; Valine; Virus Replication

2014
Automated cell-based luminescence assay for profiling antiviral compound activity against enteroviruses.
    Scientific reports, 2019, 04-15, Volume: 9, Issue:1

    Topics: Animals; Antiviral Agents; Chlorocebus aethiops; Cytopathogenic Effect, Viral; Enterovirus; Enterovirus Infections; HeLa Cells; Humans; Isoxazoles; Luminescent Measurements; Microbial Sensitivity Tests; Oxadiazoles; Oxazoles; Phenylalanine; Pyrrolidinones; Valine; Vero Cells

2019