Page last updated: 2024-09-02

u 73343 and arachidonic acid

u 73343 has been researched along with arachidonic acid in 4 studies

Compound Research Comparison

Studies
(u 73343)
Trials
(u 73343)
Recent Studies (post-2010)
(u 73343)
Studies
(arachidonic acid)
Trials
(arachidonic acid)
Recent Studies (post-2010) (arachidonic acid)
970619,2954863,040

Protein Interaction Comparison

ProteinTaxonomyu 73343 (IC50)arachidonic acid (IC50)
60 kDa heat shock protein, mitochondrialHomo sapiens (human)4.5
Fatty acid-binding protein, adipocyteHomo sapiens (human)2.75
10 kDa heat shock protein, mitochondrialHomo sapiens (human)4.5
60 kDa chaperonin Escherichia coli7.3
10 kDa chaperonin Escherichia coli7.3
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)1.0715
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)0.6026

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Farndale, RW; Heemskerk, JW; Sage, SO1
Arai, J; Okada, S; Shimizu, T; Wakiguchi, H; Yamaguchi, N; Yokotani, K1
Campbell, WB; Edwards, EM; Falck, JR; Holmes, BB; Tang, X1
George, S; Häfner, AK; Hofmann, B; Hörnig, M; Karas, M; Maier, T; Markoutsa, S; Rödl, CB; Steinhilber, D; Werz, O; Wisniewska, JM1

Other Studies

4 other study(ies) available for u 73343 and arachidonic acid

ArticleYear
Effects of U73122 and U73343 on human platelet calcium signalling and protein tyrosine phosphorylation.
    Biochimica et biophysica acta, 1997, Jan-10, Volume: 1355, Issue:1

    Topics: Arachidonic Acid; Aspirin; Blood Platelets; Blood Proteins; Calcium; Collagen; Estrenes; Humans; Phosphodiesterase Inhibitors; Phosphorylation; Phosphotyrosine; Protein-Tyrosine Kinases; Pyrrolidinones; Signal Transduction; Thapsigargin; Thrombin; Thromboxane A2; Type C Phospholipases

1997
Brain phospholipase C/diacylglycerol lipase are involved in bombesin BB2 receptor-mediated activation of sympatho-adrenomedullary outflow in rats.
    European journal of pharmacology, 2005, May-09, Volume: 514, Issue:2-3

    Topics: Adrenal Medulla; Animals; Arachidonic Acid; Bombesin; Brain; Cyclohexanones; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epinephrine; Estrenes; Gastrin-Releasing Peptide; Injections, Intraventricular; Lipoprotein Lipase; Male; Neurokinin B; Norepinephrine; Peptides, Cyclic; Phospholipases A; Phospholipases A2; Pyrrolidinones; Quinacrine; Rats; Rats, Wistar; Receptors, Bombesin; Sympathetic Nervous System; Type C Phospholipases

2005
Role of phospholipase C and diacylglyceride lipase pathway in arachidonic acid release and acetylcholine-induced vascular relaxation in rabbit aorta.
    American journal of physiology. Heart and circulatory physiology, 2006, Volume: 290, Issue:1

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Arachidonic Acid; Arachidonic Acids; Carbamates; Cells, Cultured; Cyclohexanones; Diazomethane; Endothelium, Vascular; Estrenes; In Vitro Techniques; Indomethacin; Isoenzymes; Lipoprotein Lipase; Methacholine Chloride; Nitroarginine; Phospholipases A; Phospholipases A2; Pyrrolidinones; Rabbits; Type C Phospholipases; Vasodilation

2006
Inhibition of 5-lipoxygenase by U73122 is due to covalent binding to cysteine 416.
    Biochimica et biophysica acta, 2012, Volume: 1821, Issue:2

    Topics: Adult; Animals; Arachidonate 5-Lipoxygenase; Arachidonic Acid; Cysteine; Estrenes; HeLa Cells; Humans; Lipoxygenase Inhibitors; Mice; Models, Molecular; Mutant Proteins; Protein Binding; Protein Structure, Secondary; Pyrrolidinones; Sequence Homology, Amino Acid; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Sulfhydryl Compounds

2012