urea and quinoxalines

urea has been researched along with quinoxalines in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19902 (16.67)18.7374
1990's2 (16.67)18.2507
2000's4 (33.33)29.6817
2010's2 (16.67)24.3611
2020's2 (16.67)2.80

Authors

AuthorsStudies
Ryley, JF; Wilson, RG1
Harkness, DR; Stadtman, ER1
Bauer, PM; Buga, GM; Fukuto, JM; Ignarro, LJ; Wei, LH1
Belonga, KL; Carter, DB; Im, HK; Im, WB; Jacobsen, EJ; Mickelson, JW; Petke, JD; Sethy, VH; Stelzer, LS; Tang, AH; TenBrink, RE; VonVoigtlander, PF; Zhong, WZ1
Brown, T; Bunton, D; MacDonald, A; McGrath, JC; Shaw, AM; Tracey, A1
Bohme, GA; Boireau, A; Damour, D; Debono, MW; Genevois-Borella, A; Imperato, A; Jimonet, P; Mignani, S; Pratt, J; Randle, JC; Ribeill, Y; Stutzmann, JM; Vuilhorgne, M1
Bonci, A; Borgland, SL; Fields, HL; Sarti, F; Taha, SA1
Li, J; Li, X; Qiu, B; Shen, J; Wang, X; Xiong, B; Zhang, L1
Bickle, QD; Cowan, N; Ingram-Sieber, K; Keiser, J; Mansour, NR; Panic, G; Spangenberg, T; Vargas, M; Wells, TN1
Anderson, MO; Cil, O; Diez-Cecilia, E; Lee, S; Verkman, AS1
Chen, MW; Li, X; Zhao, ZB; Zhao, ZK; Zhou, YG1
Contreras, JI; Ezell, EL; Garrison, JC; Kizhake, S; Mallareddy, JR; Napoleon, JV; Natarajan, A; Radhakrishnan, P; Rajesh, C; Rana, S; Sagar, S; Singh, S; Sonawane, YA1

Other Studies

12 other study(ies) available for urea and quinoxalines

ArticleYear
Comparative studies with anticoccidials and three species of chicken coccidia in vivo and in vitro.
    The Journal of parasitology, 1972, Volume: 58, Issue:4

    Topics: Amprolium; Animals; Antiprotozoal Agents; Benzoates; Chickens; Coccidiosis; Culture Techniques; Eimeria; Kidney; Niacinamide; Poultry Diseases; Quinolines; Quinoxalines; Urea

1972
Bacterial degradation of riboflavin. VI. Enzymatic conversion of riboflavin to 1-ribityl-2,3-diketo-1,2,3,4-tetrahydro-6, 7-dimethylquinoxaline, urea, and carbon dioxide.
    The Journal of biological chemistry, 1965, Volume: 240, Issue:10

    Topics: Ammonia; Biphenyl Compounds; Borates; Carbon Dioxide; Copper; Flavin Mononucleotide; Flavins; In Vitro Techniques; Kinetics; Mercury; Phenanthrolines; Pseudomonas; Quinoxalines; Riboflavin; Sulfites; Urea

1965
NG-hydroxy-L-arginine and nitric oxide inhibit Caco-2 tumor cell proliferation by distinct mechanisms.
    The American journal of physiology, 1998, Volume: 275, Issue:4

    Topics: Animals; Aorta; Arginase; Arginine; Caco-2 Cells; Cell Division; Coculture Techniques; DNA; Endothelium, Vascular; Humans; Nitric Oxide; Nitric Oxide Donors; Ornithine; Ornithine Decarboxylase; Oxadiazoles; Polyamines; Putrescine; Quinoxalines; Rats; Spermidine; Spermine; Thymidine; Triazenes; Urea

1998
Piperazine imidazo[1,5-a]quinoxaline ureas as high-affinity GABAA ligands of dual functionality.
    Journal of medicinal chemistry, 1999, Apr-08, Volume: 42, Issue:7

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Anxiety; Biological Availability; Cell Line; Cerebellum; Convulsants; Cyclic GMP; Drug Evaluation, Preclinical; GABA Agonists; Imidazoles; In Vitro Techniques; Ligands; Male; Mice; Models, Molecular; Molecular Conformation; Pentylenetetrazole; Piperazines; Quinoxalines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Structure-Activity Relationship; Urea

