Page last updated: 2024-08-25

ubenimex and sincalide

ubenimex has been researched along with sincalide in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19904 (50.00)18.7374
1990's2 (25.00)18.2507
2000's0 (0.00)29.6817
2010's2 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Griesbacher, T; Hill, RG; Hughes, J; Leighton, GE1
Hill, RG; Hughes, J; Pittaway, KM1
Charpentier, B; Durieux, C; Pelaprat, D; Roques, BP1
Bui, ND; Deschodt-Lanckman, M1
Devaux, B; Rose, C; Schwartz, JC; Silhouette, B; Vargas, F1
Gibson, AM; McDermott, JR; Wilson, C1

Reviews

1 review(s) available for ubenimex and sincalide

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010

Other Studies

7 other study(ies) available for ubenimex and sincalide

ArticleYear
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Reduction of food intake by central administration of cholecystokinin octapeptide in the rat is dependent upon inhibition of brain peptidases.
    British journal of pharmacology, 1989, Volume: 96, Issue:1

    Topics: Animals; Brain; Captopril; Ceruletide; Eating; Injections, Intraventricular; Leucine; Male; Protease Inhibitors; Rats; Rats, Inbred Strains; Sincalide; Thiorphan

1989
Antinociceptive action of cholecystokinin octapeptide (CCK 8) and related peptides in rats and mice: effects of naloxone and peptidase inhibitors.
    Neuropharmacology, 1987, Volume: 26, Issue:4

    Topics: Animals; Captopril; FMRFamide; Gastrins; Leucine; Male; Mice; Naloxone; Neuropeptides; Pain; Protease Inhibitors; Rats; Rats, Inbred Strains; Reaction Time; Sincalide; Tetragastrin; Thiorphan; Tiopronin

1987
Investigation on the metabolism of CCK8 analogues by rat brain slices.
    Neuropeptides, 1986, Volume: 7, Issue:1

    Topics: Animals; Cerebral Cortex; Chloromercuribenzoates; Corpus Striatum; Hydrolysis; In Vitro Techniques; Leucine; p-Chloromercuribenzoic Acid; Peptide Fragments; Sincalide; Swine; Synaptic Membranes; Thiorphan; Tiopronin

1986
Cholecystokinin octa- and tetrapeptide degradation by synaptic membranes. I. Evidence for competition with enkephalins for in vitro common degradation pathways.
    Peptides, 1981, Volume: 2 Suppl 2

    Topics: Aminopeptidases; Animals; Cholecystokinin; Chromatography, DEAE-Cellulose; Endorphins; Enkephalin, Leucine; Enkephalins; Gastrins; Kinetics; Leucine; Male; Peptide Fragments; Rats; Sincalide; Synaptic Membranes; Tetragastrin; Tryptophan

1981
Characterization of a serine peptidase responsible for the inactivation of endogenous cholecystokinin in human brain.
    Neuropeptides, 1995, Volume: 28, Issue:3

    Topics: Amino Acid Sequence; Aminopeptidases; Animals; Cerebral Cortex; Humans; Isoflurophate; Leucine; Molecular Sequence Data; Neprilysin; Nerve Tissue Proteins; Rats; Serine Endopeptidases; Serpins; Sincalide; Thiorphan

1995
Purification and characterization of tripeptidylpeptidase-II from post-mortem human brain.
    Neurochemical research, 1993, Volume: 18, Issue:7

    Topics: Amino Acid Sequence; Aminopeptidases; Angiotensin III; Cerebral Cortex; Chromatography; Chromatography, Gel; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Humans; Hydrogen-Ion Concentration; Leucine; Molecular Sequence Data; Molecular Weight; Neurokinin A; Neuropeptides; Serine Endopeptidases; Sincalide; Substrate Specificity

1993