uracil and floxuridine

uracil has been researched along with floxuridine in 132 studies

Research

Studies (132)

TimeframeStudies, this research(%)All Research%
pre-199071 (53.79)18.7374
1990's25 (18.94)18.2507
2000's24 (18.18)29.6817
2010's11 (8.33)24.3611
2020's1 (0.76)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Forsthoefel, PF; Williams, ML1
Moffatt, JG; Owen, GR; Verheyden, JP1
Bryan, AM; Lau, K; Olafsson, PG1
Pfefferkorn, ER1
Hochhauser, SJ; Weiss, B1
Chen, ZH; Chu, E; Chu, MY; Chu, SH; Darnowski, JW; Pan, BC1
Daher, GC; Diasio, RB; el Kouni, MH; Naguib, FN; Soong, SJ; Zhang, RW1
Fujimaki, M; Kurokawa, M; Kuroki, Y; Ochiai, H; Okamoto, M; Tazawa, K; Yamashita, I1
Adachi, S; Akaza, H; Ishitsuka, H; Kanazawa, K; Miwa, M; Nitta, K; Sekiguchi, F; Tokita, H1
Imai, S; Morimoto, H; Nio, Y; Shiraishi, T; Tobe, T; Tseng, CC; Tsubono, M1
Arima, S; Fukamura, T; Haruta, J; Hashimoto, M; Jyozaki, H; Okamoto, K; Shimura, H; Umeno, T1
Kawada, S; Kondo, H; Ootani, I; Sato, T; Shibata, T; Suzuki, H1
Ando, J; Kosaka, A; Sumiyoshi, K1
Eckel, ME; McAdams, E; Pfefferkorn, ER1
Abrams, DN; Knaus, EE; Lee, YW; Mercer, JR; Wiebe, LI1
Kawaguchi, T; Saito, M; Saneyoshi, M2
Fujita, F; Fujita, M; Hirai, T; Taguchi, T1
Fujii, S1
Fujimoto, K; Ishitsuka, H; Matsuura, N; Miwa, M; Ninomiya, Y; Ryu, M1
Eda, H; Fujimoto, K; Fukuda, H; Ishitsuka, H; Miwa, M1
Lin, FH; Williams, WM1
Laurensse, EJ; Peters, GJ; Pinedo, HM1
Deddish, PA; Ravin, AW1
Klímek, M1
Anraku, N; Tomizawa, J2
Geissler, E4
Donachie, WD; Masters, M1
Bielavsky, N; Leong, GF1
Bieliavsky, N; Leong, GF1
Diez, J; Lorek, H1
Halvorson, HO; Steinberg, W1
Grossowicz, N; Mandelbaum-Shavit, F1
Caster, JH; Melechen, NE1
Kaplan, RW; Pohl, D1
Baker, BR; Kelley, JL5
Ahnström, G; Ehrenberg, L; Hussain, S; Nataraian, AT1
Miovic, M; Pizer, LI1
Fox, BW; Perkins, JP; Prusoff, WH1
Beck, CF; Ingraham, JL; Neuhard, J; Thomassen, E1
Lazdunski, A; Shapiro, BM; Siccardi, AG1
Klaffke-Lobsien, G; Scheuermann, W1
Aingorn, ED; Akifjev, AP1
Hanna, C1
Beck, A; Tan, YL1
Dávila, CA; García-Pineda, D; Reuvers, T1
Bryan, AM; Olafsson, PG1
Kvelland, I1
Pearson, PL1
Anraku, N; Iwama, Y; Tomizawa, JI1
Altshtein, AD; Avakyan, AA; Ciampor, F; Nadtochey, GA; Omelchenko, TN1
Tomasz, A1
Aubert, C; Cano, JP; Coassolo, P; Rigault, JP; Sommadossi, JP1
Goulian, M; Ingraham, HA; Tseng, BY1
Kimura, K; Suga, S1
Calabresi, P; Cha, S; Chu, MY; Chu, SH; el Kouni, MH; Iltzsch, MH; Naguib, FN1
Gunner, L; Herrick, D; Kufe, DW1
Fujii, S; Shirasaka, T1
García, E; López, R; Ronda, C1
Biriukova, IV; Zinchenko, VV1
Fujioka, A; Nakano, K; Okabe, H; Saito, H; Takeda, S; Toko, T; Unemi, N1
Aida, I; Kasuga, Y; Ohwada, M; Sato, I; Suzuki, M; Tamura, T1
Fukushima, S; Hamada, A; Kawaguchi, T; Morinaga, A; Nakano, M; Saneyoshi, M1
Fukagawa, H; Hirohashi, Y; Iwanaga, A; Iyama, A; Kitahara, K; Miyazaki, K; Mori, M; Sasatomi, E; Tsutsumi, N; Yakushiji, H1
Sirover, MA; Tallarida, RJ; Wurzer, JC1
Kumagai, K; Masuo, K; Nishida, Y; Yasui, A; Yoshitoshi, A1
Fukushima, S; Hamada, A; Kawaguchi, T; Nakano, M; Saneyoshi, M; Shimizu, S2
Fukushima, M; Nakano, K; Saito, H; Satake, H; Takechi, T; Takeda, S; Uchida, J; Unemi, N1
Fujimaki, M; Katuyama, S; Kuroki, Y; Okamoto, M; Sakamoto, T; Tazawa, K; Yamashita, I1
Hamada, A; Hasegawa, T; Kawaguchi, T; Nakano, M; Shimidzu, S1
Asaeda, A; Ide, H; Kubo, K; Matsuyama, S; Ohashi, F; Shiomi, A; Takamori, Y1
Pankiewicz, KW; Stivers, JT; Watanabe, KA1
Taguchi, T1
González Barón, M1
Hoshino, K; Ikeda, H; Koyama, T; Morishita, Y; Nakamura, M1
Basaki, Y; Chikahisa, L; Hashimoto, A; Miyadera, K; Okabe, S; Wierzba, K; Yamada, Y; Yonekura, K1
Musha, N; Oka, K; Saito, H; Sando, N; Sasaki, M; Setu, M; Setu, Y; Sunami, E1
Britten, C; Hammond, L; Hidalgo, M; Rothenberg, ML; Sharma, A; Sharma, S; Siu, L; Villalona-Calero, M; Weiss, GR1
Hirakawa, Y; Kawaguchi, Y; Kuwata, K; Matsushima, E; Nagayama, S1
Ashour, OM; el Kouni, MH; Goudgaon, NM; Naguib, FN; Schinazi, RF1
Carey, PR; Dong, J; Drohat, AC; Pankiewicz, KW; Stivers, JT1
Aiba, K; Horikoshi, N; Saotome, T; Yoshida, N1
Katayama, A; Mafune, K; Makuuchi, M1
Higashigawa, M; Kagawa, Y; Kakito, H; Kawasaki, H; Kojima, M; Ohkubo, T; Ooi, A; Sakurai, M1
Fujioka, A; Fukushima, M; Nakagawa, F; Nukatsuka, M; Ohshimo, H1
Aoyagi, K; Basaki, Y; Chikahisa, L; Hashimoto, A; Miyadera, K; Okabe, S; Wierzba, K; Yamada, Y; Yonekura, K1
Fujioka, A; Fukushima, M; Kitazato, K; Nakagawa, F; Nukatsuka, M; Ohshimo, H1
Ito, T; Nakamura, A; Sato, A; Taguchi, S; Tomita, T1
Azuma, T; Hatada, T; Inoue, Y; Kusunoki, M; Miki, C; Mohri, T; Ojima, E1
HALL, TC1
BERENS, K; SHUGAR, D1
BOND, SB; KRISS, JP1
JACOBSON, BS; LANSKY, LL; SALMON, RJ1
BOOHAR, J; HEIDELBERGER, C1
MORSE, PA; POTTER, VR1
CURRERI, AR; JOHNSON, RO; WOLBERG, WH1
Handa, R; Iijima, S; Kato, T; Kikkawa, N; Kurokawa, E; Naoi, Y; Oshima, S; Tsujie, M; Yamamoto, H1
Emura, T; Fukushima, M; Ohshimo, H; Suzuki, N; Yamaguchi, M1
Hu, P; Jiang, H; Jiang, J; Lu, J1
Fujitani, K; Hirao, M; Ikenaga, M; Kashiwazaki, M; Masuda, N; Mishima, H; Sawamura, T; Takeda, Y; Takeno, A; Tsujinaka, T1
Cao, C; Jiang, YL; McDowell, LM; Poliks, B; Potter, GS; Schaefer, J; Song, F; Stivers, JT; Studelska, DR1
Hayakawa, K; Miyake, K; Morimoto, T; Mukaihara, S; Nishino, M1
Fujioka, A; Fukushima, M; Ikeda, K; Kitazato, K; Nakagawa, F; Ohshimo, H; Okabe, H; Takechi, T1
Ikeda, S; Ishibashi, N; Matono, K; Mizobe, T; Ogata, Y; Ogo, S; Ohkita, A; Ozasa, H; Sasatomi, T; Shirouzu, K1
Hamada, T; Ichimura, W; Minagawa, N; Mino, K; Naito, H; Orimo, T; Shibazaki, W; Shinohara, T1
Peters, GJ; Prins, HJ; Temmink, OH; van Gelderop, E1
Hoshino, S; Maekawa, T; Mikami, K; Sakai, T; Shirakusa, T; Yamashita, Y1
Huh, JW; Kim, HR1
Beijnen, JH; Rosing, H; Schellens, JH; Vainchtein, LD1
Nakayama, T; Noguchi, S1
Amidon, GL; Provoda, CJ; Tsume, Y1
Bellot, GL; Koh, D; Tan, WH; Tay, LL; Wang, X1
Chong, KT; Endoh, K; Fujioka, A; Fukuoka, M; Hashimoto, A; Itou, K; Miyahara, S; Miyakoshi, H; Muto, T; Nagasawa, H; Nomura, M; Shuto, S; Taguchi, J; Takao, Y; Ueno, H; Wakasa, T; Yamamura, K; Yano, W; Yokogawa, T1
Chong, KT; Endoh, K; Fukuoka, M; Miyahara, S; Miyakoshi, H; Nagasawa, H; Nomura, M; Shuto, S; Taguchi, J; Takao, Y; Ueno, H; Wakasa, T; Yano, W; Yokogawa, T1
Hwang, SH; Kim, SG1
Condie, AG; Gerson, SL; Gorityala, S; Han, X; Qing, Y; Xu, Y; Yan, Y; Yang, S; Zhang, Y1
Doki, Y; Fujita, J; Fujitani, K; Fujiwara, Y; Hirao, M; Imamura, H; Kimura, Y; Moon, JH; Mori, M; Takiguchi, S; Tamura, S; Yano, M1
Chionh, F; Lau, D; Price, T; Tebbutt, N; Yeung, Y1
Chang, I; Chang, WJ; Chen, R; Circelli, J; Harpel, Z; Rivera, J; Wei, R; Wu, S1
BURCHENAL, JH; ELLISON, RR; ESCHER, G; KARNOFSKY, DA; KAUFMAN, R; LEVICK, SN; LI, MC; MILLER, E; SULLIVAN, RD; WOLDOW, I; YOUNG, CW1
ANSFIELD, FJ; CURRERI, AR1
NICHOL, CA; WHITE, PJ1

