Page last updated: 2024-09-02

valerates and apomorphine

valerates has been researched along with apomorphine in 3 studies

Compound Research Comparison

Studies
(valerates)
Trials
(valerates)
Recent Studies (post-2010)
(valerates)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
2,2512944579,205287780

Protein Interaction Comparison

ProteinTaxonomyvalerates (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19902 (66.67)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Maxwell, DR; Read, MA; Sumpter, EA1
Burghard, GL; Flanagan, TL; Green, H; Kaiser, C; Lester, BM; Swagzdis, JE; Zirkle, CL1
Fisher, R; Jackson, MJ; Jenner, P; Lees, AJ; Lincoln, L; Neumeyer, J; Rose, S; Sromek, AW1

Reviews

1 review(s) available for valerates and apomorphine

ArticleYear
Oral r-(-)-11-o-valeryl-n-n-propylnoraporphine reverses motor deficits in mptp-treated marmosets.
    Movement disorders : official journal of the Movement Disorder Society, 2016, Volume: 31, Issue:9

    Topics: Animals; Apomorphine; Aporphines; Behavior, Animal; Callithrix; Disease Models, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Female; Male; MPTP Poisoning; Valerates

2016

Other Studies

2 other study(ies) available for valerates and apomorphine

ArticleYear
Pharmacology of M & B 18,706, a drug which selectively reduces decerebrate rigidity.
    British journal of pharmacology, 1974, Volume: 50, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Apomorphine; Cats; Cerebellar Ataxia; Cerebellum; Chlorpromazine; Decerebrate State; Dextroamphetamine; Diazepam; Dimethylamines; Dogs; Electromyography; Ischemia; Locomotion; Muscle Relaxants, Central; Muscle Rigidity; Phenothiazines; Rats; Reflex; Spinal Cord; Tranquilizing Agents; Valerates

1974
Metabolism of diphenidol. Urinary products in humans and dogs.
    Journal of medicinal chemistry, 1972, Volume: 15, Issue:11

    Topics: Administration, Oral; Amino Acids; Animals; Antiemetics; Apomorphine; Butanols; Carbon Isotopes; Chromatography, Paper; Chromatography, Thin Layer; Dogs; Female; Glucuronates; Humans; Hydrolysis; Male; Piperidines; Valerates

1972