Page last updated: 2024-09-03

u 99194a and sb 277011

u 99194a has been researched along with sb 277011 in 4 studies

Compound Research Comparison

Studies
(u 99194a)
Trials
(u 99194a)
Recent Studies (post-2010)
(u 99194a)
Studies
(sb 277011)
Trials
(sb 277011)
Recent Studies (post-2010) (sb 277011)
6201098041

Protein Interaction Comparison

ProteinTaxonomyu 99194a (IC50)sb 277011 (IC50)
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.6598

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gál, K; Gyertyán, I1
Gyertyán, I; Sághy, K1
Barth, V; Giros, B; Gleason, SD; Johansson, AM; Need, AB; Nomikos, GG; Overshiner, C; Perry, K; Tzavara, ET; Wade, M; Witkin, JM1
Newton, CL; Strange, PG; Wood, MD1

Other Studies

4 other study(ies) available for u 99194a and sb 277011

ArticleYear
Dopamine D3 receptor ligands show place conditioning effect but do not influence cocaine-induced place preference.
    Neuroreport, 2003, Jan-20, Volume: 14, Issue:1

    Topics: Animals; Avoidance Learning; Benzazepines; Benzopyrans; Cocaine; Conditioning, Classical; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Indans; Male; Naphthalenes; Nitriles; Oxazines; Piperazines; Pyrrolidines; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Reward; Spatial Behavior; Substance-Related Disorders; Tetrahydroisoquinolines; Tetrahydronaphthalenes

2003
Effects of dopamine D3 receptor antagonists on spontaneous and agonist-reduced motor activity in NMRI mice and Wistar rats: comparative study with nafadotride, U 99194A and SB 277011.
    Behavioural pharmacology, 2004, Volume: 15, Issue:4

    Topics: Animals; Benzopyrans; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Antagonism; Indans; Injections, Subcutaneous; Male; Mice; Motor Activity; Naphthalenes; Nitriles; Oxazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Species Specificity; Tetrahydroisoquinolines; Tetrahydronaphthalenes

2004
In vivo occupancy of dopamine D3 receptors by antagonists produces neurochemical and behavioral effects of potential relevance to attention-deficit-hyperactivity disorder.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 344, Issue:2

    Topics: Animals; Attention Deficit Disorder with Hyperactivity; Behavior, Animal; Brain; Brain Chemistry; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indans; Male; Microdialysis; Molecular Structure; Nitriles; Pattern Recognition, Visual; Protein Binding; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Dopamine D3; Tetrahydroisoquinolines

2013
Examining the Effects of Sodium Ions on the Binding of Antagonists to Dopamine D2 and D3 Receptors.
    PloS one, 2016, Volume: 11, Issue:7

    Topics: Animals; Binding, Competitive; Biphenyl Compounds; Cell Line, Tumor; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Indans; Indoles; Ions; Ligands; Molecular Structure; Mutation; Nitriles; Piperazines; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Sf9 Cells; Sodium; Spodoptera; Tetrahydroisoquinolines

2016