Page last updated: 2024-08-25

uk 68798 and l 706000

uk 68798 has been researched along with l 706000 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's3 (60.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Contreras-Jurado, C; Furini, S; García-Ferreiro, R; Gómez-Varela, D; Pardo, LA; Stühmer, W1
Bianucci, AM; Calderone, V; Coi, A; Massarelli, I; Testai, L1
Baskin, EP; Lynch, JJ1
de Groot, MJ; Helliwell, R; Leishman, D; Mitcheson, J; Perry, M; Sanguinetti, MC; Tristani-Firouzi, M1
Gardner, A; Sanguinetti, MC; Wu, W1

Other Studies

5 other study(ies) available for uk 68798 and l 706000

ArticleYear
Different relevance of inactivation and F468 residue in the mechanisms of hEag1 channel blockage by astemizole, imipramine and dofetilide.
    FEBS letters, 2006, Sep-18, Volume: 580, Issue:21

    Topics: Astemizole; Benzopyrans; Ether-A-Go-Go Potassium Channels; Humans; Imipramine; Ion Channel Gating; Models, Molecular; Phenethylamines; Piperidines; Point Mutation; Potassium Channel Blockers; Structure-Activity Relationship; Sulfonamides

2006
Identification of "toxicophoric" features for predicting drug-induced QT interval prolongation.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:11

    Topics: Amino Acid Sequence; Heart; Humans; Models, Molecular; Molecular Sequence Data; Molecular Structure; Protein Subunits; Sequence Alignment; Structure-Activity Relationship; Trans-Activators; Transcriptional Regulator ERG

2008
Comparative effects of increased extracellular potassium and pacing frequency on the class III activities of methanesulfonanilide IKr blockers dofetilide, D-sotalol, E-4031, and MK-499.
    Journal of cardiovascular pharmacology, 1994, Volume: 24, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; Benzopyrans; Electric Stimulation; Ferrets; Male; Phenethylamines; Piperidines; Potassium; Potassium Channel Blockers; Pyridines; Refractory Period, Electrophysiological; Sotalol; Sulfonamides

1994
Structural determinants of HERG channel block by clofilium and ibutilide.
    Molecular pharmacology, 2004, Volume: 66, Issue:2

    Topics: Amino Acid Substitution; Animals; Anti-Arrhythmia Agents; Aspartic Acid; Benzopyrans; Binding Sites; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Oocytes; Phenethylamines; Phenylalanine; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Pyridines; Quaternary Ammonium Compounds; Serine; Sulfonamides; Tyrosine; Xenopus laevis

2004
The Link between Inactivation and High-Affinity Block of hERG1 Channels.
    Molecular pharmacology, 2015, Volume: 87, Issue:6

    Topics: Animals; Benzopyrans; Cisapride; Ether-A-Go-Go Potassium Channels; Female; Humans; Ion Channel Gating; Oocytes; Patch-Clamp Techniques; Phenethylamines; Piperidines; Point Mutation; Potassium Channel Blockers; Protein Multimerization; Protein Subunits; Sulfonamides; Xenopus laevis

2015