Reviews

9 review(s) available for uracil and floxuridine

ArticleYear
[Gastrointestinal cancer and oral anticancer agents].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1999, Volume: 26, Issue:3

    Topics: Administration, Oral; Antimetabolites, Antineoplastic; Antineoplastic Agents; Camptothecin; Drug Combinations; Floxuridine; Fluorouracil; Gastrointestinal Neoplasms; Humans; Irinotecan; Organoplatinum Compounds; Oxonic Acid; Prodrugs; Pyridines; Tegafur; Uracil

1999
[Oral fluoropyrimidines in oncology].
    Anales de la Real Academia Nacional de Medicina, 1998, Volume: 115, Issue:3

    Topics: Administration, Oral; Antidotes; Antimetabolites, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Capecitabine; Clinical Trials as Topic; Combined Modality Therapy; Deoxycytidine; Female; Floxuridine; Fluorouracil; Humans; Leucovorin; Male; Neoplasm Recurrence, Local; Neoplasms; Tegafur; Time Factors; Uracil

1998
New anticancer agents.
    Cancer chemotherapy and biological response modifiers, 1999, Volume: 18

    Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Cyclin-Dependent Kinases; DNA; Floxuridine; Humans; Microtubules; Organoplatinum Compounds; Signal Transduction; Thymidylate Synthase; Uracil

1999
[Oral cancer chemotherapy in the clinic].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2000, Volume: 27, Issue:11

    Topics: Administration, Oral; Antimetabolites, Antineoplastic; Antineoplastic Agents, Alkylating; Antineoplastic Agents, Hormonal; Antineoplastic Combined Chemotherapy Protocols; Floxuridine; Hematologic Neoplasms; Humans; Melphalan; Quality of Life; Tamoxifen; Tegafur; Uracil

2000
Adrenalectomy for solitary adrenal metastasis from colorectal carcinoma.
    Japanese journal of clinical oncology, 2000, Volume: 30, Issue:9

    Topics: Adrenal Gland Neoplasms; Adrenalectomy; Antineoplastic Combined Chemotherapy Protocols; Chemotherapy, Adjuvant; Floxuridine; Humans; Lung Neoplasms; Male; Middle Aged; Mitomycin; Pneumonectomy; Rectal Neoplasms; Tegafur; Uracil

2000
[Chemotherapy of gastric cancer--a review of clinical trials in Japan].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2002, Volume: 29, Issue:9

    Topics: Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Clinical Trials as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Drug Administration Schedule; Drug Combinations; Floxuridine; Humans; Japan; Methotrexate; Mitomycin; Stomach Neoplasms; Survival Analysis; Tegafur; Uracil

2002
[Effectiveness of chemoradiotherapy for three cases of squamous cell anal carcinoma].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2004, Volume: 31, Issue:11

    Topics: Aged; Antineoplastic Combined Chemotherapy Protocols; Anus Neoplasms; Carcinoma, Squamous Cell; Chemotherapy, Adjuvant; Cisplatin; Combined Modality Therapy; Female; Floxuridine; Fluorouracil; Humans; Lymphatic Metastasis; Middle Aged; Radiotherapy, Adjuvant; Tegafur; Uracil

2004
Therapeutic usefulness of postoperative adjuvant chemotherapy with Tegafur-Uracil (UFT) in patients with breast cancer: focus on the results of clinical studies in Japan.
    The oncologist, 2010, Volume: 15, Issue:1

    Topics: Administration, Oral; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Capecitabine; Chemotherapy, Adjuvant; Cisplatin; Clinical Trials as Topic; Deoxycytidine; Drug Combinations; Female; Floxuridine; Fluorouracil; Humans; Japan; Methotrexate; Oxonic Acid; Tegafur; Uracil

2010
Oral versus intravenous fluoropyrimidines for colorectal cancer.
    The Cochrane database of systematic reviews, 2017, Jul-28, Volume: 7

    Topics: Administration, Oral; Adult; Antineoplastic Agents; Camptothecin; Capecitabine; Chemotherapy, Adjuvant; Colorectal Neoplasms; Disease-Free Survival; Female; Floxuridine; Fluorouracil; Humans; Injections, Intravenous; Irinotecan; Male; Neoadjuvant Therapy; Organoplatinum Compounds; Palliative Care; Pyridines; Pyrimidines; Randomized Controlled Trials as Topic; Tegafur; Uracil

2017

Trials

3 trial(s) available for uracil and floxuridine

ArticleYear
[5-FU concentrations in the blood and tumor tissue after 5'-DFUR or UFT administration in the patients with uterine cervical cancer].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1995, Volume: 22, Issue:2

    Topics: Administration, Oral; Antineoplastic Combined Chemotherapy Protocols; Female; Floxuridine; Fluorouracil; Humans; Lymph Nodes; Middle Aged; Tegafur; Uracil; Uterine Cervical Neoplasms

1995
Important role of the dihydrouracil/uracil ratio in marked interpatient variations of fluoropyrimidine pharmacokinetics and pharmacodynamics.
    Journal of clinical pharmacology, 2004, Volume: 44, Issue:11

    Topics: Adult; Antimetabolites, Antineoplastic; Chorionic Gonadotropin; Female; Floxuridine; Fluorouracil; Gestational Trophoblastic Disease; Humans; Leukocyte Count; Metabolic Clearance Rate; Neutrophils; Prodrugs; Prospective Studies; Uracil

2004
Randomized Controlled Trial of Adjuvant Chemotherapy with Fluoropyrimidines
    Anticancer research, 2017, Volume: 37, Issue:6

    Topics: Adult; Aged; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Chemotherapy, Adjuvant; Female; Floxuridine; Fluorouracil; Humans; Male; Middle Aged; Neoplasm Staging; Stomach Neoplasms; Survival Analysis; Tegafur; Uracil

2017

Other Studies

120 other study(ies) available for uracil and floxuridine

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
The effects of 5-fluorouracil and 5-fluorodeoxyuridine used alone and in combination with normal nucleic acid precursors on development of mice in lines selected for low and high expression of Strong's luxoid gene.
    Teratology, 1975, Volume: 11, Issue:1

    Topics: Abnormalities, Drug-Induced; Animals; Body Weight; Cell Survival; Drug Synergism; Female; Fetal Death; Floxuridine; Fluorouracil; Forelimb; Genes; Hindlimb; Mice; Mutation; Nucleic Acids; Pregnancy; Protein Precursors; Thymidine; Thymine; Tibia; Toes; Uracil

1975
4'-substituted nucleosides. 3. Synthesis of some 4'-fluorouridine derivatives.
    The Journal of organic chemistry, 1976, Sep-03, Volume: 41, Issue:18

    Topics: Anti-Bacterial Agents; Chemical Phenomena; Chemistry; Floxuridine; Uracil

1976
A differential scanning calorimetric-thin-layer chromatographic study of 5-halo-2'-deoxynucleosides.
    Journal of chromatography, 1976, Sep-15, Volume: 124, Issue:2

    Topics: Bromodeoxyuridine; Chemical Phenomena; Chemistry; Chromatography, Thin Layer; Deoxyuridine; Floxuridine; Idoxuridine; Uracil

1976
Toxoplasma gondii: the enzymic defect of a mutant resistant to 5-fluorodeoxyuridine.
    Experimental parasitology, 1978, Volume: 44, Issue:1

    Topics: Animals; Cell Line; Drug Resistance, Microbial; Floxuridine; Mutation; Pentosyltransferases; Toxoplasma; Uracil; Uridine Kinase; Uridine Phosphorylase

