uridine has been researched along with thioinosine in 116 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 61 (52.59) | 18.7374 |
1990's | 31 (26.72) | 18.2507 |
2000's | 22 (18.97) | 29.6817 |
2010's | 2 (1.72) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Jakobs, ES; Lauzon, GJ; Paterson, AR; Weinstein, WM | 1 |
Bibi, O; Eilam, Y | 1 |
Cass, CE; Naik, SR; Paterson, AR | 1 |
Bibi, O; Cabantchik, ZI; Heichal, O; Katz, J | 1 |
Cabantchik, ZI; Eilam, Y | 1 |
Lauzon, GJ; Paterson, AR | 1 |
Bernard, O; Cass, CE; Kim, SC; Paterson, AR | 1 |
Cass, CE; Paterson, AR | 1 |
Hammond, JR; Jones, KW | 2 |
Aran, JM; Krafft, GA; Plagemann, PG; Ziemnicka-Merchant, B | 1 |
Doherty, AJ; Griffith, DA; Jarvis, SM | 1 |
Finney, KJ; Harris, AL; Ince, P; Moorghen, M; Watson, AJ | 1 |
Hammond, JR | 4 |
Gengenbacher, HM; Holstege, A; Hoppmann, J; Jehle, L | 1 |
al-Jaser, MH; Baer, HP; Ogbunude, PO | 1 |
Belt, JA; Crawford, CR; Ng, CY; Ullman, B | 1 |
Conant, AR; Griffith, DA; Jarvis, SM | 1 |
Cass, CE; Hodgson, KC; Hogue, DL | 1 |
Barrett, J; Beechey, RB; Harris, DI; Linstead, D | 1 |
Plagemann, PG; Woffendin, C | 5 |
Doherty, AJ; Griffith, DA; Jarvis, SM; Williams, TC | 1 |
Hammond, JR; Johnstone, RM | 1 |
Geiger, JD; Johnston, ME | 1 |
Belt, JA; Noel, LD | 2 |
Tse, CM; Wu, JS; Young, JD | 1 |
Belt, JA; Jarvis, SM; Paterson, AR; Wu, JS; Young, JD | 1 |
Jarvis, SM; Young, JD | 4 |
Baldwin, SA; Davies, A; Henderson, PJ; Kwong, FY; Tse, CM; Young, JD | 1 |
Jarvis, SM | 2 |
Jarvis, SM; Lee, CW | 1 |
Geiger, JD; Johnston, ME; Yago, V | 1 |
Darnowski, JW; Handschumacher, RE; Holdridge, C | 1 |
Choy, MY; Jarvis, SM; Kwong, FY; Tse, CM; Young, JD | 1 |
Jarvis, SM; Martin, BW | 1 |
Kraupp, M; Plagemann, PG | 1 |
Belt, JA; Gati, WP; Jakobs, ES; Jarvis, SM; Paterson, AR; Young, JD | 1 |
Abidi, TF; Plagemann, PG; Stollar, V; Woffendin, C | 1 |
Belt, JA; Jarvis, SM; Paterson, AR; Tse, CM; Wu, JS; Young, JD | 1 |
Plagemann, PG; Wohlhueter, RM | 2 |
Jarvis, SM; Martin, BW; Ng, AS | 1 |
Janmohamed, NS; Jarvis, SM; Young, JD | 1 |
Paterson, AR; Pickard, MA | 1 |
Gati, WP; Ogbunude, PO; Paterson, AR | 1 |
Kanner, N; Koren, R; Shohami, E | 1 |
Cass, CE; Dahlig-Harley, E; Eilam, Y; Paterson, AR | 1 |
Belt, JA | 2 |
Chen, SF; Parks, RE; Stoeckler, JD | 1 |
Henderson, JF; Moyer, JD; Paterson, AR | 1 |
Jarvis, SM; Kwong, FY; Wu, JS; Young, JD | 1 |
Cass, CE; Koren, R; Paterson, AR | 1 |
Janmohamed, SN; Jarvis, SM; Young, JD | 1 |
Lee, CM; Shi, MM; Wu, JS; Young, JD | 1 |
Ellory, JC; Fincham, DA; Jarvis, SM; Paterson, AR; Young, JD | 1 |
Wu, JS; Young, JD | 1 |
Jarvis, SM; Paterson, AR; Robins, MJ; Young, JD | 1 |
Clanachan, AS; Hammond, JR; Jarvis, SM; Paterson, AR | 3 |
Jarvis, SM; McBride, D; Young, JD | 1 |
Cass, CE; Dahlig, E; Lau, EY; Paterson, AR | 1 |
Sasvari-Szekely, M; Solymossy, M; Staub, M; Szikla, K | 1 |
Barankiewicz, J; Kossenjans, W; Rymaszewski, Z; Uyesaka, J | 1 |
Goh, LB; Lee, CW; Tu, Y | 1 |
Casillas, T; Delicado, EG; Miras-Portugal, MT; Sen, RP | 1 |
Lee, CW | 1 |
Doherty, AJ; Jarvis, SM | 1 |
Cass, CE; Guilbert, L; Meckling-Gill, KA | 1 |
Fujiwara, T; Iseki, K; Kobayashi, M; Miyazaki, K; Naasani, I; Sugawara, M | 1 |
Cass, CE; Fang, X; Mowles, DA; Parkinson, FE; Young, JD | 1 |
Cai, J; Lee, CW | 1 |
Goh, LB; Lee, CW | 1 |
Baldwin, SA; Boleti, H; Cass, CE; Coe, IR; Young, JD | 1 |
Abidi, F; Baldwin, SA; Cass, CE; Griffiths, M; Phillips, SE; Yao, SY; Young, JD | 1 |
Belt, JA; Crawford, CR; Naeve, C; Patel, DH | 1 |
Glue, P; Jarvis, SM; Thorn, JA | 1 |
Burke, T; Ferguson, PJ; Hammond, JR; Lee, S | 1 |
Detke, S | 1 |
Baldwin, SA; Cass, CE; Graham, KA; Hammond, JR; Mani, RS; Marjan, JM; Young, JD | 1 |
Bakken, AH; Lum, PY; Ngo, LY; Unadkat, JD | 1 |
Camarasa, J; Camins, A; Escubedo, E; Jiménez, A; Lladó, S; Pallàs, M; Pubill, D | 1 |
Baldwin, SA; Cass, CE; Hyde, RJ; McConkey, GA; McRobert, L; Parker, MD; Yao, SY; Young, JD | 1 |
Baldwin, SA; Carpenter, P; Cass, CE; Chen, XZ; Graham, K; Hyde, RJ; Karpinski, E; Loewen, SK; Mowles, DA; Ng, AM; Ritzel, MW; Ritzel, RG; Smith, KM; Yao, SY; Young, JD | 1 |
Baldwin, SA; Cass, CE; Chomey, EG; Sundaram, M; Yao, SY; Young, JD | 1 |
Ngo, LY; Patil, SD; Unadkat, JD | 1 |
Leung, GP; Tse, CM; Ward, JL; Wong, PY | 1 |
Baldwin, SA; Cass, CE; Ng, AM; Sundaram, M; Yao, SY; Young, JD | 1 |
Casado, FJ; del Santo, B; Felipe, A; Pastor-Anglada, M; Tarafa, G | 1 |
Baldwin, SA; Cass, CE; Ng, AM; Vickers, MF; Visser, F; Young, JD | 1 |
Baldwin, SA; Cass, CE; Duszyk, M; Man, SF; Ng, AM; Sawicka, J; Szkotak, AJ; Young, JD | 1 |
Bakken, AH; Lai, Y; Lum, PY; Schneider, G; SenGupta, DJ; Shubochkina, E; Unadkat, JD | 1 |
Ahmadi, B; Hammond, JR; Vyas, S | 1 |
Akaike, T; Kato, R; Maeda, T; Tamai, I | 2 |
Cass, CE; Clarke, ML; Damaraju, VL; Lang, T; Mowles, D; Smith, KM; Tackaberry, T; Tomkinson, B; Young, JD; Zhang, J | 1 |
Flanagan, SA; Meckling, KA | 1 |
Baldwin, SA; Barron, GM; Carpenter, P; Cass, CE; Damaraju, VL; Elwi, AN; Hunter, C; Mackey, JR; Santos, C; Sawyer, MB; Sun, X; Young, JD | 1 |
Nagata, K; Nakahata, N; Ohkubo, S | 1 |
Djuricic, B; Markovic, I; Redzic, Z; Segal, M | 1 |
Burdziński, G; Filipiak, P; Gdaniec, Z; Hug, GL; Pedzinski, T; Wenska, G | 1 |
Kimura, E; Nagai, J; Suzuki, S; Takano, M; Yumoto, R | 1 |
Hosokawa, M; Iwakawa, S; Ueda, K | 1 |
1 review(s) available for uridine and thioinosine
Article | Year |
---|---|
Nucleoside transport in animal cells.
