Page last updated: 2024-08-26

u 73122 and piperidines

u 73122 has been researched along with piperidines in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (22.22)18.2507
2000's12 (44.44)29.6817
2010's9 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chung, FZ; Hill, DR; Madden, Z; Pinnock, RD; Suman-Chauhan, N; Webdale, L; Woodruff, GN1
Barrington, M; Kotsonis, P; Majewski, H; Murphy, TV1
Goodman, HM; McCullough, JR; Mitra, S; Ugur, M; Ugur, O; Yamaguchi, H1
Bell, MI; Lee, K; Richardson, PJ1
Kurz, T; Richardt, G; Schneider, I; Tölg, R1
Kato, K; Kawamura, H; Kozawa, O; Matsui, N; Matsuno, H; Niwa, M; Otsuka, T; Uematsu, T1
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L1
Trudeau, LE1
Boyd, DF; Mathie, A; Millar, JA; Watkins, CS1
Aragona, F; Malendowicz, LK; Nussdorfer, GG; Rebuffat, P; Tortorella, C1
Cabeza, R; Méndez-Díaz, M; Murillo-Rodríguez, E; Navarro, L; Prospéro-García, O1
Cheng, JS; Chou, KJ; Fang, HC; Jan, CR; Law, YP; Lee, KC; Su, W; Tseng, LL; Wang, JL1
Benard, V; Gendreau, S; Missy, K; Payrastre, B; Plantavid, M; Soulet, C1
Cheng, BL; Coy, DH; Datta, R; Rossowski, WJ; Taylor, JE1
Dirnagl, U; Dreier, JP; Kleeberg, J; Major, S; Petzold, GC1
Boon, A; Bridges, D; Deadwyler, SA; Grigorenko, E; Hampson, RE; McCloud, S; Zhuang, SY1
Hattori, M; Komori, S; Matsuyama, H; Nishimura, M; Sakamoto, T; Uchiyama, M; Unno, T1
Arai, S; Oka, S; Sugiura, T; Tokumura, A; Waku, K1
Campiglia, P; De Falco, V; Fenzi, G; Illario, M; Monaco, S; Pastore, L; Rossi, G; Rusciano, MR; Salzano, M; Santoro, M; Sapio, MR; Vitale, M1
Dietrich, A; Fuchs, B; Ghofrani, HA; Grimminger, F; Gudermann, T; Rupp, M; Schermuly, RT; Seeger, W; Weissmann, N1
Jiang, X; Qin, Z; Tao, J; Wang, F; Wang, J; Zhang, L; Zhang, Y1
Ashby, MC; Isaac, JT; Matta, JA; Roche, KW; Sanz-Clemente, A1
Chiou, LC; Fu, SY; Ho, YC; Lee, HJ; Liao, HT; Liao, YY; Mackie, K; Teng, SF; Tung, LW1
Brenowitz, SD; Sedlacek, M; Tipton, PW1
Nakamura, K; Shimizu, T; Tanaka, K; Taniuchi, K; Yokotani, K1
Conde, K; Kelly, MJ; Meza, C; Sinchak, K; Wagner, EJ1
Kamishikiryo, J; Morita, T; Nakamura, T1

Other Studies

27 other study(ies) available for u 73122 and piperidines

ArticleYear
Characterization of tachykinin mediated increases in [Ca2+]i in Chinese hamster ovary cells expressing human tachykinin NK3 receptors.
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: Animals; Benzamides; Calcium; Calcium-Transporting ATPases; CHO Cells; Cricetinae; Cricetulus; Estrenes; Fura-2; Humans; Inositol Phosphates; Manganese; Neurokinin A; Peptide Fragments; Piperidines; Pyrrolidinones; Receptors, Neurokinin-3; Ryanodine; Second Messenger Systems; Structure-Activity Relationship; Substance P; Tachykinins; Terpenes; Thapsigargin; Type C Phospholipases

1994
Noradrenaline release and the effect of endogenous activation of the phospholipase C/protein kinase C signalling pathway in rat atria.
    British journal of pharmacology, 1997, Volume: 121, Issue:6

    Topics: Androstadienes; Animals; Atrial Function; Diacylglycerol Kinase; Electric Stimulation; Enzyme Activation; Enzyme Inhibitors; Estrenes; Heart Atria; Male; Norepinephrine; Phosphotransferases (Alcohol Group Acceptor); Piperidines; Protein Kinase C; Pyrrolidinones; Quinazolines; Quinazolinones; Rats; Rats, Sprague-Dawley; Signal Transduction; Type C Phospholipases; Wortmannin

1997
(S)-Albuterol increases intracellular free calcium by muscarinic receptor activation and a phospholipase C-dependent mechanism in airway smooth muscle.
    Molecular pharmacology, 1998, Volume: 53, Issue:3