1978
Escherichia coli mutants deficient in deoxyuridine triphosphatase.
    Journal of bacteriology, 1978, Volume: 134, Issue:1

    Topics: Coliphages; Deoxyuracil Nucleotides; Escherichia coli; Floxuridine; Genes; Genetic Linkage; Mutation; Pyrophosphatases; Recombination, Genetic; Transduction, Genetic; Uracil

1978
Enhancement of 5-fluoro-2'-deoxyuridine antineoplastic activity by 5-benzyloxybenzyloxybenzylacyclouridine in a human colon carcinoma cell line.
    Cancer research, 1992, Apr-01, Volume: 52, Issue:7

    Topics: Antimetabolites, Antineoplastic; Cell Division; Cell Line; Colonic Neoplasms; Deoxyuridine; DNA Replication; Drug Synergism; Floxuridine; Humans; Kinetics; Recombinant Proteins; Thymidylate Synthase; Uracil; Uridine Monophosphate

1992
Inhibition of fluoropyrimidine catabolism by benzyloxybenzyluracil. Possible relevance to regional chemotherapy.
    Biochemical pharmacology, 1991, Jun-15, Volume: 41, Issue:12

    Topics: Animals; Floxuridine; Fluorouracil; Liver; Male; Perfusion; Rats; Rats, Inbred Strains; Uracil

1991
[Antitumor activity of T-506, a novel synthetic FUDR derivative, on murine colon cancer and its hepatic metastasis].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1991, Volume: 18, Issue:8

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Colonic Neoplasms; Floxuridine; Fluorodeoxyuridylate; Liver Neoplasms; Mice; Mice, Inbred BALB C; Tegafur; Uracil

1991
[Comparative studies on the antitumor activity of fluorinated pyrimidine derivatives against human bladder, cervical and ovarian cancer xenografts in nude mice].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1991, Volume: 18, Issue:10

    Topics: Administration, Oral; Animals; Antineoplastic Combined Chemotherapy Protocols; Female; Floxuridine; Fluorouracil; Humans; Mice; Mice, Nude; Ovarian Neoplasms; Tegafur; Uracil; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms

1991
[Chemotherapy with fluoropyrimidines for MOPC-104E plasmacytoma transplanted in mice with CCl4 induced chronic liver dysfunction].
    Nihon Gan Chiryo Gakkai shi, 1990, Mar-20, Volume: 25, Issue:3

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Carbon Tetrachloride Poisoning; Chemical and Drug Induced Liver Injury; Floxuridine; Fluorouracil; Male; Mice; Mice, Inbred BALB C; Neoplasm Transplantation; Plasmacytoma; Tegafur; Uracil

1990
[Study of tissue drug concentration of fluorinated pyrimidine anticancer drugs--comparison of 5'DFUR and UFT].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1990, Volume: 17, Issue:9

    Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Colon; Colonic Neoplasms; Drug Administration Schedule; Floxuridine; Humans; Lymph Nodes; Tegafur; Uracil

1990
[Two cases of obstructive jaundice due to extrahepatic carcinoma of the bile duct with marked response to daily oral administration of etoposide].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1990, Volume: 17, Issue:12

    Topics: Administration, Oral; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Cholestasis, Extrahepatic; Common Bile Duct Neoplasms; Etoposide; Female; Floxuridine; Humans; Male; Middle Aged; Picibanil; Remission Induction; Tegafur; Uracil

1990
[The serum and tissue concentration of FT-207, 5'-DFUR and 5-FU in patients with breast cancer by preoperative administration of UFT and 5'-DFUR].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1989, Volume: 16, Issue:2

    Topics: Antineoplastic Combined Chemotherapy Protocols; Breast; Breast Neoplasms; Floxuridine; Fluorouracil; Humans; Lymph Nodes; Preoperative Care; Tegafur; Tissue Distribution; Uracil

1989
Toxoplasma gondii: the biochemical basis of resistance to emimycin.
    Experimental parasitology, 1989, Volume: 69, Issue:2

    Topics: Animals; Anti-Bacterial Agents; Drug Resistance; Floxuridine; Nucleic Acids; Pentosyltransferases; Pyrazines; Toxoplasma; Uracil; Xanthine; Xanthines

1989
Tumour uptake of radiolabelled pyrimidine bases and pyrimidine nucleosides in animal models. IX. Radiolabelled 1-(2'-fluoro-2'-deoxy-beta-D-ribofuranosyl)uracil and 1-(2'-chloro-2'-deoxy-beta-D-ribofuranosyl)uracil.
    The British journal of radiology, 1986, Volume: 59, Issue:699

    Topics: Animals; Carbon Radioisotopes; Carcinoma 256, Walker; Chlorine; Deoxyuridine; Floxuridine; Lung Neoplasms; Mice; Radioisotopes; Rats; Rats, Inbred Strains; Tissue Distribution; Uracil; Uridine

1986
Potentiation by acyclothymidine esters of the antitumor effect of orally administered 5-fluoro-2'-deoxyuridine esters on L1210 in mice.
    Japanese journal of cancer research : Gann, 1986, Volume: 77, Issue:5

    Topics: Administration, Oral; Animals; Antineoplastic Combined Chemotherapy Protocols; Drug Synergism; Floxuridine; Leukemia L1210; Mice; Pentosyltransferases; Thymidine Phosphorylase; Uracil

1986
[Evaluation by multiple regression analysis of factors influencing the chemosensitivity of human tumors xenografted into nude mice].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1987, Volume: 14, Issue:3 Pt 1

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Cell Division; Colony-Forming Units Assay; Doxorubicin; Floxuridine; Humans; Mice; Mice, Nude; Mitomycin; Mitomycins; Neoplasm Transplantation; Nimustine; Nitrosourea Compounds; Regression Analysis; Tegafur; Tumor Stem Cell Assay; Uracil

1987
[BOF-A1 and BOF-A2, new 5-FU degradation-inhibitory agents].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1987, Volume: 14, Issue:7

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Floxuridine; Fluorouracil; Liver; Mice; Pyridines; Pyrimidines; Rats; Sarcoma 180; Sarcoma, Experimental; Sarcoma, Yoshida; Tegafur; Uracil

1987
[Antitumor activity and toxicity to the immune system and intestine, of the fluorinated pyrimidines FUra, 5'-DFUR, tegafur and UFT].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1988, Volume: 15, Issue:5

    Topics: Animals; Antibody Formation; Antineoplastic Combined Chemotherapy Protocols; Body Weight; Bone Marrow; Female; Floxuridine; Intestines; Leukopenia; Lung Neoplasms; Male; Mice; Mice, Inbred C3H; Mice, Inbred Strains; Spleen; Tegafur; Thymus Gland; Uracil

1988
[Comparative studies on the antitumor activity of the fluorinated pyrimidines 5'-DFUR, tegafur, UFT and FUra on various murine tumors].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1988, Volume: 15, Issue:5

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Colonic Neoplasms; Floxuridine; Fluorouracil; Leukemia P388; Liver Neoplasms, Experimental; Lung Neoplasms; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Inbred Strains; Neoplasms, Experimental; Sarcoma 180; Tegafur; Uracil

1988
Catabolism of 5-fluoro-2'-deoxyuridine by isolated rat intestinal epithelial cells.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1988, Volume: 189, Issue:3

    Topics: Animals; Epithelium; Floxuridine; Fluorouracil; In Vitro Techniques; Intestinal Mucosa; Kinetics; Male; Pentosyltransferases; Pyrimidine Phosphorylases; Rats; Rats, Inbred Strains; Thymidine; Uracil

1988
Potentiation of the antitumor effect of 5-fluoro-2'-deoxyuridine esters in combination with acyclothymidine esters on L1210 in mice via oral administration.
    Journal of pharmaceutical sciences, 1988, Volume: 77, Issue:11

    Topics: Animals; Antineoplastic Agents; Chemical Phenomena; Chemistry, Physical; Dogs; Drug Synergism; Floxuridine; Leukemia L1210; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Pyridines; Rats; Rats, Inbred Strains; Species Specificity; Uracil

1988
A sensitive non-radioactive assay for pyrimidine nucleoside phosphorylase using reversed-phase high performance liquid chromatography.
    Clinica chimica acta; international journal of clinical chemistry, 1988, Volume: 178, Issue:1

    Topics: Cell Line, Transformed; Chromatography, High Pressure Liquid; Floxuridine; Fluorouracil; Humans; Kinetics; Pentosyltransferases; Pyrimidine Phosphorylases; Tumor Cells, Cultured; Uracil; Uridine

1988
Relation of macromolecular synthesis in streptococci to efficiency of transformation by markers of homospecific and heterospecific origin.
    Journal of bacteriology, 1974, Volume: 117, Issue:3

    Topics: Bacterial Proteins; Carbon Radioisotopes; Chloramphenicol; Dactinomycin; DNA, Bacterial; Drug Resistance, Microbial; Erythromycin; Floxuridine; Hot Temperature; Lincomycin; Mutation; Nucleic Acids; Phenylalanine; Phosphorus Radioisotopes; Rifampin; RNA, Bacterial; Streptococcus; Streptomycin; Thymidine; Transformation, Genetic; Tritium; Uracil

1974
Thymidine incoporation into mammalian strain L-cells after the action of 5-fluorodoxyuridine and the effect of uracil.
    Neoplasma, 1965, Volume: 12, Issue:5