Topics: Animals; Biological Transport, Active; Diazepam; Dilazep; Dipyridamole; Erythrocyte Membrane; Erythrocytes; Humans; Inosine; Kinetics; Membrane Proteins; Models, Molecular; Nucleosides; Papaverine; Species Specificity; Thioinosine; Uridine | 1983 |
115 other study(ies) available for uridine and thioinosine
Article | Year |
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Drug sequence-dependent toxicity and small bowel mucosal injury in mice treated with low doses of 3-deazauridine and 1-beta-D-arabinofuranosylcytosine.
Topics: 3-Deazauridine; Animals; Cytarabine; Female; Intestinal Mucosa; Intestine, Small; Male; Mice; Thioinosine; Time Factors; Uridine | 1979 |
Distinct properties of uridine transport systems in growing, quiescent and serum-stimulated hamster embryo cells.
Topics: Animals; Biological Transport, Active; Blood; Cell Division; Cell Line; Cell Transformation, Neoplastic; Cricetinae; Kinetics; Methylcholanthrene; Phenylmercury Compounds; Thioinosine; Uridine | 1977 |
Inhibition of uridine uptake in HeLa cells by nitrobenzylthioinosine and related compounds.
Topics: Depression, Chemical; Diffusion; HeLa Cells; Humans; Inosine; Kinetics; Thioinosine; Time Factors; Uridine; Uridine Kinase | 1977 |
Nucleoside transport in mammalian cell membranes. III. Kinetic and chemical modification studies of cytosine-arabinoside and uridine transport in hamster cells in culture.
Topics: Affinity Labels; Biological Transport, Active; Cell Line; Cytarabine; Ethylmaleimide; Kinetics; Phenylmercury Compounds; Thioinosine; Uridine | 1978 |
Nucleoside transport in mammalian cell membranes: a specific inhibitory mechanism of high affinity probes.
Topics: Binding Sites; Binding, Competitive; Biological Transport, Active; Cell Line; Cell Membrane; Dextrans; Hydroxymercuribenzoates; Inosine; Kinetics; Models, Biological; Structure-Activity Relationship; Sulfhydryl Reagents; Thioinosine; Uridine | 1977 |
Binding of the nucleoside transport inhibitor nitrobenzylthioinosine to HeLa cells.
Topics: Binding Sites; Binding, Competitive; Biological Transport, Active; Depression, Chemical; Guanosine; HeLa Cells; Humans; In Vitro Techniques; Inosine; Kinetics; Thioinosine; Thionucleosides; Thymidine; Time Factors; Uridine | 1977 |
Transport of nucleosides.
Topics: Biological Transport, Active; Cell Division; Cell Membrane; HeLa Cells; Inosine; Kinetics; Nucleosides; Thioinosine; Thymidine; Time Factors; Uridine | 1975 |
Nitrobenzylthionionosine binding sites in the erythrocyte membrane.
Topics: Binding Sites; Binding, Competitive; Biological Transport, Active; Cell Membrane; Erythrocytes; Humans; Inosine; Kinetics; Nitrobenzenes; Pronase; Protein Binding; Thioinosine; Trypsin; Uridine | 1976 |
Heterogeneity of [3H]dipyridamole binding to CNS membranes: correlation with [3H]nitrobenzylthioinosine binding and [3H]uridine influx studies.
Topics: Animals; Biological Transport; Cerebral Cortex; Dipyridamole; Female; Filtration; Glass; Guinea Pigs; Male; Rabbits; Synaptosomes; Thioinosine; Tritium; Uridine | 1992 |
Effects of chemical modification of nitrobenzylthioinosine on its binding to high-affinity membrane binding sites and inhibition of nucleoside transport.
Topics: Animals; Binding Sites; Biological Transport; Cell Membrane; Erythrocyte Membrane; Formycins; Humans; Mice; Nucleosides; Rats; Structure-Activity Relationship; Thioinosine; Tumor Cells, Cultured; Uridine | 1992 |
Nucleoside transport in cultured LLC-PK1 epithelia.
Topics: Affinity Labels; Animals; Biological Transport; Cell Line; Dilazep; Epithelium; Kidney Cortex; Kidney Medulla; Kinetics; Microvilli; Nucleosides; Swine; Thioinosine; Uridine | 1992 |
Organ culture as a model for investigating the effects of antimetabolites and nucleoside transport inhibitors on rodent colonic mucosa.
Topics: Animals; Biological Transport; Colon; Dipyridamole; DNA; Hydroxyurea; Intestinal Mucosa; Male; Models, Biological; Nucleosides; Organ Culture Techniques; Pyrimidines; Rats; Rats, Inbred Strains; Thioinosine; Thymidine; Time Factors; Tritium; Uridine | 1991 |
Effect of membrane lipid composition on the functional activity of a reconstituted nucleoside transporter derived from Ehrlich ascites cells.
Topics: Animals; Biological Transport; Carcinoma, Ehrlich Tumor; Carrier Proteins; Cell Membrane; Kinetics; Membrane Lipids; Membrane Proteins; Mice; Nucleoside Transport Proteins; Phospholipids; Protein Binding; Proteolipids; Thioinosine; Uridine | 1991 |
Facilitated diffusion and sodium-dependent transport of purine and pyrimidine nucleosides in rat liver.
Topics: Animals; Biological Transport; Diffusion; Dipyridamole; In Vitro Techniques; Liver; Male; Nucleosides; Perfusion; Purine Nucleosides; Pyrimidine Nucleosides; Rats; Rats, Inbred Strains; Sodium; Thioinosine; Uridine | 1991 |
Leishmania donovani: characteristics of adenosine and inosine transporters in promastigotes of two different strains.
Topics: Adenosine; Animals; Biological Transport; Diffusion; Dilazep; Inosine; Kinetics; Leishmania donovani; Nucleosides; Thioinosine; Thymidine; Uridine | 1991 |
Identification and reconstitution of the nucleoside transporter of CEM human leukemia cells.
