Page last updated: 2024-08-25

uk 68798 and almokalant

uk 68798 has been researched along with almokalant in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (44.44)18.2507
2000's3 (33.33)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Du, LP; Li, MY; Tsai, KC; Xia, L; You, QD1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Abrahamsson, C; Bäärnhielm, C; Carlsson, L; Danielsson, B; Duker, G; Ljung, B; Palmer, M1
Abrahamsson, C; Carlsson, L; Duker, G; Lundberg, C1
Brown-Woodman, PD; Danielsson, BR; Snow, MD; Webster, WS1
Plöen, L; Ritzen, EM; Setchell, BP1
Carmeliet, E; Vereecke, J1
Amos, GJ; Carlsson, L; Duker, G; Jacobson, I1
Abi-Gerges, N; Boyett, MR; Davies, MR; Di Veroli, GY; Zhang, H1

Other Studies

9 other study(ies) available for uk 68798 and almokalant

ArticleYear
The pharmacophore hypotheses of I(Kr) potassium channel blockers: novel class III antiarrhythmic agents.
    Bioorganic & medicinal chemistry letters, 2004, Sep-20, Volume: 14, Issue:18

    Topics: Anti-Arrhythmia Agents; Models, Biological; Models, Molecular; Potassium Channel Blockers; Potassium Channels; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2004
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Induction of rhythm abnormalities in the fetal rat heart. A tentative mechanism for the embryotoxic effect of the class III antiarrhythmic agent almokalant.
    Cardiovascular research, 1994, Volume: 28, Issue:3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Cells, Cultured; Culture Techniques; Female; Fetal Death; Fetal Heart; Heart; Heart Rate; Myocardium; Phenethylamines; Pregnancy; Propanolamines; Rats; Rats, Sprague-Dawley; Sotalol; Sulfonamides

1994
Electrophysiological and inotropic effects of H 234/09 (almokalant) in vitro: a comparison with two other novel IK blocking drugs, UK-68,798 (dofetilide) and E-4031.
    Cardiovascular research, 1993, Volume: 27, Issue:5

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Cats; Dose-Response Relationship, Drug; Heart; In Vitro Techniques; Male; Myocardial Contraction; Papillary Muscles; Phenethylamines; Piperidines; Propanolamines; Purkinje Fibers; Pyridines; Rabbits; Stimulation, Chemical; Sulfonamides

1993
Teratogenic potential of almokalant, dofetilide, and d-sotalol: drugs with potassium channel blocking activity.
    Teratology, 1996, Volume: 53, Issue:3

    Topics: Abnormalities, Drug-Induced; Animals; Anti-Arrhythmia Agents; Cleft Palate; Dose-Response Relationship, Drug; Embryonic and Fetal Development; Female; Heart Rate, Fetal; Limb Deformities, Congenital; Male; Organ Culture Techniques; Phenethylamines; Potassium Channel Blockers; Pregnancy; Pregnancy Outcome; Propanolamines; Rats; Rats, Sprague-Dawley; Sotalol; Sulfonamides

1996
Reduction in fluid secretion by rat testis by drugs that block potassium channels.
    Journal of reproduction and fertility, 1998, Volume: 112, Issue:1

    Topics: Analysis of Variance; Androgen-Binding Protein; Animals; Anti-Arrhythmia Agents; Body Weight; Inositol; Magnesium; Male; Organ Size; Phenethylamines; Potassium; Potassium Channel Blockers; Propanolamines; Rats; Rats, Sprague-Dawley; Semen; Sodium; Spermatogenesis; Sulfonamides; Testis

1998
The effect of external pH on the delayed rectifying K+ current in cardiac ventricular myocytes.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 439, Issue:6

    Topics: Acids; Animals; Electrophysiology; Extracellular Space; Guinea Pigs; Hydrogen-Ion Concentration; Myocardium; Phenethylamines; Potassium Channel Blockers; Potassium Channels; Propanolamines; Rabbits; Sulfonamides; Time Factors; Ventricular Function

2000
Block of HERG-carried K+ currents by the new repolarization delaying agent H 345/52.
    Journal of cardiovascular electrophysiology, 2003, Volume: 14, Issue:6

    Topics: Action Potentials; Alkanes; Animals; Anti-Arrhythmia Agents; Binding, Competitive; Bridged Bicyclo Compounds; Cation Transport Proteins; Cell Line; DNA-Binding Proteins; Dose-Response Relationship, Drug; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Fibroblasts; Heart; Humans; Inhibitory Concentration 50; Membrane Potentials; Mice; Models, Animal; Patch-Clamp Techniques; Phenethylamines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Predictive Value of Tests; Propanolamines; Sulfonamides; Time Factors; Trans-Activators; Transcriptional Regulator ERG

2003
High-throughput screening of drug-binding dynamics to HERG improves early drug safety assessment.
    American journal of physiology. Heart and circulatory physiology, 2013, Jan-01, Volume: 304, Issue:1

    Topics: Action Potentials; Animals; CHO Cells; Cisapride; Computer Simulation; Cricetinae; Cricetulus; Dogs; Dose-Response Relationship, Drug; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; High-Throughput Screening Assays; Humans; Kinetics; Long QT Syndrome; Markov Chains; Models, Cardiovascular; Patch-Clamp Techniques; Phenethylamines; Potassium Channel Blockers; Propanolamines; Protein Binding; Risk Assessment; Sulfonamides; Torsades de Pointes; Toxicity Tests; Transfection

2013