Page last updated: 2024-09-03

uh 301 and citalopram

uh 301 has been researched along with citalopram in 3 studies

Compound Research Comparison

Studies
(uh 301)
Trials
(uh 301)
Recent Studies (post-2010)
(uh 301)
Studies
(citalopram)
Trials
(citalopram)
Recent Studies (post-2010) (citalopram)
52085,3481,4242,350

Protein Interaction Comparison

ProteinTaxonomyuh 301 (IC50)citalopram (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)2.196
AromataseRattus norvegicus (Norway rat)0.0018
Sodium-dependent noradrenaline transporter Homo sapiens (human)2.196
Alpha-1D adrenergic receptorHomo sapiens (human)3.289
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
Sodium-dependent serotonin transporterHomo sapiens (human)0.0227
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.0027
Histamine H1 receptorHomo sapiens (human)3.194
5-hydroxytryptamine receptor 2BHomo sapiens (human)1.839
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.1869
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.398
TransporterRattus norvegicus (Norway rat)8.8

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arborelius, L; Grillner, P; Hacksell, U; Hertel, P; Höök, BB; Nomikos, GG; Svensson, TH1
Hjorth, S1
Arborelius, L; Grillner, P; Hacksell, U; Hertel, P; Höök, BB; Nomikos, GG; Salmi, P; Svensson, TH1

Other Studies

3 other study(ies) available for uh 301 and citalopram

ArticleYear
5-HT1A receptor antagonists increase the activity of serotonergic cells in the dorsal raphe nucleus in rats treated acutely or chronically with citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Citalopram; Electrophysiology; Extracellular Space; Male; Neurons; Piperazines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Synaptic Transmission

1995
Serotonin 5-HT1A autoreceptor blockade potentiates the ability of the 5-HT reuptake inhibitor citalopram to increase nerve terminal output of 5-HT in vivo: a microdialysis study.
    Journal of neurochemistry, 1993, Volume: 60, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Chromatography, High Pressure Liquid; Citalopram; Dialysis; Feedback; Hippocampus; Male; Microchemistry; Nerve Endings; Penbutolol; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists

1993
The 5-HT1A receptor antagonist (S)-UH-301 augments the increase in extracellular concentrations of 5-HT in the frontal cortex produced by both acute and chronic treatment with citalopram.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Body Temperature; Citalopram; Extracellular Space; Male; Microdialysis; Raphe Nuclei; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996