    Topics: Floxuridine; In Vitro Techniques; L Cells; Thymidine; Uracil

1965
Molecular mechanisms of genetic recombination of bacteriophage. V. Two kinds of joining of parental DNA molecules.
    Journal of molecular biology, 1965, Volume: 12, Issue:3

    Topics: Centrifugation; Cesium; Chemical Phenomena; Chemistry Techniques, Analytical; Chemistry, Physical; Chloramphenicol; Coliphages; DNA, Viral; Floxuridine; Genetics; Hybridization, Genetic; In Vitro Techniques; Mutation; Phosphorus Isotopes; Temperature; Uracil

1965
[Investigations on the mechanism of induction of lysogenic bacteria. IX. The temperature dependence of induction by thymine deficiency and mitomycin C].
    Biochimica et biophysica acta, 1966, Jan-18, Volume: 114, Issue:1

    Topics: Coliphages; Escherichia coli; Floxuridine; In Vitro Techniques; Mitomycins; Mutation; Temperature; Thymine; Uracil

1966
Repression and the control of cyclic enzyme synthesis in Bacillus subtilis.
    Nature, 1966, Jan-29, Volume: 209, Issue:5022

    Topics: Alkaline Phosphatase; Bacillus subtilis; Enzyme Repression; Floxuridine; Glycoside Hydrolases; Ornithine Carbamoyltransferase; Periodicity; Sucrase; Transferases; Uracil

1966
The effect of FUDR on segmentation and incorporation of uracil-H3 in amphibian embryos. USNRDL-TR-1087.
    Research and development technical report. United States. Naval Radiological Defense Laboratory, San Francisco, 1967, Jan-11

    Topics: Amphibians; Animals; Cell Division; DNA; Floxuridine; Tritium; Uracil

1967
The effect of FUDR on segmentation and incorporation of 3-H-uracil in amphibian embryos.
    Experimental cell research, 1967, Volume: 47, Issue:1

    Topics: Amphibians; Animals; Autoradiography; Carbon Isotopes; DNA; Embryo, Nonmammalian; Floxuridine; Micromanipulation; RNA; Spectrophotometry; Tritium; Uracil

1967
[Effects of DNA inhibitors on the multiplication of bacteriophage Ox 174].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1967, Volume: 161, Issue:3

    Topics: Coliphages; DNA; Escherichia coli; Floxuridine; Thymine; Uracil

1967
Timing of enzyme synthesis during outgrowth of spores of Bacillus cereus. II. Relationship between ordered enzyme synthesis and deoxyribonucleic acid replication.
    Journal of bacteriology, 1968, Volume: 95, Issue:2

    Topics: Adenine; Amino Acid Oxidoreductases; Bacillus cereus; Bromodeoxyuridine; Carbon Isotopes; Centrifugation, Density Gradient; DNA Replication; DNA, Bacterial; Enzyme Induction; Floxuridine; Glucosidases; Lyases; Mitomycins; Mutation; RNA, Messenger; Spores; Thymine; Tritium; Uracil

1968
Effect of folinate on thymidine uptake by Pediococcus cerevisiae.
    Journal of bacteriology, 1968, Volume: 95, Issue:4

    Topics: Aminopterin; Carbon Isotopes; Deoxyuridine; Floxuridine; Glucose; Hydrogen-Ion Concentration; Iodoacetates; Leucovorin; Methotrexate; Pediococcus; Temperature; Thymidine; Thymine; Tritium; Uracil

1968
Requirements for macromolecular synthesis in the establishment of beta-galactosidase repression in zygotes.
    Journal of bacteriology, 1968, Volume: 95, Issue:5

    Topics: Aminopterin; Bacterial Proteins; Borates; Carbon Isotopes; Chloramphenicol; Conjugation, Genetic; Enzyme Repression; Escherichia coli; Floxuridine; Galactosidases; Genetics, Microbial; Molecular Biology; Recombination, Genetic; RNA, Bacterial; Streptomycin; Tryptophan; Uracil

1968
[Influence of bromouracil on mutation induction and inactivation by UV and x-rays in the phage kappa].
    Biophysik, 1968, Volume: 4, Issue:3

    Topics: Bacteriophages; Bromine; Bromodeoxyuridine; Centrifugation, Density Gradient; DNA, Viral; Floxuridine; Mutagens; Mutation; Radiation Genetics; Serratia marcescens; Ultraviolet Rays; Uracil

1968
Irreversible enzyme inhibitors. CLXIX. Inhibition of FUDR phosphorylase from Walker 256 rat tumor by 6-substituted uracils.
    Journal of medicinal chemistry, 1970, Volume: 13, Issue:3

    Topics: Animals; Binding Sites; Carcinoma 256, Walker; Floxuridine; Rats; Transferases; Uracil

1970
Irreversible enzyme inhibitors. CLXX. Inhibition of FUDR phosphorylase from Walker 256 rat tumor by 1-substituted uracils.
    Journal of medicinal chemistry, 1970, Volume: 13, Issue:3

    Topics: Animals; Binding Sites; Carcinoma 256, Walker; Floxuridine; Rats; Transferases; Uracil

1970
Irreversible enzyme inhibitors. CLXXI. Inhibition of FUDR phosphorylase from Walker 256 rat tumor by 5-substituted uracils.
    Journal of medicinal chemistry, 1970, Volume: 13, Issue:3

    Topics: Animals; Binding Sites; Carcinoma 256, Walker; Floxuridine; Rats; Transferases; Uracil

1970
On the killing and mutagenic action in E. coli associated with the Auger effect during 125-I decay.
    Mutation research, 1970, Volume: 10, Issue:3

    Topics: Escherichia coli; Floxuridine; Iodine Isotopes; Mutation; Radiation Genetics; Radiometry; Tritium; Uracil; Uridine

1970
Effect of trimethoprim on macromolecular synthesis in Escherichia coli.
    Journal of bacteriology, 1971, Volume: 106, Issue:3

    Topics: Adenine; Bacterial Proteins; Carbon Isotopes; DNA, Bacterial; Escherichia coli; Floxuridine; Folic Acid Antagonists; Isoleucine; Ligases; Nucleotides; Purines; Pyrimidines; RNA, Bacterial; RNA, Transfer; Spectrophotometry; Thymidine; Tritium; Uracil; Valine

1971
Irreversible enzyme inhibitors. 188. Inhibition of mammalian thymidine phosphorylase.
    Journal of medicinal chemistry, 1971, Volume: 14, Issue:9

    Topics: Aniline Compounds; Animals; Benzyl Compounds; Binding Sites; Bromine; Chlorine; Cyclohexanes; Escherichia coli; Ethers; Floxuridine; Liver; Methylamines; Naphthalenes; Nitro Compounds; Pentosyltransferases; Phenethylamines; Rabbits; Species Specificity; Structure-Activity Relationship; Sulfides; Sulfonamides; Sulfones; Thymidine; Uracil

1971
Inhibitory action of thymine ribonucleoside and other pyrimidine derivatives on the cleavage of 5-iodo-deoxy-uridine by mouse-liver extract.
    Chemico-biological interactions, 1970, Volume: 1, Issue:4

    Topics: Animals; Chromatography, Thin Layer; Deoxyribonucleosides; Depression, Chemical; Female; Floxuridine; Hydrogen-Ion Concentration; Idoxuridine; Iodine Isotopes; Kinetics; Liver; Mice; Nucleosides; Pentosyltransferases; Pyrimidines; Rats; Ribonucleosides; Thymidine; Thymine; Uracil; Uridine

1970
Metabolism of pyrimidines and pyrimidine nucleosides by Salmonella typhimurium.
    Journal of bacteriology, 1972, Volume: 110, Issue:1

    Topics: Aminohydrolases; Cytidine; Cytosine; Deoxyuridine; Floxuridine; Flucytosine; Fluorouracil; Genetics, Microbial; Genotype; Mutation; Nucleosides; Nucleotidyltransferases; Pentosyltransferases; Phosphotransferases; Pyrimidines; Salmonella typhimurium; Thymidine; Uracil; Uracil Nucleotides; Uridine

1972
Interrelationship between membrane protein composition and deoxyribonucleic acid synthesis in Escherichia coli.
    Biochemistry, 1972, Apr-25, Volume: 11, Issue:9

    Topics: Amino Acids; Azo Compounds; Bacterial Proteins; Carbon Isotopes; Cell Membrane; DNA, Bacterial; Electrophoresis; Escherichia coli; Floxuridine; Genetics, Microbial; Hydroxyurea; Isotope Labeling; Leucine; Mitomycins; Mutation; Nalidixic Acid; Penicillins; Sodium Dodecyl Sulfate; Temperature; Thymine; Tritium; Uracil

1972
[Influence of 5-aminouracil on the DNA synthesis in root tip meristemes].
    Hoppe-Seyler's Zeitschrift fur physiologische Chemie, 1972, Volume: 353, Issue:5

    Topics: DNA; Floxuridine; Methylation; Plants; Uracil

1972
DNA synthesis related to genome activation in human lymphocytes cultured in vitro.
    Experimental cell research, 1972, Volume: 75, Issue:2

    Topics: Autoradiography; Chromosome Aberrations; Chromosomes; Colchicine; Dactinomycin; DNA; Female; Floxuridine; Humans; Lymphocyte Activation; Lymphocytes; Male; Mitosis; Thymidine; Tritium; Uracil; Uridine

1972
Incorporation of idoxuridine analogs into corneal herpes simplex virus.
    Annals of ophthalmology, 1972, Volume: 4, Issue:11

