Page last updated: 2024-09-02

u 73343 and thapsigargin

u 73343 has been researched along with thapsigargin in 14 studies

Compound Research Comparison

Studies
(u 73343)
Trials
(u 73343)
Recent Studies (post-2010)
(u 73343)
Studies
(thapsigargin)
Trials
(thapsigargin)
Recent Studies (post-2010) (thapsigargin)
97065,2343918

Protein Interaction Comparison

ProteinTaxonomyu 73343 (IC50)thapsigargin (IC50)
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1Oryctolagus cuniculus (rabbit)0.002

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (28.57)18.2507
2000's10 (71.43)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fukuda, Y; Sakaki, Y; Yamashita, M1
Hashimoto, T; Ishii, T; Ohmori, H1
Farndale, RW; Heemskerk, JW; Sage, SO1
Farndale, RW; Feijge, MA; Heemskerk, JW; Sage, SO1
Chen, TH; Cheng, H; Hsu, WH; Yibchok-Anun, S1
Eglen, RM; MacLennan, SJ; Martin, GR; Reynen, PH1
Bellon, G; Fawzi, A; Kefalides, NA; Monboisse, JC; Robinet, A; Ziaie, Z1
Scofield, MA; Wangemann, P; Wonneberger, K1
Kato, M; Sakuma, Y; Sudo, T1
Fukuhara, S; Inagaki, C; Oshiro, A; Otani, H; Yagi, Y1
Abu-Basha, EA; Cheng, H; Ding, J; Hsu, WH; Ioudina, M; Yibchok-anun, S1
Hjertos, B; Slusarski, DC; Westfall, TA1
Baly, C; Caillol, M; Durieux, D; Grébert, D; Levasseur, G; Salesse, R1
Chang, CH; Chang, HT; Chen, WC; Chou, CT; Hsieh, CH; Hsu, SS; Jan, CR; Lin, KL; Liu, CS; Liu, SI; Wang, JL1

Other Studies

14 other study(ies) available for u 73343 and thapsigargin

ArticleYear
Muscarinic and purinergic Ca2+ mobilizations in the neural retina of early embryonic chick.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1996, Volume: 14, Issue:6

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Calcium; Carbachol; Chick Embryo; Enzyme Inhibitors; Estrenes; GTP-Binding Proteins; Lithium; Muscarinic Agonists; Neurons; Pertussis Toxin; Phosphodiesterase Inhibitors; Purinergic Agonists; Pyrrolidinones; Receptors, Muscarinic; Receptors, Purinergic; Retina; Signal Transduction; Thapsigargin; Virulence Factors, Bordetella

1996
Release of Ca2+ is the crucial step for the potentiation of IPSCs in the cultured cerebellar Purkinje cells of the rat.
    The Journal of physiology, 1996, Dec-15, Volume: 497 ( Pt 3)

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcium; Calcium Channels; Chelating Agents; Cycloleucine; Egtazic Acid; Enzyme Inhibitors; Estrenes; Evoked Potentials; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Heparin; Neuroprotective Agents; Phosphodiesterase Inhibitors; Purkinje Cells; Pyrrolidinones; Rats; Receptors, Metabotropic Glutamate; Ruthenium Red; Synapses; Thapsigargin; Type C Phospholipases

1996
Effects of U73122 and U73343 on human platelet calcium signalling and protein tyrosine phosphorylation.
    Biochimica et biophysica acta, 1997, Jan-10, Volume: 1355, Issue:1

    Topics: Arachidonic Acid; Aspirin; Blood Platelets; Blood Proteins; Calcium; Collagen; Estrenes; Humans; Phosphodiesterase Inhibitors; Phosphorylation; Phosphotyrosine; Protein-Tyrosine Kinases; Pyrrolidinones; Signal Transduction; Thapsigargin; Thrombin; Thromboxane A2; Type C Phospholipases

1997
Human platelet activation is inhibited upstream of the activation of phospholipase A2 by U73343.
    Biochemical pharmacology, 1997, May-09, Volume: 53, Issue:9

    Topics: Blood Platelets; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Estrenes; Humans; Phospholipases A; Phospholipases A2; Platelet Aggregation Inhibitors; Protein-Tyrosine Kinases; Pyrrolidinones; Thapsigargin; Thrombin

1997
Mechanisms of AVP-induced glucagon release in clonal alpha-cells in-R1-G9: involvement of Ca(2+)-dependent and -independent pathways.
    British journal of pharmacology, 2000, Volume: 129, Issue:2

    Topics: Amino Acid Chloromethyl Ketones; Animals; Arginine Vasopressin; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Line; Clone Cells; Cricetinae; Cyclic AMP; Enzyme Inhibitors; Estrenes; Glucagon; Inositol 1,4,5-Trisphosphate; Nimodipine; Phosphodiesterase Inhibitors; Pyrrolidinones; Renal Agents; Serine Proteinase Inhibitors; Thapsigargin

2000
Characterization of human recombinant alpha(2A)-adrenoceptors expressed in Chinese hamster lung cells using intracellular Ca(2+) changes: evidence for cross-talk between recombinant alpha(2A)- and native alpha(1)-adrenoceptors.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aniline Compounds; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Calcium; Cell Line; Cricetinae; Dexmedetomidine; Dose-Response Relationship, Drug; Doxazosin; Estrenes; Fluorescence; Gene Expression; Humans; Imidazoles; Norepinephrine; Prazosin; Pyrrolidinones; Quinoxalines; Radioligand Assay; Receptor Cross-Talk; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Signal Transduction; Tetrahydronaphthalenes; Thapsigargin; Xanthenes; Yohimbine