    Topics: Adrenergic beta-Agonists; Albuterol; Animals; Calcium; Cattle; Estrenes; Piperidines; Propanolamines; Pyrrolidinones; Receptors, Muscarinic; Stereoisomerism; Trachea; Type C Phospholipases

1998
Characterization of the mechanism of action of tachykinins in rat striatal cholinergic interneurons.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Chelating Agents; Corpus Striatum; Diazonium Compounds; Electric Stimulation; Estrenes; Excitatory Amino Acid Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Interneurons; Male; Membrane Potentials; Patch-Clamp Techniques; Phenoxyacetates; Phosphodiesterase Inhibitors; Photochemistry; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tachykinins; Tetrodotoxin

1998
Alpha 1-adrenergic receptor-mediated increase in the mass of phosphatidic acid and 1,2-diacylglycerol in ischemic rat heart.
    Cardiovascular research, 1999, Volume: 42, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Analysis of Variance; Animals; Chromatography, Thin Layer; Desipramine; Diacylglycerol Kinase; Diglycerides; Estrenes; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Norepinephrine; Perfusion; Phosphatidic Acids; Piperidines; Prazosin; Propranolol; Pyrrolidinones; Quinazolines; Quinazolinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Time Factors; Type C Phospholipases

1999
Endothelin-1 stimulates heat shock protein 27 induction in osteoblasts: involvement of p38 MAP kinase.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Animals; Antihypertensive Agents; Blotting, Northern; Carcinogens; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation, Enzymologic; Genistein; Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Oligopeptides; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phorbol Esters; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Propranolol; Protein Kinase C; Pyridines; Pyrrolidinones; RNA, Messenger; Skull; Staurosporine

1999
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium

2000
Neurotensin regulates intracellular calcium in ventral tegmental area astrocytes: evidence for the involvement of multiple receptors.
    Neuroscience, 2000, Volume: 97, Issue:2

    Topics: Adamantane; Animals; Animals, Newborn; Astrocytes; Calcium; Cells, Cultured; Estrenes; Gadolinium; Imidazoles; Neurotensin; Peptide Fragments; Piperidines; Pyrrolidinones; Rats; Receptors, Neurotensin; Thapsigargin; Type C Phospholipases; Ventral Tegmental Area

2000
The role of Ca2+ stores in the muscarinic inhibition of the K+ current IK(SO) in neonatal rat cerebellar granule cells.
    The Journal of physiology, 2000, Dec-01, Volume: 529 Pt 2

    Topics: Animals; Animals, Newborn; Calcium; Calcium Signaling; Cells, Cultured; Cerebellum; Chelating Agents; Dioxoles; Egtazic Acid; Electric Conductivity; Estrenes; Female; Male; Membrane Potentials; Muscarinic Antagonists; Piperidines; Potassium; Potassium Channels; Protein Isoforms; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M3; Receptors, Muscarinic; Thapsigargin

2000
Signaling pathways involved in the A and B receptor-mediated cortisol secretagogue effect of endothelins in the human adrenal cortex.
    International journal of molecular medicine, 2001, Volume: 7, Issue:3

    Topics: Adenine; Androstadienes; Cells, Cultured; Endothelin Receptor Antagonists; Endothelins; Enzyme Inhibitors; Estrenes; Flavonoids; Humans; Hydrocortisone; Indomethacin; Naphthalenes; Nifedipine; Oligopeptides; Peptides, Cyclic; Phosphoinositide-3 Kinase Inhibitors; Piperidines; Protein Kinase C; Pyrazoles; Pyrrolidinones; Receptors, Endothelin; Signal Transduction; Type C Phospholipases; Tyrphostins; Wortmannin; Zona Fasciculata; Zona Reticularis

2001
Anandamide-induced sleep is blocked by SR141716A, a CB1 receptor antagonist and by U73122, a phospholipase C inhibitor.
    Neuroreport, 2001, Jul-20, Volume: 12, Issue:10

    Topics: Animals; Arachidonic Acids; Cannabinoids; Endocannabinoids; Estrenes; Injections, Intraventricular; Male; Phosphodiesterase Inhibitors; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Sleep Stages; Type C Phospholipases; Ventral Tegmental Area

2001
CP55,940 increases intracellular Ca2+ levels in Madin-Darby canine kidney cells.
    Life sciences, 2001, Aug-17, Volume: 69, Issue:13

    Topics: Animals; Calcium; Cannabinoids; Cell Line; Cyclohexanols; Dogs; Estrenes; Extracellular Space; Indicators and Reagents; Inositol 1,4,5-Trisphosphate; Kidney; Morpholines; Piperidines; Pyrazoles; Pyrrolidinones; Receptors, Cannabinoid; Receptors, Drug

2001
Characterisation of Rac activation in thrombin- and collagen-stimulated human blood platelets.
    FEBS letters, 2001, Nov-02, Volume: 507, Issue:3

