Page last updated: 2024-08-25

uk 68798 and hmr 1556

uk 68798 has been researched along with hmr 1556 in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (66.67)29.6817
2010's4 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Du, LP; Li, MY; Tsai, KC; Xia, L; You, QD1
Gerlach, U; Nakashima, H; Nattel, S; Schmidt, D1
Bleich, M; Brendel, J; Busch, AE; Knobloch, K; Rosenstein, B; Wirth, KJ1
Ducouret, P; Ducroq, J; Gérard, JL; Puddu, PE; Rouet, R; Sallé, L; Tabourel, C1
Backx, PH; Dorian, P; Hu, XD; Puglisi, JL; So, PP1
Baczkó, I; Lengyel, C; Papp, JG; Tábori, K; Varró, A1
Thomsen, MB1
Backx, PH; Dorian, P; So, PP1
Ducroq, J; Legrand, JC; Puddu, PE; Rouet, R; Sallé, L1
Carbonell-Pascual, B; Ferrero, JM; Harmati, G; Jost, N; Kohajda, Z; Koncz, I; Kristóf, A; Nánási, PP; Papp, JG; Papp, R; Varró, A; Virág, L1
Csík, N; Farkas, A; Farkas, AS; Farkas, S; Forster, T; Orosz, S; Papp, JG; Sarusi, A; Varró, A1
Bányász, T; Hegyi, B; Horváth, B; Kistamás, K; Magyar, J; Nánási, PP; Ruzsnavszky, F; Szentandrássy, N; Váczi, K; Varró, A1

Other Studies

12 other study(ies) available for uk 68798 and hmr 1556

ArticleYear
The pharmacophore hypotheses of I(Kr) potassium channel blockers: novel class III antiarrhythmic agents.
    Bioorganic & medicinal chemistry letters, 2004, Sep-20, Volume: 14, Issue:18

    Topics: Anti-Arrhythmia Agents; Models, Biological; Models, Molecular; Potassium Channel Blockers; Potassium Channels; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2004
In vivo electrophysiological effects of a selective slow delayed-rectifier potassium channel blocker in anesthetized dogs: potential insights into class III actions.
    Cardiovascular research, 2004, Mar-01, Volume: 61, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Chromans; Dogs; Electrocardiography; Electrophysiology; Female; Male; Myocardium; Nadolol; Phenethylamines; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Sulfonamides

2004
Atrial-selective antiarrhythmic actions of novel Ikur vs. Ikr, Iks, and IKAch class Ic drugs and beta blockers in pigs.
    Medical science monitor : international medical journal of experimental and clinical research, 2004, Volume: 10, Issue:7

    Topics: Adrenergic beta-Antagonists; Amiodarone; Animals; Anti-Arrhythmia Agents; Atrial Function; Atropine; Biphenyl Compounds; Chromans; Flecainide; Heart Atria; Hydantoins; Imidazoles; Imidazolidines; Male; Phenethylamines; Piperazines; Potassium Channel Blockers; Potassium Channels; Propafenone; Propanolamines; Sotalol; Sulfonamides; Swine; Ventricular Function

2004
Electrophysiological effects of azimilide in an in vitro model of simulated-ischemia and reperfusion in guinea-pig ventricular myocardium.
    European journal of pharmacology, 2005, Aug-22, Volume: 518, Issue:2-3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Chromans; Dose-Response Relationship, Drug; Female; Guinea Pigs; Heart Ventricles; Hydantoins; Imidazolidines; In Vitro Techniques; Male; Myocardial Ischemia; Myocardial Reperfusion Injury; Phenethylamines; Piperazines; Potassium Channel Blockers; Sulfonamides; Time Factors

2005
Blockade of IKs by HMR 1556 increases the reverse rate-dependence of refractoriness prolongation by dofetilide in isolated rabbit ventricles.
    British journal of pharmacology, 2006, Volume: 148, Issue:3

    Topics: Action Potentials; Animals; Chromans; Delayed Rectifier Potassium Channels; Electrophysiology; In Vitro Techniques; Kinetics; Phenethylamines; Potassium Channel Blockers; Rabbits; Sulfonamides; Ventricular Function

2006
Combined pharmacological block of I(Kr) and I(Ks) increases short-term QT interval variability and provokes torsades de pointes.
    British journal of pharmacology, 2007, Volume: 151, Issue:7

    Topics: Animals; Blood Pressure; Chromans; Delayed Rectifier Potassium Channels; Dogs; Dose-Response Relationship, Drug; Drug Synergism; Electrocardiography; Female; Heart Conduction System; Heart Rate; Infusions, Intravenous; Long QT Syndrome; Male; Phenethylamines; Potassium; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Rabbits; Sodium; Species Specificity; Sulfonamides; Torsades de Pointes

2007
Double pharmacological challenge on repolarization opens new avenues for drug safety research.
    British journal of pharmacology, 2007, Volume: 151, Issue:7

    Topics: Animals; Chromans; Delayed Rectifier Potassium Channels; Dogs; Drug Synergism; Drug-Related Side Effects and Adverse Reactions; Electrocardiography; Humans; Long QT Syndrome; Phenethylamines; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Rabbits; Risk Factors; Sulfonamides; Torsades de Pointes

2007
Slow delayed rectifier K+ current block by HMR 1556 increases dispersion of repolarization and promotes Torsades de Pointes in rabbit ventricles.
    British journal of pharmacology, 2008, Volume: 155, Issue:8

    Topics: Animals; Chromans; Heart Ventricles; Male; Phenethylamines; Potassium Channel Blockers; Rabbits; Sulfonamides; Torsades de Pointes; Veratridine

2008
I(Kr) vs. I(Ks) blockade and arrhythmogenicity in normoxic rabbit Purkinje fibers: does it really make a difference?
    Fundamental & clinical pharmacology, 2011, Volume: 25, Issue:3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Chromans; Delayed Rectifier Potassium Channels; Epinephrine; Hydantoins; Imidazolidines; In Vitro Techniques; Male; Phenethylamines; Piperazines; Potassium Channel Blockers; Potassium Channels, Voltage-Gated; Purkinje Fibers; Rabbits; Sotalol; Sulfonamides

2011
Analysis of the contribution of I(to) to repolarization in canine ventricular myocardium.
    British journal of pharmacology, 2011, Volume: 164, Issue:1

    Topics: Action Potentials; Animals; Chromans; Dogs; Female; Heart Conduction System; Heart Ventricles; Male; Myocardium; Myocytes, Cardiac; Patch-Clamp Techniques; Phenethylamines; Potassium Channel Blockers; Potassium Channels; Sulfonamides; Ventricular Function

2011
Assessment of efficacy of proarrhythmia biomarkers in isolated rabbit hearts with attenuated repolarization reserve.
    Journal of cardiovascular pharmacology, 2014, Volume: 64, Issue:3

    Topics: Animals; Arrhythmias, Cardiac; Biomarkers; Chromans; Dose-Response Relationship, Drug; Electrocardiography; Female; Phenethylamines; Rabbits; Sulfonamides; Torsades de Pointes

2014
Contribution of ion currents to beat-to-beat variability of action potential duration in canine ventricular myocytes.
    Pflugers Archiv : European journal of physiology, 2015, Volume: 467, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium; Cardiotonic Agents; Cells, Cultured; Chromans; Dogs; Feedback, Physiological; Female; Heart Ventricles; Ion Channels; Ion Transport; Isoproterenol; Lidocaine; Male; Myocytes, Cardiac; Nisoldipine; Phenethylamines; Potassium Channel Blockers; Sulfonamides; Tetrodotoxin; Veratridine

2015