    Topics: Animals; Autoradiography; Bromodeoxyuridine; Cornea; DNA, Viral; Epithelium; Floxuridine; Fluorouracil; Herpes Simplex; Idoxuridine; Keratitis, Dendritic; Ophthalmic Solutions; Rabbits; Thymidine; Tritium; Uracil

1972
Complex formation of uracil, 2'-deoxyuridine and their 5-halogenated derivatives.
    Biochimica et biophysica acta, 1973, Apr-11, Volume: 299, Issue:4

    Topics: Bromodeoxyuridine; Bromouracil; Chemical Phenomena; Chemistry; Copper; Deoxyuridine; Drug Stability; Floxuridine; Fluorouracil; Idoxuridine; Mathematics; Nickel; Potentiometry; Silver; Uracil

1973
Effects of 5-fluoro-2'-deoxyuridine on bacterial growth. Its use for DNA labelling.
    Antonie van Leeuwenhoek, 1973, Volume: 39, Issue:3

    Topics: Bacillus; Bacillus cereus; Bacillus subtilis; Deoxyribonucleosides; DNA, Bacterial; Escherichia coli; Floxuridine; Micrococcus; Pseudomonas; Pseudomonas fluorescens; Thymine; Tritium; Uracil

1973
The influence of 5-halo substituents on the thermal depyrimidination of the glycosidic bond in 2'-deoxyuridines.
    Archives of biochemistry and biophysics, 1974, Volume: 165, Issue:1

    Topics: Bromodeoxyuridine; Calorimetry; Deoxyuridine; Floxuridine; Guanosine; Iodine; Molecular Conformation; Temperature; Thermodynamics; Thymidine; Thymine; Uracil

1974
Bromodeoxyuridine-labeled bacteriophage T4D. I. Growth parameters and frequency of markers recovered from BUdR-labeled and from non-labeled phages studied in mass lysates.
    Hereditas, 1972, Volume: 72, Issue:2

    Topics: Bromodeoxyuridine; Centrifugation, Density Gradient; Coliphages; Crosses, Genetic; Culture Media; DNA Viruses; DNA, Viral; Escherichia coli; Floxuridine; Light; Recombination, Genetic; Uracil

1972
The behavior of chromosomes.
    Advances in the biosciences, 1973, Volume: 10

    Topics: Acridines; Caffeine; Chloroquine; Depression, Chemical; DNA; DNA Repair; DNA Replication; Floxuridine; Humans; Male; Meiosis; Sex Chromosomes; Spermatogenesis; Spermatozoa; Uracil; Urea

1973
Molecular mechanisms of genetic recombination in bacteriophage. VI. A mutant defective in the joining of DNA molecules.
    Journal of molecular biology, 1966, Nov-14, Volume: 21, Issue:2

    Topics: Centrifugation, Density Gradient; Coliphages; Deoxyribonucleases; DNA, Viral; Floxuridine; Molecular Biology; Mutation; Nucleotidyltransferases; Phosphoric Monoester Hydrolases; Phosphorus Isotopes; Thymidine; Uracil

1966
Effects of inhibitors of DNA synthesis on haemagglutinin and infectious SV 15 virus formation in green monkey kidney cells.
    Acta virologica, 1969, Volume: 13, Issue:6

    Topics: Adenoviridae; Animals; Culture Techniques; Cytopathogenic Effect, Viral; Deoxyuridine; DNA, Viral; Floxuridine; Haplorhini; Hemagglutination Inhibition Tests; Hemagglutinins, Viral; Kidney; Microscopy, Electron; Uracil; Virus Cultivation; Virus Replication

1969
Cellular metabolism in genetic transformation of pneumococci: requirement for protein synthesis during induction of competence.
    Journal of bacteriology, 1970, Volume: 101, Issue:3

    Topics: Amino Acids; Bacterial Proteins; Carbon Isotopes; Chloramphenicol; Culture Media; Depression, Chemical; DNA, Bacterial; Floxuridine; Glucose; Iodoacetates; Macromolecular Substances; Mutation; Phenylalanine; Puromycin; Rifampin; RNA, Bacterial; Streptococcus pneumoniae; Thymidine; Transformation, Genetic; Uracil

1970
Irreversible enzyme inhibitors. 202. Candidate active-site-directed irreversible inhibitors of 5-fluoro-2'-deoxyuridine phosphorylase from Walker 256 rat tumor derived from 1-benzyl-5-(3-ethoxybenzyl)uracil.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:5

    Topics: Animals; Antineoplastic Agents; Binding Sites; Carcinoma 256, Walker; Chemical Phenomena; Chemistry; Floxuridine; Pentosyltransferases; Rats; Uracil; Uridine Phosphorylase

1982
Quantitative analysis of 5-fluorouracil and 5,6-dihydrofluorouracil in plasma by gas chromatography mass spectrometry.
    Biomedical mass spectrometry, 1982, Volume: 9, Issue:8

    Topics: Chromatography, High Pressure Liquid; Floxuridine; Fluorouracil; Gas Chromatography-Mass Spectrometry; Humans; Time Factors; Uracil

1982
Nucleotide levels and incorporation of 5-fluorouracil and uracil into DNA of cells treated with 5-fluorodeoxyuridine.
    Molecular pharmacology, 1982, Volume: 21, Issue:1

    Topics: Deoxyribonucleotides; DNA; Floxuridine; Fluorouracil; Humans; Lymphocytes; Uracil; Uracil Nucleotides

1982
[Pharmacological and pharmacodynamic aspects of cancer chemotherapy, with special reference to 5-fluorouracil and its derivatives].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1982, Volume: 9, Issue:8

    Topics: Antineoplastic Combined Chemotherapy Protocols; Drug Combinations; Floxuridine; Fluorouracil; Humans; Kinetics; Neoplasms; Tegafur; Uracil

1982
Potentiation of 5-fluoro-2'-deoxyuridine antineoplastic activity by the uridine phosphorylase inhibitors benzylacyclouridine and benzyloxybenzylacyclouridine.
    Cancer research, 1984, Volume: 44, Issue:5

    Topics: Animals; Cell Line; Cell Survival; Drug Evaluation, Preclinical; Drug Synergism; Female; Floxuridine; Humans; Kinetics; Lung Neoplasms; Mice; Mice, Inbred Strains; Pancreatic Neoplasms; Pentosyltransferases; Uracil; Uridine Phosphorylase

1984
Uracil enhancement of 5-fluorodexoyuridine incorporation into human breast carcinoma deoxyribonucleic acid.
    Biochemical pharmacology, 1984, Jul-15, Volume: 33, Issue:14

    Topics: Breast Neoplasms; Cells, Cultured; DNA, Neoplasm; Female; Floxuridine; Humans; RNA, Neoplasm; Uracil

1984
[Development of fluoropyrimidine derivatives].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1984, Volume: 11, Issue:11

    Topics: Animals; DNA Replication; Floxuridine; Fluorouracil; Mice; Phosphorylation; Pyrimidine Nucleotides; Rats; Sarcoma, Experimental; Tegafur; Uracil

1984
Selective replication of diplophage Dp-4 deoxyribonucleic acid in 6-(p-hydroxyphenylazo)-uracil treated Streptococcus pneumoniae.
    FEBS letters, 1980, Feb-25, Volume: 111, Issue:1

    Topics: Bacteriophages; DNA Replication; DNA, Bacterial; DNA, Viral; Floxuridine; Hydroxyphenylazouracil; Hydroxyurea; Kinetics; Nalidixic Acid; Streptococcus pneumoniae; Uracil; Virus Replication

1980
[Genetic control of pathways of pyrimidine metabolism in Aspergillus nidulans. 1. Isolation and genetic analysis of 6-azauracil resistant mutants].
    Genetika, 1980, Volume: 16, Issue:9

    Topics: Aspergillus nidulans; Chromosome Mapping; Drug Resistance; Floxuridine; Fluorouracil; Genes, Dominant; Genes, Recessive; Mutation; Pyrimidines; Uracil

1980
[Augmentation of chemotherapeutic efficaciousness of UFT by oral l-leucovorin--growth-inhibitory activity of combination against human tumor xenograft].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1995, Volume: 22, Issue:13

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Colonic Neoplasms; Female; Floxuridine; Humans; Leucovorin; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Transplantation; Tegafur; Transplantation, Heterologous; Uracil

1995
Differential effects of acyclothymidine, a potent pyrimidine nucleoside phosphorylase inhibitor, on the pharmacokinetics of doxifluridine in rabbits via oral administration.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:12

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Chromatography, High Pressure Liquid; Drug Interactions; Floxuridine; Fluorouracil; Male; Pentosyltransferases; Pyrimidine Phosphorylases; Rabbits; Uracil

1993
[A comparative study on the serum and tissue 5-FU concentrations in patients with hepatocellular carcinoma after preoperative oral administration of UFT and 5'-DFUR].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1994, Volume: 21, Issue:5

    Topics: Administration, Oral; Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Hepatocellular; Chemotherapy, Adjuvant; Drug Administration Schedule; Female; Floxuridine; Fluorouracil; Humans; Liver; Liver Neoplasms; Male; Middle Aged; Tegafur; Uracil

1994
New mechanism of action of the cancer chemotherapeutic agent 5-fluorouracil in human cells.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:1