Topics: Affinity Labels; Biological Transport; Blood Proteins; Carrier Proteins; Erythrocyte Membrane; Glycoside Hydrolases; Humans; Kinetics; Leukemia, T-Cell; Mannosyl-Glycoprotein Endo-beta-N-Acetylglucosaminidase; Membrane Proteins; Molecular Weight; Nucleoside Transport Proteins; Phospholipids; Thioinosine; Tumor Cells, Cultured; Uridine | 1990 |
Differential inhibition of nucleoside transport systems in mammalian cells by a new series of compounds related to lidoflazine and mioflazine.
Topics: Affinity Labels; Animals; Biological Transport; Cardiovascular Agents; Cattle; Cells, Cultured; Erythrocytes; Humans; Kidney; Lidoflazine; Nucleosides; Piperazines; Placenta; Rabbits; Rats; Sodium; Thioinosine; Uridine | 1990 |
Effects of inhibition of N-linked glycosylation by tunicamycin on nucleoside transport polypeptides of L1210 leukemia cells.
Topics: Animals; Biological Transport; Carrier Proteins; Electrophoresis, Polyacrylamide Gel; Glycosylation; Leukemia L1210; Membrane Proteins; Nucleoside Transport Proteins; Nucleosides; Protein Binding; Thioinosine; Tumor Cells, Cultured; Tunicamycin; Uridine | 1990 |
Nucleoside uptake by Trichomonas vaginalis.
Topics: Adenosine; Animals; Binding, Competitive; Biological Transport; Carrier Proteins; Cytidine; Dilazep; DNA; Guanosine; Inosine; Kinetics; Nucleosides; RNA; Thioinosine; Thionucleosides; Thymidine; Trichomonas vaginalis; Uridine | 1988 |
Dideoxycytidine permeation and salvage by mouse leukemia cells and human erythrocytes.
Topics: Animals; Blood Proteins; Carrier Proteins; Dipyridamole; Erythrocytes; Humans; Hydroxyurea; Leukemia, Experimental; Membrane Proteins; Mice; Nucleoside Transport Proteins; Permeability; Solubility; Structure-Activity Relationship; Thioinosine; Uridine; Zalcitabine | 1989 |
Characterization of sodium-dependent and sodium-independent nucleoside transport systems in rabbit brush-border and basolateral plasma-membrane vesicles from the renal outer cortex.
Topics: Animals; Biological Transport; Cations, Monovalent; Cell Compartmentation; Cell Membrane; Glucose; In Vitro Techniques; Kidney Cortex; Kidney Tubules, Proximal; Microvilli; Nucleosides; Rabbits; Sodium; Thioinosine; Uridine; Valinomycin | 1989 |
Na+-dependent and -independent transport of uridine and its phosphorylation in mouse spleen cells.
Topics: Animals; Biological Transport; Carrier Proteins; Dipyridamole; In Vitro Techniques; Kinetics; Membrane Proteins; Mice; Nucleoside Transport Proteins; Nucleosides; Phosphorylation; Purines; Pyrimidines; Sodium; Spleen; Thioinosine; Uridine | 1989 |
Solubilization and reconstitution of a nucleoside-transport system from Ehrlich ascites-tumour cells.
Topics: Adenosine; Animals; Binding Sites; Biological Transport, Active; Carcinoma, Ehrlich Tumor; Cell Membrane; Dipyridamole; Erythrocyte Membrane; Glucosides; Humans; Mice; Thioinosine; Tumor Cells, Cultured; Uridine | 1989 |
Sodium-dependent uptake of nucleosides by dissociated brain cells from the rat.
Topics: Adenosine; Animals; Brain; Dilazep; Dipyridamole; Kinetics; Male; Nucleosides; Ouabain; Rats; Rats, Inbred Strains; Sodium; Thioinosine; Uridine | 1989 |
Isolation and characterization of a mutant of L1210 murine leukemia deficient in nitrobenzylthioinosine-insensitive nucleoside transport.
Topics: Animals; Biological Transport; Carrier Proteins; Cytarabine; Floxuridine; Inosine; Leukemia L1210; Membrane Proteins; Mice; Mutation; Nucleoside Transport Proteins; Nucleosides; Thioinosine; Thymidine; Tubercidin; Tumor Cells, Cultured; Uridine | 1988 |
Evidence for the asymmetrical binding of p-chloromercuriphenyl sulphonate to the human erythrocyte nucleoside transporter.
Topics: 4-Chloromercuribenzenesulfonate; Biological Transport, Active; Blood Proteins; Dithiothreitol; Erythrocyte Membrane; Guanosine; Humans; Membrane Proteins; Nucleoside Transport Proteins; Phenylmercury Compounds; Structure-Activity Relationship; Thioinosine; Thionucleosides; Uridine | 1985 |
Nucleoside transport in Walker 256 rat carcinosarcoma and S49 mouse lymphoma cells. Differences in sensitivity to nitrobenzylthioinosine and thiol reagents.
Topics: 4-Chloromercuribenzenesulfonate; Animals; Biological Transport; Carcinoma 256, Walker; Cell Line; Dipyridamole; Inosine; Kinetics; Lymphoma; Mice; Nucleosides; Rats; Sulfhydryl Compounds; Thioinosine; Uridine | 1985 |
Photoaffinity labeling of the human erythrocyte glucose transporter with 8-azidoadenosine.
Topics: Adenosine; Affinity Labels; Azides; Blood Proteins; Coformycin; Cytochalasin B; Dose-Response Relationship, Drug; Erythrocytes; Humans; Kinetics; Membrane Proteins; Molecular Weight; Monosaccharide Transport Proteins; Nucleoside Transport Proteins; Pentostatin; Phenylisopropyladenosine; Phloretin; Photochemistry; Receptors, Cell Surface; Receptors, Purinergic; Thioinosine; Uridine | 1986 |
Nucleoside transport in rat erythrocytes: two components with differences in sensitivity to inhibition by nitrobenzylthioinosine and p-chloromercuriphenyl sulfonate.
Topics: 4-Chloromercuribenzenesulfonate; Animals; Biological Transport; Dipyridamole; Erythrocyte Membrane; Erythrocytes; Inosine; Kinetics; Male; Phenylmercury Compounds; Rats; Rats, Inbred Strains; Thioinosine; Uridine | 1986 |
Purification of the human erythrocyte nucleoside transporter by immunoaffinity chromatography.
Topics: Antibodies, Monoclonal; Blood Proteins; Blotting, Western; Carrier Proteins; Chromatography, Affinity; Electrophoresis, Polyacrylamide Gel; Erythrocytes; Glucose; Humans; Membrane Proteins; Nucleoside Transport Proteins; Peptide Fragments; Protein Binding; Thioinosine; Uridine | 1988 |
Inhibition by nucleosides of glucose-transport activity in human erythrocytes.
Topics: Biological Transport; Cytochalasin B; Erythrocyte Membrane; Erythrocytes; Galactosemias; Glucose; Humans; Monosaccharide Transport Proteins; Nucleosides; Thioinosine; Thymidine; Uridine | 1988 |
Nucleoside transport in rat cerebral-cortical synaptosomes. Evidence for two types of nucleoside transporters.
