u 73343 has been researched along with thapsigargin in 14 studies
Studies (u 73343) | Trials (u 73343) | Recent Studies (post-2010) (u 73343) | Studies (thapsigargin) | Trials (thapsigargin) | Recent Studies (post-2010) (thapsigargin) |
---|---|---|---|---|---|
97 | 0 | 6 | 5,234 | 3 | 918 |
Protein | Taxonomy | u 73343 (IC50) | thapsigargin (IC50) |
---|---|---|---|
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | 0.002 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 4 (28.57) | 18.2507 |
2000's | 10 (71.43) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Fukuda, Y; Sakaki, Y; Yamashita, M | 1 |
Hashimoto, T; Ishii, T; Ohmori, H | 1 |
Farndale, RW; Heemskerk, JW; Sage, SO | 1 |
Farndale, RW; Feijge, MA; Heemskerk, JW; Sage, SO | 1 |
Chen, TH; Cheng, H; Hsu, WH; Yibchok-Anun, S | 1 |
Eglen, RM; MacLennan, SJ; Martin, GR; Reynen, PH | 1 |
Bellon, G; Fawzi, A; Kefalides, NA; Monboisse, JC; Robinet, A; Ziaie, Z | 1 |
Scofield, MA; Wangemann, P; Wonneberger, K | 1 |
Kato, M; Sakuma, Y; Sudo, T | 1 |
Fukuhara, S; Inagaki, C; Oshiro, A; Otani, H; Yagi, Y | 1 |
Abu-Basha, EA; Cheng, H; Ding, J; Hsu, WH; Ioudina, M; Yibchok-anun, S | 1 |
Hjertos, B; Slusarski, DC; Westfall, TA | 1 |
Baly, C; Caillol, M; Durieux, D; Grébert, D; Levasseur, G; Salesse, R | 1 |
Chang, CH; Chang, HT; Chen, WC; Chou, CT; Hsieh, CH; Hsu, SS; Jan, CR; Lin, KL; Liu, CS; Liu, SI; Wang, JL | 1 |
14 other study(ies) available for u 73343 and thapsigargin
Article | Year |
---|---|
Muscarinic and purinergic Ca2+ mobilizations in the neural retina of early embryonic chick.
Topics: Acetylcholine; Adenosine Triphosphate; Animals; Calcium; Carbachol; Chick Embryo; Enzyme Inhibitors; Estrenes; GTP-Binding Proteins; Lithium; Muscarinic Agonists; Neurons; Pertussis Toxin; Phosphodiesterase Inhibitors; Purinergic Agonists; Pyrrolidinones; Receptors, Muscarinic; Receptors, Purinergic; Retina; Signal Transduction; Thapsigargin; Virulence Factors, Bordetella | 1996 |
Release of Ca2+ is the crucial step for the potentiation of IPSCs in the cultured cerebellar Purkinje cells of the rat.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Calcium Channels; Chelating Agents; Cycloleucine; Egtazic Acid; Enzyme Inhibitors; Estrenes; Evoked Potentials; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Heparin; Neuroprotective Agents; Phosphodiesterase Inhibitors; Purkinje Cells; Pyrrolidinones; Rats; Receptors, Metabotropic Glutamate; Ruthenium Red; Synapses; Thapsigargin; Type C Phospholipases | 1996 |
Effects of U73122 and U73343 on human platelet calcium signalling and protein tyrosine phosphorylation.
Topics: Arachidonic Acid; Aspirin; Blood Platelets; Blood Proteins; Calcium; Collagen; Estrenes; Humans; Phosphodiesterase Inhibitors; Phosphorylation; Phosphotyrosine; Protein-Tyrosine Kinases; Pyrrolidinones; Signal Transduction; Thapsigargin; Thrombin; Thromboxane A2; Type C Phospholipases | 1997 |
Human platelet activation is inhibited upstream of the activation of phospholipase A2 by U73343.
Topics: Blood Platelets; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Estrenes; Humans; Phospholipases A; Phospholipases A2; Platelet Aggregation Inhibitors; Protein-Tyrosine Kinases; Pyrrolidinones; Thapsigargin; Thrombin | 1997 |
Mechanisms of AVP-induced glucagon release in clonal alpha-cells in-R1-G9: involvement of Ca(2+)-dependent and -independent pathways.
Topics: Amino Acid Chloromethyl Ketones; Animals; Arginine Vasopressin; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Clone Cells; Cricetinae; Cyclic AMP; Enzyme Inhibitors; Estrenes; Glucagon; Inositol 1,4,5-Trisphosphate; Nimodipine; Phosphodiesterase Inhibitors; Pyrrolidinones; Renal Agents; Serine Proteinase Inhibitors; Thapsigargin | 2000 |
Characterization of human recombinant alpha(2A)-adrenoceptors expressed in Chinese hamster lung cells using intracellular Ca(2+) changes: evidence for cross-talk between recombinant alpha(2A)- and native alpha(1)-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aniline Compounds; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Calcium; Cell Line; Cricetinae; Dexmedetomidine; Dose-Response Relationship, Drug; Doxazosin; Estrenes; Fluorescence; Gene Expression; Humans; Imidazoles; Norepinephrine; Prazosin; Pyrrolidinones; Quinoxalines; Radioligand Assay; Receptor Cross-Talk; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Signal Transduction; Tetrahydronaphthalenes; Thapsigargin; Xanthenes; Yohimbine | 2000 |
A peptide of the alpha 3(IV) chain of type IV collagen modulates stimulated neutrophil function via activation of cAMP-dependent protein kinase and Ser/Thr protein phosphatase.