    Topics: Benzylamines; Blood Platelets; Calcium; cdc42 GTP-Binding Protein; Cells, Cultured; Chromones; Collagen; Enzyme Activation; Enzyme Inhibitors; Epoprostenol; Estrenes; Humans; Indoles; Morpholines; Oligopeptides; p21-Activated Kinases; Phosphatidylinositol 3-Kinases; Piperidines; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Kinase C; Protein Serine-Threonine Kinases; Pyrrolidinones; rac GTP-Binding Proteins; Thiazoles; Thrombin; Type C Phospholipases

2001
Human urotensin II-induced aorta ring contractions are mediated by protein kinase C, tyrosine kinases and Rho-kinase: inhibition by somatostatin receptor antagonists.
    European journal of pharmacology, 2002, Mar-08, Volume: 438, Issue:3

    Topics: Alkaloids; Animals; Aorta, Thoracic; Benzophenanthridines; Calcium Channel Blockers; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Genistein; Humans; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Peptide Fragments; Peptides, Cyclic; Phenanthridines; Piperidines; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Somatostatin; rho-Associated Kinases; Tyrphostins; Urotensins; Vasoconstriction

2002
ET-1 induces cortical spreading depression via activation of the ETA receptor/phospholipase C pathway in vivo.
    American journal of physiology. Heart and circulatory physiology, 2004, Volume: 286, Issue:4

    Topics: Animals; Arachidonic Acid; Astrocytes; Cell Communication; Cortical Spreading Depression; Endothelin A Receptor Antagonists; Endothelin-1; Endothelins; Estrenes; Male; Muscle, Smooth, Vascular; Oligopeptides; Parietal Lobe; Peptide Fragments; Peptides, Cyclic; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Rats; Rats, Wistar; Receptor, Endothelin A; Signal Transduction; Type C Phospholipases

2004
Cannabinoids produce neuroprotection by reducing intracellular calcium release from ryanodine-sensitive stores.
    Neuropharmacology, 2005, Volume: 48, Issue:8

    Topics: Animals; Benzoxazines; Calcium; Cell Culture Techniques; Cell Death; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclohexanols; Dantrolene; Drug Interactions; Estrenes; Fetus; Hippocampus; Macrocyclic Compounds; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Neuroprotective Agents; Okadaic Acid; Oxazoles; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptor, Cannabinoid, CB1; Rimonabant; Ryanodine; Thionucleotides

2005
Characterization of muscarinic receptor-mediated cationic currents in longitudinal smooth muscle cells of mouse small intestine.
    Journal of pharmacological sciences, 2006, Volume: 100, Issue:3

    Topics: Animals; Carbachol; Cations; Cholinergic Agonists; Diamines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Guinea Pigs; In Vitro Techniques; Intestine, Small; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Mice; Muscarinic Antagonists; Myocytes, Smooth Muscle; Pertussis Toxin; Piperidines; Pyrrolidinones; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Type C Phospholipases

2006
Depolarization-induced rapid generation of 2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand, in rat brain synaptosomes.
    Journal of biochemistry, 2007, Volume: 141, Issue:5

    Topics: Animals; Arachidonic Acids; Brain; Calcimycin; Calcium Channel Blockers; Camphanes; Diglycerides; Endocannabinoids; Estrenes; Fatty Acids; Glycerides; Male; Membrane Potentials; Neuromuscular Depolarizing Agents; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Cannabinoid; Rimonabant; Synaptosomes

2007
The Ca2+-calmodulin-dependent kinase II is activated in papillary thyroid carcinoma (PTC) and mediates cell proliferation stimulated by RET/PTC.
    Endocrine-related cancer, 2010, Volume: 17, Issue:1

    Topics: Amino Acid Sequence; Animals; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calmodulin; Carcinoma, Papillary; Cell Division; Enzyme Activation; Estrenes; Extracellular Signal-Regulated MAP Kinases; Humans; MAP Kinase Signaling System; Molecular Sequence Data; Mutation; Neoplasm Proteins; Oncogene Protein p21(ras); Piperidines; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-ret; Pyrrolidinones; Quinazolines; Rats; Thyroid Neoplasms; Type C Phospholipases

2010
Diacylglycerol regulates acute hypoxic pulmonary vasoconstriction via TRPC6.
    Respiratory research, 2011, Feb-04, Volume: 12

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Diacylglycerol Kinase; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Hypoxia; In Vitro Techniques; Lung; Mice; Mice, Inbred C57BL; Mice, Knockout; Perfusion; Piperidines; Pulmonary Circulation; Pyrrolidinones; Quinazolinones; Signal Transduction; Time Factors; TRPC Cation Channels; TRPC6 Cation Channel; Type C Phospholipases; Vasoconstriction; Vasoconstrictor Agents

