Page last updated: 2024-09-03

u 99194a and gr 103691

u 99194a has been researched along with gr 103691 in 5 studies

Compound Research Comparison

Studies
(u 99194a)
Trials
(u 99194a)
Recent Studies (post-2010)
(u 99194a)
Studies
(gr 103691)
Trials
(gr 103691)
Recent Studies (post-2010) (gr 103691)
6201028017

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's1 (20.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clifford, JJ; Waddington, JL1
Audinot, V; Bervoets, K; Brocco, M; Dekeyne, A; Desposte, I; Gluck, L; Gobert, A; Lejeune, F; Millan, MJ; Newman-Tancredi, A; Rivet, JM1
Chen, JC; Chen, PC; Chiang, YC1
Anderson, NJ; Chappell, AM; Christian, DT; Diaz, MR; McCool, BA1
Newton, CL; Strange, PG; Wood, MD1

Other Studies

5 other study(ies) available for u 99194a and gr 103691

ArticleYear
Heterogeneity of behavioural profile between three new putative selective D3 dopamine receptor antagonists using an ethologically based approach.
    Psychopharmacology, 1998, Volume: 136, Issue:3

    Topics: Animals; Behavior, Animal; Biphenyl Compounds; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Grooming; Haloperidol; Indans; Male; Motor Activity; Naphthalenes; Piperazines; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Stereotyped Behavior

1998
A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:1

    Topics: 2-Naphthylamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Biphenyl Compounds; Body Temperature; Catalepsy; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Furans; Humans; Indans; Naphthalenes; Oxazines; Piperazines; Prolactin; Pyrrolidines; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3

1998
D(3) dopamine receptors are down-regulated in amphetamine sensitized rats and their putative antagonists modulate the locomotor sensitization to amphetamine.
    Brain research, 2003, May-16, Volume: 972, Issue:1-2

    Topics: Amphetamine; Animals; Behavior, Animal; Binding, Competitive; Biphenyl Compounds; Central Nervous System Stimulants; Dopamine Agonists; Dopamine Antagonists; Down-Regulation; Drug Interactions; Indans; Male; Motor Activity; Piperazines; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; RNA, Ribosomal, 18S; Tetrahydronaphthalenes; Time Factors; Tritium

2003
Dopamine D3-like receptors modulate anxiety-like behavior and regulate GABAergic transmission in the rat lateral/basolateral amygdala.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2011, Volume: 36, Issue:5

    Topics: Amygdala; Animals; Anxiety; Benzopyrans; Biphenyl Compounds; Disease Models, Animal; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Exploratory Behavior; gamma-Aminobutyric Acid; In Vitro Techniques; Indans; Inhibitory Postsynaptic Potentials; Male; Maze Learning; Microinjections; Neurons; Oxazines; Patch-Clamp Techniques; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Synaptic Transmission

2011
Examining the Effects of Sodium Ions on the Binding of Antagonists to Dopamine D2 and D3 Receptors.
    PloS one, 2016, Volume: 11, Issue:7

    Topics: Animals; Binding, Competitive; Biphenyl Compounds; Cell Line, Tumor; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Indans; Indoles; Ions; Ligands; Molecular Structure; Mutation; Nitriles; Piperazines; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Sf9 Cells; Sodium; Spodoptera; Tetrahydroisoquinolines

2016
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