1999
5-hydroxytryptamine- and U46619-mediated vasoconstriction in bovine pulmonary conventional and supernumerary arteries: effect of endogenous nitric oxide.
    Clinical science (London, England : 1979), 2000, Volume: 98, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arteries; Cattle; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Lung; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Quinoxalines; Serotonin; Serotonin Antagonists; Urea; Vasoconstrictor Agents

2000
4,10-Dihydro-4-oxo-4H-imidazo[1,2-a]indeno[1,2-e]pyrazin-2-carboxylic acid derivatives: highly potent and selective AMPA receptors antagonists with in vivo activity.
    Bioorganic & medicinal chemistry letters, 2000, May-15, Volume: 10, Issue:10

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Drug Evaluation, Preclinical; Inhibitory Concentration 50; Isoquinolines; Mice; Mice, Inbred DBA; Pyrazines; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Tetrazoles; Urea

2000
Orexin A in the VTA is critical for the induction of synaptic plasticity and behavioral sensitization to cocaine.
    Neuron, 2006, Feb-16, Volume: 49, Issue:4

    Topics: Analysis of Variance; Anesthetics, Local; Animals; Animals, Newborn; Behavior, Animal; Benzoxazoles; Calcium Channel Blockers; Cocaine; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Immunohistochemistry; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Lysine; Male; Motor Activity; N-Methylaspartate; Naphthyridines; Neuronal Plasticity; Neurons; Neuropeptides; Orexins; Patch-Clamp Techniques; Protein Kinase C; Quinoxalines; Rats; Rats, Sprague-Dawley; Synapses; Thionucleotides; Time Factors; Tyrosine 3-Monooxygenase; Urea; Ventral Tegmental Area

2006
Quinoxalinylurea derivatives as a novel class of JSP-1 inhibitors.
    Bioorganic & medicinal chemistry letters, 2007, Apr-15, Volume: 17, Issue:8

    Topics: Allosteric Site; Dual-Specificity Phosphatases; Enzyme Inhibitors; Inhibitory Concentration 50; Mitogen-Activated Protein Kinase Phosphatases; Phosphoprotein Phosphatases; Protein Phosphatase 1; Protein Tyrosine Phosphatases; Quinoxalines; Structure-Activity Relationship; Urea

2007
Orally active antischistosomal early leads identified from the open access malaria box.
    PLoS neglected tropical diseases, 2014, Volume: 8, Issue:1

    Topics: Administration, Oral; Animals; Anthelmintics; Disease Models, Animal; Female; Inhibitory Concentration 50; Mice; Parasite Load; Parasitic Sensitivity Tests; Quinoxalines; Schistosoma mansoni; Schistosomiasis mansoni; Urea

2014
Nanomolar-Potency 1,2,4-Triazoloquinoxaline Inhibitors of the Kidney Urea Transporter UT-A1.
    Journal of medicinal chemistry, 2018, 04-12, Volume: 61, Issue:7

    Topics: Animals; Diuresis; Diuretics; Dogs; Humans; Kidney; Madin Darby Canine Kidney Cells; Male; Membrane Transport Proteins; Models, Molecular; Molecular Conformation; Molecular Docking Simulation; Osmolar Concentration; Quinoxalines; Rats; Rats, Wistar; Structure-Activity Relationship; Urea; Urea Transporters

2018
Biomimetic asymmetric reduction of benzoxazinones and quinoxalinones using ureas as transfer catalysts.
    Chemical communications (Cambridge, England), 2020, Jul-07, Volume: 56, Issue:53

    Topics: Benzoxazines; Biomimetic Materials; Catalysis; Cell Cycle Proteins; Coordination Complexes; Hydrogen Bonding; Models, Chemical; Molecular Conformation; NAD; Niacinamide; Oxidation-Reduction; Quinoxalines; Ruthenium; Substrate Specificity; Transcription Factors; Urea

2020
Structure activity relationship (SAR) study identifies a quinoxaline urea analog that modulates IKKβ phosphorylation for pancreatic cancer therapy.
    European journal of medicinal chemistry, 2021, Oct-15, Volume: 222

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; I-kappa B Kinase; Mice; Molecular Structure; Pancreatic Neoplasms; Phosphorylation; Protein Kinase Inhibitors; Quinoxalines; Structure-Activity Relationship; Urea

2021