Topics: Adenosine; Amino Acid Sequence; Autoantigens; Calcium; Carbazoles; Chelating Agents; Collagen; Collagen Type IV; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Antagonists; Egtazic Acid; Enzyme Inhibitors; Estrenes; Humans; Indoles; Marine Toxins; Molecular Sequence Data; Neutrophils; Okadaic Acid; Oxazoles; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphoprotein Phosphatases; Pyrroles; Pyrrolidinones; Respiratory Burst; Signal Transduction; Thapsigargin; Trifluoperazine | 2000 |
Evidence for a calcium-sensing receptor in the vascular smooth muscle cells of the spiral modiolar artery.
Topics: Arteries; Base Sequence; Calcium; Calcium Channel Blockers; Cations, Divalent; Cochlea; DNA, Complementary; Enzyme Inhibitors; Estrenes; Molecular Sequence Data; Muscle, Smooth, Vascular; Nickel; Nifedipine; Pyrrolidinones; Receptors, Calcium-Sensing; Receptors, Cell Surface; Ryanodine; Thapsigargin; Type C Phospholipases; Vasodilator Agents | 2000 |
Bradykinin and angiotensin II-induced [Ca2+]i rise in cultured rat pituitary folliculo-stellate cells.
Topics: Angiotensin II; Animals; Bradykinin; Caffeine; Calcium; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Galanin; Male; Neuropeptides; Neurotensin; Phosphodiesterase Inhibitors; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Pyrrolidinones; Rats; Rats, Wistar; Ryanodine; Thapsigargin; Type C Phospholipases; Vasoconstrictor Agents | 2001 |
Protease-activated receptor-2-mediated Ca2+ signaling in guinea pig tracheal epithelial cells.
Topics: Animals; Calcium Signaling; Chelating Agents; Enzyme Inhibitors; Epithelial Cells; Estrenes; Fura-2; Guinea Pigs; Manganese; Oligopeptides; Pyrrolidinones; Receptor, PAR-2; Receptors, Thrombin; Thapsigargin; Trachea; Trypsin; Type C Phospholipases | 2002 |
Mechanisms of bradykinin-induced glucagon release in clonal alpha-cells In-R1-G9: involvement of Ca(2+)-dependent and -independent pathways.
Topics: Animals; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Chelating Agents; Clone Cells; Cricetinae; Egtazic Acid; Endoplasmic Reticulum; Enzyme Inhibitors; Estrenes; Glucagon; Glucagonoma; GTP-Binding Proteins; Heparin; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Mesocricetus; Microinjections; Pancreatic Neoplasms; Pertussis Toxin; Phospholipase D; Pyrrolidinones; Receptor, Bradykinin B2; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thapsigargin; Tumor Cells, Cultured; Type C Phospholipases | 2002 |
Requirement for intracellular calcium modulation in zebrafish dorsal-ventral patterning.
Topics: Animals; beta Catenin; Body Patterning; Calcium; Cytoskeletal Proteins; Diphosphonates; Dose-Response Relationship, Drug; Embryo, Nonmammalian; Enzyme Inhibitors; Estrenes; Gene Expression Regulation, Developmental; Models, Biological; Phenotype; Phosphatidylinositols; Pyrrolidinones; Signal Transduction; Thapsigargin; Trans-Activators; Type C Phospholipases; Zebrafish; Zebrafish Proteins | 2003 |
Anatomical and functional evidence for a role of arginine-vasopressin (AVP) in rat olfactory epithelium cells.
Topics: Animals; Animals, Newborn; Arginine Vasopressin; Boron Compounds; Cadmium Chloride; Calcium; Calcium Channel Blockers; Cells, Cultured; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Estrenes; Extracellular Space; Fura-2; Immunohistochemistry; Male; Neurons; Olfactory Mucosa; Oxytocin; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Oxytocin; Receptors, Vasopressin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thapsigargin; Time Factors; Verapamil | 2004 |
Nonylphenol-induced Ca2+ elevation and Ca2+-independent cell death in human osteosarcoma cells.
Topics: Calcium; Calcium Channel Blockers; Cell Death; Cell Line, Tumor; Cell Proliferation; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; Estrenes; Fluorescent Dyes; Fura-2; Humans; Osteoblasts; Osteosarcoma; Phenols; Pyrrolidinones; Spectrometry, Fluorescence; Tetrazolium Salts; Thapsigargin; Type C Phospholipases | 2005 |