u 73122 has been researched along with piperidines in 27 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (22.22) | 18.2507 |
2000's | 12 (44.44) | 29.6817 |
2010's | 9 (33.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Chung, FZ; Hill, DR; Madden, Z; Pinnock, RD; Suman-Chauhan, N; Webdale, L; Woodruff, GN | 1 |
Barrington, M; Kotsonis, P; Majewski, H; Murphy, TV | 1 |
Goodman, HM; McCullough, JR; Mitra, S; Ugur, M; Ugur, O; Yamaguchi, H | 1 |
Bell, MI; Lee, K; Richardson, PJ | 1 |
Kurz, T; Richardt, G; Schneider, I; Tölg, R | 1 |
Kato, K; Kawamura, H; Kozawa, O; Matsui, N; Matsuno, H; Niwa, M; Otsuka, T; Uematsu, T | 1 |
Lee, K; Pinnock, RD; Preston, Z; Richardson, PJ; Widdowson, L | 1 |
Trudeau, LE | 1 |
Boyd, DF; Mathie, A; Millar, JA; Watkins, CS | 1 |
Aragona, F; Malendowicz, LK; Nussdorfer, GG; Rebuffat, P; Tortorella, C | 1 |
Cabeza, R; Méndez-Díaz, M; Murillo-Rodríguez, E; Navarro, L; Prospéro-García, O | 1 |
Cheng, JS; Chou, KJ; Fang, HC; Jan, CR; Law, YP; Lee, KC; Su, W; Tseng, LL; Wang, JL | 1 |
Benard, V; Gendreau, S; Missy, K; Payrastre, B; Plantavid, M; Soulet, C | 1 |
Cheng, BL; Coy, DH; Datta, R; Rossowski, WJ; Taylor, JE | 1 |
Dirnagl, U; Dreier, JP; Kleeberg, J; Major, S; Petzold, GC | 1 |
Boon, A; Bridges, D; Deadwyler, SA; Grigorenko, E; Hampson, RE; McCloud, S; Zhuang, SY | 1 |
Hattori, M; Komori, S; Matsuyama, H; Nishimura, M; Sakamoto, T; Uchiyama, M; Unno, T | 1 |
Arai, S; Oka, S; Sugiura, T; Tokumura, A; Waku, K | 1 |
Campiglia, P; De Falco, V; Fenzi, G; Illario, M; Monaco, S; Pastore, L; Rossi, G; Rusciano, MR; Salzano, M; Santoro, M; Sapio, MR; Vitale, M | 1 |
Dietrich, A; Fuchs, B; Ghofrani, HA; Grimminger, F; Gudermann, T; Rupp, M; Schermuly, RT; Seeger, W; Weissmann, N | 1 |
Jiang, X; Qin, Z; Tao, J; Wang, F; Wang, J; Zhang, L; Zhang, Y | 1 |
Ashby, MC; Isaac, JT; Matta, JA; Roche, KW; Sanz-Clemente, A | 1 |
Chiou, LC; Fu, SY; Ho, YC; Lee, HJ; Liao, HT; Liao, YY; Mackie, K; Teng, SF; Tung, LW | 1 |
Brenowitz, SD; Sedlacek, M; Tipton, PW | 1 |
Nakamura, K; Shimizu, T; Tanaka, K; Taniuchi, K; Yokotani, K | 1 |
Conde, K; Kelly, MJ; Meza, C; Sinchak, K; Wagner, EJ | 1 |
Kamishikiryo, J; Morita, T; Nakamura, T | 1 |
27 other study(ies) available for u 73122 and piperidines
Article | Year |
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Characterization of tachykinin mediated increases in [Ca2+]i in Chinese hamster ovary cells expressing human tachykinin NK3 receptors.
Topics: Animals; Benzamides; Calcium; Calcium-Transporting ATPases; CHO Cells; Cricetinae; Cricetulus; Estrenes; Fura-2; Humans; Inositol Phosphates; Manganese; Neurokinin A; Peptide Fragments; Piperidines; Pyrrolidinones; Receptors, Neurokinin-3; Ryanodine; Second Messenger Systems; Structure-Activity Relationship; Substance P; Tachykinins; Terpenes; Thapsigargin; Type C Phospholipases | 1994 |
Noradrenaline release and the effect of endogenous activation of the phospholipase C/protein kinase C signalling pathway in rat atria.
Topics: Androstadienes; Animals; Atrial Function; Diacylglycerol Kinase; Electric Stimulation; Enzyme Activation; Enzyme Inhibitors; Estrenes; Heart Atria; Male; Norepinephrine; Phosphotransferases (Alcohol Group Acceptor); Piperidines; Protein Kinase C; Pyrrolidinones; Quinazolines; Quinazolinones; Rats; Rats, Sprague-Dawley; Signal Transduction; Type C Phospholipases; Wortmannin | 1997 |
(S)-Albuterol increases intracellular free calcium by muscarinic receptor activation and a phospholipase C-dependent mechanism in airway smooth muscle.