2011
Activation of M3 muscarinic receptors inhibits T-type Ca(2+) channel currents via pertussis toxin-sensitive novel protein kinase C pathway in small dorsal root ganglion neurons.
    Cellular signalling, 2011, Volume: 23, Issue:6

    Topics: Animals; Calcium Channels, T-Type; Calcium Signaling; Cholera Toxin; Cobra Neurotoxin Proteins; Estrenes; Ganglia, Spinal; Indoles; Maleimides; Mice; Mice, Inbred ICR; Muscarinic Antagonists; Neurons; Pain Measurement; Pertussis Toxin; Piperidines; Protein Kinase C; Pyrrolidinones; Receptor, Muscarinic M3; Type C Phospholipases

2011
mGluR5 and NMDA receptors drive the experience- and activity-dependent NMDA receptor NR2B to NR2A subunit switch.
    Neuron, 2011, Apr-28, Volume: 70, Issue:2

    Topics: Adaptation, Physiological; Animals; Animals, Newborn; Electric Stimulation; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Knockout; Models, Biological; N-Methylaspartate; Piperidines; Pyramidal Cells; Pyridines; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synapses; Thiazoles; Time Factors; Visual Cortex

2011
Activation of orexin 1 receptors in the periaqueductal gray of male rats leads to antinociception via retrograde endocannabinoid (2-arachidonoylglycerol)-induced disinhibition.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Oct-12, Volume: 31, Issue:41

    Topics: Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Benzoxazoles; Biphenyl Compounds; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Disease Models, Animal; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Intracellular Signaling Peptides and Proteins; Lactones; Male; Morpholines; Naphthalenes; Naphthyridines; Neural Inhibition; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Orlistat; Pain; Pain Measurement; Patch-Clamp Techniques; Periaqueductal Gray; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea

2011
Sustained firing of cartwheel cells in the dorsal cochlear nucleus evokes endocannabinoid release and retrograde suppression of parallel fiber synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Nov-02, Volume: 31, Issue:44

    Topics: Action Potentials; Anesthetics, Local; Animals; Animals, Newborn; Biophysics; Calcium; Cannabinoid Receptor Modulators; Cochlear Nucleus; Dendrites; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; In Vitro Techniques; Male; Mice; Mice, Inbred CBA; Mice, Inbred ICR; Nerve Fibers; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Piperidines; Pyrazoles; Pyrrolidinones; Quinoxalines; Refractory Period, Electrophysiological; Synaptic Transmission; Tetrodotoxin; Time Factors

2011
Brain phospholipase C, diacylglycerol lipase and monoacylglycerol lipase are involved in (±)-epibatidine-induced activation of central adrenomedullary outflow in rats.
    European journal of pharmacology, 2012, Sep-15, Volume: 691, Issue:1-3

    Topics: Adrenal Medulla; Animals; Arachidonic Acids; Benzodioxoles; Brain; Bridged Bicyclo Compounds, Heterocyclic; Catecholamines; Cyclohexanones; Esterases; Estrenes; Lipoprotein Lipase; Male; Monoacylglycerol Lipases; Neurons; Nicotinic Agonists; Organophosphonates; Paraventricular Hypothalamic Nucleus; Piperidines; Pyridines; Pyrrolidinones; Rats; Rats, Wistar; Type C Phospholipases

2012
Estradiol Rapidly Attenuates ORL-1 Receptor-Mediated Inhibition of Proopiomelanocortin Neurons via Gq-Coupled, Membrane-Initiated Signaling.
    Neuroendocrinology, 2016, Volume: 103, Issue:6

    Topics: Animals; Drug Interactions; Enzyme Inhibitors; Estradiol; Estrenes; Estrogens; Female; Hypothalamus; In Vitro Techniques; Membrane Potentials; Neurons; Nociceptin; Nociceptin Receptor; Opioid Peptides; Ovariectomy; Piperidines; Pro-Opiomelanocortin; Pyrrolidinones; Rats; Rats, Long-Evans; Receptors, Opioid; Signal Transduction; Sodium Channel Blockers; Stilbamidines; Tetrodotoxin

2016
Prazosin-stimulated release of hepatic triacylglyceride lipase from primary cultured rat hepatocytes is involved in the regulation of cAMP-dependent protein kinase through activation of the Ca(2+)/calmodulin-dependent protein kinase-II.
    Pharmacological reports : PR, 2016, Volume: 68, Issue:3

    Topics: Animals; Benzophenanthridines; Benzylamines; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Estrenes; Hepatocytes; Lipoprotein Lipase; Macrocyclic Compounds; Male; Oxazoles; Piperidines; Prazosin; Primary Cell Culture; Pyrrolidinones; Quinazolinones; Rats; Sulfonamides; Time Factors; Trifluoperazine

2016