Page last updated: 2024-09-02

valerates and desipramine

valerates has been researched along with desipramine in 3 studies

Compound Research Comparison

Studies
(valerates)
Trials
(valerates)
Recent Studies (post-2010)
(valerates)
Studies
(desipramine)
Trials
(desipramine)
Recent Studies (post-2010) (desipramine)
2,2512944575,775487414

Protein Interaction Comparison

ProteinTaxonomyvalerates (IC50)desipramine (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)9.18
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)0.0003
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.35
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0034
Alpha-2B adrenergic receptorHomo sapiens (human)0.0003
Alpha-2C adrenergic receptorHomo sapiens (human)0.0003
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.35
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.0031
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 6Rattus norvegicus (Norway rat)0.35
Histamine H1 receptorRattus norvegicus (Norway rat)0.0008
Sodium-dependent serotonin transporterHomo sapiens (human)0.1961
5-hydroxytryptamine receptor 7 Rattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 5ARattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 5BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.35
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0003
Histamine H2 receptorCavia porcellus (domestic guinea pig)3.8
Sodium-dependent dopamine transporter Homo sapiens (human)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.4035
Sodium channel protein type 5 subunit alphaHomo sapiens (human)1.52
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.35
Solute carrier family 22 member 2Rattus norvegicus (Norway rat)10
TransporterRattus norvegicus (Norway rat)7.8

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19903 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Maxwell, DR; Sumpter, EA1
Iversen, LL; Johnston, GA1
Nakazawa, K1

Other Studies

3 other study(ies) available for valerates and desipramine

ArticleYear
A comparison of the actions of some drugs on decerebrate rigidity, muscle spindle activity and alpha-adrenoceptors.
    British journal of pharmacology, 1974, Volume: 50, Issue:3

    Topics: Animals; Blood Pressure; Cats; Chlorpromazine; Decerebrate State; Desipramine; Dimethylamines; Dose-Response Relationship, Drug; Methotrimeprazine; Muscle Rigidity; Muscle Spindles; Nictitating Membrane; Norepinephrine; Phenothiazines; Receptors, Adrenergic; Serotonin Antagonists; Structure-Activity Relationship; Valerates

1974
GABA uptake in rat central nervous system: comparison of uptake in slices and homogenates and the effects of some inhibitors.
    Journal of neurochemistry, 1971, Volume: 18, Issue:10

    Topics: Aminobutyrates; Animals; Caproates; Carnitine; Centrifugation, Density Gradient; Cerebellum; Cerebral Cortex; Chlorpromazine; Cysteamine; Desipramine; Dithiothreitol; Ethylmaleimide; Haloperidol; Hippocampus; Imipramine; Ornithine; Pimelic Acids; Propionates; Rats; Spinal Cord; Sulfanilamides; Synaptic Vesicles; Taurine; Tritium; Valerates

1971
Studies on the demethylation, hydroxylation and N-oxidation of imipramine in rat liver.
    Biochemical pharmacology, 1970, Volume: 19, Issue:4

    Topics: Amino Alcohols; Animals; Carbon Isotopes; Chlorides; Chromatography, Paper; Dealkylation; Desipramine; Ethylamines; Imipramine; Liver; Magnesium; Male; Metabolism; Methylation; Oxidation-Reduction; Oxides; Phenobarbital; Proadifen; Rats; Valerates

1970