Topics: Adrenergic beta-Agonists; Albuterol; Animals; Calcium; Cattle; Estrenes; Piperidines; Propanolamines; Pyrrolidinones; Receptors, Muscarinic; Stereoisomerism; Trachea; Type C Phospholipases | 1998 |
Characterization of the mechanism of action of tachykinins in rat striatal cholinergic interneurons.
Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Chelating Agents; Corpus Striatum; Diazonium Compounds; Electric Stimulation; Estrenes; Excitatory Amino Acid Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Interneurons; Male; Membrane Potentials; Patch-Clamp Techniques; Phenoxyacetates; Phosphodiesterase Inhibitors; Photochemistry; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tachykinins; Tetrodotoxin | 1998 |
Alpha 1-adrenergic receptor-mediated increase in the mass of phosphatidic acid and 1,2-diacylglycerol in ischemic rat heart.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Analysis of Variance; Animals; Chromatography, Thin Layer; Desipramine; Diacylglycerol Kinase; Diglycerides; Estrenes; Male; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Norepinephrine; Perfusion; Phosphatidic Acids; Piperidines; Prazosin; Propranolol; Pyrrolidinones; Quinazolines; Quinazolinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Time Factors; Type C Phospholipases | 1999 |
Endothelin-1 stimulates heat shock protein 27 induction in osteoblasts: involvement of p38 MAP kinase.
Topics: Animals; Antihypertensive Agents; Blotting, Northern; Carcinogens; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation, Enzymologic; Genistein; Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Oligopeptides; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phorbol Esters; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Propranolol; Protein Kinase C; Pyridines; Pyrrolidinones; RNA, Messenger; Skull; Staurosporine | 1999 |
Tachykinins increase [3H]acetylcholine release in mouse striatum through multiple receptor subtypes.
Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Choline O-Acetyltransferase; Corpus Striatum; Electrophysiology; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; In Situ Hybridization; Indoles; Interneurons; Membrane Potentials; Mice; Mice, Inbred C57BL; Neurokinin A; Oligopeptides; omega-N-Methylarginine; Peptide Fragments; Phenanthridines; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; RNA, Messenger; Signal Transduction; Substance P; Tachykinins; Tetrodotoxin; Tritium | 2000 |
Neurotensin regulates intracellular calcium in ventral tegmental area astrocytes: evidence for the involvement of multiple receptors.
Topics: Adamantane; Animals; Animals, Newborn; Astrocytes; Calcium; Cells, Cultured; Estrenes; Gadolinium; Imidazoles; Neurotensin; Peptide Fragments; Piperidines; Pyrrolidinones; Rats; Receptors, Neurotensin; Thapsigargin; Type C Phospholipases; Ventral Tegmental Area | 2000 |
The role of Ca2+ stores in the muscarinic inhibition of the K+ current IK(SO) in neonatal rat cerebellar granule cells.
Topics: Animals; Animals, Newborn; Calcium; Calcium Signaling; Cells, Cultured; Cerebellum; Chelating Agents; Dioxoles; Egtazic Acid; Electric Conductivity; Estrenes; Female; Male; Membrane Potentials; Muscarinic Antagonists; Piperidines; Potassium; Potassium Channels; Protein Isoforms; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M3; Receptors, Muscarinic; Thapsigargin | 2000 |
Signaling pathways involved in the A and B receptor-mediated cortisol secretagogue effect of endothelins in the human adrenal cortex.
Topics: Adenine; Androstadienes; Cells, Cultured; Endothelin Receptor Antagonists; Endothelins; Enzyme Inhibitors; Estrenes; Flavonoids; Humans; Hydrocortisone; Indomethacin; Naphthalenes; Nifedipine; Oligopeptides; Peptides, Cyclic; Phosphoinositide-3 Kinase Inhibitors; Piperidines; Protein Kinase C; Pyrazoles; Pyrrolidinones; Receptors, Endothelin; Signal Transduction; Type C Phospholipases; Tyrphostins; Wortmannin; Zona Fasciculata; Zona Reticularis | 2001 |
Anandamide-induced sleep is blocked by SR141716A, a CB1 receptor antagonist and by U73122, a phospholipase C inhibitor.
Topics: Animals; Arachidonic Acids; Cannabinoids; Endocannabinoids; Estrenes; Injections, Intraventricular; Male; Phosphodiesterase Inhibitors; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Sleep Stages; Type C Phospholipases; Ventral Tegmental Area | 2001 |
CP55,940 increases intracellular Ca2+ levels in Madin-Darby canine kidney cells.