Topics: Animals; Biological Transport; Cerebral Cortex; Dilazep; Dipyridamole; Male; Nucleosides; Rats; Rats, Inbred Strains; Synaptosomes; Thioinosine; Uridine | 1988 |
Species differences in sensitivity of nucleoside transport in erythrocytes and cultured cells to inhibition by nitrobenzylthioinosine, dipyridamole, dilazep and lidoflazine.
Topics: Animals; Azepines; Biological Transport; Carrier Proteins; Cells, Cultured; Dilazep; Dipyridamole; Erythrocytes; Humans; Inosine; Lidoflazine; Membrane Proteins; Nucleoside Transport Proteins; Piperazines; Species Specificity; Thioinosine; Uridine | 1988 |
Pharmacological characterization of rapidly accumulated adenosine by dissociated brain cells from adult rat.
Topics: Adenosine; Adenosine Monophosphate; Animals; Binding, Competitive; Brain; Dilazep; Dipyridamole; Inosine; Kinetics; Male; Rats; Rats, Inbred Strains; Serum Albumin, Bovine; Thioinosine; Uridine | 1988 |
Effects of Ca2+-channel antagonists on nucleoside and nucleobase transport in human erythrocytes and cultured mammalian cells.
Topics: Animals; Biological Transport; Calcium Channel Blockers; Cell Line; Erythrocytes; HeLa Cells; Humans; Leukemia P388; Lidoflazine; Liver Neoplasms, Experimental; Mice; Nucleosides; Rats; Species Specificity; Thioinosine; Uridine | 1987 |
Concentrative uridine transport by murine splenocytes: kinetics, substrate specificity, and sodium dependency.
Topics: Animals; Biological Transport, Active; Kinetics; Leukemia L1210; Mice; Mice, Inbred C57BL; Sodium; Spleen; Substrate Specificity; Thioinosine; Thymidine; Uridine | 1987 |
Nucleoside transporter of pig erythrocytes. Kinetic properties, isolation and reaction with nitrobenzylthioinosine and dipyridamole.
Topics: Affinity Labels; Animals; Biological Transport; Carbohydrates; Carrier Proteins; Dipyridamole; Electrophoresis, Polyacrylamide Gel; Erythrocytes; Humans; Inosine; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Photochemistry; Swine; Thioinosine; Uridine | 1987 |
Purification and reconstitution studies of the nucleoside transporter from pig erythrocytes.
Topics: Affinity Labels; Animals; Carrier Proteins; Chromatography, DEAE-Cellulose; Electrophoresis, Polyacrylamide Gel; Erythrocytes; Glucosides; Guanosine; Membrane Proteins; Molecular Weight; Nucleoside Transport Proteins; Photochemistry; Solubility; Swine; Thioinosine; Thionucleosides; Uridine | 1987 |
Effects of temperature on the transport of nucleosides in guinea pig erythrocytes.
Topics: Affinity Labels; Animals; Biological Transport; Carbon Radioisotopes; Erythrocytes; Guinea Pigs; Kinetics; Temperature; Thermodynamics; Thioinosine; Uridine | 1986 |
Inhibition of nucleoside and nucleobase transport and nitrobenzylthioinosine binding by dilazep and hexobendine.
Topics: Animals; Azepines; Benzoates; Biological Transport; Carbon Radioisotopes; Cell Line; Cricetinae; Cricetulus; Dilazep; Dipyridamole; Erythrocytes; Hexobendine; Humans; Hypoxanthine; Hypoxanthines; Inosine; Mice; Nucleosides; Rats; Thioinosine; Uridine | 1986 |
Nitrobenzylthioinosine-sensitive nucleoside transport system: mechanism of inhibition by dipyridamole.
Topics: Animals; Binding, Competitive; Dipyridamole; Erythrocytes; Female; Guinea Pigs; Humans; Inosine; Kinetics; Thioinosine; Uridine | 1986 |
Photoaffinity labelling of a nitrobenzylthioinosine-binding polypeptide from cultured Novikoff hepatoma cells.
Topics: Adenosine; Affinity Labels; Animals; Binding Sites; Biological Transport; Cell Membrane; Cells, Cultured; Dipyridamole; Electrophoresis, Polyacrylamide Gel; Inosine; Liver Neoplasms, Experimental; Neoplasm Proteins; Rats; Thioinosine; Uridine | 1986 |
Nucleoside and nucleobase transport and metabolism in wild type and nucleoside transport-deficient Aedes albopictus cells.
Topics: Adenine; Adenosine Triphosphate; Aedes; Animals; Biological Transport; Carrier Proteins; Hypoxanthine; Hypoxanthines; Kinetics; Membrane Proteins; Mutation; Nucleoside Transport Proteins; Nucleosides; Thioinosine; Thymidine; Uracil; Uridine | 1987 |
Reconstitution studies of the human erythrocyte nucleoside transporter.
Topics: Biological Transport, Active; Blood Proteins; Erythrocytes; Glucose; Guanosine; Humans; Membrane Proteins; Molecular Weight; Nucleoside Transport Proteins; Octoxynol; Phospholipids; Photolysis; Polyethylene Glycols; Sonication; Stereoisomerism; Thioinosine; Thionucleosides; Time Factors; Uridine | 1985 |
Nitrobenzylthioinosine-sensitive and -resistant nucleoside transport in normal and transformed rat cells.
Topics: Animals; Binding Sites; Biological Transport; Carcinoma 256, Walker; Dipyridamole; Inosine; Kidney; Liver; Liver Neoplasms, Experimental; Male; Mathematics; Nucleosides; Rats; Thioinosine; Uridine | 1985 |
2-Chloroadenosine, a permeant for the nucleoside transporter.
Topics: 2-Chloroadenosine; Adenine; Adenosine; Biological Transport; Blood Proteins; Carrier Proteins; Erythrocyte Membrane; Erythrocytes; Humans; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Thioinosine; Uridine | 1985 |
Proteolytic cleavage of [3H]nitrobenzylthioinosine-labelled nucleoside transporter in human erythrocytes.
Topics: Affinity Labels; Blood Proteins; Carrier Proteins; Chymotrypsin; Cytochalasin B; Erythrocyte Membrane; Humans; Membrane Proteins; Monosaccharide Transport Proteins; Nucleoside Transport Proteins; Thioinosine; Trypsin; Uridine | 1985 |
Use of 4-nitrobenzylthioinosine in the measurement of rates of nucleoside transport in human erythrocytes.
Topics: Biological Transport; Carbon Isotopes; Erythrocytes; Humans; Inosine; Kinetics; Methods; Nitrobenzenes; Nucleosides; Sulfides; Thioinosine; Uridine | 1972 |
Dephosphorylation of nitrobenzylthioinosine 5'-monophosphate by ecto 5'-nucleotidase of HeLa cells.
Topics: 5'-Nucleotidase; Animals; Binding Sites; Cell Membrane; Erythrocytes; HeLa Cells; Humans; Inosine; Kinetics; Male; Mice; Nucleotidases; Protein Binding; Thioinosine; Thionucleotides; Uridine | 1984 |
S-substituted derivatives of 6-mercaptopurine ribosides interact both with the transport and metabolic phosphorylation of uridine by virus-transformed hamster fibroblasts.
Topics: Animals; Cell Line; Cell Transformation, Viral; Cricetinae; Cytarabine; Deoxyglucose; Inosine; Kinetics; Mesocricetus; Phosphorylation; Sarcoma Viruses, Murine; Thioinosine; Uridine | 1980 |
Binding of nitrobenzylthioinosine to high-affinity sites on the nucleoside-transport mechanism of HeLa cells.