    Topics: Binding, Competitive; Cell Count; Cells, Cultured; DNA; DNA Glycosylases; Fibroblasts; Floxuridine; Fluorouracil; Humans; Kinetics; N-Glycosyl Hydrolases; Uracil; Uracil-DNA Glycosidase

1994
The significance of preoperative chemotherapy for early gastric carcinoma.
    Surgery today, 1993, Volume: 23, Issue:10

    Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Chemotherapy, Adjuvant; Drug Administration Schedule; Female; Floxuridine; Fluorouracil; Humans; Male; Middle Aged; Neoplasm Staging; Preoperative Care; Prognosis; Stomach Neoplasms; Tegafur; Uracil

1993
Modulation of the pharmacokinetics of 5'-deoxy-5-fluorouridine and 5-fluorouracil in rats by oral co-administration of acyclothymidine.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:5

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Drug Interactions; Enzyme Inhibitors; Floxuridine; Fluorouracil; Intestines; Liver; Male; Pentosyltransferases; Pyrimidine Phosphorylases; Rats; Uracil

1996
Acyclothymidine alleviates intestinal toxicity of 5'-deoxy-5-fluorouridine without loss of antitumor activity in mice.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:10

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Body Weight; Carcinoma, Lewis Lung; Drug Synergism; Enzyme Inhibitors; Floxuridine; Intestines; Isomerism; Mice; Thymidine Phosphorylase; Uracil

1996
[Antimetastatic effects of UFT on murine liver metastasis model using L5178YHM lymphoma].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1996, Volume: 23, Issue:14

    Topics: Animals; Body Weight; Drug Combinations; Floxuridine; Leukemia L5178; Liver Neoplasms; Male; Mice; Tegafur; Uracil

1996
Inhibitory effects of fluorinated pyrimidines, 5'-DFUR, UFT and T-506, in a model of hepatic metastasis of mouse colon 26 adenocarcinoma-assessment of inhibitory activity and adverse reactions at the maximum tolerated dose.
    Clinical & experimental metastasis, 1997, Volume: 15, Issue:3

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Body Weight; Colonic Neoplasms; Dose-Response Relationship, Drug; Drug Combinations; Female; Floxuridine; Fluorodeoxyuridylate; Liver Neoplasms, Experimental; Male; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Tegafur; Uracil

1997
Inhibition of 5'-deoxy-5-fluorouridine phosphorolysis by acyclothymidine in tumor cell homogenates.
    Biological & pharmaceutical bulletin, 1997, Volume: 20, Issue:8

    Topics: Animals; Antineoplastic Agents; Enzyme Inhibitors; Floxuridine; Humans; Kinetics; Mice; Mice, Inbred C57BL; Thymidine Phosphorylase; Tumor Cells, Cultured; Uracil

1997
Induction of fragile sites by fluorodeoxyuridine and caffeine accompanies with misincorpolation of endogenous uridine nucleotide into DNA of feline fibroblasts.
    The Journal of veterinary medical science, 1998, Volume: 60, Issue:12

    Topics: Animals; Caffeine; Cats; Cells, Cultured; Chromosome Fragile Sites; Chromosome Fragility; DNA; DNA Glycosylases; Female; Fibroblasts; Floxuridine; N-Glycosyl Hydrolases; Uracil; Uracil Nucleotides; Uracil-DNA Glycosidase

1998
Kinetic mechanism of damage site recognition and uracil flipping by Escherichia coli uracil DNA glycosylase.
    Biochemistry, 1999, Jan-19, Volume: 38, Issue:3

    Topics: Binding Sites; DNA Damage; DNA Glycosylases; DNA Repair; Escherichia coli; Floxuridine; Kinetics; Macromolecular Substances; N-Glycosyl Hydrolases; Spectrometry, Fluorescence; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Substrate Specificity; Thermodynamics; Uracil; Uracil-DNA Glycosidase

1999
[Effective chemo-endocrine combination therapy for obstructive-jaundice caused by multiple liver metastasis of recurrent breast cancer--a case report].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1999, Volume: 26, Issue:7

    Topics: Aged; Antineoplastic Agents, Hormonal; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cholestasis; Cyclophosphamide; Doxorubicin; Drainage; Female; Floxuridine; Fluorouracil; Humans; Liver Neoplasms; Lung Neoplasms; Mastectomy, Radical; Medroxyprogesterone Acetate; Tamoxifen; Tegafur; Toremifene; Uracil

1999
UFT and its metabolites inhibit the angiogenesis induced by murine renal cell carcinoma, as determined by a dorsal air sac assay in mice.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 1999, Volume: 5, Issue:8

    Topics: 4-Butyrolactone; Animals; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Renal Cell; Cell Division; Diffusion Chambers, Culture; Dose-Response Relationship, Drug; Floxuridine; Fluorouracil; Hydroxybutyrates; Kidney Neoplasms; Male; Mice; Mice, Inbred BALB C; Neoplasm Transplantation; Neovascularization, Pathologic; Tegafur; Tumor Cells, Cultured; Uracil

1999
[Long-term complete response in a case of unresectable rectal cancer following chemoradiation].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2000, Volume: 27, Issue:1

    Topics: Adenocarcinoma; Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Combined Modality Therapy; Drug Administration Schedule; Floxuridine; Fluorouracil; Humans; Male; Middle Aged; Radiotherapy Dosage; Rectal Neoplasms; Remission Induction; Tegafur; Uracil

2000
[Comparison of pharmacokinetics of 5-FU and alpha-fluoro-beta-alanine, a metabolite of 5-FU, in plasma after administration of UFT, tegafur, 5-FU or doxifluridine to rats].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2000, Volume: 27, Issue:6

    Topics: Administration, Oral; Animals; Antineoplastic Combined Chemotherapy Protocols; beta-Alanine; Floxuridine; Fluorouracil; Male; Rats; Rats, Sprague-Dawley; Tegafur; Uracil

2000
Effect of administration of 5-(phenylselenenyl)acyclouridine, an inhibitor of uridine phosphorylase, on the anti-tumor efficacy of 5-fluoro-2'-deoxyuridine against murine colon tumor C26-10.
    Biochemical pharmacology, 2000, Sep-01, Volume: 60, Issue:5

    Topics: Animals; Antimetabolites, Antineoplastic; Drug Interactions; Enzyme Inhibitors; Female; Floxuridine; Mice; Mice, Inbred BALB C; Organoselenium Compounds; Transplantation, Heterologous; Tumor Cells, Cultured; Uracil; Uridine Phosphorylase

2000
Raman spectroscopy of uracil DNA glycosylase-DNA complexes: insights into DNA damage recognition and catalysis.
    Biochemistry, 2000, Oct-31, Volume: 39, Issue:43

    Topics: Base Composition; Catalysis; DNA Damage; DNA Glycosylases; DNA Repair; DNA-Binding Proteins; DNA, Bacterial; Escherichia coli; Floxuridine; Furans; Glycosides; Hydrogen Bonding; Hydrogen-Ion Concentration; Macromolecular Substances; N-Glycosyl Hydrolases; Nucleic Acid Conformation; Solvents; Spectrum Analysis, Raman; Uracil; Uracil-DNA Glycosidase

2000
Plasma, intestine and tumor levels of 5-fluorouracil in mice bearing L1210 ascites tumor following oral administration of 5-fluorouracil, UFT (mixed compound of tegafur and uracil), carmofur and 5'-deoxy-5-fluorouridine.
    Biological & pharmaceutical bulletin, 2001, Volume: 24, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Carcinoma, Ehrlich Tumor; Drug Combinations; Floxuridine; Fluorouracil; Intestinal Mucosa; Leukemia L1210; Male; Mice; Tegafur; Uracil

2001
[Antimetastatic and antitumor effects of fluoropyrimidines alone and combined with taxanes in a murine model of breast cancer metastatic to the lung].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2002, Volume: 29, Issue:1

    Topics: Aminoacridines; Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Bridged-Ring Compounds; Disease Models, Animal; Drug Combinations; Female; Floxuridine; Humans; Lung Neoplasms; Mice; Mice, Inbred ICR; Mice, SCID; Neoplasm Transplantation; Taxoids; Tegafur; Uracil

2002
gamma-Hydroxybutyric acid and 5-fluorouracil, metabolites of UFT, inhibit the angiogenesis induced by vascular endothelial growth factor.
    Angiogenesis, 2001, Volume: 4, Issue:3

    Topics: Angiogenesis Inhibitors; Animals; Antimetabolites, Antineoplastic; Breast Neoplasms; Carcinoma; Carcinoma, Renal Cell; Chemotaxis; Colonic Neoplasms; DNA Replication; Drug Combinations; Endothelial Growth Factors; Endothelium, Vascular; Female; Fibroblast Growth Factor 2; Floxuridine; Fluorouracil; Humans; Intercellular Signaling Peptides and Proteins; Kidney Neoplasms; Lung Neoplasms; Lymphokines; Mice; Mice, Inbred BALB C; Mice, Inbred ICR; Neoplasm Proteins; Neovascularization, Pathologic; Prodrugs; Prostheses and Implants; Recombinant Proteins; Sodium Oxybate; Stomach Neoplasms; Tegafur; Tumor Cells, Cultured; Uracil; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Xenograft Model Antitumor Assays

2001
[The antitumor activity of DPD inhibitory-fluoropyrimidine (DIF) and non-DIF alone or in combination with paclitaxel against orthotopically implanted human breast cancer].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2002, Volume: 29, Issue:5

