Page last updated: 2024-09-03

u 99194a and raclopride

u 99194a has been researched along with raclopride in 6 studies

Compound Research Comparison

Studies
(u 99194a)
Trials
(u 99194a)
Recent Studies (post-2010)
(u 99194a)
Studies
(raclopride)
Trials
(raclopride)
Recent Studies (post-2010) (raclopride)
620101,802132419

Protein Interaction Comparison

ProteinTaxonomyu 99194a (IC50)raclopride (IC50)
D(2) dopamine receptorHomo sapiens (human)0.052
D(2) dopamine receptorMus musculus (house mouse)0.032
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0279

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (16.67)18.2507
2000's3 (50.00)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carlsson, A; Haadsma-Svensson, SR; Smith, MW; Svensson, K; Waters, N1
Hillefors, M; von Euler, G1
Cunningham, CL; Dickinson, SD; Lee, EL; Rindal, K1
Bastianetto, S; Danik, M; Mennicken, F; Quirion, R; Williams, S1
Brudzynski, SM; Komadoski, M; St Pierre, J1
Liang, SL; Pan, JT1

Other Studies

6 other study(ies) available for u 99194a and raclopride

ArticleYear
The dopamine D3-receptor: a postsynaptic receptor inhibitory on rat locomotor activity.
    Journal of neural transmission. General section, 1993, Volume: 94, Issue:1

    Topics: Aminoquinolines; Animals; Apomorphine; CHO Cells; Corpus Striatum; Cricetinae; Dextroamphetamine; Dopamine; Dopamine Antagonists; Drug Interactions; Indans; Male; Methyltyrosines; Models, Biological; Motor Activity; Nucleus Accumbens; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Recombinant Fusion Proteins; Reserpine; Salicylamides; Spiperone; Stimulation, Chemical

1993
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
    Neurochemistry international, 2001, Volume: 38, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes

2001
Lack of effect of dopamine receptor blockade on expression of ethanol-induced conditioned place preference in mice.
    Psychopharmacology, 2003, Volume: 165, Issue:3

    Topics: Animals; Association Learning; Benzazepines; Conditioning, Classical; Dopamine Antagonists; Dose-Response Relationship, Drug; Ethanol; Indans; Male; Mice; Mice, Inbred DBA; Motivation; Motor Activity; Raclopride; Receptors, Dopamine

2003
Prototypical antipsychotic drugs protect hippocampal neuronal cultures against cell death induced by growth medium deprivation.
    BMC neuroscience, 2006, Mar-30, Volume: 7

    Topics: Animals; Anisoles; Antipsychotic Agents; Benzazepines; Butaclamol; Caspase Inhibitors; Cell Death; Cells, Cultured; Chlorpromazine; Clozapine; Domperidone; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Ginkgo biloba; Haloperidol; Hippocampus; Indans; Isoxazoles; Neurons; Neuroprotective Agents; Peptides; Piperidines; Plant Extracts; Propylamines; Raclopride; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, N-Methyl-D-Aspartate; Remoxipride; Risperidone; Sulpiride

2006
Quinpirole-induced 50 kHz ultrasonic vocalization in the rat: role of D2 and D3 dopamine receptors.
    Behavioural brain research, 2012, Jan-15, Volume: 226, Issue:2

    Topics: Animals; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indans; Male; Microinjections; Nucleus Accumbens; Quinpirole; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Vocalization, Animal

2012
An endogenous dopaminergic tone acting on dopamine D3 receptors may be involved in diurnal changes of tuberoinfundibular dopaminergic neuron activity and prolactin secretion in estrogen-primed ovariectomized rats.
    Brain research bulletin, 2012, Feb-10, Volume: 87, Issue:2-3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Analysis of Variance; Animals; Benzopyrans; Chromatography, High Pressure Liquid; Circadian Rhythm; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopaminergic Neurons; Dose-Response Relationship, Drug; Drug Combinations; Enzyme Inhibitors; Estrogens; Female; Gene Expression Regulation; Hydrazines; Hypothalamic Area, Lateral; Indans; Oligodeoxyribonucleotides, Antisense; Ovariectomy; Oxazines; Prolactin; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; RNA, Messenger; Time Factors

2012