Topics: 4-Chloromercuribenzenesulfonate; Binding Sites; Biological Transport; Cell Membrane; Drug Synergism; Ethylmaleimide; HeLa Cells; Humans; Inosine; Kinetics; Nucleosides; Thioinosine; Uridine | 1981 |
Nucleoside translocation in sheep reticulocytes and fetal erythrocytes: a proposed model for the nucleoside transporter.
Topics: 4-Chloromercuribenzenesulfonate; Animals; Binding Sites; Biological Transport; Cell Membrane Permeability; Erythrocytes; Fetal Blood; Kinetics; Models, Biological; Nucleosides; Reticulocytes; Sheep; Thioinosine; Trypsin; Uridine | 1982 |
Nitrobenzylthioinosine-insensitive uridine transport in human lymphoblastoid and murine leukemia cells.
Topics: 4-Chloromercuribenzenesulfonate; Animals; Biological Transport, Active; Humans; In Vitro Techniques; Inosine; Leukemia L1210; Lymphocytes; Mice; Nucleosides; Thioinosine; Uridine | 1983 |
Heterogeneity of nucleoside transport in mammalian cells. Two types of transport activity in L1210 and other cultured neoplastic cells.
Topics: 4-Chloromercuribenzenesulfonate; Animals; Biological Transport; Cell Line; Diffusion; Dipyridamole; Leukemia L1210; Mice; Neoplasms, Experimental; Nucleosides; Rats; Thioinosine; Uridine | 1983 |
Transport of deoxycoformycin in human erythrocytes. Measurement by adenosine deaminase titration and radioisotope assays.
Topics: Adenosine Deaminase Inhibitors; Biological Transport; Coformycin; Dipyridamole; Erythrocytes; Humans; Kinetics; Nucleoside Deaminases; Nucleosides; Pentostatin; Ribonucleosides; Thioinosine; Tritium; Uridine | 1984 |
Effect of an inhibitor of nucleoside transport on the disposition of uridine in mice.
Topics: Animals; Biological Transport; Inosine; Liver; Mice; Mice, Inbred ICR; Nucleosides; Thioinosine; Tissue Distribution; Uridine | 1984 |
Identification of the erythrocyte nucleoside transporter as a band 4.5 polypeptide. Photoaffinity labeling studies using nitrobenzylthioinosine.
Topics: Affinity Labels; Blood Proteins; Carrier Proteins; Electrophoresis, Polyacrylamide Gel; Erythrocyte Membrane; Inosine; Kinetics; Membrane Proteins; Molecular Weight; Nucleoside Transport Proteins; Photolysis; Thioinosine; Uridine | 1983 |
The kinetics of dissociation of the inhibitor of nucleoside transport, nitrobenzylthioinosine, from the high-affinity binding sites of cultured hamster cells.
Topics: Animals; Binding Sites; Biological Transport; Cell Division; Cell Line; Cell Membrane; Cell Transformation, Viral; Clone Cells; Cricetinae; Dilazep; Fibroblasts; Inosine; Kinetics; Mesocricetus; Nucleosides; Thioinosine; Uridine | 1983 |
Kinetics of nitrobenzylthioinosine binding to the human erythrocyte nucleoside transporter.
Topics: Adenosine; Binding Sites; Carrier Proteins; Dipyridamole; Erythrocyte Membrane; Humans; In Vitro Techniques; Inosine; Kinetics; Models, Biological; Nucleosides; Protein Binding; Thioinosine; Uridine | 1983 |
Nucleoside transport. Photoaffinity labelling of high-affinity nitrobenzylthioinosine binding sites in rat and guinea pig lung.
Topics: Adenosine; Affinity Labels; Animals; Binding Sites; Biological Transport; Cell Membrane; Dipyridamole; Guinea Pigs; Inosine; Kinetics; Lung; Male; Nucleosides; Rats; Rats, Inbred Strains; Thioinosine; Uridine | 1984 |
Nucleoside transport in human erythrocytes. Nitrobenzylthioinosine binding and uridine transport activities have similar radiation target sizes.
Topics: Biological Transport; Dose-Response Relationship, Radiation; Erythrocyte Membrane; Freezing; Humans; Inosine; Kinetics; Thioinosine; Uridine | 1984 |
Nucleoside transport in cultured mammalian cells. Multiple forms with different sensitivity to inhibition by nitrobenzylthioinosine or hypoxanthine.
Topics: Animals; Biological Transport; Cell Line; Cricetinae; Cricetulus; Female; Hypoxanthine; Hypoxanthines; Inosine; Kinetics; L Cells; Leukemia L1210; Leukemia P388; Liver Neoplasms, Experimental; Lymphoma; Mice; Ovary; Rats; Thioinosine; Tritium; Uridine | 1984 |
Photoaffinity labelling of nucleoside-transport proteins in plasma membranes isolated from rat and guinea-pig liver.
Topics: Affinity Labels; Animals; Carrier Proteins; Cell Fractionation; Cell Membrane; Erythrocyte Membrane; Guinea Pigs; In Vitro Techniques; Liver; Male; Membrane Proteins; Nucleosides; Rats; Rats, Inbred Strains; Thioinosine; Uridine | 1984 |
Photoaffinity labeling of the human erythrocyte nucleoside transporter by N6-(p-Azidobenzyl)adenosine and nitrobenzylthioinosine. Evidence that the transporter is a band 4.5 polypeptide.
Topics: Affinity Labels; Azides; Dithiothreitol; Erythrocyte Membrane; Erythrocytes; Humans; Inosine; Nucleosides; Photochemistry; Thioinosine; Time Factors; Ultraviolet Rays; Uridine | 1983 |
Benzodiazepine inhibition of nucleoside transport in human erythrocytes.
Topics: Benzodiazepines; Binding, Competitive; Biological Transport; Erythrocytes; Humans; Kinetics; Thioinosine; Uridine | 1983 |
Nucleoside transport in human erythrocytes. A simple carrier with directional symmetry in fresh cells, but with directional asymmetry in cells from outdated blood.
Topics: Binding Sites; Biological Transport, Active; Blood Preservation; Erythrocytes; Humans; In Vitro Techniques; Kinetics; Thioinosine; Time Factors; Uridine | 1983 |
Erythrocyte nucleoside transport: asymmetrical binding of nitrobenzylthioinosine to nucleoside permeation sites.
Topics: Animals; Binding Sites; Binding, Competitive; Biological Transport; Cell Membrane Permeability; Deoxycytidine; Dipyridamole; Erythrocytes; Humans; Inosine; Kinetics; Nucleosides; Sheep; Thioinosine; Uridine | 1982 |
Species differences in nucleoside transport. A study of uridine transport and nitrobenzylthioinosine binding by mammalian erythrocytes.
Topics: Animals; Binding Sites; Biological Transport; Dogs; Erythrocytes; Guinea Pigs; Humans; In Vitro Techniques; Inosine; Kinetics; Mice; Rabbits; Rats; Species Specificity; Swine; Thioinosine; Uridine | 1982 |
A common basis for inhibition of nucleoside transport by dipyridamole and nitrobenzylthioinosine?
Topics: Binding, Competitive; Dipyridamole; HeLa Cells; Humans; Inosine; Lidoflazine; Nucleosides; Thioinosine; Uridine | 1980 |
Nucleoside transport in human and sheep erythrocytes. Evidence that nitrobenzylthioinosine binds specifically to functional nucleoside-transport sites.