Topics: Animals; Calcium; Cannabinoids; Cell Line; Cyclohexanols; Dogs; Estrenes; Extracellular Space; Indicators and Reagents; Inositol 1,4,5-Trisphosphate; Kidney; Morpholines; Piperidines; Pyrazoles; Pyrrolidinones; Receptors, Cannabinoid; Receptors, Drug | 2001 |
Characterisation of Rac activation in thrombin- and collagen-stimulated human blood platelets.
Topics: Benzylamines; Blood Platelets; Calcium; cdc42 GTP-Binding Protein; Cells, Cultured; Chromones; Collagen; Enzyme Activation; Enzyme Inhibitors; Epoprostenol; Estrenes; Humans; Indoles; Morpholines; Oligopeptides; p21-Activated Kinases; Phosphatidylinositol 3-Kinases; Piperidines; Platelet Aggregation Inhibitors; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Kinase C; Protein Serine-Threonine Kinases; Pyrrolidinones; rac GTP-Binding Proteins; Thiazoles; Thrombin; Type C Phospholipases | 2001 |
Human urotensin II-induced aorta ring contractions are mediated by protein kinase C, tyrosine kinases and Rho-kinase: inhibition by somatostatin receptor antagonists.
Topics: Alkaloids; Animals; Aorta, Thoracic; Benzophenanthridines; Calcium Channel Blockers; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Genistein; Humans; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Peptide Fragments; Peptides, Cyclic; Phenanthridines; Piperidines; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptors, Somatostatin; rho-Associated Kinases; Tyrphostins; Urotensins; Vasoconstriction | 2002 |
ET-1 induces cortical spreading depression via activation of the ETA receptor/phospholipase C pathway in vivo.
Topics: Animals; Arachidonic Acid; Astrocytes; Cell Communication; Cortical Spreading Depression; Endothelin A Receptor Antagonists; Endothelin-1; Endothelins; Estrenes; Male; Muscle, Smooth, Vascular; Oligopeptides; Parietal Lobe; Peptide Fragments; Peptides, Cyclic; Phosphodiesterase Inhibitors; Piperidines; Pyrrolidinones; Rats; Rats, Wistar; Receptor, Endothelin A; Signal Transduction; Type C Phospholipases | 2004 |
Cannabinoids produce neuroprotection by reducing intracellular calcium release from ryanodine-sensitive stores.
Topics: Animals; Benzoxazines; Calcium; Cell Culture Techniques; Cell Death; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclohexanols; Dantrolene; Drug Interactions; Estrenes; Fetus; Hippocampus; Macrocyclic Compounds; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Neuroprotective Agents; Okadaic Acid; Oxazoles; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptor, Cannabinoid, CB1; Rimonabant; Ryanodine; Thionucleotides | 2005 |
Characterization of muscarinic receptor-mediated cationic currents in longitudinal smooth muscle cells of mouse small intestine.
Topics: Animals; Carbachol; Cations; Cholinergic Agonists; Diamines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Guinea Pigs; In Vitro Techniques; Intestine, Small; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Mice; Muscarinic Antagonists; Myocytes, Smooth Muscle; Pertussis Toxin; Piperidines; Pyrrolidinones; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Type C Phospholipases | 2006 |
Depolarization-induced rapid generation of 2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand, in rat brain synaptosomes.
Topics: Animals; Arachidonic Acids; Brain; Calcimycin; Calcium Channel Blockers; Camphanes; Diglycerides; Endocannabinoids; Estrenes; Fatty Acids; Glycerides; Male; Membrane Potentials; Neuromuscular Depolarizing Agents; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Cannabinoid; Rimonabant; Synaptosomes | 2007 |
The Ca2+-calmodulin-dependent kinase II is activated in papillary thyroid carcinoma (PTC) and mediates cell proliferation stimulated by RET/PTC.
Topics: Amino Acid Sequence; Animals; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calmodulin; Carcinoma, Papillary; Cell Division; Enzyme Activation; Estrenes; Extracellular Signal-Regulated MAP Kinases; Humans; MAP Kinase Signaling System; Molecular Sequence Data; Mutation; Neoplasm Proteins; Oncogene Protein p21(ras); Piperidines; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-ret; Pyrrolidinones; Quinazolines; Rats; Thyroid Neoplasms; Type C Phospholipases | 2010 |
Diacylglycerol regulates acute hypoxic pulmonary vasoconstriction via TRPC6.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Diacylglycerol Kinase; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Hypoxia; In Vitro Techniques; Lung; Mice; Mice, Inbred C57BL; Mice, Knockout; Perfusion; Piperidines; Pulmonary Circulation; Pyrrolidinones; Quinazolinones; Signal Transduction; Time Factors; TRPC Cation Channels; TRPC6 Cation Channel; Type C Phospholipases; Vasoconstriction; Vasoconstrictor Agents | 2011 |
Activation of M3 muscarinic receptors inhibits T-type Ca(2+) channel currents via pertussis toxin-sensitive novel protein kinase C pathway in small dorsal root ganglion neurons.