2000
A peptide of the alpha 3(IV) chain of type IV collagen modulates stimulated neutrophil function via activation of cAMP-dependent protein kinase and Ser/Thr protein phosphatase.
    Cellular signalling, 2000, Volume: 12, Issue:5

    Topics: Adenosine; Amino Acid Sequence; Autoantigens; Calcium; Carbazoles; Chelating Agents; Collagen; Collagen Type IV; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Antagonists; Egtazic Acid; Enzyme Inhibitors; Estrenes; Humans; Indoles; Marine Toxins; Molecular Sequence Data; Neutrophils; Okadaic Acid; Oxazoles; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphoprotein Phosphatases; Pyrroles; Pyrrolidinones; Respiratory Burst; Signal Transduction; Thapsigargin; Trifluoperazine

2000
Evidence for a calcium-sensing receptor in the vascular smooth muscle cells of the spiral modiolar artery.
    The Journal of membrane biology, 2000, Jun-01, Volume: 175, Issue:3

    Topics: Arteries; Base Sequence; Calcium; Calcium Channel Blockers; Cations, Divalent; Cochlea; DNA, Complementary; Enzyme Inhibitors; Estrenes; Molecular Sequence Data; Muscle, Smooth, Vascular; Nickel; Nifedipine; Pyrrolidinones; Receptors, Calcium-Sensing; Receptors, Cell Surface; Ryanodine; Thapsigargin; Type C Phospholipases; Vasodilator Agents

2000
Bradykinin and angiotensin II-induced [Ca2+]i rise in cultured rat pituitary folliculo-stellate cells.
    Journal of neuroendocrinology, 2001, Volume: 13, Issue:11

    Topics: Angiotensin II; Animals; Bradykinin; Caffeine; Calcium; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Galanin; Male; Neuropeptides; Neurotensin; Phosphodiesterase Inhibitors; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Pyrrolidinones; Rats; Rats, Wistar; Ryanodine; Thapsigargin; Type C Phospholipases; Vasoconstrictor Agents

2001
Protease-activated receptor-2-mediated Ca2+ signaling in guinea pig tracheal epithelial cells.
    Life sciences, 2002, Jun-21, Volume: 71, Issue:5

    Topics: Animals; Calcium Signaling; Chelating Agents; Enzyme Inhibitors; Epithelial Cells; Estrenes; Fura-2; Guinea Pigs; Manganese; Oligopeptides; Pyrrolidinones; Receptor, PAR-2; Receptors, Thrombin; Thapsigargin; Trachea; Trypsin; Type C Phospholipases

2002
Mechanisms of bradykinin-induced glucagon release in clonal alpha-cells In-R1-G9: involvement of Ca(2+)-dependent and -independent pathways.
    Molecular and cellular endocrinology, 2002, Jun-28, Volume: 192, Issue:1-2

    Topics: Animals; Bradykinin; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Chelating Agents; Clone Cells; Cricetinae; Egtazic Acid; Endoplasmic Reticulum; Enzyme Inhibitors; Estrenes; Glucagon; Glucagonoma; GTP-Binding Proteins; Heparin; Imidazoles; Inositol 1,4,5-Trisphosphate Receptors; Mesocricetus; Microinjections; Pancreatic Neoplasms; Pertussis Toxin; Phospholipase D; Pyrrolidinones; Receptor, Bradykinin B2; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Thapsigargin; Tumor Cells, Cultured; Type C Phospholipases

2002
Requirement for intracellular calcium modulation in zebrafish dorsal-ventral patterning.
    Developmental biology, 2003, Jul-15, Volume: 259, Issue:2

    Topics: Animals; beta Catenin; Body Patterning; Calcium; Cytoskeletal Proteins; Diphosphonates; Dose-Response Relationship, Drug; Embryo, Nonmammalian; Enzyme Inhibitors; Estrenes; Gene Expression Regulation, Developmental; Models, Biological; Phenotype; Phosphatidylinositols; Pyrrolidinones; Signal Transduction; Thapsigargin; Trans-Activators; Type C Phospholipases; Zebrafish; Zebrafish Proteins

2003
Anatomical and functional evidence for a role of arginine-vasopressin (AVP) in rat olfactory epithelium cells.
    The European journal of neuroscience, 2004, Volume: 20, Issue:3

    Topics: Animals; Animals, Newborn; Arginine Vasopressin; Boron Compounds; Cadmium Chloride; Calcium; Calcium Channel Blockers; Cells, Cultured; Chelating Agents; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Estrenes; Extracellular Space; Fura-2; Immunohistochemistry; Male; Neurons; Olfactory Mucosa; Oxytocin; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Oxytocin; Receptors, Vasopressin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thapsigargin; Time Factors; Verapamil

2004
Nonylphenol-induced Ca2+ elevation and Ca2+-independent cell death in human osteosarcoma cells.
    Toxicology letters, 2005, Dec-30, Volume: 160, Issue:1

    Topics: Calcium; Calcium Channel Blockers; Cell Death; Cell Line, Tumor; Cell Proliferation; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; Estrenes; Fluorescent Dyes; Fura-2; Humans; Osteoblasts; Osteosarcoma; Phenols; Pyrrolidinones; Spectrometry, Fluorescence; Tetrazolium Salts; Thapsigargin; Type C Phospholipases

2005