Topics: Animals; Binding Sites; Biological Transport; Cell Membrane Permeability; Erythrocyte Membrane; Erythrocytes; Humans; In Vitro Techniques; Inosine; Kinetics; Nitrobenzenes; Nucleosides; Sheep; Thioinosine; Uridine | 1980 |
Nucleoside transport and metabolism in lymphocytes, polymorphonuclear cells and cerebral synaptosomes.
Topics: Adenosine; Animals; Biological Transport; Cerebral Cortex; Child; Deoxycytidine; Dilazep; Dipyridamole; DNA; Humans; Kinetics; Lymphocytes; Neutrophils; Nucleosides; Palatine Tonsil; Papaverine; Rats; Synaptosomes; Thioinosine; Thymidine; Uridine | 1994 |
Inhibition of nucleoside transport by reactive oxygen species in bovine heart microvascular endothelial cells.
Topics: Adenosine; Animals; Biological Transport; Cattle; Cell Line; Dipyridamole; Endothelium, Vascular; Heart; Hydrogen Peroxide; Hypochlorous Acid; Inosine; Kinetics; Nucleosides; Reactive Oxygen Species; Thioinosine; Uridine; Vitamin K | 1994 |
Sensitivity to inhibition by N-ethylmaleimide: a property of nitrobenzylthioinosine-sensitive equilibrative nucleoside transporter of murine myeloma cells.
Topics: Animals; Biological Transport; Carrier Proteins; Cell Line; Ethylmaleimide; Kinetics; Membrane Proteins; Mice; Nucleoside Transport Proteins; Thioinosine; Tumor Cells, Cultured; Uridine | 1995 |
Evidence that adenine nucleotides modulate nucleoside-transporter function. Characterization of uridine transport in chromaffin cells and plasma membrane vesicles.
Topics: Adenine Nucleotides; Adrenal Medulla; Affinity Labels; Animals; Biological Transport; Carrier Proteins; Cattle; Cell Membrane; Cells, Cultured; Dipyridamole; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Thioinosine; Uridine | 1994 |
Functional reconstitution of pharmacologically distinct subtypes of nucleoside transporters in liposomal membranes.
Topics: Animals; Carrier Proteins; Glucosides; Kinetics; Lipids; Liposomes; Male; Membrane Proteins; Mice; Nucleoside Transport Proteins; Thioinosine; Uridine | 1994 |
Decrease in equilibrative uridine transport during monocytic differentiation of HL-60 leukaemia: involvement of protein kinase C.
Topics: Affinity Labels; Alkaloids; Binding Sites; Biological Transport; Cell Differentiation; Dilazep; Dipyridamole; Humans; Kinetics; Leukemia; Monocytes; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Thioinosine; Thymidine; Tumor Cells, Cultured; Uracil; Uridine | 1994 |
Interaction of the mioflazine derivative R75231 with the nucleoside transporter: evidence for positive cooperativity.
Topics: Adenosine; Animals; Binding, Competitive; Carrier Proteins; Cerebral Cortex; Erythrocyte Membrane; Half-Life; Humans; In Vitro Techniques; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Piperazines; Rabbits; Synaptosomes; Thioinosine; Uridine | 1993 |
Na(+)-dependent and -independent uridine uptake in an established renal epithelial cell line, OK, from the opossum kidney.
Topics: Animals; Carrier Proteins; Cell Line; Cellular Senescence; Epithelium; Kidney Tubules, Proximal; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Opossums; Purine Nucleosides; Sodium; Thioinosine; Uridine | 1993 |
CSF-1 stimulates nucleoside transport in S1 macrophages.
Topics: 3-O-Methylglucose; Adenosine; Animals; Binding Sites; Biological Transport; Bone Marrow; Cell Division; Cell Line, Transformed; Diffusion; Kinetics; Macrophage Colony-Stimulating Factor; Macrophages; Methylglucosides; Mice; Nucleosides; S Phase; Thioinosine; Uridine | 1993 |
Transport mechanisms of nucleosides and the derivative, 6-mercaptopurine riboside across rate intestinal brush-border membranes.
Topics: Adenosine; Animals; Biological Transport; Carrier Proteins; Intestinal Mucosa; Intestine, Small; Kinetics; Male; Microvilli; Molecular Structure; Rats; Rats, Wistar; Sodium; Symporters; Thioinosine; Uridine | 1996 |
Functional characterization of a recombinant sodium-dependent nucleoside transporter with selectivity for pyrimidine nucleosides (cNT1rat) by transient expression in cultured mammalian cells.
Topics: Adenosine; Amino Acid Sequence; Animals; Base Sequence; Biological Transport; Carrier Proteins; Cells, Cultured; Dilazep; Dipyridamole; Genes, myc; Guanosine; Haplorhini; Intestines; Kidney; Membrane Transport Proteins; Molecular Sequence Data; Nucleosides; Pyrimidine Nucleosides; Rats; Recombinant Proteins; Thioinosine; Transfection; Uridine | 1996 |
Tamoxifen inhibits nitrobenzylthioinosine-sensitive equilibrative uridine transport in human MCF-7 breast cancer cells.
Topics: Animals; Breast Neoplasms; Carrier Proteins; Cells, Cultured; Humans; Kinetics; Membrane Proteins; Mice; Neoplasms; Nucleoside Transport Proteins; Nucleosides; Protein Binding; Sodium; Spleen; Tamoxifen; Thioinosine; Uridine | 1996 |
Enhancement of the functional stability of solubilized nucleoside transporters by substrates and inhibitors.
Topics: Adenosine; Animals; Binding Sites; Carrier Proteins; Membrane Proteins; Mice; Nucleoside Transport Proteins; Thioinosine; Uridine | 1997 |
Reduction of equilibrative nitrobenzylthioinosine-sensitive nucleoside transporter in tamoxifen-treated MCF-7 cells: an oestrogen-reversible phenomenon.
Topics: Binding Sites; Biological Transport; Breast Neoplasms; Carrier Proteins; Cell Division; Estradiol; Humans; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Protein Binding; Substrate Specificity; Tamoxifen; Thioinosine; Tumor Cells, Cultured; Uridine | 1997 |
Molecular identification of the equilibrative NBMPR-sensitive (es) nucleoside transporter and demonstration of an equilibrative NBMPR-insensitive (ei) transport activity in human erythroleukemia (K562) cells.
Topics: Adenosine; Affinity Labels; Binding Sites; Blotting, Northern; Carrier Proteins; Cell Division; Cell Line; DNA, Complementary; Electrophoresis, Polyacrylamide Gel; Erythrocytes; Gene Amplification; Humans; In Vitro Techniques; Leukemia, Erythroblastic, Acute; Membrane Proteins; Nucleoside Transport Proteins; Polymerase Chain Reaction; Protein Binding; Thioinosine; Thymidine; Tubercidin; Uridine | 1997 |
Molecular cloning and characterization of a nitrobenzylthioinosine-insensitive (ei) equilibrative nucleoside transporter from human placenta.
Topics: Adenosine; Amino Acid Sequence; Animals; Biological Transport; Cardiotonic Agents; Carrier Proteins; Cloning, Molecular; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Gene Expression; Humans; Kinetics; Membrane Proteins; Molecular Sequence Data; Nuclear Proteins; Nucleoside Transport Proteins; Oocytes; Placenta; RNA, Messenger; Sequence Alignment; Sequence Analysis, DNA; Thioinosine; Uridine; Vasodilator Agents; Xenopus | 1997 |
Cloning of the human equilibrative, nitrobenzylmercaptopurine riboside (NBMPR)-insensitive nucleoside transporter ei by functional expression in a transport-deficient cell line.