Topics: Animals; Calcium Channels, T-Type; Calcium Signaling; Cholera Toxin; Cobra Neurotoxin Proteins; Estrenes; Ganglia, Spinal; Indoles; Maleimides; Mice; Mice, Inbred ICR; Muscarinic Antagonists; Neurons; Pain Measurement; Pertussis Toxin; Piperidines; Protein Kinase C; Pyrrolidinones; Receptor, Muscarinic M3; Type C Phospholipases | 2011 |
mGluR5 and NMDA receptors drive the experience- and activity-dependent NMDA receptor NR2B to NR2A subunit switch.
Topics: Adaptation, Physiological; Animals; Animals, Newborn; Electric Stimulation; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Knockout; Models, Biological; N-Methylaspartate; Piperidines; Pyramidal Cells; Pyridines; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synapses; Thiazoles; Time Factors; Visual Cortex | 2011 |
Activation of orexin 1 receptors in the periaqueductal gray of male rats leads to antinociception via retrograde endocannabinoid (2-arachidonoylglycerol)-induced disinhibition.
Topics: Analysis of Variance; Animals; Animals, Newborn; Arachidonic Acids; Benzoxazines; Benzoxazoles; Biphenyl Compounds; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Disease Models, Animal; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; gamma-Aminobutyric Acid; Glycerides; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Intracellular Signaling Peptides and Proteins; Lactones; Male; Morpholines; Naphthalenes; Naphthyridines; Neural Inhibition; Neural Pathways; Neuropeptides; Orexin Receptors; Orexins; Orlistat; Pain; Pain Measurement; Patch-Clamp Techniques; Periaqueductal Gray; Piperidines; Pyrazoles; Pyrrolidinones; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Urea | 2011 |
Sustained firing of cartwheel cells in the dorsal cochlear nucleus evokes endocannabinoid release and retrograde suppression of parallel fiber synapses.
Topics: Action Potentials; Anesthetics, Local; Animals; Animals, Newborn; Biophysics; Calcium; Cannabinoid Receptor Modulators; Cochlear Nucleus; Dendrites; Electric Stimulation; Endocannabinoids; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; In Vitro Techniques; Male; Mice; Mice, Inbred CBA; Mice, Inbred ICR; Nerve Fibers; Neural Inhibition; Neurons; Patch-Clamp Techniques; Picrotoxin; Piperidines; Pyrazoles; Pyrrolidinones; Quinoxalines; Refractory Period, Electrophysiological; Synaptic Transmission; Tetrodotoxin; Time Factors | 2011 |
Brain phospholipase C, diacylglycerol lipase and monoacylglycerol lipase are involved in (±)-epibatidine-induced activation of central adrenomedullary outflow in rats.
Topics: Adrenal Medulla; Animals; Arachidonic Acids; Benzodioxoles; Brain; Bridged Bicyclo Compounds, Heterocyclic; Catecholamines; Cyclohexanones; Esterases; Estrenes; Lipoprotein Lipase; Male; Monoacylglycerol Lipases; Neurons; Nicotinic Agonists; Organophosphonates; Paraventricular Hypothalamic Nucleus; Piperidines; Pyridines; Pyrrolidinones; Rats; Rats, Wistar; Type C Phospholipases | 2012 |
Estradiol Rapidly Attenuates ORL-1 Receptor-Mediated Inhibition of Proopiomelanocortin Neurons via Gq-Coupled, Membrane-Initiated Signaling.
Topics: Animals; Drug Interactions; Enzyme Inhibitors; Estradiol; Estrenes; Estrogens; Female; Hypothalamus; In Vitro Techniques; Membrane Potentials; Neurons; Nociceptin; Nociceptin Receptor; Opioid Peptides; Ovariectomy; Piperidines; Pro-Opiomelanocortin; Pyrrolidinones; Rats; Rats, Long-Evans; Receptors, Opioid; Signal Transduction; Sodium Channel Blockers; Stilbamidines; Tetrodotoxin | 2016 |
Prazosin-stimulated release of hepatic triacylglyceride lipase from primary cultured rat hepatocytes is involved in the regulation of cAMP-dependent protein kinase through activation of the Ca(2+)/calmodulin-dependent protein kinase-II.
Topics: Animals; Benzophenanthridines; Benzylamines; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Estrenes; Hepatocytes; Lipoprotein Lipase; Macrocyclic Compounds; Male; Oxazoles; Piperidines; Prazosin; Primary Cell Culture; Pyrrolidinones; Quinazolinones; Rats; Sulfonamides; Time Factors; Trifluoperazine | 2016 |