u 99194a has been researched along with sb 277011 in 4 studies
Studies (u 99194a) | Trials (u 99194a) | Recent Studies (post-2010) (u 99194a) | Studies (sb 277011) | Trials (sb 277011) | Recent Studies (post-2010) (sb 277011) |
---|---|---|---|---|---|
62 | 0 | 10 | 98 | 0 | 41 |
Protein | Taxonomy | u 99194a (IC50) | sb 277011 (IC50) |
---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 1.6598 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (50.00) | 29.6817 |
2010's | 2 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Gál, K; Gyertyán, I | 1 |
Gyertyán, I; Sághy, K | 1 |
Barth, V; Giros, B; Gleason, SD; Johansson, AM; Need, AB; Nomikos, GG; Overshiner, C; Perry, K; Tzavara, ET; Wade, M; Witkin, JM | 1 |
Newton, CL; Strange, PG; Wood, MD | 1 |
4 other study(ies) available for u 99194a and sb 277011
Article | Year |
---|---|
Dopamine D3 receptor ligands show place conditioning effect but do not influence cocaine-induced place preference.
Topics: Animals; Avoidance Learning; Benzazepines; Benzopyrans; Cocaine; Conditioning, Classical; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Haloperidol; Indans; Male; Naphthalenes; Nitriles; Oxazines; Piperazines; Pyrrolidines; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Reward; Spatial Behavior; Substance-Related Disorders; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2003 |
Effects of dopamine D3 receptor antagonists on spontaneous and agonist-reduced motor activity in NMRI mice and Wistar rats: comparative study with nafadotride, U 99194A and SB 277011.
Topics: Animals; Benzopyrans; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Antagonism; Indans; Injections, Subcutaneous; Male; Mice; Motor Activity; Naphthalenes; Nitriles; Oxazines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Species Specificity; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2004 |
In vivo occupancy of dopamine D3 receptors by antagonists produces neurochemical and behavioral effects of potential relevance to attention-deficit-hyperactivity disorder.
Topics: Animals; Attention Deficit Disorder with Hyperactivity; Behavior, Animal; Brain; Brain Chemistry; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indans; Male; Microdialysis; Molecular Structure; Nitriles; Pattern Recognition, Visual; Protein Binding; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Dopamine D3; Tetrahydroisoquinolines | 2013 |
Examining the Effects of Sodium Ions on the Binding of Antagonists to Dopamine D2 and D3 Receptors.
Topics: Animals; Binding, Competitive; Biphenyl Compounds; Cell Line, Tumor; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Indans; Indoles; Ions; Ligands; Molecular Structure; Mutation; Nitriles; Piperazines; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Sf9 Cells; Sodium; Spodoptera; Tetrahydroisoquinolines | 2016 |