Topics: Affinity Labels; Amino Acid Sequence; Biological Transport; Carrier Proteins; Cloning, Molecular; Equilibrative-Nucleoside Transporter 2; Gene Expression; Humans; Membrane Proteins; Molecular Sequence Data; Nuclear Proteins; Nucleosides; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Thioinosine; Tumor Cells, Cultured; Uridine | 1998 |
Ribavirin uptake by human erythrocytes and the involvement of nitrobenzylthioinosine-sensitive (es)-nucleoside transporters.
Topics: Adenosine; Animals; Antiviral Agents; Carrier Proteins; Equilibrative-Nucleoside Transporter 2; Erythrocyte Membrane; Erythrocytes; Horses; Humans; In Vitro Techniques; Membrane Proteins; Ribavirin; Thioinosine; Uridine | 1998 |
Interaction of 2',2'-difluorodeoxycytidine (gemcitabine) and formycin B with the Na+-dependent and -independent nucleoside transporters of Ehrlich ascites tumor cells.
Topics: Animals; Antimetabolites, Antineoplastic; Carcinoma, Ehrlich Tumor; Carrier Proteins; Deoxycytidine; Formycins; Gemcitabine; Male; Membrane Proteins; Mice; Nucleoside Transport Proteins; Sodium; Thioinosine; Uridine | 1998 |
Cloning of the Candida albicans nucleoside transporter by complementation of nucleoside transport-deficient Saccharomyces.
Topics: Adenosine; Amino Acid Sequence; Base Sequence; Candida albicans; Carrier Proteins; Cloning, Molecular; Dipyridamole; Genetic Complementation Test; Guanosine; Membrane Proteins; Molecular Sequence Data; Nucleoside Transport Proteins; Purine Nucleosides; Saccharomyces cerevisiae; Substrate Specificity; Thioinosine; Uridine | 1998 |
Demonstration of equilibrative nucleoside transporters (hENT1 and hENT2) in nuclear envelopes of cultured human choriocarcinoma (BeWo) cells by functional reconstitution in proteoliposomes.
Topics: Affinity Labels; Binding Sites; Carrier Proteins; Cell Membrane; Cell Nucleus; Choriocarcinoma; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Humans; Membrane Proteins; Nuclear Envelope; Proteolipids; RNA, Messenger; Thioinosine; Tumor Cells, Cultured; Uridine | 1998 |
Human intestinal es nucleoside transporter: molecular characterization and nucleoside inhibitory profiles.
Topics: Animals; Carrier Proteins; Gene Library; Humans; Intestine, Small; Membrane Proteins; Nucleoside Transport Proteins; Nucleosides; Plasmids; Reverse Transcriptase Polymerase Chain Reaction; Thioinosine; Uridine; Xenopus laevis | 2000 |
Interaction of a series of draflazine analogues with equilibrative nucleoside transporters: species differences and transporter subtype selectivity.
Topics: Animals; Carcinoma, Ehrlich Tumor; Carrier Proteins; Cell Membrane; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Erythrocytes; Humans; In Vitro Techniques; Membrane Proteins; Mice; Piperazines; Radioligand Assay; Species Specificity; Thioinosine; Tumor Cells, Cultured; Uridine | 2000 |
Further characterization of an adenosine transport system in the mitochondrial fraction of rat testis.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Benzodiazepinones; Biological Transport; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Guanosine; Hexobendine; Hydrogen-Ion Concentration; Inosine; Isoquinolines; Kinetics; Male; Mitochondria; Osmolar Concentration; Phenylisopropyladenosine; Rats; Rats, Sprague-Dawley; Sodium; Subcellular Fractions; Temperature; Testis; Thioinosine; Thionucleosides; Time Factors; Tritium; Uridine | 2000 |
Identification of a nucleoside/nucleobase transporter from Plasmodium falciparum, a novel target for anti-malarial chemotherapy.
Topics: Adenine; Amino Acid Sequence; Animals; Antimalarials; Biological Transport; Blotting, Southern; Carrier Proteins; Cations; Cell Membrane; Cloning, Molecular; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Kinetics; Molecular Sequence Data; Nucleobase, Nucleoside, Nucleotide, and Nucleic Acid Transport Proteins; Nucleosides; Phylogeny; Piperazines; Plasmodium falciparum; Platelet Aggregation Inhibitors; Protein Structure, Secondary; Protozoan Proteins; Sequence Homology, Amino Acid; Substrate Specificity; Thioinosine; Time Factors; Uridine; Vasodilator Agents; Xenopus | 2000 |
Molecular identification and characterization of novel human and mouse concentrative Na+-nucleoside cotransporter proteins (hCNT3 and mCNT3) broadly selective for purine and pyrimidine nucleosides (system cib).
Topics: Amino Acid Sequence; Animals; Biological Transport; Carrier Proteins; Cell Differentiation; Dilazep; Dipyridamole; Electric Conductivity; Evolution, Molecular; HL-60 Cells; Humans; Membrane Transport Proteins; Mice; Models, Molecular; Molecular Sequence Data; Purine Nucleosides; Pyrimidine Nucleosides; Recombinant Proteins; Sequence Homology, Amino Acid; Sodium; Substrate Specificity; Symporters; Thioinosine; Uridine | 2001 |
Identification of Cys140 in helix 4 as an exofacial cysteine residue within the substrate-translocation channel of rat equilibrative nitrobenzylthioinosine (NBMPR)-insensitive nucleoside transporter rENT2.
Topics: Amino Acid Sequence; Animals; Carrier Proteins; Cysteine; Equilibrative Nucleoside Transport Proteins; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Kinetics; Molecular Sequence Data; Nucleoside Transport Proteins; Oocytes; Rats; Sequence Alignment; Thioinosine; Transcription, Genetic; Uridine; Xenopus | 2001 |
Ontogenic and longitudinal activity of Na(+)-nucleoside transporters in the human intestine.
Topics: Adult; Biological Transport; Carrier Proteins; Cell Membrane; Cytidine; Cytoplasmic Vesicles; Drug Design; Female; Fetus; Gene Expression Regulation, Developmental; Guanosine; Humans; Inosine; Intestine, Small; Male; Membrane Transport Proteins; Microvilli; Organ Specificity; Protein Isoforms; Sodium; Thioinosine; Uridine | 2001 |
Characterization of nucleoside transport systems in cultured rat epididymal epithelium.
Topics: Animals; Biological Transport; Carrier Proteins; Cells, Cultured; Epididymis; Epithelial Cells; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Guanosine; Male; Membrane Proteins; Membrane Transport Proteins; Nucleosides; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Sodium; Thioinosine; Thymidine; Tritium; Uridine | 2001 |
Equilibrative nucleoside transporters: mapping regions of interaction for the substrate analogue nitrobenzylthioinosine (NBMPR) using rat chimeric proteins.
Topics: Affinity Labels; Animals; Biological Transport; Carrier Proteins; Equilibrative Nucleoside Transport Proteins; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Oocytes; Peptide Mapping; Purine Nucleosides; Rats; Recombinant Fusion Proteins; Thioinosine; Uridine; Xenopus | 2001 |
Developmental regulation of the concentrative nucleoside transporters CNT1 and CNT2 in rat liver.