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Dihydrouracil Dehydrogenase (NADP); Female; Floxuridine; Humans; Mice; Mice, Inbred ICR; Neoplasm Transplantation; Oxidoreductases; Paclitaxel; Pyrimidines; Tegafur; Uracil

2002
[A case of colon metastasis to the lung treated successfully with combined chemotherapy of CPT-11 and 5'-DFUR].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2002, Volume: 29, Issue:10

    Topics: Adenocarcinoma; Antineoplastic Combined Chemotherapy Protocols; Camptothecin; Drug Administration Schedule; Drug Combinations; Floxuridine; Fluorouracil; Humans; Irinotecan; Lung Neoplasms; Male; Middle Aged; Rectal Neoplasms; Tegafur; Uracil

2002
A comparative study of 5-fluorouracil (FU), 5-fluorodeoxyuridine (FUDR), and methotrexate (MTX)-progress report.
    Cancer chemotherapy reports, 1962, Volume: 16

    Topics: Antineoplastic Agents; Floxuridine; Fluorouracil; Folic Acid Antagonists; Methotrexate; Nucleosides; Nucleotides; Research Report; Uracil

1962
[Studies on the mechanism of induction. IV. The effect of 5-bromouracil on induction with 5-fluorouracil and 5-fluorodeoxyuridine].
    Acta biologica et medica Germanica, 1963, Volume: 10

    Topics: Bromouracil; Coliphages; Escherichia coli; Floxuridine; Fluorouracil; Uracil

1963
[Studies on the mechanism of induction. III. The effect of uracil on the induction effect of 5-fluorouracil and 5-fluorodeoxyuridine].
    Acta biologica et medica Germanica, 1963, Volume: 10

    Topics: Coliphages; Culture Media; Escherichia coli; Floxuridine; Fluorouracil; Uracil

1963
Ultraviolet absorption spectra and structure of halogenated uracils and their glycosides.
    Acta biochimica Polonica, 1963, Volume: 10

    Topics: Floxuridine; Fluorouracil; Glycosides; Nucleosides; Uracil

1963
[STUDIES ON THE MECHANISM OF INDUCTION. V. EXPERIMENTS ON ANALYSIS OF THE INDUCTIVE EFFECT OF HALOGENATED BASES AND THEIR DESOXYRIBONUCLEOSIDES].
    Acta biologica et medica Germanica, 1963, Volume: 11

    Topics: Coliphages; Culture Media; Cytosine Nucleotides; Deoxyribonucleosides; Escherichia coli; Floxuridine; Fluorouracil; Halogenation; Uracil; Uracil Nucleotides

1963
THE EFFECT OF NATURAL AND UNNNATURAL PYRIMIDINES AND PYRIMIDINE NUCLEOSIDES ON THE PHOSPHOROLYSIS OF 5-IODODEOXYURIDINE BY MOUSE LIVER EXTRACT.
    Biochemical pharmacology, 1964, Volume: 13

    Topics: Animals; Chromatography; Deoxyuridine; Floxuridine; Fluorouracil; Idoxuridine; Iodine Isotopes; Liver; Liver Extracts; Metabolism; Mice; Nucleosides; Pharmacology; Phosphotransferases; Pyrimidine Nucleosides; Pyrimidines; Research; Thymidine; Thymine; Uracil

1964
ANTIMITOTIC EFFECTS OF CHLORAMPHENICOL AND OTHER INHIBITORY AGENTS IN CHLAMYDOMONAS.
    Experimental cell research, 1964, Volume: 36

    Topics: Antimitotic Agents; Cell Division; Cell Nucleus; Chlamydia; Chlamydomonas; Chloramphenicol; Chlorides; DNA; Floxuridine; Fluorouracil; Glycols; Mercaptoethanol; Nucleosides; Pharmacology; Proteins; Radiation Effects; Research; RNA; Uracil

1964
FLUORINATED PYRIMIDINES. 23. FURTHER STUDIES ON NUCLEOSIDE PHOSPHORYLASE.
    Biochimica et biophysica acta, 1964, Dec-16, Volume: 91

    Topics: Adenocarcinoma; Animals; Carbon Isotopes; Carcinoma, Ehrlich Tumor; Enzyme Inhibitors; Floxuridine; Liver; Nucleosides; Nucleotidyltransferases; Pentosyltransferases; Pyrimidines; Research; Uracil

1964
MOLECULAR MECHANISMS OF GENETIC RECOMBINATION IN BACTERIOPHAGE. 3. JOINING OF PARENTAL POLYNUCLEOTIDES OF PHAGE T4 IN THE PRESENCE OF 5-FLUORODEOXYURIDINE.
    Journal of molecular biology, 1965, Volume: 11

    Topics: Bacteriophage T4; Bacteriophages; Centrifugation; Coliphages; DNA; DNA, Viral; Floxuridine; Genetics; Metabolism; Models, Theoretical; Molecular Biology; Pharmacology; Phosphorus Isotopes; Polynucleotides; Recombination, Genetic; Research; Tritium; Uracil

1965
PYRIMIDINE METABOLISM IN TISSUE CULTURE CELLS DERIVED FROM RAT HEPATOMAS. I. SUSPENSION CELL CULTURES DERIVED FROM THE NOVIKOFF HEPATOMA.
    Cancer research, 1965, Volume: 25

    Topics: Animals; Carcinoma, Hepatocellular; Cell Culture Techniques; Floxuridine; Fluorouracil; Glycine; Liver Neoplasms; Liver Neoplasms, Experimental; Metabolism; Methotrexate; Mutation; Neoplasms; Neoplasms, Experimental; Nucleosides; Pharmacology; Pyrimidines; Rats; Research; Serine; Thymidine; Thymidine Kinase; Thymine; Tissue Culture Techniques; Toxicology; Uracil

1965
Studies on the feasibility of adjuvant chemotherapy with 5-fluorouracil (FU) and 5-fluoro-2'-deoxyuridine (FUDR) in the immediate postoperative period.
    Archives of surgery (Chicago, Ill. : 1960), 1962, Volume: 85

    Topics: Antineoplastic Agents; Chemotherapy, Adjuvant; Deoxyuridine; Floxuridine; Fluorouracil; Humans; Postoperative Period; Pyrimidines; Uracil

1962
[A case of hepatic metastasis and local recurrence from rectal cancer responding to hepatic arterial infusion and systemic chemotherapy].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2003, Volume: 30, Issue:11

    Topics: Adenocarcinoma; Aged; Antineoplastic Combined Chemotherapy Protocols; Camptothecin; Drug Administration Schedule; Drug Combinations; Floxuridine; Fluorouracil; Hepatic Artery; Humans; Infusions, Intra-Arterial; Irinotecan; Leucovorin; Liver Neoplasms; Male; Neoplasm Recurrence, Local; Rectal Neoplasms; Tegafur; Uracil

2003
A novel combination antimetabolite, TAS-102, exhibits antitumor activity in FU-resistant human cancer cells through a mechanism involving FTD incorporation in DNA.
    International journal of oncology, 2004, Volume: 25, Issue:3

    Topics: Animals; Antimetabolites, Antineoplastic; Cell Line, Tumor; Colonic Neoplasms; DNA Damage; DNA, Neoplasm; Drug Combinations; Drug Resistance, Neoplasm; Floxuridine; Fluorouracil; Humans; Mice; Mice, Nude; Neoplasm Transplantation; Pyrrolidines; Rats; Rats, Nude; Stomach Neoplasms; Thymine; Trifluridine; Uracil; Xenograft Model Antitumor Assays

2004
Recognition of an unnatural difluorophenyl nucleotide by uracil DNA glycosylase.
    Biochemistry, 2004, Dec-14, Volume: 43, Issue:49

    Topics: Amino Acid Substitution; Binding Sites; Catalysis; DNA Glycosylases; Enzyme Stability; Escherichia coli Proteins; Floxuridine; Fluorine; Hydrogen Bonding; Leucine; Models, Molecular; Nuclear Magnetic Resonance, Biomolecular; Nucleic Acid Heteroduplexes; Solutions; Spectrometry, Fluorescence; Substrate Specificity; Thermodynamics; Uracil; Uracil-DNA Glycosidase

2004
Effects of oral 5-fluorouracil drugs on hepatic fat content in patients with colon cancer.
    Academic radiology, 2005, Volume: 12, Issue:6

    Topics: Adult; Aged; Aged, 80 and over; Antimetabolites, Antineoplastic; Chemotherapy, Adjuvant; Chi-Square Distribution; Colonic Neoplasms; Fatty Liver; Female; Floxuridine; Fluorouracil; Humans; Male; Middle Aged; Retrospective Studies; Tegafur; Tomography, X-Ray Computed; Uracil

2005
Correlations between antitumor activities of fluoropyrimidines and DPD activity in lung tumor xenografts.
    Oncology reports, 2005, Volume: 14, Issue:1

    Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Capecitabine; Cell Line, Tumor; Deoxycytidine; Dihydrouracil Dehydrogenase (NADP); Floxuridine; Fluorouracil; Humans; Lung Neoplasms; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Orotate Phosphoribosyltransferase; Oxonic Acid; Pyridines; Tegafur; Thymidine Phosphorylase; Treatment Outcome; Uracil; Xenograft Model Antitumor Assays

2005
The MMP-9 expression determined the efficacy of postoperative adjuvant chemotherapy using oral fluoropyrimidines in stage II or III colorectal cancer.
    Cancer chemotherapy and pharmacology, 2006, Volume: 57, Issue:5