Topics: Animals; Animals, Newborn; Biological Transport, Active; Cell Differentiation; Dexamethasone; Embryonic and Fetal Development; Female; Fetus; Gene Expression Regulation, Developmental; Hepatocytes; In Vitro Techniques; Liver; Membrane Transport Modulators; Membrane Transport Proteins; Pregnancy; Rats; Rats, Wistar; RNA, Messenger; Thioinosine; Triiodothyronine; Uridine | 2001 |
Mutation of residue 33 of human equilibrative nucleoside transporters 1 and 2 alters sensitivity to inhibition of transport by dilazep and dipyridamole.
Topics: Amino Acid Sequence; Animals; Biological Transport; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Humans; Membrane Transport Proteins; Mice; Molecular Sequence Data; Mutagenesis, Site-Directed; Rats; Recombinant Proteins; Structure-Activity Relationship; Thioinosine; Uridine; Xenopus laevis | 2002 |
Regulation of K(+) current in human airway epithelial cells by exogenous and autocrine adenosine.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine; Affinity Labels; Amiloride; Autocrine Communication; Cell Line; Cell Polarity; Clotrimazole; Diuretics; Epithelial Cells; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Growth Inhibitors; Humans; Membrane Transport Proteins; Patch-Clamp Techniques; Potassium; Potassium Channels; Quinazolines; Receptors, Purinergic P1; Respiratory Mucosa; Theobromine; Thioinosine; Triazoles; Uridine; Xanthines | 2001 |
A single glycine mutation in the equilibrative nucleoside transporter gene, hENT1, alters nucleoside transport activity and sensitivity to nitrobenzylthioinosine.
Topics: Alanine; Animals; Biological Transport; Cell Line; Conserved Sequence; Dogs; Equilibrative Nucleoside Transporter 1; Genetic Vectors; Glycine; Guanosine; Humans; Inosine; Membrane Transport Modulators; Membrane Transport Proteins; Mutagenesis, Site-Directed; Point Mutation; Saccharomyces cerevisiae; Thioinosine; Thionucleotides; Transfection; Uridine | 2002 |
Complex effects of sulfhydryl reagents on ligand interactions with nucleoside transporters: evidence for multiple populations of ENT1 transporters with differential sensitivities to N-ethylmaleimide.
Topics: Adenosine; Animals; Binding Sites; Biological Transport; Carcinoma, Ehrlich Tumor; Carrier Proteins; Cell Membrane; Detergents; Dithiothreitol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Equilibrative Nucleoside Transporter 1; Erythrocytes; Ethylmaleimide; Humans; Kinetics; Ligands; Mice; Nucleoside Transport Proteins; Protein Binding; Protein Structure, Secondary; Protein Transport; Sulfhydryl Reagents; Thioinosine; Time Factors; Uridine | 2002 |
Nucleoside transport at the blood-testis barrier studied with primary-cultured sertoli cells.
Topics: Algorithms; Animals; Biological Transport, Active; Blood-Testis Barrier; Cell Line; Cells, Cultured; Kinetics; Male; Mice; Nucleosides; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA; Sertoli Cells; Sodium; Thioinosine; Uridine | 2005 |
Characterization of novel Na+-dependent nucleobase transport systems at the blood-testis barrier.
Topics: Adenine; Animals; Biological Transport; Blood-Testis Barrier; Cytosine; Guanine; Hypoxanthine; Kinetics; Male; Meglumine; Nucleobase Transport Proteins; Nucleoside Transport Proteins; Purine Nucleosides; Pyrimidine Nucleosides; Rats; Rats, Inbred Strains; Sertoli Cells; Sodium; Thioinosine; Thymine; Uracil; Uridine | 2006 |
The role of human nucleoside transporters in cellular uptake of 4'-thio-beta-D-arabinofuranosylcytosine and beta-D-arabinosylcytosine.
Topics: Animals; Arabinonucleosides; Biological Transport; Cell Line, Tumor; Cell Survival; Cytarabine; Cytidine; Dose-Response Relationship, Drug; Equilibrative-Nucleoside Transporter 2; Female; HeLa Cells; Humans; Membrane Potentials; Nucleoside Transport Proteins; Oocytes; Saccharomyces cerevisiae; Thioinosine; Transfection; Tritium; Uridine; Xenopus laevis | 2006 |
Nucleoside transporter expression and activity is regulated during granulocytic differentiation of NB4 cells in response to all-trans-retinoic acid.
Topics: Affinity Labels; Biological Transport; Cell Differentiation; Cell Membrane; Granulocytes; Guanosine; Humans; Kinetics; Leukemia, Promyelocytic, Acute; Neutrophils; Nucleoside Transport Proteins; Subcellular Fractions; Thioinosine; Tretinoin; Tumor Cells, Cultured; Uridine | 2007 |
Localization of broadly selective equilibrative and concentrative nucleoside transporters, hENT1 and hCNT3, in human kidney.
Topics: Antibodies, Monoclonal; Antibody Specificity; Biomarkers; Blotting, Western; Cells, Cultured; Equilibrative Nucleoside Transporter 1; Fluorescent Antibody Technique; Humans; Immunohistochemistry; Kidney; Kidney Tubules, Collecting; Kidney Tubules, Proximal; Kinetics; Loop of Henle; Membrane Transport Proteins; Membranes; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thioinosine; Uridine | 2007 |
Adenosine uptake-dependent C6 cell growth inhibition.
Topics: 5'-Nucleotidase; Adenine Nucleotides; Adenosine; Adenosine Deaminase; Adenosine Diphosphate; Adenosine Kinase; Adenosine Monophosphate; Animals; Brain Neoplasms; Cell Count; Cell Line, Tumor; Cell Proliferation; Cyclic AMP; Dipyridamole; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Glioma; Hydrolysis; Rats; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles; Thioinosine; Uridine | 2007 |
Kinetics of nucleoside uptake by the basolateral side of the sheep choroid plexus epithelium perfused in situ.
Topics: Adenosine; Animals; Cell Polarity; Cell Survival; Choroid Plexus; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Epithelial Cells; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Inosine; Kinetics; Membrane Transport Proteins; Models, Biological; Nucleoside Transport Proteins; Nucleosides; Perfusion; Sheep; Sodium; Thioinosine; Thymidine; Uridine | 2008 |
Photocycloaddition of the T1 excited state of thioinosine to uridine and adenosine.
Topics: Absorption; Acetylation; Adenosine; Oxygen; Photochemical Processes; Temperature; Thioinosine; Uridine | 2009 |
Human erythrocyte nucleoside transporter ENT1 functions at ice-cold temperatures.
Topics: Cold Temperature; Dose-Response Relationship, Drug; Equilibrative Nucleoside Transporter 1; Erythrocyte Membrane; Glucose Transporter Type 1; Humans; Ribavirin; Thioinosine; Uridine | 2010 |
Cellular Uptake of Decitabine by Equilibrative Nucleoside Transporters in HCT116 Cells.
Topics: Antimetabolites, Antineoplastic; Azacitidine; Carrier Proteins; Colorectal Neoplasms; Decitabine; DNA Methylation; Equilibrative Nucleoside Transporter 1; Gene Expression; HCT116 Cells; Humans; Melanoma-Specific Antigens; Real-Time Polymerase Chain Reaction; RNA, Messenger; Thioinosine; Uridine | 2015 |