    Topics: Administration, Oral; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Chemotherapy, Adjuvant; Colorectal Neoplasms; Disease-Free Survival; Female; Floxuridine; Humans; Liver Neoplasms; Lung Neoplasms; Lymph Node Excision; Lymphatic Metastasis; Male; Matrix Metalloproteinase 9; Neoplasm Invasiveness; Neoplasm Recurrence, Local; Neoplasm Staging; Postoperative Period; Retrospective Studies; Survival Rate; Tegafur; Uracil

2006
[Case report--postoperative continuous intraarterial infusion of small doses of 5-FU successfully controlled residual tumor and liver metastasis of stage IV gastric cancer].
    Gan to kagaku ryoho. Cancer & chemotherapy, 2005, Volume: 32, Issue:10

    Topics: Aged; Antineoplastic Combined Chemotherapy Protocols; Disease-Free Survival; Doxorubicin; Drug Combinations; Floxuridine; Fluorouracil; Gastrectomy; Humans; Infusions, Intra-Arterial; Liver Neoplasms; Lymph Node Excision; Lymph Nodes; Lymphatic Metastasis; Male; Methotrexate; Mitomycin; Neoplasm Staging; Picibanil; Proteoglycans; Stomach Neoplasms; Tegafur; Uracil

2005
The Hollow Fibre Assay as a model for in vivo pharmacodynamics of fluoropyrimidines in colon cancer cells.
    British journal of cancer, 2007, Jan-15, Volume: 96, Issue:1

    Topics: Administration, Oral; Animals; Apoptosis; Capecitabine; Cell Cycle; Cell Line, Tumor; Colonic Neoplasms; Deoxycytidine; Drug Combinations; Drug Synergism; Enzyme Inhibitors; Flow Cytometry; Floxuridine; Fluorouracil; Humans; Mice; Mice, Inbred BALB C; Pyrrolidines; Sensitivity and Specificity; Thymidine Phosphorylase; Thymine; Treatment Outcome; Trifluridine; Tumor Cells, Cultured; Uracil; Xenograft Model Antitumor Assays

2007
Immunochemotherapy with PSK and fluoropyrimidines improves long-term prognosis for curatively resected colorectal cancer.
    Cancer biotherapy & radiopharmaceuticals, 2008, Volume: 23, Issue:4

    Topics: Aged; Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; Colorectal Neoplasms; Combined Modality Therapy; Drug Combinations; Female; Floxuridine; Fluorouracil; Humans; Immunotherapy; Kaplan-Meier Estimate; Male; Middle Aged; Prognosis; Proportional Hazards Models; Proteoglycans; Retrospective Studies; Tegafur; Uracil

2008
Postoperative chemotherapy after neoadjuvant chemoradiation and surgery for rectal cancer: is it essential for patients with ypT0-2N0?
    Journal of surgical oncology, 2009, Oct-01, Volume: 100, Issue:5

    Topics: Adenocarcinoma; Adult; Aged; Aged, 80 and over; Antimetabolites, Antineoplastic; Chemotherapy, Adjuvant; Disease-Free Survival; Female; Floxuridine; Fluorouracil; Follow-Up Studies; Humans; Male; Middle Aged; Neoadjuvant Therapy; Neoplasm Recurrence, Local; Rectal Neoplasms; Retrospective Studies; Tegafur; Uracil

2009
A new, validated HPLC-MS/MS method for the simultaneous determination of the anti-cancer agent capecitabine and its metabolites: 5'-deoxy-5-fluorocytidine, 5'-deoxy-5-fluorouridine, 5-fluorouracil and 5-fluorodihydrouracil, in human plasma.
    Biomedical chromatography : BMC, 2010, Volume: 24, Issue:4

    Topics: 1-Propanol; Acetonitriles; Antimetabolites, Antineoplastic; Capecitabine; Chemical Precipitation; Chromatography, High Pressure Liquid; Deoxycytidine; Drug Stability; Floxuridine; Fluorouracil; Furans; Humans; Linear Models; Pyrimidines; Reproducibility of Results; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Trichloroacetic Acid; Uracil; Vidarabine

2010
The achievement of mass balance by simultaneous quantification of floxuridine prodrug, floxuridine, 5-fluorouracil, 5-dihydrouracil, α-fluoro-β-ureidopropionate, α-fluoro-β-alanine using LC-MS.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2011, Apr-15, Volume: 879, Issue:13-14

    Topics: Analysis of Variance; Antimetabolites, Antineoplastic; beta-Alanine; Cell Extracts; Cell Line, Tumor; Chromatography, High Pressure Liquid; Floxuridine; Fluorouracil; Humans; Linear Models; Mass Spectrometry; Reproducibility of Results; Uracil; Urea

2011
Reliability of tumor primary cultures as a model for drug response prediction: expression profiles comparison of tissues versus primary cultures from colorectal cancer patients.
    Journal of cancer research and clinical oncology, 2012, Volume: 138, Issue:3

    Topics: Adenocarcinoma; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Camptothecin; Capecitabine; Cisplatin; Colorectal Neoplasms; Deoxycytidine; Down-Regulation; Doxorubicin; Etoposide; Floxuridine; Fluorescent Antibody Technique; Fluorouracil; Gene Expression Profiling; Gene Expression Regulation, Neoplastic; Genomic Instability; Humans; Irinotecan; Metaphase; Paclitaxel; Polymerase Chain Reaction; Predictive Value of Tests; Protein Array Analysis; Reproducibility of Results; Tegafur; Tissue Array Analysis; Tumor Cells, Cultured; Up-Regulation; Uracil

2012
Discovery of a novel class of potent human deoxyuridine triphosphatase inhibitors remarkably enhancing the antitumor activity of thymidylate synthase inhibitors.
    Journal of medicinal chemistry, 2012, Apr-12, Volume: 55, Issue:7

    Topics: Animals; Antineoplastic Agents; Cell Proliferation; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Drug Synergism; Floxuridine; HeLa Cells; Humans; Mice; Models, Molecular; Neoplasm Transplantation; Protein Conformation; Pyrophosphatases; Pyrrolidines; Stereoisomerism; Structure-Activity Relationship; Sulfonamides; Thymidylate Synthase; Transplantation, Heterologous; Uracil

2012
Synthesis and discovery of N-carbonylpyrrolidine- or N-sulfonylpyrrolidine-containing uracil derivatives as potent human deoxyuridine triphosphatase inhibitors.
    Journal of medicinal chemistry, 2012, Apr-12, Volume: 55, Issue:7

    Topics: Antineoplastic Agents; Cell Proliferation; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Drug Synergism; Floxuridine; HeLa Cells; Humans; Models, Molecular; Protein Conformation; Pyrophosphatases; Pyrrolidines; Small Molecule Libraries; Stereoisomerism; Structure-Activity Relationship; Thymidylate Synthase; Uracil

2012
The association between the duration of fluoropyrimidine-based adjuvant chemotherapy and survival in stage II or III gastric cancer.
    World journal of surgical oncology, 2016, Apr-02, Volume: 14

    Topics: Adenocarcinoma; Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Capecitabine; Chemotherapy, Adjuvant; Cisplatin; Drug Combinations; Female; Floxuridine; Follow-Up Studies; Humans; Lymphatic Metastasis; Male; Middle Aged; Neoplasm Invasiveness; Neoplasm Staging; Organoplatinum Compounds; Oxaliplatin; Oxonic Acid; Prognosis; Retrospective Studies; Stomach Neoplasms; Survival Rate; Tegafur; Time Factors; Uracil

2016
Inhibition of uracil DNA glycosylase sensitizes cancer cells to 5-fluorodeoxyuridine through replication fork collapse-induced DNA damage.
    Oncotarget, 2016, Sep-13, Volume: 7, Issue:37

    Topics: Antineoplastic Agents; Apoptosis; Cell Cycle Checkpoints; Cell Line, Tumor; DNA Damage; DNA Replication; Drug Resistance; Floxuridine; Histones; Humans; Neoplasms; RNA, Small Interfering; Uracil; Uracil-DNA Glycosidase

2016
Effects of six pyrimidine analogs on the growth of Tetrahymena thermophila and their implications in pyrimidine metabolism.
    PloS one, 2023, Volume: 18, Issue:9

    Topics: Antimetabolites; Cytarabine; Floxuridine; Fluorouracil; Gemcitabine; Nucleosides; Pyrimidines; Tetrahymena thermophila; Thymine; Uracil

2023
The clinical evaluation of 5-fluorouracil and 5-fluoro-2'-deoxyuridine in solid tumors in adults: a progress report.
    Cancer chemotherapy reports, 1960, Volume: 6

    Topics: Antineoplastic Agents; Deoxyuridine; Fluorouracil; Neoplasms; Nucleosides; Nucleotides; Research Report; Uracil

1960
Comparison of 5-fluorouracil and 5-fluoro-2'-deoxyuridine in the treatment of far-advanced breast and colon lesions.
    Cancer chemotherapy reports, 1962, Volume: 16

    Topics: Antineoplastic Agents; Breast Neoplasms; Colonic Neoplasms; Deoxyuridine; Fluorouracil; Humans; Nucleosides; Nucleotides; Uracil

1962
Effects of uracil and thymidine on the development of resistance to 5-fluorouracil in Pediococcus cerevisiae.
    Journal of bacteriology, 1963, Volume: 85

    Topics: Deoxyuridine; Fluorouracil; Pediococcus; Thymidine; Uracil

1963